CO6180480A2 - Pirimidinilpirazoles como principios activos insecticidas y parasiticidas - Google Patents
Pirimidinilpirazoles como principios activos insecticidas y parasiticidasInfo
- Publication number
- CO6180480A2 CO6180480A2 CO09063290A CO09063290A CO6180480A2 CO 6180480 A2 CO6180480 A2 CO 6180480A2 CO 09063290 A CO09063290 A CO 09063290A CO 09063290 A CO09063290 A CO 09063290A CO 6180480 A2 CO6180480 A2 CO 6180480A2
- Authority
- CO
- Colombia
- Prior art keywords
- haloalkyl
- alkyl
- optionally substituted
- alkoxy
- halogen
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
- C07D401/14—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing three or more hetero rings
-
- A—HUMAN NECESSITIES
- A01—AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
- A01N—PRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
- A01N43/00—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds
- A01N43/48—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with two nitrogen atoms as the only ring hetero atoms
- A01N43/54—1,3-Diazines; Hydrogenated 1,3-diazines
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P33/00—Antiparasitic agents
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D403/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00
- C07D403/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings
- C07D403/04—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings directly linked by a ring-member-to-ring-member bond
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D403/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00
- C07D403/14—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing three or more hetero rings
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Health & Medical Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
- General Health & Medical Sciences (AREA)
- Veterinary Medicine (AREA)
- Medicinal Chemistry (AREA)
- Engineering & Computer Science (AREA)
- General Chemical & Material Sciences (AREA)
- Pharmacology & Pharmacy (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Animal Behavior & Ethology (AREA)
- Tropical Medicine & Parasitology (AREA)
- Public Health (AREA)
- Agronomy & Crop Science (AREA)
- Pest Control & Pesticides (AREA)
- Plant Pathology (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Dentistry (AREA)
- Wood Science & Technology (AREA)
- Zoology (AREA)
- Environmental Sciences (AREA)
- Agricultural Chemicals And Associated Chemicals (AREA)
- Plural Heterocyclic Compounds (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Nitrogen Condensed Heterocyclic Rings (AREA)
- Low-Molecular Organic Synthesis Reactions Using Catalysts (AREA)
Abstract
1.- Compuestos de la fórmula (I),en la que X representa fenilo, 2-piridilo, 3-piridilo o 2-pirimidinilo, en cada caso sustituido con uno o varios sustituyentes seleccionados de halógeno, alquilo, haloalquilo, alcoxi alcoxialquilo, alcoxialcoxi, cicloalquilo alquenoxi, alquinoxi, benciloxi, cicloalquilalcoxi, haloalcoxi, haloalcoxialquilo, alquilsulfanilo, haloalquilsulfanilo, alquilsulfinilo, haloalquilsulfinilo, alquilsulfonilo, haloalquilsulfonilo, ciano, alquilcarbonilo, alcoxicarbonilo, alcoxicarbonilalquilo, carboxilo, carboxamida dialquilcarboxamida, trialquilsililo, nitro, amino, alquilamino,dialquilamino, alquilsulfonilamino, dialquilsulfonilamino, -CH=NO-H, -CH=NO-alquilo, -CH=NO-haloalquilo, -C(CH3)NO-H, -C(CH3)=NO-alquilo, -C(CH3)=NO-haloalquilo, formilo, bencilo (eventualmente sustituido, a su vez, con uno o varios átomos de halógeno), fenoxi o pirid-2-iloxi (los dos últimos eventualmente sustituidos con uno o varios seleccionados de alquilo, halógeno y/o haloalquilo) y fenilo (eventualmente sustituido con uno o varios átomos de halógeno), en donde grupos alquilo, haloalquilo, alcoxi y/o haloalcoxi vecinos, junto con los átomos de carbono a los que están unidos, pueden formar un sistema cíclico de cinco a seis miembros que contiene 0 a 2 átomos de oxígeno y cuya parte de alquilo puede estar eventualmente sustituida con uno o varios átomos de flúor, R1 representa alquilo (eventualmente mono- o disustituido con sustituyentes seleccionados, de modo independiente entre sí, de alcoxi, haloalcoxi, alquilsulfanilo, haloalquilsulfonilo, alquilsulfinilo, haloalquilsulfinilo, alquilsulfonilo, haloalquilsulfonilo, alquilcarbonilo, alcoxicarbonilo, hidroxi, cicloalquilo, fenilo (a su vez, eventualmente sustituido con uno o varios átomos de halógeno) y heterociclilo), cicloalquilo (eventualmente sustituido con uno o varios grupos haloalquilo y/o átomos de halógeno), haloalquilo (eventualmente sustituido con alcoxi), ciano, formilo, -CH=NO-H, -CH=NO-alquilo, -CH= NO-haloalquilo, -C(CH3)=NO-H, -C(CH3)=NO-alquilo, -C(CH3)=NO-haloalquilo o bencilo ...
Applications Claiming Priority (2)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| DE102006060230 | 2006-12-20 | ||
| DE102007003036A DE102007003036A1 (de) | 2006-12-20 | 2007-01-20 | Pyrimidinylpyrazole |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| CO6180480A2 true CO6180480A2 (es) | 2010-07-19 |
Family
ID=39226311
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| CO09063290A CO6180480A2 (es) | 2006-12-20 | 2009-06-18 | Pirimidinilpirazoles como principios activos insecticidas y parasiticidas |
Country Status (22)
| Country | Link |
|---|---|
| US (1) | US20100144672A1 (es) |
| EP (2) | EP2275422A1 (es) |
| JP (1) | JP2010513345A (es) |
| KR (1) | KR20090090393A (es) |
| CN (1) | CN101611030A (es) |
| AR (1) | AR064463A1 (es) |
| AT (1) | ATE502029T1 (es) |
| AU (1) | AU2007338425A1 (es) |
| BR (1) | BRPI0720518A2 (es) |
| CA (1) | CA2672989A1 (es) |
| CL (1) | CL2007003735A1 (es) |
| CO (1) | CO6180480A2 (es) |
| DE (2) | DE102007003036A1 (es) |
| DK (1) | DK2125789T3 (es) |
| MX (1) | MX2009006567A (es) |
| PL (1) | PL2125789T3 (es) |
| PT (1) | PT2125789E (es) |
| RU (1) | RU2009127515A (es) |
| SI (1) | SI2125789T1 (es) |
| TW (1) | TW200835443A (es) |
| WO (1) | WO2008077483A1 (es) |
| ZA (1) | ZA200904229B (es) |
Families Citing this family (21)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| WO2010017902A1 (de) * | 2008-08-14 | 2010-02-18 | Bayer Cropscience Aktiengesellschaft | Insektizide 4-phenyl-1h-pyrazole |
| EP2266973A1 (de) * | 2009-05-29 | 2010-12-29 | Bayer CropScience AG | Pyrazinylpyrazole |
| IN2012DN02679A (es) * | 2009-10-12 | 2015-09-04 | Bayer Cropscience Ag | |
| AU2010318059A1 (en) | 2009-11-11 | 2012-06-07 | Bayer Cropscience Ag | Novel diazinylpyrazolyl compounds |
| EP2571359A4 (en) * | 2010-05-20 | 2013-10-23 | Merck Sharp & Dohme | NOVEL PROLYLCARBOXYPEPTIDASE HEMMER |
| CA2826059A1 (en) * | 2011-02-09 | 2012-08-16 | Pierre Joseph Marcel Jung | Insecticidal compounds |
| TW201238487A (en) * | 2011-02-25 | 2012-10-01 | Dow Agrosciences Llc | Pesticidal compositions and processes related thereto |
| AU2012342564A1 (en) | 2011-11-21 | 2014-06-12 | Basf Se | Process for preparing N-substituted 1H-pyrazole-5-carboxylate compounds and derivatives thereof |
| KR20150050527A (ko) | 2012-05-04 | 2015-05-08 | 바스프 에스이 | 치환된 피라졸-함유 화합물 및 이의 살충제로서의 용도 |
| AU2014300673B2 (en) | 2013-06-27 | 2017-12-14 | Pfizer Inc. | Heteroaromatic compounds and their use as dopamine D1 ligands |
| TWI648260B (zh) * | 2013-11-05 | 2019-01-21 | 德商拜耳作物科學股份有限公司 | 用於控制節肢動物的新穎化合物（一） |
| CN108137531A (zh) * | 2015-09-25 | 2018-06-08 | 先正达参股股份有限公司 | 具有含硫取代基的杀有害生物活性杂环衍生物 |
| CN106632300B (zh) * | 2016-09-29 | 2019-11-12 | 华东理工大学 | 具有杀虫活性的多取代异噁唑类化合物及其制备方法 |
| CN109400591B (zh) * | 2018-12-26 | 2022-01-14 | 西华大学 | 4-(2-呋喃基)嘧啶类化合物及其制备方法和应用 |
| CN113481255B (zh) * | 2021-06-17 | 2023-08-15 | 南京师范大学 | 含纤维素原料的酶解方法 |
| CN113854036B (zh) * | 2021-09-28 | 2023-04-07 | 江西省农业科学院农业应用微生物研究所（江西省农村能源研究中心） | 一种茶树菇病虫害绿色防控方法 |
| WO2024121261A1 (en) | 2022-12-09 | 2024-06-13 | Syngenta Crop Protection Ag | Insecticidal compound based on pyrazole derivatives |
| WO2024121264A1 (en) | 2022-12-09 | 2024-06-13 | Syngenta Crop Protection Ag | Insecticidal compound based on pyrazole derivatives |
| WO2024121263A1 (en) | 2022-12-09 | 2024-06-13 | Syngenta Crop Protection Ag | Insecticidal compound based on pyrazole derivatives |
| WO2024121262A1 (en) | 2022-12-09 | 2024-06-13 | Syngenta Crop Protection Ag | Insecticidal compound based on pyrazole derivatives |
| WO2024175804A1 (en) * | 2023-02-24 | 2024-08-29 | Katholieke Universiteit Leuven | Nuclear transport modulators |
Family Cites Families (10)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| NL253320A (es) * | 1959-07-03 | |||
| FR2326421A1 (fr) | 1975-09-30 | 1977-04-29 | Ugine Kuhlmann | Nouveaux trifluoromethyl-3-aryl-4 amino-5 pyrazoles et leur application comme bases diazotables pour la synthese de matieres colorantes |
| US5201938A (en) * | 1991-07-19 | 1993-04-13 | Dowelanco | N-pyrazolyl-1,2,4-triazolo[1,5-c]pyrimidine-2-sulfonamide herbicides |
| WO1993019054A1 (en) | 1992-03-26 | 1993-09-30 | Dowelanco | N-heterocyclic nitro anilines as fungicides |
| DE4405207A1 (de) | 1994-02-18 | 1995-08-24 | Bayer Ag | N-Pyrazolylaniline und N-Pyrazolylaminopyridine |
| JPH08208620A (ja) | 1995-02-03 | 1996-08-13 | Takeda Chem Ind Ltd | アミノピラゾール誘導体、その製造法および用途 |
| CA2297780A1 (en) | 1998-06-10 | 1999-12-16 | Boulder Scientific Company | Synthesis of aryl boronic acids |
| DE10108480A1 (de) | 2001-02-22 | 2002-09-05 | Bayer Ag | Pyrazolylpyrimidine |
| KR100969088B1 (ko) | 2002-03-05 | 2010-07-09 | 메리얼 리미티드 | 살충제로서의 5-치환된-알킬아미노피라졸 유도체 |
| US20080009531A1 (en) | 2004-05-20 | 2008-01-10 | Bayer Pharmaceuticals Corporation | 5-Anilino-4-Heteroarylpyrazole Derivatives Useful for the Treatment of Diabetes |
-
2007
- 2007-01-20 DE DE102007003036A patent/DE102007003036A1/de not_active Withdrawn
- 2007-12-12 DK DK07856587.6T patent/DK2125789T3/da active
- 2007-12-12 PL PL07856587T patent/PL2125789T3/pl unknown
- 2007-12-12 MX MX2009006567A patent/MX2009006567A/es active IP Right Grant
- 2007-12-12 EP EP10173541A patent/EP2275422A1/de not_active Withdrawn
- 2007-12-12 BR BRPI0720518-0A patent/BRPI0720518A2/pt not_active IP Right Cessation
- 2007-12-12 WO PCT/EP2007/010839 patent/WO2008077483A1/de active Application Filing
- 2007-12-12 EP EP07856587A patent/EP2125789B1/de not_active Not-in-force
- 2007-12-12 US US12/520,477 patent/US20100144672A1/en not_active Abandoned
- 2007-12-12 SI SI200730623T patent/SI2125789T1/sl unknown
- 2007-12-12 AU AU2007338425A patent/AU2007338425A1/en not_active Abandoned
- 2007-12-12 DE DE502007006748T patent/DE502007006748D1/de active Active
- 2007-12-12 RU RU2009127515/04A patent/RU2009127515A/ru not_active Application Discontinuation
- 2007-12-12 CA CA002672989A patent/CA2672989A1/en not_active Abandoned
- 2007-12-12 JP JP2009541836A patent/JP2010513345A/ja not_active Withdrawn
- 2007-12-12 PT PT07856587T patent/PT2125789E/pt unknown
- 2007-12-12 KR KR1020097014888A patent/KR20090090393A/ko not_active Application Discontinuation
- 2007-12-12 AT AT07856587T patent/ATE502029T1/de active
- 2007-12-12 CN CNA2007800515010A patent/CN101611030A/zh active Pending
- 2007-12-19 AR ARP070105741A patent/AR064463A1/es not_active Application Discontinuation
- 2007-12-19 TW TW096148542A patent/TW200835443A/zh unknown
- 2007-12-20 CL CL200703735A patent/CL2007003735A1/es unknown
-
2009
- 2009-06-17 ZA ZA200904229A patent/ZA200904229B/xx unknown
- 2009-06-18 CO CO09063290A patent/CO6180480A2/es not_active Application Discontinuation
Also Published As
| Publication number | Publication date |
|---|---|
| JP2010513345A (ja) | 2010-04-30 |
| ATE502029T1 (de) | 2011-04-15 |
| CA2672989A1 (en) | 2008-07-03 |
| EP2125789B1 (de) | 2011-03-16 |
| PT2125789E (pt) | 2011-05-18 |
| SI2125789T1 (sl) | 2011-07-29 |
| KR20090090393A (ko) | 2009-08-25 |
| MX2009006567A (es) | 2009-07-02 |
| BRPI0720518A2 (pt) | 2013-12-31 |
| PL2125789T3 (pl) | 2011-08-31 |
| ZA200904229B (en) | 2010-10-27 |
| DK2125789T3 (da) | 2011-07-18 |
| RU2009127515A (ru) | 2011-02-10 |
| WO2008077483A1 (de) | 2008-07-03 |
| DE502007006748D1 (de) | 2011-04-28 |
| DE102007003036A1 (de) | 2008-06-26 |
| EP2125789A1 (de) | 2009-12-02 |
| AR064463A1 (es) | 2009-04-01 |
| CL2007003735A1 (es) | 2008-05-16 |
| EP2275422A1 (de) | 2011-01-19 |
| TW200835443A (en) | 2008-09-01 |
| US20100144672A1 (en) | 2010-06-10 |
| CN101611030A (zh) | 2009-12-23 |
| AU2007338425A1 (en) | 2008-07-03 |
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Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| FC | Application refused |