DK204388D0 - Substituerede piperidiner til anvendelse som opioidantagonister og fremgangsmaade til fremstilling af saadenne forbindelser - Google Patents
Substituerede piperidiner til anvendelse som opioidantagonister og fremgangsmaade til fremstilling af saadenne forbindelserInfo
- Publication number
- DK204388D0 DK204388D0 DK204388A DK204388A DK204388D0 DK 204388 D0 DK204388 D0 DK 204388D0 DK 204388 A DK204388 A DK 204388A DK 204388 A DK204388 A DK 204388A DK 204388 D0 DK204388 D0 DK 204388D0
- Authority
- DK
- Denmark
- Prior art keywords
- procedures
- compounds
- making
- opioid antagonists
- substituted piperidines
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D211/00—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings
- C07D211/04—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom
- C07D211/06—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members
- C07D211/08—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members with hydrocarbon or substituted hydrocarbon radicals directly attached to ring carbon atoms
- C07D211/10—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members with hydrocarbon or substituted hydrocarbon radicals directly attached to ring carbon atoms with radicals containing only carbon and hydrogen atoms attached to ring carbon atoms
- C07D211/14—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members with hydrocarbon or substituted hydrocarbon radicals directly attached to ring carbon atoms with radicals containing only carbon and hydrogen atoms attached to ring carbon atoms with hydrocarbon or substituted hydrocarbon radicals attached to the ring nitrogen atom
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D409/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms
- C07D409/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms containing two hetero rings
- C07D409/06—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms containing two hetero rings linked by a carbon chain containing only aliphatic carbon atoms
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/04—Centrally acting analgesics, e.g. opioids
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/30—Drugs for disorders of the nervous system for treating abuse or dependence
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P3/00—Drugs for disorders of the metabolism
- A61P3/04—Anorexiants; Antiobesity agents
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P7/00—Drugs for disorders of the blood or the extracellular fluid
- A61P7/10—Antioedematous agents; Diuretics
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D211/00—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings
- C07D211/04—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom
- C07D211/06—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members
- C07D211/08—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members with hydrocarbon or substituted hydrocarbon radicals directly attached to ring carbon atoms
- C07D211/18—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members with hydrocarbon or substituted hydrocarbon radicals directly attached to ring carbon atoms with substituted hydrocarbon radicals attached to ring carbon atoms
- C07D211/20—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members with hydrocarbon or substituted hydrocarbon radicals directly attached to ring carbon atoms with substituted hydrocarbon radicals attached to ring carbon atoms with hydrocarbon radicals, substituted by singly bound oxygen or sulphur atoms
- C07D211/22—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members with hydrocarbon or substituted hydrocarbon radicals directly attached to ring carbon atoms with substituted hydrocarbon radicals attached to ring carbon atoms with hydrocarbon radicals, substituted by singly bound oxygen or sulphur atoms by oxygen atoms
Landscapes
- Health & Medical Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Life Sciences & Earth Sciences (AREA)
- General Health & Medical Sciences (AREA)
- Veterinary Medicine (AREA)
- Public Health (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Chemical Kinetics & Catalysis (AREA)
- General Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Engineering & Computer Science (AREA)
- Pharmacology & Pharmacy (AREA)
- Animal Behavior & Ethology (AREA)
- Biomedical Technology (AREA)
- Diabetes (AREA)
- Hematology (AREA)
- Neurology (AREA)
- Neurosurgery (AREA)
- Obesity (AREA)
- Addiction (AREA)
- Psychiatry (AREA)
- Child & Adolescent Psychology (AREA)
- Pain & Pain Management (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Hydrogenated Pyridines (AREA)
- Plural Heterocyclic Compounds (AREA)
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US3912187A | 1987-04-16 | 1987-04-16 |
Publications (2)
| Publication Number | Publication Date |
|---|---|
| DK204388D0 true DK204388D0 (da) | 1988-04-14 |
| DK204388A DK204388A (da) | 1989-01-05 |
Family
ID=21903800
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| DK204388A DK204388A (da) | 1987-04-16 | 1988-04-14 | Substituerede piperidiner til anvendelse som opioidantagonister og fremgangsmaade til fremstilling af saadenne forbindelser |
Country Status (21)
| Country | Link |
|---|---|
| EP (1) | EP0287339B1 (da) |
| JP (1) | JP2661699B2 (da) |
| KR (1) | KR960015087B1 (da) |
| CN (1) | CN1017992B (da) |
| AR (1) | AR245933A1 (da) |
| AT (1) | ATE110057T1 (da) |
| AU (1) | AU596290B2 (da) |
| CA (1) | CA1321792C (da) |
| DE (1) | DE3851081T2 (da) |
| DK (1) | DK204388A (da) |
| EG (1) | EG18864A (da) |
| ES (1) | ES2058265T3 (da) |
| HU (1) | HU202492B (da) |
| IE (1) | IE64508B1 (da) |
| IL (1) | IL86061A (da) |
| MX (1) | MX11117A (da) |
| NZ (1) | NZ224236A (da) |
| PH (1) | PH24752A (da) |
| PT (1) | PT87233B (da) |
| SU (1) | SU1598869A3 (da) |
| ZA (1) | ZA882640B (da) |
Families Citing this family (24)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| EP0299549A3 (en) * | 1987-07-09 | 1989-02-08 | Duphar International Research B.V | Tertiary 2,5-dialkyl-3-phenyl-piperidine derivatives having opiate-antagonistic activity |
| ZA922180B (en) * | 1991-03-29 | 1993-09-27 | Lilly Co Eli | Piperidine derivatives |
| US5985880A (en) * | 1996-06-05 | 1999-11-16 | Delta Pharmaceuticals | Compositions and methods for reducing respiratory depression and attendant side effects of mu opioid compounds |
| US5807858A (en) * | 1996-06-05 | 1998-09-15 | Delta Pharmaceutical, Inc. | Compositions and methods for reducing respiratory depression |
| US5574159A (en) * | 1992-02-03 | 1996-11-12 | Delta Pharmaceuticals, Inc. | Opioid compounds and methods for making therefor |
| GB9202238D0 (en) * | 1992-02-03 | 1992-03-18 | Wellcome Found | Compounds |
| US5681830A (en) * | 1992-02-03 | 1997-10-28 | Delta Pharmaceuticals, Inc. | Opioid compounds |
| MY111348A (en) * | 1993-07-30 | 1999-11-30 | Ardent Pharmaceuticals Inc | Opioid diarylmethylpiperazines and piperidines |
| GB9725114D0 (en) * | 1997-11-28 | 1998-01-28 | Pfizer Ltd | Treatment of pruritus |
| GB9810671D0 (en) | 1998-05-18 | 1998-07-15 | Pfizer Ltd | Anti-pruritic agents |
| GB9815618D0 (en) | 1998-07-18 | 1998-09-16 | Univ Manchester | Treatment of dyskinesia |
| TWI244481B (en) | 1998-12-23 | 2005-12-01 | Pfizer | 3-azabicyclo[3.1.0]hexane derivatives useful in therapy |
| GB9912413D0 (en) | 1999-05-28 | 1999-07-28 | Pfizer Ltd | Compounds useful in therapy |
| GB9912417D0 (en) * | 1999-05-28 | 1999-07-28 | Pfizer Ltd | Compounds useful in therapy |
| GB9912411D0 (en) * | 1999-05-28 | 1999-07-28 | Pfizer Ltd | Compounds useful in therapy |
| GB9912416D0 (en) * | 1999-05-28 | 1999-07-28 | Pfizer Ltd | Compounds useful in therapy |
| GB9912415D0 (en) * | 1999-05-28 | 1999-07-28 | Pfizer Ltd | Compounds useful in therapy |
| GB9912410D0 (en) | 1999-05-28 | 1999-07-28 | Pfizer Ltd | Compounds useful in therapy |
| MXPA02005335A (es) * | 1999-11-29 | 2003-01-28 | Adolor Corp | Metodos y composiciones novedosos que incluyen opioides y antagonistas de los mismos. |
| GB0015562D0 (en) * | 2000-06-23 | 2000-08-16 | Pfizer Ltd | Heterocycles |
| CA2463264C (en) | 2001-10-22 | 2009-05-26 | Pfizer Products Inc. | 3-azabicyclo (3.1.0) hexane derivatives as opioid receptor antagonists |
| WO2004026305A1 (en) * | 2002-09-19 | 2004-04-01 | Eli Lilly And Company | Diaryl ethers as opioid receptor antagonist |
| US7538110B2 (en) | 2005-10-27 | 2009-05-26 | Adolor Corporation | Opioid antagonists |
| AU2012284127A1 (en) * | 2011-07-18 | 2013-05-02 | Adolor Corporation | Processes for the preparation of peripheral opioid antagonist compounds and intermediates thereto |
Family Cites Families (1)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| AR206937A1 (es) * | 1974-09-06 | 1976-08-31 | Lilly Co Eli | Procedimiento para preparar compuestos de 1-sustituido-4-alquil-4-fenil-piperidina |
-
1988
- 1988-04-13 AT AT88303302T patent/ATE110057T1/de not_active IP Right Cessation
- 1988-04-13 AR AR88310556A patent/AR245933A1/es active
- 1988-04-13 CA CA000563995A patent/CA1321792C/en not_active Expired - Fee Related
- 1988-04-13 DE DE3851081T patent/DE3851081T2/de not_active Expired - Fee Related
- 1988-04-13 ES ES88303302T patent/ES2058265T3/es not_active Expired - Lifetime
- 1988-04-13 EP EP88303302A patent/EP0287339B1/en not_active Expired - Lifetime
- 1988-04-13 NZ NZ224236A patent/NZ224236A/xx unknown
- 1988-04-13 IL IL86061A patent/IL86061A/xx not_active IP Right Cessation
- 1988-04-13 PH PH36789A patent/PH24752A/en unknown
- 1988-04-14 KR KR1019880004245A patent/KR960015087B1/ko not_active IP Right Cessation
- 1988-04-14 AU AU14624/88A patent/AU596290B2/en not_active Ceased
- 1988-04-14 PT PT87233A patent/PT87233B/pt active IP Right Grant
- 1988-04-14 SU SU884355530A patent/SU1598869A3/ru active
- 1988-04-14 DK DK204388A patent/DK204388A/da not_active Application Discontinuation
- 1988-04-14 EG EG21388A patent/EG18864A/xx active
- 1988-04-14 ZA ZA882640A patent/ZA882640B/xx unknown
- 1988-04-14 IE IE112588A patent/IE64508B1/en not_active IP Right Cessation
- 1988-04-14 MX MX1111788A patent/MX11117A/es unknown
- 1988-04-15 HU HU881968A patent/HU202492B/hu not_active IP Right Cessation
- 1988-04-15 JP JP63094395A patent/JP2661699B2/ja not_active Expired - Lifetime
- 1988-04-15 CN CN88102191A patent/CN1017992B/zh not_active Expired
Also Published As
| Publication number | Publication date |
|---|---|
| IL86061A0 (en) | 1988-09-30 |
| KR880012551A (ko) | 1988-11-28 |
| DE3851081D1 (de) | 1994-09-22 |
| DK204388A (da) | 1989-01-05 |
| JPS63277661A (ja) | 1988-11-15 |
| EG18864A (en) | 1995-06-29 |
| NZ224236A (en) | 1990-08-28 |
| ES2058265T3 (es) | 1994-11-01 |
| HUT46892A (en) | 1988-12-28 |
| EP0287339B1 (en) | 1994-08-17 |
| CN1017992B (zh) | 1992-08-26 |
| CA1321792C (en) | 1993-08-31 |
| PT87233B (pt) | 1992-07-31 |
| MX11117A (es) | 1993-11-01 |
| IE64508B1 (en) | 1995-08-09 |
| SU1598869A3 (ru) | 1990-10-07 |
| IL86061A (en) | 1992-07-15 |
| IE881125L (en) | 1988-10-16 |
| JP2661699B2 (ja) | 1997-10-08 |
| AR245933A1 (es) | 1994-03-30 |
| CN88102191A (zh) | 1988-11-02 |
| DE3851081T2 (de) | 1995-02-16 |
| PT87233A (pt) | 1988-05-01 |
| EP0287339A3 (en) | 1991-05-15 |
| AU1462488A (en) | 1988-10-20 |
| KR960015087B1 (ko) | 1996-10-24 |
| EP0287339A2 (en) | 1988-10-19 |
| PH24752A (en) | 1990-10-01 |
| ZA882640B (en) | 1989-12-27 |
| ATE110057T1 (de) | 1994-09-15 |
| HU202492B (en) | 1991-03-28 |
| AU596290B2 (en) | 1990-04-26 |
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Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| AHB | Application shelved due to non-payment |