CL2008000703A1 - Compuestos derivados de pirimidinas sustituidas; procedimiento para la preparacion de dichos compuestos; composicion farmaceutica que comprende a dichos compuestos; y su uso para tratar transtornos hematologicos. - Google Patents

Compuestos derivados de pirimidinas sustituidas; procedimiento para la preparacion de dichos compuestos; composicion farmaceutica que comprende a dichos compuestos; y su uso para tratar transtornos hematologicos.

Info

Publication number: CL2008000703A1
Authority: CL; Chile
Prior art keywords: compounds; pyrimidins; substituted; procedure; preparation
Prior art date: 2007-03-16

Application number

CL200800703A

Other languages

English (en)

Inventor

Stephan Siegel Dr Andreas W Dr

Original Assignee

Bayer Healthcare Ag

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

2007-03-16

Filing date

2008-03-10

Publication date

2008-09-26

2008-03-10 Application filed by Bayer Healthcare Ag filed Critical Bayer Healthcare Ag

2008-09-26 Publication of CL2008000703A1 publication Critical patent/CL2008000703A1/es

Classifications

- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D487/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
- C07D487/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
- C07D487/04—Ortho-condensed systems
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- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
- A61K31/505—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
- A61K31/519—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim ortho- or peri-condensed with heterocyclic rings
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Heart & Thoracic Surgery (AREA)
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CL200800703A 2007-03-16 2008-03-10 Compuestos derivados de pirimidinas sustituidas; procedimiento para la preparacion de dichos compuestos; composicion farmaceutica que comprende a dichos compuestos; y su uso para tratar transtornos hematologicos. CL2008000703A1 (es)

Applications Claiming Priority (1)

Application Number	Priority Date	Filing Date	Title
DE102007012645A DE102007012645A1 (de)	2007-03-16	2007-03-16	Substituierte Imidazo- und Triazolopyrimidine

Publications (1)

Publication Number	Publication Date
CL2008000703A1 true CL2008000703A1 (es)	2008-09-26

Family

ID=39688187

Family Applications (1)

Application Number	Title	Priority Date	Filing Date
CL200800703A CL2008000703A1 (es)	2007-03-16	2008-03-10	Compuestos derivados de pirimidinas sustituidas; procedimiento para la preparacion de dichos compuestos; composicion farmaceutica que comprende a dichos compuestos; y su uso para tratar transtornos hematologicos.

Country Status (13)

Country	Link
US (2)	US8273752B2 (es)
EP (1)	EP2137188B1 (es)
JP (1)	JP5400626B2 (es)
AR (1)	AR065719A1 (es)
CA (1)	CA2680697C (es)
CL (1)	CL2008000703A1 (es)
DE (1)	DE102007012645A1 (es)
ES (1)	ES2387223T3 (es)
PA (1)	PA8772101A1 (es)
PE (1)	PE20081806A1 (es)
TW (1)	TW200904819A (es)
UY (1)	UY30956A1 (es)
WO (1)	WO2008113469A2 (es)

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* Cited by examiner, † Cited by third party
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DE102007012645A1 (de)	2007-03-16	2008-09-18	Bayer Healthcare Ag	Substituierte Imidazo- und Triazolopyrimidine
DE102008023801A1 (de) *	2008-05-15	2009-11-19	Bayer Schering Pharma Aktiengesellschaft	Substituierte Imidazo- und Triazolopyrimidine, Imidazo- und Pyrazolopyrazine und Imidazotriazine
DE102008035552A1 (de) *	2008-07-30	2010-02-04	Bayer Schering Pharma Aktiengesellschaft	Substituierte Pyridine und ihre Verwendung
CA2752114C (en) *	2009-02-13	2017-06-20	Bayer Pharma Aktiengesellschaft	Fused pyrimidines as akt inhibitors
JP5503930B2 (ja) *	2009-09-18	2014-05-28	住友化学株式会社	３−アミノ−１−ｔｅｒｔ−ブトキシカルボニルピペリジンの精製方法およびそのクエン酸塩
PH12012500355A1 (en) *	2009-09-24	2019-11-29	Hoffmann La Roche	Imidazopyridine or imidazopyrimidine derivatives as phosphodiesterase 10a inhibitors
WO2011044637A1 (en)	2009-10-15	2011-04-21	Monash University	Affinity ligands and methods for protein purification
EP2526102B1 (en)	2010-01-22	2017-03-08	Fundación Centro Nacional de Investigaciones Oncológicas Carlos III	Inhibitors of PI3 kinase
WO2011107494A1 (de)	2010-03-03	2011-09-09	Sanofi	Neue aromatische glykosidderivate, diese verbindungen enthaltende arzneimittel und deren verwendung
CN102791692B (zh) *	2010-03-12	2015-05-27	日本曹达株式会社	叔丁氧基羰基胺化合物的制造方法
CN102985424B (zh) *	2010-04-14	2015-03-11	阵列生物制药公司	5,7-取代的-咪唑并[1,2-c]嘧啶
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US8530413B2 (en)	2010-06-21	2013-09-10	Sanofi	Heterocyclically substituted methoxyphenyl derivatives with an oxo group, processes for preparation thereof and use thereof as medicaments
TW201215388A (en)	2010-07-05	2012-04-16	Sanofi Sa	(2-aryloxyacetylamino)phenylpropionic acid derivatives, processes for preparation thereof and use thereof as medicaments
TW201221505A (en)	2010-07-05	2012-06-01	Sanofi Sa	Aryloxyalkylene-substituted hydroxyphenylhexynoic acids, process for preparation thereof and use thereof as a medicament
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EA201691594A1 (ru)	2014-02-13	2017-02-28	Инсайт Корпорейшн	Циклопропиламины в качестве ингибиторов lsd1
US9527835B2 (en)	2014-02-13	2016-12-27	Incyte Corporation	Cyclopropylamines as LSD1 inhibitors
LT3105218T (lt)	2014-02-13	2019-12-10	Incyte Corp	Ciklopropilaminai kaip lsd1 inhibitoriai
EP3392244A1 (en)	2014-02-13	2018-10-24	Incyte Corporation	Cyclopropylamines as lsd1 inhibitors
CN106255689B (zh)	2014-03-19	2019-09-17	勃林格殷格翰国际有限公司	杂芳基syk抑制剂
US9695180B2 (en)	2014-07-10	2017-07-04	Incyte Corporation	Substituted imidazo[1,2-a]pyrazines as LSD1 inhibitors
WO2016007722A1 (en)	2014-07-10	2016-01-14	Incyte Corporation	Triazolopyridines and triazolopyrazines as lsd1 inhibitors
WO2016007731A1 (en)	2014-07-10	2016-01-14	Incyte Corporation	Imidazopyridines and imidazopyrazines as lsd1 inhibitors
WO2016007727A1 (en)	2014-07-10	2016-01-14	Incyte Corporation	Triazolopyridines and triazolopyrazines as lsd1 inhibitors
EP3626720A1 (en)	2015-04-03	2020-03-25	Incyte Corporation	Heterocyclic compounds as lsd1 inhibitors
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2007
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2008
- 2008-03-04 EP EP08716201A patent/EP2137188B1/de not_active Not-in-force
- 2008-03-04 US US12/529,711 patent/US8273752B2/en not_active Expired - Fee Related
- 2008-03-04 ES ES08716201T patent/ES2387223T3/es active Active
- 2008-03-04 CA CA2680697A patent/CA2680697C/en not_active Expired - Fee Related
- 2008-03-04 WO PCT/EP2008/001682 patent/WO2008113469A2/de active Application Filing
- 2008-03-04 JP JP2009553944A patent/JP5400626B2/ja not_active Expired - Fee Related
- 2008-03-10 PE PE2008000448A patent/PE20081806A1/es not_active Application Discontinuation
- 2008-03-10 PA PA20088772101A patent/PA8772101A1/es unknown
- 2008-03-10 CL CL200800703A patent/CL2008000703A1/es unknown
- 2008-03-11 UY UY30956A patent/UY30956A1/es not_active Application Discontinuation
- 2008-03-13 AR ARP080101031A patent/AR065719A1/es unknown
- 2008-03-14 TW TW097108955A patent/TW200904819A/zh unknown
2012
- 2012-09-24 US US13/625,086 patent/US9051323B2/en not_active Expired - Fee Related

Also Published As

Publication number	Publication date
AR065719A1 (es)	2009-06-24
US9051323B2 (en)	2015-06-09
US20130040946A1 (en)	2013-02-14
PA8772101A1 (es)	2009-02-09
US8273752B2 (en)	2012-09-25
CA2680697C (en)	2016-09-20
UY30956A1 (es)	2008-10-31
EP2137188B1 (de)	2012-06-06
EP2137188A2 (de)	2009-12-30
JP5400626B2 (ja)	2014-01-29
TW200904819A (en)	2009-02-01
JP2010521506A (ja)	2010-06-24
US20100113441A1 (en)	2010-05-06
WO2008113469A8 (de)	2009-09-24
ES2387223T3 (es)	2012-09-18
PE20081806A1 (es)	2009-02-07
WO2008113469A2 (de)	2008-09-25
DE102007012645A1 (de)	2008-09-18
WO2008113469A3 (de)	2008-11-13
CA2680697A1 (en)	2008-09-25

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