CO4750837A1 - Derivados de acido boronico - Google Patents
Derivados de acido boronicoInfo
- Publication number
- CO4750837A1 CO4750837A1 CO96039770A CO96039770A CO4750837A1 CO 4750837 A1 CO4750837 A1 CO 4750837A1 CO 96039770 A CO96039770 A CO 96039770A CO 96039770 A CO96039770 A CO 96039770A CO 4750837 A1 CO4750837 A1 CO 4750837A1
- Authority
- CO
- Colombia
- Prior art keywords
- acid derivatives
- boronic acid
- formula
- residue
- compound
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07K—PEPTIDES
- C07K5/00—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof
- C07K5/04—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof containing only normal peptide links
- C07K5/06—Dipeptides
- C07K5/06191—Dipeptides containing heteroatoms different from O, S, or N
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K38/00—Medicinal preparations containing peptides
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Health & Medical Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
- Biochemistry (AREA)
- Biophysics (AREA)
- General Health & Medical Sciences (AREA)
- Genetics & Genomics (AREA)
- Medicinal Chemistry (AREA)
- Molecular Biology (AREA)
- Proteomics, Peptides & Aminoacids (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Abstract
Un compuesto de la fórmula I:caracterizado porque cada uno de Q1 y Q2 es OH o Q1 y Q2 forman conjuntamente un residuo de la fórmula (a)en la forma libre o, cuando cada uno de Q1 y Q2 es OH, también en la forma de sal.
Applications Claiming Priority (1)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
GBGB9515489.4A GB9515489D0 (en) | 1995-07-28 | 1995-07-28 | Organic compounds |
Publications (1)
Publication Number | Publication Date |
---|---|
CO4750837A1 true CO4750837A1 (es) | 1999-03-31 |
Family
ID=10778404
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
CO96039770A CO4750837A1 (es) | 1995-07-28 | 1996-07-26 | Derivados de acido boronico |
Country Status (5)
Country | Link |
---|---|
AU (1) | AU6737996A (es) |
CO (1) | CO4750837A1 (es) |
GB (1) | GB9515489D0 (es) |
WO (1) | WO1997005161A1 (es) |
ZA (1) | ZA966396B (es) |
Families Citing this family (5)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US7030141B2 (en) * | 2001-11-29 | 2006-04-18 | Christopher Franklin Bigge | Inhibitors of factor Xa and other serine proteases involved in the coagulation cascade |
KR20030080810A (ko) * | 2002-04-11 | 2003-10-17 | 주식회사 엘지생명과학 | 아미노피리도아릴 그룹을 가진 선택적 트롬빈 억제제 |
US7371729B2 (en) | 2002-09-09 | 2008-05-13 | Trigen Limited | Boronic acid salts useful in parenteral formulations |
ATE376551T1 (de) | 2002-09-09 | 2007-11-15 | Trigen Ltd | Peptidborsäuren und deren verwendung in der herstellung von salzen derselben |
ES2543588T3 (es) | 2002-12-03 | 2015-08-20 | Pharmacyclics Llc | Derivados de 2-(2-hidroxibifenil-3-il)-1H-benzoimidazol-5-carboxamidina como inhibidores del factor VIIa |
Family Cites Families (3)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
GB9017694D0 (en) * | 1990-08-13 | 1990-09-26 | Sandoz Ltd | Improvements in or relating to organic chemistry |
MY131622A (en) * | 1993-03-03 | 2007-08-30 | Novartis Ag | Organic compounds |
GB9401483D0 (en) * | 1994-01-26 | 1994-03-23 | Sandoz Ltd | Organic compounds |
-
1995
- 1995-07-28 GB GBGB9515489.4A patent/GB9515489D0/en active Pending
-
1996
- 1996-07-26 ZA ZA9606396A patent/ZA966396B/xx unknown
- 1996-07-26 CO CO96039770A patent/CO4750837A1/es unknown
- 1996-07-26 AU AU67379/96A patent/AU6737996A/en not_active Abandoned
- 1996-07-26 WO PCT/EP1996/003314 patent/WO1997005161A1/en active Application Filing
Also Published As
Publication number | Publication date |
---|---|
ZA966396B (en) | 1998-01-26 |
AU6737996A (en) | 1997-02-26 |
WO1997005161A1 (en) | 1997-02-13 |
GB9515489D0 (en) | 1995-09-27 |
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