DE69908951D1 - Kristallformen von osanetant - Google Patents
Kristallformen von osanetantInfo
- Publication number
- DE69908951D1 DE69908951D1 DE69908951T DE69908951T DE69908951D1 DE 69908951 D1 DE69908951 D1 DE 69908951D1 DE 69908951 T DE69908951 T DE 69908951T DE 69908951 T DE69908951 T DE 69908951T DE 69908951 D1 DE69908951 D1 DE 69908951D1
- Authority
- DE
- Germany
- Prior art keywords
- osanetant
- crystal forms
- crystal
- forms
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Expired - Fee Related
Links
- 239000013078 crystal Substances 0.000 title 1
- DZOJBGLFWINFBF-UMSFTDKQSA-N osanetant Chemical compound C([C@](C1)(CCCN2CCC(CC2)(N(C(C)=O)C)C=2C=CC=CC=2)C=2C=C(Cl)C(Cl)=CC=2)CCN1C(=O)C1=CC=CC=C1 DZOJBGLFWINFBF-UMSFTDKQSA-N 0.000 title 1
- 229950009875 osanetant Drugs 0.000 title 1
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D211/00—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings
- C07D211/04—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom
- C07D211/06—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members
- C07D211/36—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D211/56—Nitrogen atoms
- C07D211/58—Nitrogen atoms attached in position 4
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Health & Medical Sciences (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Life Sciences & Earth Sciences (AREA)
- General Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Pharmacology & Pharmacy (AREA)
- Engineering & Computer Science (AREA)
- Animal Behavior & Ethology (AREA)
- General Health & Medical Sciences (AREA)
- Public Health (AREA)
- Veterinary Medicine (AREA)
- Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Hydrogenated Pyridines (AREA)
- Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
Applications Claiming Priority (3)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
FR9810107 | 1998-08-05 | ||
FR9810107A FR2782082B3 (fr) | 1998-08-05 | 1998-08-05 | Formes cristallines de (r)-(+)-n-[[3-[1-benzoyl-3-(3,4- dichlorophenyl)piperidin-3-yl]prop-1-yl]-4-phenylpiperidin-4 -yl]-n-methylacetamide (osanetant) et procede pour la preparation dudit compose |
PCT/FR1999/001914 WO2000007987A1 (fr) | 1998-08-05 | 1999-08-03 | Formes cristallines du osanetant |
Publications (2)
Publication Number | Publication Date |
---|---|
DE69908951D1 true DE69908951D1 (de) | 2003-07-24 |
DE69908951T2 DE69908951T2 (de) | 2004-05-19 |
Family
ID=9529458
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
DE69908951T Expired - Fee Related DE69908951T2 (de) | 1998-08-05 | 1999-08-03 | Kristallformen von osanetant |
Country Status (32)
Country | Link |
---|---|
US (1) | US7041679B2 (de) |
EP (1) | EP1102747B1 (de) |
JP (1) | JP3807938B2 (de) |
KR (1) | KR100571944B1 (de) |
CN (1) | CN1114592C (de) |
AR (1) | AR019953A1 (de) |
AT (1) | ATE243197T1 (de) |
AU (1) | AU748177B2 (de) |
BR (1) | BR9913357A (de) |
CA (1) | CA2339007A1 (de) |
CO (1) | CO5070576A1 (de) |
DE (1) | DE69908951T2 (de) |
DK (1) | DK1102747T3 (de) |
DZ (1) | DZ3074A1 (de) |
EA (1) | EA003205B1 (de) |
EE (1) | EE04274B1 (de) |
ES (1) | ES2200535T3 (de) |
FR (1) | FR2782082B3 (de) |
HK (1) | HK1035535A1 (de) |
HU (1) | HUP0103134A3 (de) |
IS (1) | IS5821A (de) |
MY (1) | MY121447A (de) |
NO (1) | NO320645B1 (de) |
NZ (1) | NZ509561A (de) |
PL (1) | PL345999A1 (de) |
PT (1) | PT1102747E (de) |
SK (1) | SK1742001A3 (de) |
TR (1) | TR200100261T2 (de) |
TW (1) | TW527354B (de) |
UA (1) | UA72890C2 (de) |
WO (1) | WO2000007987A1 (de) |
YU (1) | YU8601A (de) |
Families Citing this family (9)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
SE0100902D0 (sv) * | 2001-03-15 | 2001-03-15 | Astrazeneca Ab | Compounds |
SE0202539D0 (sv) | 2002-08-27 | 2002-08-27 | Astrazeneca Ab | Compounds |
US7648992B2 (en) * | 2004-07-05 | 2010-01-19 | Astrazeneca Ab | Hydantoin derivatives for the treatment of obstructive airway diseases |
SE0401762D0 (sv) * | 2004-07-05 | 2004-07-05 | Astrazeneca Ab | Novel compounds |
SE0403085D0 (sv) * | 2004-12-17 | 2004-12-17 | Astrazeneca Ab | Novel componds |
SE0403086D0 (sv) * | 2004-12-17 | 2004-12-17 | Astrazeneca Ab | Compounds |
TW200800954A (en) * | 2006-03-16 | 2008-01-01 | Astrazeneca Ab | Novel crystal modifications |
TW200831488A (en) * | 2006-11-29 | 2008-08-01 | Astrazeneca Ab | Novel compounds |
US20240336565A1 (en) * | 2021-07-02 | 2024-10-10 | Acer Therapeutics, Inc. | Solid forms of osanetant |
Family Cites Families (5)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
FR2719311B1 (fr) * | 1994-03-18 | 1998-06-26 | Sanofi Sa | Composés antagonistes sélectifs du récepteur NK3 humain et leur utilisation comme médicaments et outils de diagnostic. |
JPH1053576A (ja) * | 1996-06-07 | 1998-02-24 | Eisai Co Ltd | 塩酸ドネペジルの多形結晶およびその製造法 |
WO1998005640A2 (en) * | 1996-08-05 | 1998-02-12 | Smithkline Beecham S.P.A. | Process for the preparation of 3,3-disubstituted piperidines |
US6040316A (en) * | 1996-09-16 | 2000-03-21 | Warner-Lambert Company | 3-alkyl-3-phenyl-piperidines |
FR2757543B1 (fr) * | 1996-12-23 | 1999-04-02 | Sanofi Sa | Procede pour la cristallisation d'un derive de tetrahydropyridine et formes cristallines ainsi obtenues |
-
1998
- 1998-08-05 FR FR9810107A patent/FR2782082B3/fr not_active Expired - Lifetime
-
1999
- 1999-07-25 DZ DZ990156A patent/DZ3074A1/xx active
- 1999-07-28 AR ARP990103741A patent/AR019953A1/es unknown
- 1999-08-03 PT PT99936672T patent/PT1102747E/pt unknown
- 1999-08-03 BR BR9913357-1A patent/BR9913357A/pt not_active IP Right Cessation
- 1999-08-03 YU YU8601A patent/YU8601A/sh unknown
- 1999-08-03 DK DK99936672T patent/DK1102747T3/da active
- 1999-08-03 CA CA002339007A patent/CA2339007A1/en not_active Abandoned
- 1999-08-03 DE DE69908951T patent/DE69908951T2/de not_active Expired - Fee Related
- 1999-08-03 WO PCT/FR1999/001914 patent/WO2000007987A1/fr not_active Application Discontinuation
- 1999-08-03 AT AT99936672T patent/ATE243197T1/de not_active IP Right Cessation
- 1999-08-03 JP JP2000563621A patent/JP3807938B2/ja not_active Expired - Fee Related
- 1999-08-03 KR KR1020017001460A patent/KR100571944B1/ko not_active Expired - Fee Related
- 1999-08-03 NZ NZ509561A patent/NZ509561A/xx unknown
- 1999-08-03 TR TR2001/00261T patent/TR200100261T2/xx unknown
- 1999-08-03 SK SK174-2001A patent/SK1742001A3/sk unknown
- 1999-08-03 EA EA200100096A patent/EA003205B1/ru not_active IP Right Cessation
- 1999-08-03 EP EP99936672A patent/EP1102747B1/de not_active Expired - Lifetime
- 1999-08-03 HU HU0103134A patent/HUP0103134A3/hu unknown
- 1999-08-03 CN CN99810182A patent/CN1114592C/zh not_active Expired - Fee Related
- 1999-08-03 ES ES99936672T patent/ES2200535T3/es not_active Expired - Lifetime
- 1999-08-03 AU AU51685/99A patent/AU748177B2/en not_active Ceased
- 1999-08-03 UA UA2001010591A patent/UA72890C2/xx unknown
- 1999-08-03 MY MYPI99003297A patent/MY121447A/en unknown
- 1999-08-03 EE EEP200100070A patent/EE04274B1/xx not_active IP Right Cessation
- 1999-08-03 PL PL99345999A patent/PL345999A1/xx not_active Application Discontinuation
- 1999-08-04 CO CO99049286A patent/CO5070576A1/es unknown
- 1999-08-04 TW TW088113235A patent/TW527354B/zh not_active IP Right Cessation
-
2001
- 2001-01-23 IS IS5821A patent/IS5821A/is unknown
- 2001-02-01 NO NO20010553A patent/NO320645B1/no unknown
- 2001-09-04 HK HK01106232A patent/HK1035535A1/xx not_active IP Right Cessation
-
2003
- 2003-08-28 US US10/651,313 patent/US7041679B2/en not_active Expired - Fee Related
Also Published As
Similar Documents
Publication | Publication Date | Title |
---|---|---|
DE69928195D1 (de) | Komplettierung von Untrerdruck-Bohrlöchern | |
DE69941116D1 (de) | G von gdf-8 | |
CY2012029I2 (el) | Nεα μορφη της 5-ομεπραζολης | |
DE69834123D1 (de) | Rheologieänderung von elastomeren | |
DE59905858D1 (de) | Verwendung von pit-emulsionen | |
ID24481A (id) | Gastrokinetik monosiklik benzamida dari derivat-3-atau-tersubstitusi 4-(aminometil)-piperidin | |
DE60020817D1 (de) | Planung von betriebsmitteln | |
DE69913553D1 (de) | Konfigurierung von systemeinheiten | |
IT1304793B1 (it) | Miscela di stabilizzanti | |
DE50012379D1 (de) | Verwendung von nanoskaligen antischuppenwirkstoffen | |
DE69905054D1 (de) | KRISTALLINE FORMEN VON EtO2C-CH2-(R)Cgl-Aze-Pab-OH | |
ID24458A (id) | Modifikasi rheologi in-sito poliolefin | |
NO20011886D0 (no) | Utforminger av fexofenadin | |
NO994626D0 (no) | Substituerte benzamider | |
ID26514A (id) | Sumur penjernih | |
ATE196764T1 (de) | Kristallform von 5-methylisoxazol-4-carbonsäure- (4-trifluormethyl)-anilid | |
DE69907146T2 (de) | Direkte oxidation von cycloalkanen | |
IT1304794B1 (it) | Miscela di stabilizzanti | |
DE69531048D1 (de) | Verwendung von steroidsulphatase-hemmern | |
DE69806558D1 (de) | Stabilisierung von 3-Isothiazolonlösungen | |
DE69908951D1 (de) | Kristallformen von osanetant | |
DE69840875D1 (de) | Verwaltung von datenstrukturen | |
DE69922558D1 (de) | Herstellung von Aluminiumoxid | |
ID28032A (id) | TRISIKLIK PIPERIDIN-Δ3-SEBAGAI ANTAGONIS-α2 | |
DE69927626D1 (de) | Ausführung von Permutationen |
Legal Events
Date | Code | Title | Description |
---|---|---|---|
8364 | No opposition during term of opposition | ||
8327 | Change in the person/name/address of the patent owner |
Owner name: SANOFI-AVENTIS, PARIS, FR |
|
8339 | Ceased/non-payment of the annual fee |