ES458249A1 - Procedimiento para preparar derivados de 6-(m-aminofenil)-2,3,5,6-tetrahidroimidazo (2,1-b)tiazol. - Google Patents
Procedimiento para preparar derivados de 6-(m-aminofenil)-2,3,5,6-tetrahidroimidazo (2,1-b)tiazol.Info
- Publication number
- ES458249A1 ES458249A1 ES458249A ES458249A ES458249A1 ES 458249 A1 ES458249 A1 ES 458249A1 ES 458249 A ES458249 A ES 458249A ES 458249 A ES458249 A ES 458249A ES 458249 A1 ES458249 A1 ES 458249A1
- Authority
- ES
- Spain
- Prior art keywords
- tetrahidroimidazo
- aminophenil
- thiazol
- procedure
- preparing derivatives
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Expired
Links
- FZWLAAWBMGSTSO-UHFFFAOYSA-N Thiazole Chemical compound C1=CSC=N1 FZWLAAWBMGSTSO-UHFFFAOYSA-N 0.000 title 1
- 239000002253 acid Substances 0.000 abstract 2
- IQGVBROUGQZILV-UHFFFAOYSA-N 3-(2,3,5,6-tetrahydroimidazo[2,1-b][1,3]thiazol-6-yl)aniline Chemical class NC1=CC=CC(C2N=C3SCCN3C2)=C1 IQGVBROUGQZILV-UHFFFAOYSA-N 0.000 abstract 1
- JUJWROOIHBZHMG-UHFFFAOYSA-N Pyridine Chemical group C1=CC=NC=C1 JUJWROOIHBZHMG-UHFFFAOYSA-N 0.000 abstract 1
- 125000006297 carbonyl amino group Chemical group [H]N([*:2])C([*:1])=O 0.000 abstract 1
- 150000001875 compounds Chemical class 0.000 abstract 1
- 238000004519 manufacturing process Methods 0.000 abstract 1
- 231100000252 nontoxic Toxicity 0.000 abstract 1
- 230000003000 nontoxic effect Effects 0.000 abstract 1
- 150000003839 salts Chemical class 0.000 abstract 1
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D213/00—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members
- C07D213/02—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members
- C07D213/04—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom
- C07D213/60—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D213/78—Carbon atoms having three bonds to hetero atoms, with at the most one bond to halogen, e.g. ester or nitrile radicals
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P33/00—Antiparasitic agents
- A61P33/10—Anthelmintics
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D213/00—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members
- C07D213/02—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members
- C07D213/04—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom
- C07D213/60—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D213/78—Carbon atoms having three bonds to hetero atoms, with at the most one bond to halogen, e.g. ester or nitrile radicals
- C07D213/79—Acids; Esters
- C07D213/80—Acids; Esters in position 3
Landscapes
- Organic Chemistry (AREA)
- Chemical & Material Sciences (AREA)
- Health & Medical Sciences (AREA)
- Veterinary Medicine (AREA)
- Chemical Kinetics & Catalysis (AREA)
- General Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Tropical Medicine & Parasitology (AREA)
- Pharmacology & Pharmacy (AREA)
- Life Sciences & Earth Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- General Health & Medical Sciences (AREA)
- Public Health (AREA)
- Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Abstract
Procedimiento para preparar derivados de 6-(m-aminofenil)-2,3,5,6-tetrahidroimidazo[2,1-b]tiazol, en particular la forma dl(racémica) ó `1 de un compuesto de fórmula *** en la que Hal es F, Cl, Br ó I y el grupo ¿CONH está unido a la posición 3 ó 4 de anillo piridina; y sus sales de adición de ácido atóxicas; caracterizado porque comprende reaccionar la forma dl(racémica) ó l de m-aminotetramisol con un ácido de fórmula: ***
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| GB17883/76A GB1516938A (en) | 1976-05-01 | 1976-05-01 | Halopyridylamides of m-aminotetramisole and their use as anthelmintics |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| ES458249A1 true ES458249A1 (es) | 1978-06-01 |
Family
ID=10102899
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| ES458249A Expired ES458249A1 (es) | 1976-05-01 | 1977-04-28 | Procedimiento para preparar derivados de 6-(m-aminofenil)-2,3,5,6-tetrahidroimidazo (2,1-b)tiazol. |
Country Status (24)
| Country | Link |
|---|---|
| US (1) | US4112102A (es) |
| JP (1) | JPS52133998A (es) |
| AR (1) | AR215629A1 (es) |
| AT (1) | AT355572B (es) |
| BE (1) | BE854073A (es) |
| CA (1) | CA1067082A (es) |
| CH (1) | CH620218A5 (es) |
| CS (1) | CS189598B2 (es) |
| DD (1) | DD130149A5 (es) |
| DE (1) | DE2718976A1 (es) |
| DK (1) | DK142583B (es) |
| ES (1) | ES458249A1 (es) |
| FI (1) | FI60712C (es) |
| FR (1) | FR2349592A1 (es) |
| GB (1) | GB1516938A (es) |
| IE (1) | IE45140B1 (es) |
| IL (1) | IL51875A0 (es) |
| LU (1) | LU77233A1 (es) |
| NL (1) | NL162389C (es) |
| NZ (1) | NZ183876A (es) |
| PH (1) | PH11989A (es) |
| PT (1) | PT66491B (es) |
| SE (1) | SE432423B (es) |
| YU (1) | YU102377A (es) |
Families Citing this family (2)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| EP0041322A1 (en) | 1980-05-30 | 1981-12-09 | Beecham Group Plc | m-Pyrazolylamido tetramisole derivatives, compositions thereof, processes for production of such compounds and compositions and their use in treating helminthiasis |
| WO2018231704A1 (en) * | 2017-06-12 | 2018-12-20 | Dow Agrosciences, Llc | 6-bromonicotinamide and processes of preparation |
Family Cites Families (7)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| NL131034C (es) * | 1964-05-11 | |||
| US3673205A (en) * | 1970-03-25 | 1972-06-27 | American Cyanamid Co | 6-(m-AMINO AND SUBSTITUTED-AMINO PHENYL)-2,3,5,6-TETRAHYDRO{8 2,1-b{9 THIAZOLES AND METHOD OF USE |
| GB1365515A (en) * | 1971-09-03 | 1974-09-04 | American Cyanamid Co | 6-tetrahydro imidazol/2 1-b/thiazoles |
| CA982136A (en) * | 1971-09-07 | 1976-01-20 | Larry D. Spicer | 6-(aminophenyl)-2,3,5,6-tetrahydro(2,1-b)thiazoles |
| JPS4839492A (es) * | 1971-09-23 | 1973-06-09 | ||
| CH556871A (de) * | 1971-09-24 | 1974-12-13 | American Cyanamid Co | Verfahren zur herstellung von substituierten 6-phenylimidazo (2,1-b)thiazolen. |
| FR2153206A2 (en) * | 1971-09-24 | 1973-05-04 | American Cyanamid Co | Phenyl - dihydroimidazo (2,1-b) thiazole derivs - anthelmintics |
-
1976
- 1976-05-01 GB GB17883/76A patent/GB1516938A/en not_active Expired
-
1977
- 1977-03-28 SE SE7703553A patent/SE432423B/xx unknown
- 1977-04-13 IL IL51875A patent/IL51875A0/xx unknown
- 1977-04-15 NZ NZ183876A patent/NZ183876A/xx unknown
- 1977-04-18 PH PH19684A patent/PH11989A/en unknown
- 1977-04-20 YU YU01023/77A patent/YU102377A/xx unknown
- 1977-04-26 CA CA276,958A patent/CA1067082A/en not_active Expired
- 1977-04-27 JP JP4900777A patent/JPS52133998A/ja active Granted
- 1977-04-28 FI FI771362A patent/FI60712C/fi not_active IP Right Cessation
- 1977-04-28 PT PT66491A patent/PT66491B/pt unknown
- 1977-04-28 BE BE177110A patent/BE854073A/xx not_active IP Right Cessation
- 1977-04-28 DE DE19772718976 patent/DE2718976A1/de not_active Withdrawn
- 1977-04-28 CS CS772804A patent/CS189598B2/cs unknown
- 1977-04-28 DD DD7700198638A patent/DD130149A5/xx unknown
- 1977-04-28 AR AR267385A patent/AR215629A1/es active
- 1977-04-28 ES ES458249A patent/ES458249A1/es not_active Expired
- 1977-04-28 NL NL7704662.A patent/NL162389C/xx not_active IP Right Cessation
- 1977-04-28 DK DK186877AA patent/DK142583B/da unknown
- 1977-04-29 FR FR7713038A patent/FR2349592A1/fr active Granted
- 1977-04-29 IE IE866/77A patent/IE45140B1/en unknown
- 1977-04-29 AT AT305677A patent/AT355572B/de not_active IP Right Cessation
- 1977-04-29 US US05/792,142 patent/US4112102A/en not_active Expired - Lifetime
- 1977-04-29 CH CH539477A patent/CH620218A5/fr not_active IP Right Cessation
- 1977-04-29 LU LU77233A patent/LU77233A1/xx unknown
Also Published As
| Publication number | Publication date |
|---|---|
| FI771362A (es) | 1977-11-02 |
| AU2437377A (en) | 1977-09-29 |
| ATA305677A (de) | 1979-08-15 |
| IE45140B1 (en) | 1982-06-30 |
| CA1067082A (en) | 1979-11-27 |
| AR215629A1 (es) | 1979-10-31 |
| BE854073A (fr) | 1977-10-28 |
| SE7703553L (sv) | 1977-11-02 |
| FR2349592A1 (fr) | 1977-11-25 |
| PH11989A (en) | 1978-10-05 |
| CS189598B2 (en) | 1979-04-30 |
| PT66491B (en) | 1978-09-29 |
| LU77233A1 (es) | 1977-08-18 |
| JPS52133998A (en) | 1977-11-09 |
| CH620218A5 (es) | 1980-11-14 |
| NL162389C (nl) | 1980-05-16 |
| FI60712B (fi) | 1981-11-30 |
| DD130149A5 (de) | 1978-03-08 |
| NL7704662A (nl) | 1977-11-03 |
| GB1516938A (en) | 1978-07-05 |
| IL51875A0 (en) | 1977-06-30 |
| DK186877A (es) | 1977-11-02 |
| AT355572B (de) | 1980-03-10 |
| DK142583C (es) | 1981-07-27 |
| NL162389B (nl) | 1979-12-17 |
| FI60712C (fi) | 1982-03-10 |
| NZ183876A (en) | 1979-03-16 |
| DK142583B (da) | 1980-11-24 |
| JPS5713554B2 (es) | 1982-03-17 |
| US4112102A (en) | 1978-09-05 |
| SE432423B (sv) | 1984-04-02 |
| IE45140L (en) | 1977-11-01 |
| PT66491A (en) | 1977-05-01 |
| FR2349592B1 (es) | 1980-09-19 |
| YU102377A (en) | 1982-06-30 |
| DE2718976A1 (de) | 1977-11-17 |
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Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| FD1A | Patent lapsed |
Effective date: 19990601 |