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DK1319007T3 - Kondenserede heterocykliske succinimidforbindelser og analoger deraf, modulatorer af nukleær hormonreceptorfunktion - Google Patents

Kondenserede heterocykliske succinimidforbindelser og analoger deraf, modulatorer af nukleær hormonreceptorfunktion

Info

Publication number
DK1319007T3
DK1319007T3 DK01948503T DK01948503T DK1319007T3 DK 1319007 T3 DK1319007 T3 DK 1319007T3 DK 01948503 T DK01948503 T DK 01948503T DK 01948503 T DK01948503 T DK 01948503T DK 1319007 T3 DK1319007 T3 DK 1319007T3
Authority
DK
Denmark
Prior art keywords
modulators
analogs
hormone receptor
receptor function
condensed heterocyclic
Prior art date
Application number
DK01948503T
Other languages
English (en)
Inventor
Mark E Salvati
Soren Giese
Aberra Fura
Wenying Li
Ramesh N Patel
Ronald L Hanson
James Aaron Balog
Dacia A Pickering
Original Assignee
Bristol Myers Squibb Co
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Bristol Myers Squibb Co filed Critical Bristol Myers Squibb Co
Application granted granted Critical
Publication of DK1319007T3 publication Critical patent/DK1319007T3/da

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    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D487/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
    • C07D487/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
    • C07D487/08—Bridged systems
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D491/00—Heterocyclic compounds containing in the condensed ring system both one or more rings having oxygen atoms as the only ring hetero atoms and one or more rings having nitrogen atoms as the only ring hetero atoms, not provided for by groups C07D451/00 - C07D459/00, C07D463/00, C07D477/00 or C07D489/00
    • C07D491/02—Heterocyclic compounds containing in the condensed ring system both one or more rings having oxygen atoms as the only ring hetero atoms and one or more rings having nitrogen atoms as the only ring hetero atoms, not provided for by groups C07D451/00 - C07D459/00, C07D463/00, C07D477/00 or C07D489/00 in which the condensed system contains two hetero rings
    • C07D491/08—Bridged systems
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
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    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/40—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with one nitrogen as the only ring hetero atom, e.g. sulpiride, succinimide, tolmetin, buflomedil
    • A61K31/407—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with one nitrogen as the only ring hetero atom, e.g. sulpiride, succinimide, tolmetin, buflomedil condensed with other heterocyclic ring systems, e.g. ketorolac, physostigmine
    • A—HUMAN NECESSITIES
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    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
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    • A61K31/655—Azo (—N=N—), diazo (=N2), azoxy (>N—O—N< or N(=O)—N<), azido (—N3) or diazoamino (—N=N—N<) compounds
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    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/66—Phosphorus compounds
    • A61K31/675—Phosphorus compounds having nitrogen as a ring hetero atom, e.g. pyridoxal phosphate
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    • A—HUMAN NECESSITIES
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    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D487/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
    • C07D487/12—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains three hetero rings
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    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D491/00—Heterocyclic compounds containing in the condensed ring system both one or more rings having oxygen atoms as the only ring hetero atoms and one or more rings having nitrogen atoms as the only ring hetero atoms, not provided for by groups C07D451/00 - C07D459/00, C07D463/00, C07D477/00 or C07D489/00
    • C07D491/12—Heterocyclic compounds containing in the condensed ring system both one or more rings having oxygen atoms as the only ring hetero atoms and one or more rings having nitrogen atoms as the only ring hetero atoms, not provided for by groups C07D451/00 - C07D459/00, C07D463/00, C07D477/00 or C07D489/00 in which the condensed system contains three hetero rings
    • C07D491/18—Bridged systems
    • C—CHEMISTRY; METALLURGY
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    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D491/00—Heterocyclic compounds containing in the condensed ring system both one or more rings having oxygen atoms as the only ring hetero atoms and one or more rings having nitrogen atoms as the only ring hetero atoms, not provided for by groups C07D451/00 - C07D459/00, C07D463/00, C07D477/00 or C07D489/00
    • C07D491/22—Heterocyclic compounds containing in the condensed ring system both one or more rings having oxygen atoms as the only ring hetero atoms and one or more rings having nitrogen atoms as the only ring hetero atoms, not provided for by groups C07D451/00 - C07D459/00, C07D463/00, C07D477/00 or C07D489/00 in which the condensed system contains four or more hetero rings
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
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    • C07D495/12—Heterocyclic compounds containing in the condensed system at least one hetero ring having sulfur atoms as the only ring hetero atoms in which the condensed system contains three hetero rings
    • C07D495/18—Bridged systems
    • C—CHEMISTRY; METALLURGY
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    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D519/00—Heterocyclic compounds containing more than one system of two or more relevant hetero rings condensed among themselves or condensed with a common carbocyclic ring system not provided for in groups C07D453/00 or C07D455/00

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DK01948503T 2000-09-19 2001-06-20 Kondenserede heterocykliske succinimidforbindelser og analoger deraf, modulatorer af nukleær hormonreceptorfunktion DK1319007T3 (da)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US23351900P 2000-09-19 2000-09-19
US28443801P 2001-04-18 2001-04-18
US28473001P 2001-04-18 2001-04-18

Publications (1)

Publication Number Publication Date
DK1319007T3 true DK1319007T3 (da) 2006-06-19

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DK01948503T DK1319007T3 (da) 2000-09-19 2001-06-20 Kondenserede heterocykliske succinimidforbindelser og analoger deraf, modulatorer af nukleær hormonreceptorfunktion

Country Status (36)

Country Link
US (1) US20040176324A1 (da)
EP (1) EP1319007B9 (da)
JP (1) JP4966477B2 (da)
KR (1) KR100765670B1 (da)
CN (2) CN1307181C (da)
AR (1) AR035340A1 (da)
AT (1) ATE318822T1 (da)
AU (2) AU2001269943B2 (da)
BG (1) BG107675A (da)
BR (1) BR0113980A (da)
CA (1) CA2423071A1 (da)
CZ (1) CZ2003780A3 (da)
DE (1) DE60117551T2 (da)
DK (1) DK1319007T3 (da)
EE (1) EE200300108A (da)
ES (1) ES2260244T3 (da)
GE (1) GEP20074144B (da)
HK (1) HK1054230B (da)
HR (1) HRP20030305B9 (da)
HU (1) HUP0400455A3 (da)
IL (1) IL155019A0 (da)
IS (1) IS6750A (da)
MX (1) MXPA03002412A (da)
MY (1) MY138531A (da)
NO (1) NO329931B1 (da)
NZ (1) NZ524803A (da)
PE (1) PE20020729A1 (da)
PL (1) PL361707A1 (da)
PT (1) PT1319007E (da)
SK (1) SK4982003A3 (da)
TW (1) TWI305208B (da)
UA (1) UA78686C2 (da)
UY (1) UY26808A1 (da)
WO (1) WO2002024702A1 (da)
YU (1) YU20003A (da)
ZA (1) ZA200302963B (da)

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EP1319007B1 (en) 2006-03-01
NO20031266L (no) 2003-05-13
HUP0400455A2 (hu) 2004-06-28
IS6750A (is) 2003-03-18
SK4982003A3 (en) 2004-05-04
EP1319007A1 (en) 2003-06-18
WO2002024702A1 (en) 2002-03-28
ZA200302963B (en) 2004-07-15
DE60117551D1 (de) 2006-04-27
AU2001269943B2 (en) 2006-11-09
CN1608069A (zh) 2005-04-20
KR20030028847A (ko) 2003-04-10
GEP20074144B (en) 2007-07-10
ES2260244T3 (es) 2006-11-01
CA2423071A1 (en) 2002-03-28
EE200300108A (et) 2005-02-15
PT1319007E (pt) 2006-05-31
TWI305208B (en) 2009-01-11
HUP0400455A3 (en) 2007-10-29
EP1319007B9 (en) 2007-10-10
HRP20030305A2 (en) 2005-04-30
DE60117551T2 (de) 2007-01-18
PL361707A1 (en) 2004-10-04
PE20020729A1 (es) 2002-08-11
ATE318822T1 (de) 2006-03-15
AU6994301A (en) 2002-04-02
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JP4966477B2 (ja) 2012-07-04
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