BRPI0809837A2 - "composto para tratamento de distúrbios mentais, saldo do composto para tratamento de distúrbios mentais, composição farmacéutica e uso do composto para tratamento de distúrbios mentais" - Google Patents
"composto para tratamento de distúrbios mentais, saldo do composto para tratamento de distúrbios mentais, composição farmacéutica e uso do composto para tratamento de distúrbios mentais"Info
- Publication number
- BRPI0809837A2 BRPI0809837A2 BRPI0809837-9A2A BRPI0809837A BRPI0809837A2 BR PI0809837 A2 BRPI0809837 A2 BR PI0809837A2 BR PI0809837 A BRPI0809837 A BR PI0809837A BR PI0809837 A2 BRPI0809837 A2 BR PI0809837A2
- Authority
- BR
- Brazil
- Prior art keywords
- mental disorders
- treating mental
- composite
- composition
- balance
- Prior art date
Links
- 208000020016 psychiatric disease Diseases 0.000 title 3
- 239000002131 composite material Substances 0.000 title 2
- 239000000203 mixture Substances 0.000 title 1
- 239000008194 pharmaceutical composition Substances 0.000 title 1
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
- C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
- C07D471/04—Ortho-condensed systems
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
- A61K31/505—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/18—Antipsychotics, i.e. neuroleptics; Drugs for mania or schizophrenia
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D413/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms
- C07D413/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings
- C07D413/04—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings directly linked by a ring-member-to-ring-member bond
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Health & Medical Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- General Health & Medical Sciences (AREA)
- Veterinary Medicine (AREA)
- Public Health (AREA)
- Engineering & Computer Science (AREA)
- Life Sciences & Earth Sciences (AREA)
- Pharmacology & Pharmacy (AREA)
- Medicinal Chemistry (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- General Chemical & Material Sciences (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Psychiatry (AREA)
- Biomedical Technology (AREA)
- Neurosurgery (AREA)
- Neurology (AREA)
- Epidemiology (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Nitrogen Condensed Heterocyclic Rings (AREA)
- Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
Applications Claiming Priority (2)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
CN200710098304 | 2007-04-19 | ||
PCT/CN2008/000803 WO2008128436A1 (en) | 2007-04-19 | 2008-04-18 | Novel compounds for treatment of psychotic disorders, preparation methods and uses thereof |
Publications (1)
Publication Number | Publication Date |
---|---|
BRPI0809837A2 true BRPI0809837A2 (pt) | 2014-11-11 |
Family
ID=39875078
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
BRPI0809837-9A2A BRPI0809837A2 (pt) | 2007-04-19 | 2008-04-18 | "composto para tratamento de distúrbios mentais, saldo do composto para tratamento de distúrbios mentais, composição farmacéutica e uso do composto para tratamento de distúrbios mentais" |
Country Status (9)
Country | Link |
---|---|
US (1) | US8314110B2 (pt) |
EP (1) | EP2154138B1 (pt) |
JP (1) | JP5315336B2 (pt) |
KR (1) | KR101244185B1 (pt) |
CN (1) | CN101641353B (pt) |
BR (1) | BRPI0809837A2 (pt) |
DK (1) | DK2154138T3 (pt) |
RU (1) | RU2459824C2 (pt) |
WO (1) | WO2008128436A1 (pt) |
Families Citing this family (7)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US7820816B2 (en) | 2006-08-23 | 2010-10-26 | Teva Pharmaceutical Industries Ltd. | Process for the synthesis of CMHTP and intermediates thereof |
EP2224472B8 (en) | 2007-12-17 | 2014-03-19 | JX Nippon Mining & Metals Corporation | Substrate and method for manufacturing the same |
WO2011042450A1 (en) | 2009-10-06 | 2011-04-14 | Ascendis Pharma As | Carrier linked paliperidone prodrugs |
WO2011042453A1 (en) | 2009-10-06 | 2011-04-14 | Ascendis Pharma As | Subcutaneous paliperidone composition |
DK2529757T3 (en) | 2011-05-31 | 2014-02-24 | Rovi Lab Farmaceut Sa | Paliperidonimplantatformulering |
DK2529756T3 (da) | 2011-05-31 | 2021-08-02 | Farm Rovi Lab Sa | Risperidon- og/eller paliperidon-implantatformulering |
KR101867988B1 (ko) * | 2016-11-02 | 2018-06-15 | 주식회사 엔지켐생명과학 | 팔리페리돈 중간체 및 이를 이용한 팔리페리돈의 제조방법 |
Family Cites Families (13)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US5158952A (en) * | 1988-11-07 | 1992-10-27 | Janssen Pharmaceutica N.V. | 3-[2-[4-(6-fluoro-1,2-benzisoxozol-3-yl)-1-piperidinyl]ethyl]-6,7,8,9 tetrahydro-9-hydroxy-2-methyl-4H-pyrido [1,2-a]pyrimidin-4-one, compositions and method of use |
CA2000786C (en) * | 1988-11-07 | 1999-01-26 | Cornelus G. M. Janssen | 3-piperidinyl-1,2-benzisoxazoles |
JP3124120B2 (ja) * | 1992-08-31 | 2001-01-15 | エーザイ株式会社 | 1−ヨウ化アルキル炭酸エステルの製造方法 |
CN1093762A (zh) * | 1993-04-16 | 1994-10-19 | 沈阳石油化工厂 | 氨纶高弹纤维纺丝的制造方法 |
ES2074966B1 (es) * | 1994-02-11 | 1996-06-16 | Vita Invest Sa | Procedimiento para la obtencion de 3-(2-(4-(6-fluoro-benzo(d)isoxazol-3-il)piperidin-1-il)-etil)-2-metil-6,7,8,9-tetrahidro-4h-pirido-(1,2-a)pirimidin-4-ona. |
ES2085234B1 (es) * | 1994-02-24 | 1997-01-16 | Vita Invest Sa | Agente activo sobre el sistema nervioso central, procedimiento para su preparacion y composiciones farmaceuticas que lo contienen. |
CN1160074A (zh) * | 1996-03-19 | 1997-09-24 | 谭兆兴 | 石燃气燃料制造方法 |
TW487572B (en) * | 1996-05-20 | 2002-05-21 | Janssen Pharmaceutica Nv | Aqueous suspensions of 9-hydroxyrisperidone fatty acid esters |
UA72189C2 (uk) * | 1997-11-17 | 2005-02-15 | Янссен Фармацевтика Н.В. | Фармацевтична композиція, що містить водну суспензію субмікронних ефірів 9-гідроксирисперидон жирних кислот |
JP2005060385A (ja) * | 2003-07-31 | 2005-03-10 | Dainippon Pharmaceut Co Ltd | 2−フランカルボン酸ヒドラジド化合物からなる医薬 |
US7314872B2 (en) * | 2003-08-20 | 2008-01-01 | Irm Llc | Inhibitors of cathepsin S |
AU2005247671A1 (en) * | 2004-05-25 | 2005-12-08 | Astrazeneca Ab | 3- (4- (2-dihydroisoxazol-3-ylpyridin-5-yl) phenyl) -5-triazol-1-ylmethyloxazolidin-2-one derivaives as MAO inhibitors for the treatment of bacterial infections |
JP2008513375A (ja) * | 2004-09-13 | 2008-05-01 | ピーアール ファーマシューティカルズ,インコーポレイテッド | エストラジオール代謝産物の長期間作用型の注射可能な結晶性処方物およびその使用法 |
-
2008
- 2008-04-18 CN CN2008800067502A patent/CN101641353B/zh not_active Expired - Fee Related
- 2008-04-18 EP EP08733996.6A patent/EP2154138B1/en not_active Not-in-force
- 2008-04-18 DK DK08733996.6T patent/DK2154138T3/en active
- 2008-04-18 BR BRPI0809837-9A2A patent/BRPI0809837A2/pt not_active IP Right Cessation
- 2008-04-18 RU RU2009142595/04A patent/RU2459824C2/ru not_active IP Right Cessation
- 2008-04-18 US US12/596,516 patent/US8314110B2/en not_active Expired - Fee Related
- 2008-04-18 WO PCT/CN2008/000803 patent/WO2008128436A1/zh active Application Filing
- 2008-04-18 KR KR1020097024012A patent/KR101244185B1/ko active Active
- 2008-04-18 JP JP2010503338A patent/JP5315336B2/ja not_active Expired - Fee Related
Also Published As
Publication number | Publication date |
---|---|
JP5315336B2 (ja) | 2013-10-16 |
EP2154138A1 (en) | 2010-02-17 |
RU2009142595A (ru) | 2011-05-27 |
WO2008128436A1 (en) | 2008-10-30 |
KR20100016659A (ko) | 2010-02-12 |
KR101244185B1 (ko) | 2013-03-25 |
US20100113482A1 (en) | 2010-05-06 |
RU2459824C2 (ru) | 2012-08-27 |
EP2154138B1 (en) | 2015-08-19 |
EP2154138A4 (en) | 2011-06-08 |
DK2154138T3 (en) | 2015-11-02 |
CN101641353A (zh) | 2010-02-03 |
JP2010524863A (ja) | 2010-07-22 |
CN101641353B (zh) | 2012-05-23 |
US8314110B2 (en) | 2012-11-20 |
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Legal Events
Date | Code | Title | Description |
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B07D | Technical examination (opinion) related to article 229 of industrial property law [chapter 7.4 patent gazette] | ||
B06F | Objections, documents and/or translations needed after an examination request according [chapter 6.6 patent gazette] | ||
B08F | Application dismissed because of non-payment of annual fees [chapter 8.6 patent gazette] |
Free format text: REFERENTE A 11A ANUIDADE. |
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B08K | Patent lapsed as no evidence of payment of the annual fee has been furnished to inpi [chapter 8.11 patent gazette] |
Free format text: EM VIRTUDE DO ARQUIVAMENTO PUBLICADO NA RPI 2510 DE 12-02-2019 E CONSIDERANDO AUSENCIA DE MANIFESTACAO DENTRO DOS PRAZOS LEGAIS, INFORMO QUE CABE SER MANTIDO O ARQUIVAMENTO DO PEDIDO DE PATENTE, CONFORME O DISPOSTO NO ARTIGO 12, DA RESOLUCAO 113/2013. |
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B350 | Update of information on the portal [chapter 15.35 patent gazette] |