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DK113427B - Fremgangsmåde til fremstilling af angulære cyano- eller carboxamidoderivater af polyhydronaphthalener, polyhydrophenanthrener, polyhydrochrysener eller cyclopentanopolyhydrophenanthrener eller ketaler, estere eller ethere deraf. - Google Patents

Fremgangsmåde til fremstilling af angulære cyano- eller carboxamidoderivater af polyhydronaphthalener, polyhydrophenanthrener, polyhydrochrysener eller cyclopentanopolyhydrophenanthrener eller ketaler, estere eller ethere deraf.

Info

Publication number
DK113427B
DK113427B DK104661AA DK104661A DK113427B DK 113427 B DK113427 B DK 113427B DK 104661A A DK104661A A DK 104661AA DK 104661 A DK104661 A DK 104661A DK 113427 B DK113427 B DK 113427B
Authority
DK
Denmark
Prior art keywords
polyhydrophenanthrenes
polyhydronaphthalenes
polyhydrochrysenes
cyclopentanopolyhydrophenanthrenes
ketals
Prior art date
Application number
DK104661AA
Other languages
English (en)
Inventor
W Nagata
Original Assignee
Shionogi & Co
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Shionogi & Co filed Critical Shionogi & Co
Publication of DK113427B publication Critical patent/DK113427B/da

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07J—STEROIDS
    • C07J71/00—Steroids in which the cyclopenta(a)hydrophenanthrene skeleton is condensed with a heterocyclic ring
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C29/00—Preparation of compounds having hydroxy or O-metal groups bound to a carbon atom not belonging to a six-membered aromatic ring
    • C07C29/132—Preparation of compounds having hydroxy or O-metal groups bound to a carbon atom not belonging to a six-membered aromatic ring by reduction of an oxygen containing functional group
    • C07C29/136—Preparation of compounds having hydroxy or O-metal groups bound to a carbon atom not belonging to a six-membered aromatic ring by reduction of an oxygen containing functional group of >C=O containing groups, e.g. —COOH
    • C07C29/147—Preparation of compounds having hydroxy or O-metal groups bound to a carbon atom not belonging to a six-membered aromatic ring by reduction of an oxygen containing functional group of >C=O containing groups, e.g. —COOH of carboxylic acids or derivatives thereof
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C35/00—Compounds having at least one hydroxy or O-metal group bound to a carbon atom of a ring other than a six-membered aromatic ring
    • C07C35/22—Compounds having at least one hydroxy or O-metal group bound to a carbon atom of a ring other than a six-membered aromatic ring polycyclic, at least one hydroxy group bound to a condensed ring system
    • C07C35/44—Compounds having at least one hydroxy or O-metal group bound to a carbon atom of a ring other than a six-membered aromatic ring polycyclic, at least one hydroxy group bound to a condensed ring system with a hydroxy group on a condensed ring system having more than three rings
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C62/00—Compounds having carboxyl groups bound to carbon atoms of rings other than six—membered aromatic rings and containing any of the groups OH, O—metal, —CHO, keto, ether, groups, groups, or groups
    • C07C62/18—Saturated compounds containing keto groups
    • C07C62/26—Saturated compounds containing keto groups containing singly bound oxygen-containing groups
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07J—STEROIDS
    • C07J1/00—Normal steroids containing carbon, hydrogen, halogen or oxygen, not substituted in position 17 beta by a carbon atom, e.g. estrane, androstane
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07J—STEROIDS
    • C07J21/00—Normal steroids containing carbon, hydrogen, halogen or oxygen having an oxygen-containing hetero ring spiro-condensed with the cyclopenta(a)hydrophenanthrene skeleton
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07J—STEROIDS
    • C07J5/00—Normal steroids containing carbon, hydrogen, halogen or oxygen, substituted in position 17 beta by a chain of two carbon atoms, e.g. pregnane and substituted in position 21 by only one singly bound oxygen atom, i.e. only one oxygen bound to position 21 by a single bond
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07J—STEROIDS
    • C07J63/00—Steroids in which the cyclopenta(a)hydrophenanthrene skeleton has been modified by expansion of only one ring by one or two atoms
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07J—STEROIDS
    • C07J63/00—Steroids in which the cyclopenta(a)hydrophenanthrene skeleton has been modified by expansion of only one ring by one or two atoms
    • C07J63/008—Expansion of ring D by one atom, e.g. D homo steroids
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07J—STEROIDS
    • C07J7/00—Normal steroids containing carbon, hydrogen, halogen or oxygen substituted in position 17 beta by a chain of two carbon atoms
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07J—STEROIDS
    • C07J71/00—Steroids in which the cyclopenta(a)hydrophenanthrene skeleton is condensed with a heterocyclic ring
    • C07J71/0036—Nitrogen-containing hetero ring
    • C07J71/0042—Nitrogen only
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07J—STEROIDS
    • C07J75/00—Processes for the preparation of steroids in general
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07J—STEROIDS
    • C07J9/00—Normal steroids containing carbon, hydrogen, halogen or oxygen substituted in position 17 beta by a chain of more than two carbon atoms, e.g. cholane, cholestane, coprostane
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C2603/00—Systems containing at least three condensed rings
    • C07C2603/02—Ortho- or ortho- and peri-condensed systems
    • C07C2603/04—Ortho- or ortho- and peri-condensed systems containing three rings
    • C07C2603/22—Ortho- or ortho- and peri-condensed systems containing three rings containing only six-membered rings
    • C07C2603/26—Phenanthrenes; Hydrogenated phenanthrenes
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C2603/00—Systems containing at least three condensed rings
    • C07C2603/02—Ortho- or ortho- and peri-condensed systems
    • C07C2603/40—Ortho- or ortho- and peri-condensed systems containing four condensed rings
    • C07C2603/42—Ortho- or ortho- and peri-condensed systems containing four condensed rings containing only six-membered rings
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C2603/00—Systems containing at least three condensed rings
    • C07C2603/02—Ortho- or ortho- and peri-condensed systems
    • C07C2603/40—Ortho- or ortho- and peri-condensed systems containing four condensed rings
    • C07C2603/42—Ortho- or ortho- and peri-condensed systems containing four condensed rings containing only six-membered rings
    • C07C2603/48—Chrysenes; Hydrogenated chrysenes

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Steroid Compounds (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
DK104661AA 1960-03-12 1961-03-10 Fremgangsmåde til fremstilling af angulære cyano- eller carboxamidoderivater af polyhydronaphthalener, polyhydrophenanthrener, polyhydrochrysener eller cyclopentanopolyhydrophenanthrener eller ketaler, estere eller ethere deraf. DK113427B (da)

Applications Claiming Priority (8)

Application Number Priority Date Filing Date Title
JP820860 1960-03-12
JP942160 1960-03-19
JP2012460 1960-04-04
JP2012560 1960-04-04
JP2072360 1960-04-06
JP2241760 1960-04-21
JP2261160 1960-04-25
JP2598661 1961-07-19

Publications (1)

Publication Number Publication Date
DK113427B true DK113427B (da) 1969-03-24

Family

ID=27571631

Family Applications (1)

Application Number Title Priority Date Filing Date
DK104661AA DK113427B (da) 1960-03-12 1961-03-10 Fremgangsmåde til fremstilling af angulære cyano- eller carboxamidoderivater af polyhydronaphthalener, polyhydrophenanthrener, polyhydrochrysener eller cyclopentanopolyhydrophenanthrener eller ketaler, estere eller ethere deraf.

Country Status (7)

Country Link
US (4) US3206472A (da)
CH (6) CH416602A (da)
DE (5) DE1234714B (da)
DK (1) DK113427B (da)
FR (1) FR1517665A (da)
GB (9) GB915892A (da)
NL (2) NL6512737A (da)

Families Citing this family (7)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
NL113064C (da) * 1960-03-12
US3294817A (en) * 1964-03-23 1966-12-27 American Home Prod Octahydroindolobenzazepines and compounds intermediate thereto
US3835160A (en) * 1967-06-06 1974-09-10 Schering Corp 3{40 -keto-2{40 ,3{40 -seco-1{40 -(2{40 )-yne steroidal derivatives, methods for their manufacture, and compounds produced thereby
US3898264A (en) * 1970-08-26 1975-08-05 Hoffmann La Roche Steroid total synthesis process utilizing a cyanoalkyl A-ring precursor
US5028631A (en) * 1987-11-25 1991-07-02 Schwartz Arthur G Homoandrostan-17-one and homoandrosten-17-ones
US5480913A (en) * 1989-09-27 1996-01-02 Arch Development Corporation Anti-androgen compounds
US5116865A (en) * 1990-09-05 1992-05-26 Peters Richard H 15,16-seco-19-nor progestins

Family Cites Families (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3024271A (en) * 1958-08-08 1962-03-06 Lab Francais Chimiotherapie 3, 11, 17-trioxygenated-18-nor-d-homo-13alpha-steroids and processes for their preparation
NL113064C (da) * 1960-03-12

Also Published As

Publication number Publication date
CH491886A (de) 1970-06-15
GB945518A (en) 1964-01-02
DE1234714B (de) 1967-02-23
GB984024A (en) 1965-02-24
GB915892A (en) 1963-01-16
CH416602A (de) 1966-07-15
US3407212A (en) 1968-10-22
CH430707A (de) 1967-02-28
NL6512737A (da) 1965-12-27
DE1203262B (de) 1965-10-21
GB984023A (en) 1965-02-24
GB959799A (en) 1964-06-03
US3206472A (en) 1965-09-14
DE1593385A1 (de) 1971-03-25
CH406202A (de) 1966-01-31
GB936892A (en) 1963-09-18
GB984022A (en) 1965-02-24
GB984021A (en) 1965-02-24
CH400138A (de) 1965-10-15
DE1260466B (de) 1968-02-08
NL113064C (da)
US3197485A (en) 1965-07-27
CH419113A (de) 1966-08-31
DE1172670B (de) 1964-06-25
GB959798A (en) 1964-06-03
FR1517665A (fr) 1968-03-22
US3403167A (en) 1968-09-24
DE1191808B (de) 1965-04-29

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