DK155603C - Analogifremgangsmaade til fremstilling af benzimidazolderivater - Google Patents

Analogifremgangsmaade til fremstilling af benzimidazolderivater

Info

Publication number: DK155603C
Authority: DK; Denmark
Prior art keywords: preparing; analogy procedure; benzimidazold; derivatives; benzimidazold derivatives
Prior art date: 1977-04-12

Application number

DK159478A

Other languages

English (en)

Other versions

DK159478A (da

DK155603B (da

Inventor

Jean Jacques Gallay

Manfred Kuehne

Alfred Meyer

Oswald Rechsteiner

Max Schellenbaum

Original Assignee

Ciba Geigy Ag

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

1977-04-12

Filing date

1978-04-11

Publication date

1989-09-04

1977-04-12 Priority claimed from LU77120A external-priority patent/LU77120A1/xx

1978-03-15 Priority claimed from LU79232A external-priority patent/LU79232A1/de

1978-04-11 Application filed by Ciba Geigy Ag filed Critical Ciba Geigy Ag

1978-10-13 Publication of DK159478A publication Critical patent/DK159478A/da

1989-04-24 Publication of DK155603B publication Critical patent/DK155603B/da

1989-09-04 Application granted granted Critical

1989-09-04 Publication of DK155603C publication Critical patent/DK155603C/da

Classifications

- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D235/00—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, condensed with other rings
- C07D235/02—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, condensed with other rings condensed with carbocyclic rings or ring systems
- C07D235/04—Benzimidazoles; Hydrogenated benzimidazoles
- C07D235/24—Benzimidazoles; Hydrogenated benzimidazoles with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached in position 2
- C07D235/28—Sulfur atoms
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P33/00—Antiparasitic agents
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P33/00—Antiparasitic agents
- A61P33/10—Anthelmintics

Landscapes

Organic Chemistry (AREA)
Chemical & Material Sciences (AREA)
Health & Medical Sciences (AREA)
Veterinary Medicine (AREA)
Chemical Kinetics & Catalysis (AREA)
General Chemical & Material Sciences (AREA)
Medicinal Chemistry (AREA)
Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
Tropical Medicine & Parasitology (AREA)
Pharmacology & Pharmacy (AREA)
Life Sciences & Earth Sciences (AREA)
Animal Behavior & Ethology (AREA)
General Health & Medical Sciences (AREA)
Public Health (AREA)
Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Plural Heterocyclic Compounds (AREA)
Heterocyclic Carbon Compounds Containing A Hetero Ring Having Oxygen Or Sulfur (AREA)

DK159478A 1977-04-12 1978-04-11 Analogifremgangsmaade til fremstilling af benzimidazolderivater DK155603C (da)

Applications Claiming Priority (4)

Application Number	Priority Date	Filing Date	Title
LU77120		1977-04-12
LU77120A LU77120A1 (da)	1977-04-12	1977-04-12
LU79232A LU79232A1 (de)	1978-03-15	1978-03-15	Verfahren zur herstellung von anthelmintika
LU79232		1978-03-15

Publications (3)

Publication Number	Publication Date
DK159478A DK159478A (da)	1978-10-13
DK155603B DK155603B (da)	1989-04-24
DK155603C true DK155603C (da)	1989-09-04

Family

ID=26640224

Family Applications (1)

Application Number	Title	Priority Date	Filing Date
DK159478A DK155603C (da)	1977-04-12	1978-04-11	Analogifremgangsmaade til fremstilling af benzimidazolderivater

Country Status (27)

Country	Link
US (1)	US4197307A (da)
JP (1)	JPS6019753B2 (da)
AR (1)	AR230270A1 (da)
AT (1)	AT363078B (da)
AU (1)	AU520836B2 (da)
BE (1)	BE865870A (da)
CA (1)	CA1105034A (da)
CH (1)	CH634306A5 (da)
CS (1)	CS209450B2 (da)
DE (1)	DE2815621A1 (da)
DK (1)	DK155603C (da)
FR (1)	FR2387220A1 (da)
GB (1)	GB1599970A (da)
IE (1)	IE46718B1 (da)
IL (1)	IL54474A (da)
IT (1)	IT1113128B (da)
KE (1)	KE3345A (da)
MX (1)	MX5951E (da)
MY (1)	MY8500089A (da)
NL (1)	NL187808C (da)
NZ (1)	NZ186936A (da)
PH (1)	PH18234A (da)
PL (2)	PL117396B1 (da)
SE (1)	SE444315B (da)
SU (1)	SU1097196A3 (da)
YU (1)	YU41309B (da)
ZA (1)	ZA782086B (da)

Families Citing this family (28)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
DE3132167A1 (de) *	1981-08-14	1983-03-03	Hoechst Ag, 6000 Frankfurt	"5(6)-phenylsulfonyloxy-benzimidazolderivate, verfahren zu ihrer herstellung, sie enthaltende pharmazeutische zubereitungen und ihre verwendung gegen leberegel"
MA19678A1 (fr) *	1982-01-13	1983-10-01	Ciba Geigy Ag	Agents anti-helmintiques.
GB2124904B (en) *	1982-08-13	1986-01-15	Ciba Geigy Ag	Synergistic anthelmintic compositions
US4472419A (en) *	1984-01-25	1984-09-18	American Cyanamid Company	Method of controlling plant nematodes
GB8426367D0 (en) *	1984-10-18	1984-11-21	Shell Int Research	Heteroaromatic ether herbicides
US4781920A (en) *	1984-11-13	1988-11-01	American Cyanamid Company	Anthelmintic paste compositions containing resinates of d1-6-phenyl-2,3,5,6-tetrahydroimidazo[2,1-b]thiazole
DE3508665A1 (de) *	1985-03-12	1986-09-18	Hoechst Ag, 6230 Frankfurt	Heterocyclische sulfide und ihre anwendung als immunmodulatoren
GB8519920D0 (en) *	1985-08-08	1985-09-18	Fbc Ltd	Fungicides
JPS62246587A (ja) *	1986-03-17	1987-10-27	ピ−ピ−ジ−　インダストリイズ，インコ−ポレイテツド	除草活性を有する置換ベンゾオキサゾロン（またはベンゾチアゾロン）化合物
DE3719783A1 (de) *	1987-06-13	1988-12-22	Hoechst Ag	Verfahren zur herstellung von 5-phenylsulfinyl-1h-2-(methoxycarbonylamino)- benzimidazol
AU2003236405B2 (en) *	1999-04-14	2007-10-25	Merial Ltd	Anthelmintic Composition
NZ335166A (en)	1999-04-14	2001-11-30	Ashmont Holdings Ltd	Anthelmintic composition containing triclabendazole in at least one solvent
US5538989A (en) *	1993-11-10	1996-07-23	Hoechst-Roussel Agri-Vet Company	Fenbendazole formulations
US7001889B2 (en) *	2002-06-21	2006-02-21	Merial Limited	Anthelmintic oral homogeneous veterinary pastes
US20060205681A1 (en) *	2002-06-21	2006-09-14	Maryam Moaddeb	Homogenous paste formulations
ATE402924T1 (de)	2003-03-03	2008-08-15	Mycosol Inc	Pyridiniumsalze und deren verwendung
ATE466578T1 (de) *	2004-02-03	2010-05-15	Wyeth Llc	Wurmmittel
PE20070427A1 (es) *	2005-08-30	2007-04-21	Novartis Ag	Compuestos derivados de benzimidazoles sustituidos como inhibidores de tirosina quinasas
US20080027011A1 (en) *	2005-12-20	2008-01-31	Hassan Nached	Homogeneous paste and gel formulations
AU2009245834B2 (en) *	2008-10-08	2013-11-14	Zoetis Services Llc	Benzimidazole anthelmintic compositions
CN101555231B (zh) *	2009-05-04	2011-03-23	扬州天和药业有限公司	一种制备三氯苯达唑的方法
WO2012070068A2 (en) *	2010-11-24	2012-05-31	Sequent Scientific Limited	Process for preparation of triclabendazole
SG11201406730RA (en) *	2012-04-20	2014-11-27	Merial Ltd	Parasiticidal compositions comprising benzimidazole derivatives, methods and uses thereof
CN103319416B (zh) *	2013-06-24	2015-02-25	常州佳灵药业有限公司	新型兽药三氯苯达唑亚砜及其制备方法
EP3235815A1 (de)	2016-04-19	2017-10-25	Philipps-Universität Marburg	Wirkstoffe gegen parasitäre helminthen
RU2640482C2 (ru) *	2016-04-22	2018-01-09	ФАНО России Федеральное государственное бюджетное научное учреждение Всероссийский научно-исследовательский институт фундаментальной и прикладной паразитологии животных и растений им. К.И. Скрябина (ФГБНУ "ВНИИП им. К.И. Скрябина")	Супрамолекулярный комплекс триклабендазола для лечения животных при фасциолёзе
CN113507922A (zh)	2019-03-01	2021-10-15	勃林格殷格翰动物保健美国公司	可注射的氯舒隆组合物、其方法和用途
AU2022228569A1 (en) *	2021-03-03	2023-10-12	Terns Pharmaceuticals, Inc.	Thyroid hormone receptor beta agonist compounds

Family Cites Families (12)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
US2666764A (en) *	1951-07-14	1954-01-19	Ciba Pharm Prod Inc	Process of splitting aralkylheterocyclic thioethers with aluminum bromide
FR1476558A (fr) *	1965-07-26	1967-04-14	Chimetron Sarl	Thiazolylthiobenzimidazoles et thiazolylsulfinylbenzimidazoles
CH443777A (de) *	1965-08-06	1968-02-15	Agripat Sa	Verfahren zum Schützen textiler Keratinfasern vor Insektenfrass und Mittel zur Durchführung dieses Verfahrens
US3506767A (en) *	1965-08-06	1970-04-14	Geigy Chem Corp	Benzimidazole compositions and methods of use
FR1509192A (fr) *	1966-12-01	1968-01-12		Benzylthio-2 benzimidazoles
US3480643A (en) *	1967-05-09	1969-11-25	American Cyanamid Co	Alkylsulfonylbenzimidazoles
NL7013343A (da) *	1969-09-26	1971-03-30
BE754874A (fr) *	1969-10-30	1971-01-18	Buckman Labor Inc	Composes s-chloromethyliques de 2-mercapto-benzothiazole, de 2-mercaptobenzoxazole et de 2-mercaptobenzimidazole
DE2041324A1 (de) *	1970-08-20	1972-02-24	Agfa Gevaert Ag	Neue Benzimidazolderivate,sowie ein Verfahren zu ihrer Herstellung
US3840550A (en) *	1971-05-24	1974-10-08	Ciba Geigy Corp	Certain 6-isothiocyanobenzothiazoles
US3933841A (en) *	1971-05-24	1976-01-20	Ciba-Geigy Corporation	2-Phenoxy, -phenylthio-, and -phenyl-amino-benzoxazoles having an isothiocyano substituent
BE792402A (fr) *	1971-12-07	1973-06-07	Ciba Geigy	Composes heterocycliques azotes et medicaments anthelminthiqueset antimicrobiens qui en contiennent

1978
- 1978-04-10 CH CH382678A patent/CH634306A5/de not_active IP Right Cessation
- 1978-04-10 IL IL54474A patent/IL54474A/xx unknown
- 1978-04-10 US US05/894,973 patent/US4197307A/en not_active Expired - Lifetime
- 1978-04-11 YU YU857/78A patent/YU41309B/xx unknown
- 1978-04-11 AT AT0253478A patent/AT363078B/de active
- 1978-04-11 DK DK159478A patent/DK155603C/da not_active IP Right Cessation
- 1978-04-11 GB GB14183/78A patent/GB1599970A/en not_active Expired
- 1978-04-11 BE BE186705A patent/BE865870A/xx not_active IP Right Cessation
- 1978-04-11 ZA ZA00782086A patent/ZA782086B/xx unknown
- 1978-04-11 SE SE7804057A patent/SE444315B/sv not_active IP Right Cessation
- 1978-04-11 CS CS782366A patent/CS209450B2/cs unknown
- 1978-04-11 DE DE19782815621 patent/DE2815621A1/de active Granted
- 1978-04-11 IT IT22189/78A patent/IT1113128B/it active
- 1978-04-11 IE IE704/78A patent/IE46718B1/en not_active IP Right Cessation
- 1978-04-11 NZ NZ186936A patent/NZ186936A/xx unknown
- 1978-04-11 SU SU782601448A patent/SU1097196A3/ru active
- 1978-04-11 MX MX787013U patent/MX5951E/es unknown
- 1978-04-12 FR FR7810731A patent/FR2387220A1/fr active Granted
- 1978-04-12 PL PL1978221071A patent/PL117396B1/pl unknown
- 1978-04-12 NL NLAANVRAGE7803886,A patent/NL187808C/xx not_active IP Right Cessation
- 1978-04-12 JP JP53043058A patent/JPS6019753B2/ja not_active Expired
- 1978-04-12 PH PH20998A patent/PH18234A/en unknown
- 1978-04-12 CA CA300,973A patent/CA1105034A/en not_active Expired
- 1978-04-12 PL PL1978206019A patent/PL115361B1/pl unknown
- 1978-04-12 AU AU35022/78A patent/AU520836B2/en not_active Expired
1979
- 1979-06-28 AR AR277106A patent/AR230270A1/es active
1983
- 1983-11-16 KE KE3345A patent/KE3345A/xx unknown
1985
- 1985-12-30 MY MY89/85A patent/MY8500089A/xx unknown

Also Published As

Publication number	Publication date
PL115361B1 (en)	1981-03-31
DK159478A (da)	1978-10-13
GB1599970A (en)	1981-10-07
MX5951E (es)	1984-09-06
PL206019A1 (pl)	1979-06-04
FR2387220B1 (da)	1983-06-03
PH18234A (en)	1985-05-03
IL54474A (en)	1982-04-30
MY8500089A (en)	1985-12-31
NZ186936A (en)	1980-10-24
KE3345A (en)	1983-12-16
FR2387220A1 (fr)	1978-11-10
SU1097196A3 (ru)	1984-06-07
DK155603B (da)	1989-04-24
IT7822189A0 (it)	1978-04-11
CH634306A5 (de)	1983-01-31
ZA782086B (en)	1979-03-28
AT363078B (de)	1981-07-10
DE2815621C2 (da)	1990-08-09
BE865870A (fr)	1978-10-11
YU41309B (en)	1987-02-28
CA1105034A (en)	1981-07-14
YU85778A (en)	1983-01-21
IE780704L (en)	1978-10-12
IE46718B1 (en)	1983-09-07
NL187808C (nl)	1992-01-16
NL187808B (nl)	1991-08-16
JPS6019753B2 (ja)	1985-05-17
IL54474A0 (en)	1978-07-31
DE2815621A1 (de)	1978-10-19
AU520836B2 (en)	1982-03-04
JPS53127476A (en)	1978-11-07
PL117396B1 (en)	1981-07-31
SE7804057L (sv)	1978-10-13
IT1113128B (it)	1986-01-20
CS209450B2 (en)	1981-12-31
SE444315B (sv)	1986-04-07
NL7803886A (nl)	1978-10-16
AU3502278A (en)	1979-10-18
US4197307A (en)	1980-04-08
AR230270A1 (es)	1984-03-01
ATA253478A (de)	1980-12-15

Publication	Publication Date	Title
DK151253C (da)	1988-05-16	Analogifremgangsmaade til fremstilling af 2-benzylphthalazin-4-yleddikesyrederivater
DK155603C (da)	1989-09-04	Analogifremgangsmaade til fremstilling af benzimidazolderivater
DK157019C (da)	1990-03-26	Analogifremgangsmaade til fremstilling af 2-amino-4-hydroxyquinazolinderivater
DK195378A (da)	1978-11-05	Fremgangsmaade til fremstilling af polyenforbindelser
DK147422C (da)	1985-02-11	Analogifremgangsmaade til fremstilling af phosphonoacylproliner
DK148280C (da)	1985-11-18	Analogifremgangsmaade til fremstilling af thienothiazinderivater
DK155733C (da)	1989-09-25	Fremgangsmaade til fremstilling af 4-hydroxy-2-oxo-pyrrolidinderivater
DK155367C (da)	1989-08-14	Analogifremgangsmaade til fremstilling af 2-nitroimidazolderivater
DK349478A (da)	1979-02-10	Fremgangsmaade til fremstilling af oligoimider
DK254878A (da)	1979-02-09	Fremgangsmaade til fremstilling af carbostyrilderivater
DK539578A (da)	1979-07-05	Fremgangsmaade til fremstilling af pleuromutilinglycsid-derivater
DK155279C (da)	1989-07-24	Fremgangsmaade til fremstilling af 4-hydroxy-2-oxo-pyrrolidinderivater
DK531178A (da)	1979-05-31	Fremgangsmaade til fremstilling af phenylglycinderivater
DK147068C (da)	1984-09-10	Analogifremgangsmaade til fremstilling af 1-naphthylmethyl-cinnamyl-aminderivater
DK153482C (da)	1988-12-27	Analogifremgangsmaade til fremstilling af 5-cyano-prostacyklinderivater
DK145698C (da)	1983-07-25	Analogifremgangsmaade til fremstilling af 2-alkoxyadeninderivater
DK154137C (da)	1989-04-10	Analogifremgangsmaade til fremstilling af meta-sulfonamido-benzamidderivater
DK153950C (da)	1989-02-20	Analogifremgangsmaade til fremstilling af quinolylguanidiner eller derivater deraf
DK147145C (da)	1984-10-15	Analogifremgangsmaade til fremstilling af chlorambucilderivater
DK470978A (da)	1979-05-01	R fremgangsmaade til fremstilling af pyrazinobenzoxapinderivate
DK152130C (da)	1988-08-15	Fremgangsmaade til fremstilling af benzooebaathienopyridinderivater
DK494978A (da)	1979-05-08	Fremgangsmaade til fremstilling af 2-iminoimidazolidinderivater
DK262678A (da)	1978-12-21	Fremgangsmaade til fremstilling af quinolinonderivater
DK129978A (da)	1978-09-24	Fremgangsmaade til fremstilling af morfinderivater
DK142848C (da)	1981-08-24	Analogifremgangsmaade til fremstilling af 2-acylamido-4-amino-5-benzylpyrimidinforbindelser

Legal Events

Date	Code	Title	Description
1998-05-18	PUP	Patent expired