DK1222173T3 - Fremgangsmåde til fremstilling af 4-trifluormethylsulphinylpyrazolderivat - Google Patents

Fremgangsmåde til fremstilling af 4-trifluormethylsulphinylpyrazolderivat

Info

Publication number: DK1222173T3
Authority: DK; Denmark
Prior art keywords: sub; compound; preparation; formula; trifluoromethylsulphinylpyrazole
Prior art date: 1999-10-22

Application number

DK99955978T

Other languages

English (en)

Inventor

Jean-Louis Clavel

Isabelle Pelta

Bars Sylvie Le

Philippe Charreau

Original Assignee

Bayer Cropscience Sa

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

1999-10-22

Filing date

1999-10-22

Publication date

2004-09-20

Family has litigation

First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=8167491&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=DK1222173(T3) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.

1999-10-22 Application filed by Bayer Cropscience Sa filed Critical Bayer Cropscience Sa

2004-09-20 Application granted granted Critical

2004-09-20 Publication of DK1222173T3 publication Critical patent/DK1222173T3/da

Classifications

- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
- C07D401/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
- C07D401/04—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings directly linked by a ring-member-to-ring-member bond
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D231/00—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings
- C07D231/02—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings
- C07D231/10—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
- C07D231/14—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D231/44—Oxygen and nitrogen or sulfur and nitrogen atoms

Landscapes

Chemical & Material Sciences (AREA)
Organic Chemistry (AREA)
Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
Plural Heterocyclic Compounds (AREA)
Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Low-Molecular Organic Synthesis Reactions Using Catalysts (AREA)
Agricultural Chemicals And Associated Chemicals (AREA)
Preparation Of Compounds By Using Micro-Organisms (AREA)

DK99955978T 1999-10-22 1999-10-22 Fremgangsmåde til fremstilling af 4-trifluormethylsulphinylpyrazolderivat DK1222173T3 (da)

Applications Claiming Priority (1)

Application Number	Priority Date	Filing Date	Title
PCT/EP1999/008687 WO2001030760A1 (en)	1999-10-22	1999-10-22	Process for preparing 4-trifluoromethylsulphinylpyrazole derivative

Publications (1)

Publication Number	Publication Date
DK1222173T3 true DK1222173T3 (da)	2004-09-20

Family

ID=8167491

Family Applications (1)

Application Number	Title	Priority Date	Filing Date
DK99955978T DK1222173T3 (da)	1999-10-22	1999-10-22	Fremgangsmåde til fremstilling af 4-trifluormethylsulphinylpyrazolderivat

Country Status (30)

Country	Link
US (2)	US6620943B1 (da)
EP (1)	EP1222173B1 (da)
JP (1)	JP4666863B2 (da)
KR (2)	KR100665598B1 (da)
CN (3)	CN1896066B (da)
AT (1)	ATE273961T1 (da)
AU (1)	AU783139B2 (da)
BG (1)	BG65483B1 (da)
BR (1)	BR9917518B1 (da)
CA (1)	CA2384283C (da)
CZ (1)	CZ299822B6 (da)
DE (1)	DE69919599T2 (da)
DK (1)	DK1222173T3 (da)
EA (1)	EA005077B1 (da)
ES (1)	ES2222743T3 (da)
HR (1)	HRP20020438B1 (da)
HU (1)	HU229393B1 (da)
IL (2)	IL149152A0 (da)
IN (2)	IN2005MU00818A (da)
ME (1)	MEP7808A (da)
MX (1)	MX229662B (da)
NZ (2)	NZ517770A (da)
PL (1)	PL206482B1 (da)
PT (1)	PT1222173E (da)
RO (1)	RO121209B1 (da)
TR (2)	TR200201072T2 (da)
TW (1)	TW553936B (da)
UA (1)	UA73752C2 (da)
WO (1)	WO2001030760A1 (da)
ZA (1)	ZA200201961B (da)

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DE60036290T2 (de)	1999-06-29	2008-06-05	Nihon Nohyaku Kabushiki Kaisha	Pyrazolderivate und verfahren zu ihrer herstellung und pestizide die diese als aktive inhaltsstoffe enthalten
WO2005023774A1 (en) *	2003-09-11	2005-03-17	Cheminova A/S	Process for the preparation of a trifluoromethylthioether
CN100586934C (zh) *	2003-11-07	2010-02-03	凯米诺瓦有限公司	制备三氟甲基硫醚的方法
DE102004020069C5 (de)	2004-04-24	2013-12-05	Voith Patent Gmbh	Verfahren zum Satinieren einer Papierbahn
AU2013203222B2 (en) *	2005-12-14	2015-08-20	Adama Makhteshim Ltd.	Polymorphs and amorphous forms of 5-amino-1-[2,6- dichloro-4-(trifluoromethyl)phenyl]-4- [(trifluoromethyl)sulfinyl]-1H-pyrazole-3-carbonitrile
JP5396085B2 (ja)	2005-12-14	2014-01-22	マクテシム・ケミカル・ワークス・リミテツド	５−アミノ−１−［２，６−ジクロロ−４−（トリフルオロメチル）フェニル］−４−［（トリフルオロメチル）スルフィニル］−１ｈ−ピラゾール−３−カルボニトリルの多形および非晶形
EP2069311B1 (en)	2006-04-25	2012-05-16	Gharda Chemicals Limited	Process for the preparation of fipronil, an insecticide, and related pyrazoles
CN101168529B (zh) *	2006-10-24	2011-03-23	温州大学	氟虫腈、乙虫腈及其衍生物的合成方法
AU2007316720B2 (en)	2006-11-10	2013-05-09	Basf Se	Process for the sulfinylation of a pyrazole derivative
WO2008055884A1 (en) *	2006-11-10	2008-05-15	Basf Se	Crystalline modification of fipronil
BRPI0718774A2 (pt)	2006-11-10	2013-12-03	Basf Se	"processo para a sulfinilação de um derivado de pirazol, 5-amino-1-[2,6-dicloro-4-(trifluorometil) fenil] -4-(trifluorometilsulfinil) -pirazol-3-carbonitrila, composição pesticida ou parasiticida, uso, métodos para o controle de insetos, acarídeos ou nematódeos, de proteger plantas em crescimento, para tratar, controlar, prevenir ou proteger animais, e, processo para a preparação de uma composição."
KR101540122B1 (ko) *	2006-11-10	2015-07-28	바스프 에스이	피프로닐의 결정질 변형물
AU2007316639B2 (en)	2006-11-10	2012-12-20	Basf Se	Crystalline modification of fipronil
UA110598C2 (uk)	2006-11-10	2016-01-25	Басф Се	Спосіб одержання кристалічної модифікації фіпронілу
CN102171182B (zh)	2008-10-02	2015-07-22	巴斯夫欧洲公司	生产和提纯三氟甲烷亚磺酸的方法
WO2010049746A1 (en) *	2008-10-27	2010-05-06	Dynamit Nobel Gmbh Explosivstoff-Und Systemtechnic	Process for the synthesis of fipronil
US8476459B2 (en)	2009-10-30	2013-07-02	Basf Se	Process for the preparation of 4-sulfinyl-pyrazole derivatives
AU2010100462A4 (en)	2010-03-03	2010-06-17	Keki Hormusji Gharda	A process for the synthesis of Fipronil
IT1400666B1 (it)	2010-07-07	2013-06-28	Finchimica Srl	Procedimento per la sintesi di 5-amino, 1-fenil, 3-ciano, 4-trifluorometil sulfinil pirazoli.
CN103153961A (zh)	2010-07-12	2013-06-12	塞尔休斯物业公司埃尔维塔植物保护分公司	氟虫腈制备方法
EP2663192A4 (en) *	2011-01-14	2015-06-03	Keki Hormusji Gharda	POLYMORPHISMS IN 5-AMINO-1- (2,6-DICHLOR-4-TRIFLUOROMETHYLPHENYL-) 3-CYAN-4-TRIFLUOR-METHYL-SULFINYL-PYRAZOLE
EP2714664B1 (en)	2011-05-30	2016-10-19	Keki Hormusji Gharda	Process for synthesis of fipronil
CN102633722B (zh) *	2012-03-20	2015-05-06	金坛市凌云动物保健品有限公司	一种非泼罗尼的制备方法
TWI579274B (zh) *	2012-04-20	2017-04-21	龍馬躍公司	製備１－芳基－５－烷基吡唑化合物的改良方法
CN102690232A (zh) *	2012-05-30	2012-09-26	河南中医学院	一种氟虫腈中间体的合成方法
US8993613B2 (en)	2013-04-17	2015-03-31	The Hartz Mountain Corporation	Ectoparasiticidal formulations
CN105254565A (zh) *	2015-09-30	2016-01-20	乐平市康鑫医药化工有限公司	由氰基吡唑一锅法合成硫醚的工艺方法
CN106977460A (zh) *	2017-04-19	2017-07-25	江苏托球农化股份有限公司	1‑(2,6‑二氯‑4‑三氟甲基)苯基‑3‑氰基‑4‑乙巯基‑5‑氨基吡唑的合成
EP3412658A1 (en)	2017-06-09	2018-12-12	Solvay Sa	Processes for the manufacture of sulfur-substitued pyrazole derivatives
EP3412659A1 (en)	2017-06-09	2018-12-12	Solvay Sa	Processes for the manufacture of sulfur-substituted pyrazole derivatives
CN112430213A (zh) *	2020-12-03	2021-03-02	江苏优普生物化学科技股份有限公司	一种三氟甲硫基吡唑合成工艺
CN113149909B (zh) *	2021-03-24	2022-04-19	台州达辰药业有限公司	5-氨基-3-氰基-1-(2,6-二氯-4-三氟甲基-苯基)吡唑二硫化物制备方法
CN113480482B (zh) *	2021-07-05	2022-11-18	海正药业南通有限公司	一种非泼罗尼中间体的合成方法
CN114213330A (zh) *	2021-12-29	2022-03-22	天和药业股份有限公司	一种氟虫腈精制母液的处理方法

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FR2716453B1 (fr)	1994-02-22	1996-03-29	Rhone Poulenc Agrochimie	Procédé de sulfinylation de composés hétérocycliques.
DE3602728A1 (de) *	1985-05-17	1986-11-20	Bayer Ag, 51373 Leverkusen	Schaedlingsbekaempfungsmittel auf basis von pyrazolderivaten
US5232940A (en)	1985-12-20	1993-08-03	Hatton Leslie R	Derivatives of N-phenylpyrazoles
US5547974A (en) *	1985-12-20	1996-08-20	Rhone-Poulenc Agriculture Ltd.	Derivatives of N-phenylpyrazoles
GB8713768D0 (en) *	1987-06-12	1987-07-15	May & Baker Ltd	Compositions of matter
CA2004776C (fr) *	1988-12-13	2000-04-25	Claude Wakselman	Procede de preparation de perfluoroalkylthioethers

1999
- 1999-10-22 KR KR1020027005011A patent/KR100665598B1/ko not_active Expired - Fee Related
- 1999-10-22 AU AU12707/00A patent/AU783139B2/en not_active Expired
- 1999-10-22 CZ CZ20021384A patent/CZ299822B6/cs not_active IP Right Cessation
- 1999-10-22 ME MEP-78/08A patent/MEP7808A/xx unknown
- 1999-10-22 ES ES99955978T patent/ES2222743T3/es not_active Expired - Lifetime
- 1999-10-22 PT PT99955978T patent/PT1222173E/pt unknown
- 1999-10-22 CN CN2004101300014A patent/CN1896066B/zh not_active Expired - Lifetime
- 1999-10-22 NZ NZ517770A patent/NZ517770A/en not_active IP Right Cessation
- 1999-10-22 NZ NZ527896A patent/NZ527896A/en not_active IP Right Cessation
- 1999-10-22 HU HU0203206A patent/HU229393B1/hu unknown
- 1999-10-22 CN CNB998060828A patent/CN1163488C/zh not_active Expired - Lifetime
- 1999-10-22 IL IL14915299A patent/IL149152A0/xx active IP Right Grant
- 1999-10-22 EP EP99955978A patent/EP1222173B1/en not_active Expired - Lifetime
- 1999-10-22 DE DE69919599T patent/DE69919599T2/de not_active Expired - Lifetime
- 1999-10-22 EA EA200200481A patent/EA005077B1/ru not_active IP Right Cessation
- 1999-10-22 MX MXPA02003944 patent/MX229662B/es active IP Right Grant
- 1999-10-22 TR TR2002/01072T patent/TR200201072T2/xx unknown
- 1999-10-22 BR BRPI9917518-5A patent/BR9917518B1/pt not_active IP Right Cessation
- 1999-10-22 WO PCT/EP1999/008687 patent/WO2001030760A1/en active Application Filing
- 1999-10-22 TR TR2002/02806T patent/TR200202806T2/xx unknown
- 1999-10-22 IN IN818MU2005 patent/IN2005MU00818A/en unknown
- 1999-10-22 UA UA2002054165A patent/UA73752C2/uk unknown
- 1999-10-22 RO ROA200200317A patent/RO121209B1/ro unknown
- 1999-10-22 HR HR20020438A patent/HRP20020438B1/xx not_active IP Right Cessation
- 1999-10-22 DK DK99955978T patent/DK1222173T3/da active
- 1999-10-22 US US10/111,000 patent/US6620943B1/en not_active Expired - Lifetime
- 1999-10-22 KR KR1020067017067A patent/KR100665599B1/ko not_active Expired - Fee Related
- 1999-10-22 AT AT99955978T patent/ATE273961T1/de active
- 1999-10-22 CN CN2008101863366A patent/CN101445483B/zh not_active Expired - Lifetime
- 1999-10-22 CA CA002384283A patent/CA2384283C/en not_active Expired - Fee Related
- 1999-10-22 JP JP2001533114A patent/JP4666863B2/ja not_active Expired - Fee Related
- 1999-10-22 PL PL354611A patent/PL206482B1/pl not_active IP Right Cessation
2000
- 2000-10-11 TW TW089121214A patent/TW553936B/zh not_active IP Right Cessation
2002
- 2002-03-08 ZA ZA200201961A patent/ZA200201961B/en unknown
- 2002-04-01 IN IN312MU2002 patent/IN2002MU00312A/en unknown
- 2002-04-15 IL IL149152A patent/IL149152A/en not_active IP Right Cessation
- 2002-04-17 BG BG106622A patent/BG65483B1/bg unknown
2003
- 2003-07-03 US US10/611,979 patent/US6881848B2/en not_active Expired - Fee Related

Also Published As

Publication number	Publication date
KR20060097747A (ko)	2006-09-14
BG106622A (en)	2002-12-29
CN1896066A (zh)	2007-01-17
TW553936B (en)	2003-09-21
PL354611A1 (en)	2004-02-09
EA200200481A1 (ru)	2002-10-31
JP4666863B2 (ja)	2011-04-06
KR100665599B1 (ko)	2007-01-10
HUP0203206A2 (hu)	2003-03-28
ATE273961T1 (de)	2004-09-15
HU229393B1 (en)	2013-11-28
HRP20020438B1 (en)	2011-01-31
IN192712B (da)	2004-05-15
EP1222173B1 (en)	2004-08-18
AU783139B2 (en)	2005-09-29
UA73752C2 (en)	2005-09-15
CZ299822B6 (cs)	2008-12-03
CN1896066B (zh)	2011-06-15
ZA200201961B (en)	2003-05-28
NZ527896A (en)	2004-07-30
DE69919599D1 (de)	2004-09-23
CN1332730A (zh)	2002-01-23
KR20020040899A (ko)	2002-05-30
PL206482B1 (pl)	2010-08-31
JP2003512456A (ja)	2003-04-02
BR9917518B1 (pt)	2009-08-11
ES2222743T3 (es)	2005-02-01
US6620943B1 (en)	2003-09-16
IL149152A0 (en)	2002-11-10
BG65483B1 (bg)	2008-09-30
AU1270700A (en)	2001-05-08
CN1163488C (zh)	2004-08-25
PT1222173E (pt)	2004-11-30
RO121209B1 (ro)	2007-01-30
CN101445483B (zh)	2011-03-30
HRP20020438A2 (en)	2004-08-31
IN2005MU00818A (da)	2005-11-11
HUP0203206A3 (en)	2005-11-28
MXPA02003944A (es)	2003-10-15
CA2384283A1 (en)	2001-05-03
MEP7808A (en)	2010-06-10
CA2384283C (en)	2009-02-03
IN2002MU00312A (da)	2007-06-29
MX229662B (es)	2005-08-04
WO2001030760A1 (en)	2001-05-03
CN101445483A (zh)	2009-06-03
BR9917518A (pt)	2002-06-18
DE69919599T2 (de)	2005-08-11
KR100665598B1 (ko)	2007-01-10
EA005077B1 (ru)	2004-10-28
TR200202806T2 (tr)	2003-03-21
US6881848B2 (en)	2005-04-19
US20040034234A1 (en)	2004-02-19
IL149152A (en)	2008-08-07
EP1222173A1 (en)	2002-07-17
NZ517770A (en)	2003-11-28
CZ20021384A3 (cs)	2002-08-14
TR200201072T2 (tr)	2002-07-22

Publication	Publication Date	Title
DK1222173T3 (da)	2004-09-20	Fremgangsmåde til fremstilling af 4-trifluormethylsulphinylpyrazolderivat
BR0313341A (pt)	2005-07-12	Método para a preparação de uma oxazinona fundida e método para a preparação de um composto de fórmula iii
SG114563A1 (en)	2005-09-28	Microbicidal and algicidal composition, microbicidal and algicidal process for a water system and process for producing a microbicidal and algicidal comosition
BRPI0406500A (pt)	2008-07-22	processo farmacêutico e compostos preparados pelo mesmo
KR830007662A (ko)	1983-11-04	5,6,7,7a-테트라하이드로-4H-티에노 [3,2-c]-피리딘-2-온 유도체의 제조방법
KR840008155A (ko)	1984-12-13	트리아조로[4,3,-c] 피리미딘과 트리아조로[1,5-c]피리미딘의 제조방법
DK1021416T3 (da)	2004-09-27	Fremgangsmåde til fremstilling af substituerede pyrazoler
ATE442849T1 (de)	2009-10-15	Wässrige zusammensetzung mit einem thiazol- derivat
EA199900754A1 (ru)	2000-04-24	Способ получения замещенного тиазолидиндиона
BR0009453B1 (pt)	2011-03-22	processo para a preparação de um composto.
KR860001808A (ko)	1986-03-22	이미다조〔1,5-a〕피리미딘 유도체의 제조방법
KR860008983A (ko)	1986-12-19	4- 벤조일-1- 알킬(알켄일) 피라졸의 제조방법
RS49983B (sr)	2008-09-29	Postupak dobijanja 3-acil-indola
KR960702432A (ko)	1996-04-27	P-알킬- 및p-아릴설포닐벤조산 유도체의 제조방법(process to prepare p-alkyl-and p-arylsulphonylbenzoic acid derivatives)
KR960701001A (ko)	1996-02-24	디아조메탄 유도체의 제조 방법(Process for Producing Diazomethane Derivative)
KR850008169A (ko)	1985-12-13	1-헤테로아릴-4-아릴-피라졸린-5-온의 제조방법
DE602004032024D1 (de)	2011-05-12	Behandlung hochleistungsfähiger pigmentfarbstoffe mit dispergierenden etheramin-salzen
PT859795E (pt)	2003-08-29	Processo para a preparacao de ferro-dextrano cristalino
EA200100601A1 (ru)	2001-10-22	Производные 3-(гетероциклил) бензоилпиразолов
PE20010090A1 (es)	2001-02-22	Sal de acido fosforico de una diamina aromatica
DE60302217D1 (de)	2005-12-15	Trizyklo-imidazolinen derivaten, verfahren zu deren herstellung und deren verwendung als heilmitteln
KR870001210A (ko)	1987-03-12	퀴놀론 카복실산 및 이의 유도체의 엠보네이트의 제조방법
AR023181A1 (es)	2002-09-04	Un procedimiento para preparar una fenilhidrazina
TH31600A (th)	1999-01-11	เกลือของกรดแคลวูแลนิค
DE60206051D1 (de)	2005-10-13	Verfahren zur herstellung organischen nanoröhrchen, insbesondere aus lithocholsäure und ihre anwendungen