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CO4770984A1 - Compuesto de ciclohexapeptidil bis-amina, composiciones que lo contienen y metodos de uso - Google Patents

Compuesto de ciclohexapeptidil bis-amina, composiciones que lo contienen y metodos de uso

Info

Publication number
CO4770984A1
CO4770984A1 CO96058746A CO96058746A CO4770984A1 CO 4770984 A1 CO4770984 A1 CO 4770984A1 CO 96058746 A CO96058746 A CO 96058746A CO 96058746 A CO96058746 A CO 96058746A CO 4770984 A1 CO4770984 A1 CO 4770984A1
Authority
CO
Colombia
Prior art keywords
cyclohexapeptidil
bis
methods
compositions containing
amine compound
Prior art date
Application number
CO96058746A
Other languages
English (en)
Inventor
James M Balkovec
Frances A Bouffard
James F Dropinski
Original Assignee
Merck & Co Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Priority claimed from GBGB9603241.2A external-priority patent/GB9603241D0/en
Application filed by Merck & Co Inc filed Critical Merck & Co Inc
Publication of CO4770984A1 publication Critical patent/CO4770984A1/es

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07KPEPTIDES
    • C07K7/00Peptides having 5 to 20 amino acids in a fully defined sequence; Derivatives thereof
    • C07K7/50Cyclic peptides containing at least one abnormal peptide link
    • C07K7/54Cyclic peptides containing at least one abnormal peptide link with at least one abnormal peptide link in the ring
    • C07K7/56Cyclic peptides containing at least one abnormal peptide link with at least one abnormal peptide link in the ring the cyclisation not occurring through 2,4-diamino-butanoic acid
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/10Antimycotics
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K38/00Medicinal preparations containing peptides

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • Animal Behavior & Ethology (AREA)
  • Communicable Diseases (AREA)
  • Oncology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Biochemistry (AREA)
  • Biophysics (AREA)
  • Genetics & Genomics (AREA)
  • Proteomics, Peptides & Aminoacids (AREA)
  • Molecular Biology (AREA)
  • Peptides Or Proteins (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)

Abstract

Un compuesto de fórmula:o una sal de adición de ácido del mismo.
CO96058746A 1995-11-09 1996-11-07 Compuesto de ciclohexapeptidil bis-amina, composiciones que lo contienen y metodos de uso CO4770984A1 (es)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US650595P 1995-11-09 1995-11-09
GBGB9603241.2A GB9603241D0 (en) 1996-02-16 1996-02-16 Cyclohexapeptidyl bisamine compound, compositions containing said compound and methods of use

Publications (1)

Publication Number Publication Date
CO4770984A1 true CO4770984A1 (es) 1999-04-30

Family

ID=26308720

Family Applications (1)

Application Number Title Priority Date Filing Date
CO96058746A CO4770984A1 (es) 1995-11-09 1996-11-07 Compuesto de ciclohexapeptidil bis-amina, composiciones que lo contienen y metodos de uso

Country Status (9)

Country Link
EP (1) EP0862579A1 (es)
JP (1) JP2000501076A (es)
AR (1) AR001314A1 (es)
AU (1) AU707664B2 (es)
CA (1) CA2235824A1 (es)
CO (1) CO4770984A1 (es)
HR (1) HRP960521A2 (es)
PE (1) PE16198A1 (es)
WO (1) WO1997017365A1 (es)

Families Citing this family (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JP2002532513A (ja) * 1998-12-16 2002-10-02 イーライ リリー アンド カンパニー 糖置換基を有する環式ペプチド抗真菌剤

Family Cites Families (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US6030944A (en) * 1991-10-01 2000-02-29 Merck & Co., Inc. Cyclohexapeptidyl bisamine compounds
US5378804A (en) * 1993-03-16 1995-01-03 Merck & Co., Inc. Aza cyclohexapeptide compounds
IL109615A (en) * 1993-05-17 2000-12-06 Fujisawa Pharmaceutical Co Cyclic polypeptide derivatives processes for the preparation thereof and pharmaceutical compositions containing the same

Also Published As

Publication number Publication date
AU7554096A (en) 1997-05-29
CA2235824A1 (en) 1997-05-15
PE16198A1 (es) 1998-04-11
WO1997017365A1 (en) 1997-05-15
EP0862579A1 (en) 1998-09-09
AU707664B2 (en) 1999-07-15
AR001314A1 (es) 1997-10-22
JP2000501076A (ja) 2000-02-02
HRP960521A2 (en) 1998-04-30

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