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CY2004002I2 - Παραγωγο ανδροστενονης - Google Patents

Παραγωγο ανδροστενονης

Info

Publication number
CY2004002I2
CY2004002I2 CY200400002C CY2004002C CY2004002I2 CY 2004002 I2 CY2004002 I2 CY 2004002I2 CY 200400002 C CY200400002 C CY 200400002C CY 2004002 C CY2004002 C CY 2004002C CY 2004002 I2 CY2004002 I2 CY 2004002I2
Authority
CY
Cyprus
Prior art keywords
androstenone
derivative
androstenone derivative
Prior art date
Application number
CY200400002C
Other languages
English (en)
Other versions
CY2004002I1 (el
Original Assignee
Smithkline Beecham Corporation
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=22407744&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=CY2004002(I2) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Smithkline Beecham Corporation filed Critical Smithkline Beecham Corporation
Publication of CY2004002I1 publication Critical patent/CY2004002I1/el
Publication of CY2004002I2 publication Critical patent/CY2004002I2/el

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07JSTEROIDS
    • C07J3/00Normal steroids containing carbon, hydrogen, halogen or oxygen, substituted in position 17 beta by one carbon atom
    • C07J3/005Normal steroids containing carbon, hydrogen, halogen or oxygen, substituted in position 17 beta by one carbon atom the carbon atom being part of a carboxylic function
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P5/00Drugs for disorders of the endocrine system
    • A61P5/24Drugs for disorders of the endocrine system of the sex hormones
    • A61P5/26Androgens
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07CACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C235/00Carboxylic acid amides, the carbon skeleton of the acid part being further substituted by oxygen atoms
    • C07C235/70Carboxylic acid amides, the carbon skeleton of the acid part being further substituted by oxygen atoms having carbon atoms of carboxamide groups and doubly-bound oxygen atoms bound to the same carbon skeleton
    • C07C235/82Carboxylic acid amides, the carbon skeleton of the acid part being further substituted by oxygen atoms having carbon atoms of carboxamide groups and doubly-bound oxygen atoms bound to the same carbon skeleton with the carbon atom of at least one of the carboxamide groups bound to a carbon atom of a ring other than a six-membered aromatic ring
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07JSTEROIDS
    • C07J41/00Normal steroids containing one or more nitrogen atoms not belonging to a hetero ring
    • C07J41/0033Normal steroids containing one or more nitrogen atoms not belonging to a hetero ring not covered by C07J41/0005
    • C07J41/0066Normal steroids containing one or more nitrogen atoms not belonging to a hetero ring not covered by C07J41/0005 the 17-beta position being substituted by a carbon atom forming part of an amide group
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07JSTEROIDS
    • C07J73/00Steroids in which the cyclopenta[a]hydrophenanthrene skeleton has been modified by substitution of one or two carbon atoms by hetero atoms
    • C07J73/001Steroids in which the cyclopenta[a]hydrophenanthrene skeleton has been modified by substitution of one or two carbon atoms by hetero atoms by one hetero atom
    • C07J73/005Steroids in which the cyclopenta[a]hydrophenanthrene skeleton has been modified by substitution of one or two carbon atoms by hetero atoms by one hetero atom by nitrogen as hetero atom
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07CACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C2603/00Systems containing at least three condensed rings
    • C07C2603/02Ortho- or ortho- and peri-condensed systems
    • C07C2603/04Ortho- or ortho- and peri-condensed systems containing three rings
    • C07C2603/06Ortho- or ortho- and peri-condensed systems containing three rings containing at least one ring with less than six ring members
    • C07C2603/10Ortho- or ortho- and peri-condensed systems containing three rings containing at least one ring with less than six ring members containing five-membered rings
    • C07C2603/12Ortho- or ortho- and peri-condensed systems containing three rings containing at least one ring with less than six ring members containing five-membered rings only one five-membered ring
    • C07C2603/14Benz[f]indenes; Hydrogenated benz[f]indenes

Landscapes

  • Organic Chemistry (AREA)
  • Chemical & Material Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Medicinal Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • Animal Behavior & Ethology (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Diabetes (AREA)
  • Endocrinology (AREA)
  • Steroid Compounds (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
CY200400002C 1993-09-17 2004-07-26 Παραγωγο ανδροστενονης CY2004002I2 (el)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US12328093A 1993-09-17 1993-09-17
PCT/US1994/010530 WO1995007927A1 (en) 1993-09-17 1994-09-16 Androstenone derivative

Publications (2)

Publication Number Publication Date
CY2004002I1 CY2004002I1 (el) 2009-11-04
CY2004002I2 true CY2004002I2 (el) 2009-11-04

Family

ID=22407744

Family Applications (2)

Application Number Title Priority Date Filing Date
CY0100002A CY2219B1 (en) 1993-09-17 2001-01-03 Androstenone derivative
CY200400002C CY2004002I2 (el) 1993-09-17 2004-07-26 Παραγωγο ανδροστενονης

Family Applications Before (1)

Application Number Title Priority Date Filing Date
CY0100002A CY2219B1 (en) 1993-09-17 2001-01-03 Androstenone derivative

Country Status (41)

Country Link
US (2) US5565467A (el)
EP (1) EP0719278B1 (el)
JP (1) JP2904310B2 (el)
KR (1) KR100364953B1 (el)
CN (1) CN1057771C (el)
AP (1) AP494A (el)
AT (1) ATE162199T1 (el)
AU (1) AU690925B2 (el)
BG (1) BG62363B1 (el)
BR (1) BR1100329A (el)
CA (2) CA2462061A1 (el)
CY (2) CY2219B1 (el)
CZ (1) CZ286069B6 (el)
DE (2) DE69407978T2 (el)
DK (1) DK0719278T3 (el)
EE (1) EE03241B1 (el)
ES (1) ES2113127T3 (el)
FI (1) FI115216B (el)
GR (1) GR3026144T3 (el)
HK (1) HK1004334A1 (el)
HR (1) HRP940563B1 (el)
HU (1) HU220060B (el)
IL (1) IL110978A (el)
IS (1) IS1713B (el)
LU (1) LU91027I2 (el)
MY (1) MY119778A (el)
NL (1) NL300122I2 (el)
NO (2) NO306117B1 (el)
NZ (1) NZ274642A (el)
OA (1) OA10575A (el)
PE (1) PE15095A1 (el)
PL (1) PL180002B1 (el)
RO (1) RO117455B1 (el)
RU (1) RU2140926C1 (el)
SA (1) SA94150231B1 (el)
SG (1) SG52650A1 (el)
SI (1) SI0719278T1 (el)
SK (1) SK281869B6 (el)
TW (1) TW369521B (el)
WO (1) WO1995007927A1 (el)
ZA (2) ZA947118B (el)

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US5693810A (en) * 1992-10-06 1997-12-02 Merck & Co., Inc. 17 β-carboxanilides of 4-aza-5α-androstan-3-ones as 5α-reductase inhibitors
TW408127B (en) * 1993-09-17 2000-10-11 Glaxo Inc Androstenones
US5547957A (en) * 1993-10-15 1996-08-20 Merck & Co., Inc. Method of treating androgenic alopecia with 5-α reductase inhibitors
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ES2125495T3 (es) * 1993-10-21 1999-03-01 Merck & Co Inc 4-aza-androstano 16 sustituidos inhibidores de la isoenzima 5-alfa-reductasa 1.
US5817818A (en) * 1994-09-16 1998-10-06 Glaxo Wellcome Inc. Androstenones
USRE39056E1 (en) * 1995-09-15 2006-04-04 Merck & Co, Inc. 4-Azasteroids for treatment of hyperandrogenic conditions
US5872126A (en) * 1996-09-06 1999-02-16 Merck & Co., Inc. Methods and compositions for treating preterm labor
US5935968A (en) * 1997-03-17 1999-08-10 Merck & Co., Inc. Methods for treating polycystic ovary syndrome
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WO1999021563A1 (en) * 1997-10-28 1999-05-06 Merck & Co., Inc. Prevention of precipitated acute urinary retention
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EP1321146A3 (en) * 1998-03-11 2004-06-02 Endorecherche Inc. Inhibitors of type 5 and 3 17beta-hydroxysteroid dehydrogenase and methods for their use
US5998427A (en) * 1998-05-14 1999-12-07 Glaxo Wellcome Inc. Androstenones
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KR20010101931A (ko) 1999-02-03 2001-11-15 피터 지. 스트링거 α1-아드레날린성 수용체 길항제
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US7402577B2 (en) * 2001-10-03 2008-07-22 Merck & Co., Inc. Androstane 17-beta-carboxamides as androgen receptor modulators
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CN113896607B (zh) * 2015-03-13 2024-04-16 陶氏环球技术有限责任公司 利用包含具有含有磷环的配体的铬络合物的催化剂的烯烃低聚反应方法
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KR102281252B1 (ko) 2018-05-21 2021-07-23 (주)인벤티지랩 두타스테라이드를 포함하는 마이크로 입자 및 이의 제조 방법
WO2019225924A1 (ko) * 2018-05-21 2019-11-28 (주)인벤티지랩 두타스테라이드를 포함하는 마이크로 입자 및 이의 제조 방법
CN113507931A (zh) 2018-11-21 2021-10-15 卡斯西部储备大学 调节短链脱氢酶活性的组合物和方法
KR20200074759A (ko) 2018-12-17 2020-06-25 동국제약 주식회사 두타스테라이드를 함유하는 고형제제
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IL110978A0 (en) 1994-11-28
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