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CY1105337T1 - Πρωτοτυπες διυδροπτepιδινονες, μεθοδος για την παραγωγη τους και η χρηση τους ως φαρμακευτικα μεσα - Google Patents

Πρωτοτυπες διυδροπτepιδινονες, μεθοδος για την παραγωγη τους και η χρηση τους ως φαρμακευτικα μεσα

Info

Publication number
CY1105337T1
CY1105337T1 CY20061101285T CY061101285T CY1105337T1 CY 1105337 T1 CY1105337 T1 CY 1105337T1 CY 20061101285 T CY20061101285 T CY 20061101285T CY 061101285 T CY061101285 T CY 061101285T CY 1105337 T1 CY1105337 T1 CY 1105337T1
Authority
CY
Cyprus
Prior art keywords
prototype
production
pharmaceutical agents
dihydroptepidinones
dihydropteridinones
Prior art date
Application number
CY20061101285T
Other languages
English (en)
Inventor
Matthias Hoffmann
Matthias Grauert
Steffen Breitfelder
Christian Eickmeier
Gerald Pohl
Thorsten Lehmann-Lintz
Norbert Redemann
Gisela Schnapp
Martin Steegmaier
Eckhart Bauer
Jens Jürgen QUANT
Original Assignee
Boehringer Ingelheim Pharma Gmbh & Co. Kg
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Boehringer Ingelheim Pharma Gmbh & Co. Kg filed Critical Boehringer Ingelheim Pharma Gmbh & Co. Kg
Publication of CY1105337T1 publication Critical patent/CY1105337T1/el

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D487/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
    • C07D487/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
    • C07D487/04—Ortho-condensed systems
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P29/00—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/12—Antivirals
    • A61P31/14—Antivirals for RNA viruses
    • A61P31/18—Antivirals for RNA viruses for HIV
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00—Antineoplastic agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P37/00—Drugs for immunological or allergic disorders
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P37/00—Drugs for immunological or allergic disorders
    • A61P37/02—Immunomodulators
    • A61P37/06—Immunosuppressants, e.g. drugs for graft rejection
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • Animal Behavior & Ethology (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • Immunology (AREA)
  • Virology (AREA)
  • Oncology (AREA)
  • Communicable Diseases (AREA)
  • AIDS & HIV (AREA)
  • Molecular Biology (AREA)
  • Tropical Medicine & Parasitology (AREA)
  • Transplantation (AREA)
  • Pain & Pain Management (AREA)
  • Rheumatology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Hydrogenated Pyridines (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Plural Heterocyclic Compounds (AREA)

Abstract

Η παρούσα εφεύρεση σχετίζεται με πρωτότυπες διυδροπτεριδινόνες του γενικού τύπου (I), στον οποίο οι ρίζες Χ, R1, R2, R3, R4, R5 και R7 έχουν τις σημασίες που κατονομάζονται στις αξιώσεις και στην περιγραφή, με τα ισομερή αυτών, με μέθοδο παραγωγής αυτών των διυδροπτεριδινονών καθώς και η χρήση τους ως φαρμακευτικών μέσων.
CY20061101285T 2001-09-04 2006-09-08 Πρωτοτυπες διυδροπτepιδινονες, μεθοδος για την παραγωγη τους και η χρηση τους ως φαρμακευτικα μεσα CY1105337T1 (el)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
DE10143272 2001-09-04
PCT/EP2002/009728 WO2003020722A1 (de) 2001-09-04 2002-08-30 Neue dihydropteridinone, verfahren zu deren herstellung und deren verwendung als arzneimittel

Publications (1)

Publication Number Publication Date
CY1105337T1 true CY1105337T1 (el) 2010-03-03

Family

ID=7697637

Family Applications (1)

Application Number Title Priority Date Filing Date
CY20061101285T CY1105337T1 (el) 2001-09-04 2006-09-08 Πρωτοτυπες διυδροπτepιδινονες, μεθοδος για την παραγωγη τους και η χρηση τους ως φαρμακευτικα μεσα

Country Status (30)

Country Link
EP (1) EP1427730B1 (el)
JP (1) JP3876254B2 (el)
KR (1) KR100955589B1 (el)
CN (1) CN1551881A (el)
AR (1) AR036586A1 (el)
AT (1) ATE332898T1 (el)
AU (1) AU2002337047B2 (el)
BR (1) BRPI0212137A2 (el)
CA (1) CA2458699C (el)
CO (1) CO5560575A2 (el)
CY (1) CY1105337T1 (el)
DE (1) DE50207522D1 (el)
DK (1) DK1427730T3 (el)
EA (1) EA007062B1 (el)
EC (1) ECSP045003A (el)
ES (1) ES2268093T3 (el)
HR (1) HRP20040213A2 (el)
HU (1) HUP0401293A3 (el)
IL (2) IL160440A0 (el)
MX (1) MXPA04002067A (el)
MY (1) MY129751A (el)
NO (1) NO328804B1 (el)
NZ (1) NZ531928A (el)
PL (1) PL369740A1 (el)
PT (1) PT1427730E (el)
RS (1) RS51012B (el)
UA (1) UA76512C2 (el)
UY (1) UY27427A1 (el)
WO (1) WO2003020722A1 (el)
ZA (1) ZA200401365B (el)

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