DK220386D0 - 2-(4-benzoyl-1-piperidinyl)-alkanolderivater, fremgangsmaade til fremstilling af saadanne derivater og anvendelse af disse som laegemidler - Google Patents

2-(4-benzoyl-1-piperidinyl)-alkanolderivater, fremgangsmaade til fremstilling af saadanne derivater og anvendelse af disse som laegemidler

Info

Publication number: DK220386D0
Authority: DK; Denmark
Prior art keywords: derivatives; piperidinyl; pharmaceuticals; benzoyl; procedures
Prior art date: 1985-05-14

Application number

DK220386A

Other languages

English (en)

Other versions

DK220386A (da

Inventor

Bernard Gaudilliere

Jean Rousseau

Original Assignee

Synthelabo

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

1985-05-14

Filing date

1986-05-13

Publication date

1986-05-13

1986-05-13 Application filed by Synthelabo filed Critical Synthelabo

1986-05-13 Publication of DK220386D0 publication Critical patent/DK220386D0/da

1986-11-15 Publication of DK220386A publication Critical patent/DK220386A/da

Classifications

- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D211/00—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings
- C07D211/04—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom
- C07D211/06—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members
- C07D211/36—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D211/60—Carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals
- C07D211/62—Carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals attached in position 4
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D211/00—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings
- C07D211/04—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom
- C07D211/06—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members
- C07D211/08—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members with hydrocarbon or substituted hydrocarbon radicals directly attached to ring carbon atoms
- C07D211/18—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members with hydrocarbon or substituted hydrocarbon radicals directly attached to ring carbon atoms with substituted hydrocarbon radicals attached to ring carbon atoms
- C07D211/30—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members with hydrocarbon or substituted hydrocarbon radicals directly attached to ring carbon atoms with substituted hydrocarbon radicals attached to ring carbon atoms with hydrocarbon radicals, substituted by doubly bound oxygen or sulfur atoms or by two oxygen or sulfur atoms singly bound to the same carbon atom
- C07D211/32—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members with hydrocarbon or substituted hydrocarbon radicals directly attached to ring carbon atoms with substituted hydrocarbon radicals attached to ring carbon atoms with hydrocarbon radicals, substituted by doubly bound oxygen or sulfur atoms or by two oxygen or sulfur atoms singly bound to the same carbon atom by oxygen atoms
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/28—Drugs for disorders of the nervous system for treating neurodegenerative disorders of the central nervous system, e.g. nootropic agents, cognition enhancers, drugs for treating Alzheimer's disease or other forms of dementia
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
- A61P9/08—Vasodilators for multiple indications

Landscapes

Chemical & Material Sciences (AREA)
Organic Chemistry (AREA)
Health & Medical Sciences (AREA)
Engineering & Computer Science (AREA)
Bioinformatics & Cheminformatics (AREA)
General Health & Medical Sciences (AREA)
Veterinary Medicine (AREA)
General Chemical & Material Sciences (AREA)
Medicinal Chemistry (AREA)
Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
Neurosurgery (AREA)
Pharmacology & Pharmacy (AREA)
Life Sciences & Earth Sciences (AREA)
Animal Behavior & Ethology (AREA)
Neurology (AREA)
Public Health (AREA)
Chemical Kinetics & Catalysis (AREA)
Biomedical Technology (AREA)
Hospice & Palliative Care (AREA)
Cardiology (AREA)
Heart & Thoracic Surgery (AREA)
Psychiatry (AREA)
Hydrogenated Pyridines (AREA)
Plural Heterocyclic Compounds (AREA)
Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
Organic Insulating Materials (AREA)
Compositions Of Macromolecular Compounds (AREA)
Steroid Compounds (AREA)

DK220386A 1985-05-14 1986-05-13 2-(4-benzoyl-1-piperidinyl)-alkanolderivater, fremgangsmaade til fremstilling af saadanne derivater og anvendelse af disse som laegemidler DK220386A (da)

Applications Claiming Priority (1)

Application Number	Priority Date	Filing Date	Title
FR8507270A FR2581993B1 (fr)	1985-05-14	1985-05-14	Derives de (benzoyl-4 piperidino)-2 phenyl-1 alcanols, leur preparation et leur application en therapeutique

Publications (2)

Publication Number	Publication Date
DK220386D0 true DK220386D0 (da)	1986-05-13
DK220386A DK220386A (da)	1986-11-15

Family

ID=9319247

Family Applications (1)

Application Number	Title	Priority Date	Filing Date
DK220386A DK220386A (da)	1985-05-14	1986-05-13	2-(4-benzoyl-1-piperidinyl)-alkanolderivater, fremgangsmaade til fremstilling af saadanne derivater og anvendelse af disse som laegemidler

Country Status (18)

Country	Link
US (1)	US4711899A (da)
EP (1)	EP0202164B1 (da)
JP (1)	JPS61260063A (da)
KR (1)	KR860008976A (da)
AT (1)	ATE40684T1 (da)
AU (1)	AU584701B2 (da)
DE (1)	DE3662044D1 (da)
DK (1)	DK220386A (da)
ES (2)	ES8802138A1 (da)
FI (1)	FI861995A (da)
FR (1)	FR2581993B1 (da)
GR (1)	GR861253B (da)
HU (1)	HU195640B (da)
IL (1)	IL78773A (da)
NO (1)	NO861897L (da)
NZ (1)	NZ216145A (da)
PT (1)	PT82569B (da)
ZA (1)	ZA863533B (da)

Families Citing this family (26)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
KR910006138B1 (ko) *	1986-09-30	1991-08-16	에자이 가부시끼가이샤	환상아민 유도체
JP2573195B2 (ja) *	1986-09-30	1997-01-22	エーザイ株式会社	環状アミン誘導体
US4870083A (en) *	1987-11-24	1989-09-26	Merrell Dow Pharmaceuticals Inc.	1,4-Disubstituted-piperidinyl compounds useful as analgesics and muscle relaxants
US5166211A (en) *	1987-12-17	1992-11-24	Merrell Dow Pharmaceuticals Inc.	Method of using 1,4-disubstituted piperidinyl compounds in the treatment of coronary vasospasons and variant angina
US5093341A (en) *	1987-12-17	1992-03-03	Merrell Dow Pharmaceuticals Inc.	N-aralkyl piperidine derivatives useful as antithrombolytic agents
US5064838A (en) *	1988-01-21	1991-11-12	Merrell Dow Pharmaceuticals	1,4-disubstituted-piperidinyl compounds as pain relievers
FR2640266B2 (fr) *	1988-07-12	1992-07-10	Synthelabo	Derives de (hydroxy-1 piperidinyl-2 alkyl) indolones-2, quinoleinones-2, benzo(b)azepinones-2 et benzimidazolones-2, leur preparation et leur application en therapeutique
FR2634206B1 (fr) *	1988-07-12	1992-05-15	Synthelabo	Derives de (hydroxy-1 piperidinyl-2 alkyl) indolones-2 et quinoleinones-2, leur preparation et leur application en therapeutique
GB8823776D0 (en) *	1988-10-11	1988-11-16	Scras	New 2-methoxycarbonyl sustituted n n'-di-(trimethoxybenzoyl)piperazines
GB8823775D0 (en) *	1988-10-11	1988-11-16	Scras	New 2-carbonyl substituted n n'-di-(trimethoxybenzoyl)piperazines
US5055470A (en) *	1989-06-01	1991-10-08	Bristol-Myers Squibb Co.	Method of treatment of ischemia in brain
US4994460A (en) *	1989-06-01	1991-02-19	Bristol-Myers Squibb Co.	Agents for treatment of brain ischemia
NZ236501A (en) *	1989-12-21	1992-12-23	Merrell Dow Pharma	Piperidine derivatives and antithrombotic compositions
US5292752A (en) *	1989-12-21	1994-03-08	Merrell Dow Pharmaceuticals Inc.	Antithrombotic compounds
EP0554247B1 (en) *	1990-05-10	2000-04-26	Pfizer Inc.	Neuroprotective indolone and related derivatives
US5478846A (en) *	1990-06-07	1995-12-26	Merrell Dow Pharmaceuticals Inc.	1-piperidinyl alkanoylanyl sulfonamides for treatment of cardiac arrhythmia
JP3032294B2 (ja) *	1990-06-07	2000-04-10	メレルダウファーマス―ティカルズインコーポレイテッド	１―ピペリジニルアルカノイルアリールスルホンアミド誘導体類
US5512584A (en) *	1991-04-16	1996-04-30	Basf Aktiengesellschaft	1,3,4-trisubstituted piperidine derivatives, the preparation and use thereof
FR2678269B1 (fr) *	1991-06-27	1995-01-13	Synthelabo	Derives de 1-(4-chlorophenyl)-2-[4-(2-phenylethyl)piperidin-1-yl]ethanol, leur application et leur preparation en therapeutique.
FR2688504B1 (fr) *	1992-03-13	1995-05-05	Synthelabo	Derives de 2-(piperidin-1-yl)ethanol, leur preparation et leur application en therapeutique.
US5436255A (en) *	1992-07-23	1995-07-25	Pfizer Inc.	Method of treating diseases susceptable to treatment by blocking NMDA-receptors
US5498610A (en) *	1992-11-06	1996-03-12	Pfizer Inc.	Neuroprotective indolone and related derivatives
ATE183184T1 (de) *	1994-01-31	1999-08-15	Pfizer	Neuroprotektive chroman verbindungen
FR2737494B1 (fr) *	1995-08-04	1997-08-29	Synthelabo	Derives de benzenesulfonamide, leur preparation et leur application en therapeutique
US6770659B2 (en) *	2002-08-26	2004-08-03	Sk Corporation	Benzoyl piperidine compounds
US20050158270A1 (en) *	2004-01-15	2005-07-21	Seren Frantz	Pearlizer concentrate and its use in personal care compositions

Family Cites Families (15)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
CH492709A (de) *	1968-01-11	1970-06-30	Geigy Ag J R	Verfahren zur Herstellung von neuen Piperidinderivaten
US3632767A (en) *	1968-02-12	1972-01-04	Mallinckrodt Chemical Works	Treatment of depression with 4-substituted piperidines
US3576810A (en) *	1968-06-20	1971-04-27	Robins Co Inc A H	1-substituted-3-(-4)-aroylpiperidines
BE791088A (fr) *	1971-11-09	1973-03-01	Richardson Merrell Inc	Nouveaux derives d'aryl (piperidyl-4) cetone, utiles notamment comme analgesiques et anticoagulants, et leur procede de preparation
US4101662A (en) *	1973-05-03	1978-07-18	A. H. Robins Company, Incorporated	Method for inhibiting emesis and compositions therefor
GB1535791A (en) *	1975-05-07	1978-12-13	Ferrosan Ab	Derivatives of 4-piperidinol
US4035369A (en) *	1975-10-08	1977-07-12	Janssen Pharmaceutica N.V.	1-Benzazolylalkyl-4-substituted-piperidines
CH602642A5 (da) *	1975-11-14	1978-07-31	Orgamol Sa
FR2408602A2 (fr) *	1977-11-15	1979-06-08	Synthelabo	Nouveaux derives de piperidine et leur methode de preparation
US4335127A (en) *	1979-01-08	1982-06-15	Janssen Pharmaceutica, N.V.	Piperidinylalkyl quinazoline compounds, composition and method of use
US4198419A (en) *	1979-01-10	1980-04-15	American Hoechst Corporation	Phenylthiophenylpiperidines
US4443451A (en) *	1981-07-15	1984-04-17	Janssen Pharmaceutica N.V.	Bicyclic pyrimidin-5-one derivatives
FR2534580A1 (fr) *	1982-10-13	1984-04-20	Synthelabo	Derives de phenyl-1 piperidino-2 propanol, leur preparation, et medicaments qui les contiennent
DK159420C (da) *	1983-03-09	1991-03-11	Ciba Geigy Ag	N-(piperidinyl-alkyl)-carboxamider og salte deraf, farmaceutiske praeparater indeholdende disse forbindelser samt anvendelsen af forbindelserne til fremstilling af antipsykotiske farmaceutiske praeparater
US4458076A (en) *	1983-05-31	1984-07-03	Hoechst-Roussel Pharmaceuticals	3-(4-Piperidinyl)-1,2-benzisothiazoles

1985
- 1985-05-14 FR FR8507270A patent/FR2581993B1/fr not_active Expired
1986
- 1986-05-12 DE DE8686401000T patent/DE3662044D1/de not_active Expired
- 1986-05-12 AT AT86401000T patent/ATE40684T1/de active
- 1986-05-12 EP EP86401000A patent/EP0202164B1/fr not_active Expired
- 1986-05-13 HU HU861975A patent/HU195640B/hu not_active IP Right Cessation
- 1986-05-13 IL IL78773A patent/IL78773A/xx unknown
- 1986-05-13 DK DK220386A patent/DK220386A/da not_active Application Discontinuation
- 1986-05-13 JP JP61110463A patent/JPS61260063A/ja active Pending
- 1986-05-13 GR GR861253A patent/GR861253B/el unknown
- 1986-05-13 ES ES554895A patent/ES8802138A1/es not_active Expired
- 1986-05-13 AU AU57406/86A patent/AU584701B2/en not_active Ceased
- 1986-05-13 US US06/862,715 patent/US4711899A/en not_active Expired - Fee Related
- 1986-05-13 KR KR1019860003714A patent/KR860008976A/ko not_active Application Discontinuation
- 1986-05-13 FI FI861995A patent/FI861995A/fi not_active Application Discontinuation
- 1986-05-13 NO NO861897A patent/NO861897L/no unknown
- 1986-05-13 ZA ZA863533A patent/ZA863533B/xx unknown
- 1986-05-13 NZ NZ216145A patent/NZ216145A/xx unknown
- 1986-05-13 PT PT82569A patent/PT82569B/pt unknown
1987
- 1987-06-08 ES ES557582A patent/ES8801631A1/es not_active Expired

Also Published As

Publication number	Publication date
PT82569A (fr)	1986-06-01
ES554895A0 (es)	1988-04-01
NO861897L (no)	1986-11-17
FR2581993A1 (fr)	1986-11-21
FI861995A (fi)	1986-11-15
ES557582A0 (es)	1988-02-16
ES8802138A1 (es)	1988-04-01
IL78773A0 (en)	1986-08-31
JPS61260063A (ja)	1986-11-18
PT82569B (fr)	1988-04-12
DK220386A (da)	1986-11-15
ES8801631A1 (es)	1988-02-16
GR861253B (en)	1986-09-10
EP0202164B1 (fr)	1989-02-08
HUT40790A (en)	1987-02-27
AU5740686A (en)	1986-11-20
HU195640B (en)	1988-06-28
AU584701B2 (en)	1989-06-01
US4711899A (en)	1987-12-08
DE3662044D1 (en)	1989-03-16
ZA863533B (en)	1986-12-30
FI861995A0 (fi)	1986-05-13
EP0202164A1 (fr)	1986-11-20
ATE40684T1 (de)	1989-02-15
KR860008976A (ko)	1986-12-19
IL78773A (en)	1990-09-17
FR2581993B1 (fr)	1988-03-18
NZ216145A (en)	1988-10-28

Publication	Publication Date	Title
DK220386D0 (da)	1986-05-13	2-(4-benzoyl-1-piperidinyl)-alkanolderivater, fremgangsmaade til fremstilling af saadanne derivater og anvendelse af disse som laegemidler
DK0464465T3 (da)	1995-05-22	Substituerede aminoalkylbiphenylderivater, antimykotiske præparater indeholdende disse derivater og mellemprodukter til fremstilling deraf
AU2058283A (en)	1984-05-03	2-amino-3-acylamino-6-benzylamino pyridine derivatives
DK0766696T3 (da)	1999-02-15	Thiazolidinderivater, fremstilling af disse forbindelser og lægemidler indeholdende disse forbindelser
SE8802412D0 (sv)	1988-06-28	Thiourea derivatives
DK227085D0 (da)	1985-05-22	1-halogen-1-azolyl-2,2-diaryl-ethan-derivater, salte og metalkomplekser deraf samt deres fremstilling og anvendelse
ES8707923A1 (es)	1987-09-01	Procedimiento para la obtencion de benzamidas
DK32287D0 (da)	1987-01-21	3-acylaminomethyl-imidazo(1,2-a)pyridinderivater, fremgangsmaade til fremstilling deraf samt laegemiddel indeholdende saadanne derivater
DK0816358T3 (da)	2005-03-07	4-amino-2-ureidopyrimidin-5-carboxylsyreamider, fremgangsmåde til fremstilling heraf, lægemidler indeholdende sådanne forbindelser og anvendelsen af disse
DK158729C (da)	1990-11-19	N-(3-trifluormethylphenyl)-n'-propargylpiperazin, farmaceutiske praeparater, der indeholder det, dets anvendelse, samt en fremgangsmaade til fremstilling af et farmaceutisk praeparat
DK452088D0 (da)	1988-08-12	4-amino-6,7-dimethoxy-2-(1,2,3,4-tetrahydroisoquinolin-2-yl)quinolin-forbindelser, farmaceutiske praeparater indeholdende disse og deres anvendelse til fremstilling af antiarytmiske laegemidler samt n-(1-oe1,2,3,4-tetrahydroisozuinolin-2-ylaaethyliden)-2-cyan-4,5-dimethoxyanilin-forbindelser til anvendelse som udgangsmateriale ved deres fremstilling
DK373985A (da)	1986-02-18	Substituerede pyridazinoner samt deres fremstilling og anvendelse
DE3278074D1 (de)	1988-03-10	Imidazolecarboxylic acid derivatives
DK506885D0 (da)	1985-11-04	3-amino-2,3-dihydro-1-benzoxepin-forbindelser og farmaceutiske praeparater indeholdende disse
SE8101592L (sv)	1981-09-18	Pyrazolopyridinoner och pyridinylnikotinater och forfarande for framstellning derav
FI882421A (fi)	1988-11-24	5-fenyl-1,2,3a,4,5,9b-hexahydro-3h -benz(e)indol, deras framstaellning och anvaendning som laekemedel.
DK154961C (da)	1989-06-05	2-(4'-phenoxyphenyl)-5,6-dihydro-4-pyroner og salte deraf med baser, herbicider indeholdende disse forbindelser samt fremgangsmaade til bekaempelse af ukrudt

Legal Events

Date	Code	Title	Description
1991-01-21	AHB	Application shelved due to non-payment