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DK142583B - Analogifremgangsmåde til fremstilling af dl(racem)- eller 1-formen af derivater af 6-(m-aminophenyl)-2,3,5,6-tetrahydroimidazo(2,1-b)thiazol eller syreadditionssalte heraf. - Google Patents

Analogifremgangsmåde til fremstilling af dl(racem)- eller 1-formen af derivater af 6-(m-aminophenyl)-2,3,5,6-tetrahydroimidazo(2,1-b)thiazol eller syreadditionssalte heraf. Download PDF

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Publication number
DK142583B
DK142583B DK186877AA DK186877A DK142583B DK 142583 B DK142583 B DK 142583B DK 186877A A DK186877A A DK 186877AA DK 186877 A DK186877 A DK 186877A DK 142583 B DK142583 B DK 142583B
Authority
DK
Denmark
Prior art keywords
thiazole
acid
tetrahydroimidazo
aminophenyl
compounds
Prior art date
Application number
DK186877AA
Other languages
Danish (da)
English (en)
Other versions
DK186877A (xx
DK142583C (xx
Inventor
John Eric Thorpe
Original Assignee
Pfizer
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Pfizer filed Critical Pfizer
Publication of DK186877A publication Critical patent/DK186877A/da
Publication of DK142583B publication Critical patent/DK142583B/da
Application granted granted Critical
Publication of DK142583C publication Critical patent/DK142583C/da

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D213/00Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members
    • C07D213/02Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members
    • C07D213/04Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom
    • C07D213/60Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D213/78Carbon atoms having three bonds to hetero atoms, with at the most one bond to halogen, e.g. ester or nitrile radicals
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P33/00Antiparasitic agents
    • A61P33/10Anthelmintics
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D213/00Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members
    • C07D213/02Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members
    • C07D213/04Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom
    • C07D213/60Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D213/78Carbon atoms having three bonds to hetero atoms, with at the most one bond to halogen, e.g. ester or nitrile radicals
    • C07D213/79Acids; Esters
    • C07D213/80Acids; Esters in position 3

Landscapes

  • Organic Chemistry (AREA)
  • Chemical & Material Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Tropical Medicine & Parasitology (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
DK186877AA 1976-05-01 1977-04-28 Analogifremgangsmåde til fremstilling af dl(racem)- eller 1-formen af derivater af 6-(m-aminophenyl)-2,3,5,6-tetrahydroimidazo(2,1-b)thiazol eller syreadditionssalte heraf. DK142583B (da)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
GB1788376 1976-05-01
GB17883/76A GB1516938A (en) 1976-05-01 1976-05-01 Halopyridylamides of m-aminotetramisole and their use as anthelmintics

Publications (3)

Publication Number Publication Date
DK186877A DK186877A (xx) 1977-11-02
DK142583B true DK142583B (da) 1980-11-24
DK142583C DK142583C (xx) 1981-07-27

Family

ID=10102899

Family Applications (1)

Application Number Title Priority Date Filing Date
DK186877AA DK142583B (da) 1976-05-01 1977-04-28 Analogifremgangsmåde til fremstilling af dl(racem)- eller 1-formen af derivater af 6-(m-aminophenyl)-2,3,5,6-tetrahydroimidazo(2,1-b)thiazol eller syreadditionssalte heraf.

Country Status (24)

Country Link
US (1) US4112102A (xx)
JP (1) JPS52133998A (xx)
AR (1) AR215629A1 (xx)
AT (1) AT355572B (xx)
BE (1) BE854073A (xx)
CA (1) CA1067082A (xx)
CH (1) CH620218A5 (xx)
CS (1) CS189598B2 (xx)
DD (1) DD130149A5 (xx)
DE (1) DE2718976A1 (xx)
DK (1) DK142583B (xx)
ES (1) ES458249A1 (xx)
FI (1) FI60712C (xx)
FR (1) FR2349592A1 (xx)
GB (1) GB1516938A (xx)
IE (1) IE45140B1 (xx)
IL (1) IL51875A0 (xx)
LU (1) LU77233A1 (xx)
NL (1) NL162389C (xx)
NZ (1) NZ183876A (xx)
PH (1) PH11989A (xx)
PT (1) PT66491B (xx)
SE (1) SE432423B (xx)
YU (1) YU102377A (xx)

Families Citing this family (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
EP0041322A1 (en) 1980-05-30 1981-12-09 Beecham Group Plc m-Pyrazolylamido tetramisole derivatives, compositions thereof, processes for production of such compounds and compositions and their use in treating helminthiasis
WO2018231704A1 (en) * 2017-06-12 2018-12-20 Dow Agrosciences, Llc 6-bromonicotinamide and processes of preparation

Family Cites Families (7)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
NL131034C (xx) * 1964-05-11
US3673205A (en) * 1970-03-25 1972-06-27 American Cyanamid Co 6-(m-AMINO AND SUBSTITUTED-AMINO PHENYL)-2,3,5,6-TETRAHYDRO{8 2,1-b{9 THIAZOLES AND METHOD OF USE
GB1365515A (en) * 1971-09-03 1974-09-04 American Cyanamid Co 6-tetrahydro imidazol/2 1-b/thiazoles
CA982136A (en) * 1971-09-07 1976-01-20 Larry D. Spicer 6-(aminophenyl)-2,3,5,6-tetrahydro(2,1-b)thiazoles
JPS4839492A (xx) * 1971-09-23 1973-06-09
CH556871A (de) * 1971-09-24 1974-12-13 American Cyanamid Co Verfahren zur herstellung von substituierten 6-phenylimidazo (2,1-b)thiazolen.
FR2153206A2 (en) * 1971-09-24 1973-05-04 American Cyanamid Co Phenyl - dihydroimidazo (2,1-b) thiazole derivs - anthelmintics

Also Published As

Publication number Publication date
FI771362A (xx) 1977-11-02
AU2437377A (en) 1977-09-29
ATA305677A (de) 1979-08-15
IE45140B1 (en) 1982-06-30
CA1067082A (en) 1979-11-27
AR215629A1 (es) 1979-10-31
BE854073A (fr) 1977-10-28
SE7703553L (sv) 1977-11-02
FR2349592A1 (fr) 1977-11-25
PH11989A (en) 1978-10-05
CS189598B2 (en) 1979-04-30
PT66491B (en) 1978-09-29
LU77233A1 (xx) 1977-08-18
JPS52133998A (en) 1977-11-09
CH620218A5 (xx) 1980-11-14
NL162389C (nl) 1980-05-16
FI60712B (fi) 1981-11-30
DD130149A5 (de) 1978-03-08
NL7704662A (nl) 1977-11-03
GB1516938A (en) 1978-07-05
IL51875A0 (en) 1977-06-30
DK186877A (xx) 1977-11-02
AT355572B (de) 1980-03-10
DK142583C (xx) 1981-07-27
NL162389B (nl) 1979-12-17
FI60712C (fi) 1982-03-10
NZ183876A (en) 1979-03-16
JPS5713554B2 (xx) 1982-03-17
US4112102A (en) 1978-09-05
SE432423B (sv) 1984-04-02
ES458249A1 (es) 1978-06-01
IE45140L (en) 1977-11-01
PT66491A (en) 1977-05-01
FR2349592B1 (xx) 1980-09-19
YU102377A (en) 1982-06-30
DE2718976A1 (de) 1977-11-17

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