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BR9909487A - N-pyridonyl herbicides - Google Patents

N-pyridonyl herbicides

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Publication number
BR9909487A
BR9909487A BR9909487-8A BR9909487A BR9909487A BR 9909487 A BR9909487 A BR 9909487A BR 9909487 A BR9909487 A BR 9909487A BR 9909487 A BR9909487 A BR 9909487A
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BR
Brazil
Prior art keywords
alkyl
haloalkyl
alkoxy
phenyl
halogen
Prior art date
Application number
BR9909487-8A
Other languages
Portuguese (pt)
Inventor
Kurt Nebel
Walter Kunz
Jean Wenger
Original Assignee
Novartis Ag
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Filing date
Publication date
Application filed by Novartis Ag filed Critical Novartis Ag
Publication of BR9909487A publication Critical patent/BR9909487A/en

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    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D213/00—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members
    • C07D213/02—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members
    • C07D213/04—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom
    • C07D213/60—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D213/72—Nitrogen atoms
    • C07D213/75—Amino or imino radicals, acylated by carboxylic or carbonic acids, or by sulfur or nitrogen analogues thereof, e.g. carbamates
    • A—HUMAN NECESSITIES
    • A01—AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
    • A01N—PRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
    • A01N43/00—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds
    • A01N43/34—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with one nitrogen atom as the only ring hetero atom
    • A01N43/40—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with one nitrogen atom as the only ring hetero atom six-membered rings
    • A—HUMAN NECESSITIES
    • A01—AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
    • A01N—PRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
    • A01N43/00—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds
    • A01N43/48—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with two nitrogen atoms as the only ring hetero atoms
    • A01N43/54—1,3-Diazines; Hydrogenated 1,3-diazines
    • A—HUMAN NECESSITIES
    • A01—AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
    • A01N—PRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
    • A01N43/00—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds
    • A01N43/48—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with two nitrogen atoms as the only ring hetero atoms
    • A01N43/56—1,2-Diazoles; Hydrogenated 1,2-diazoles
    • A—HUMAN NECESSITIES
    • A01—AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
    • A01N—PRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
    • A01N43/00—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds
    • A01N43/48—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with two nitrogen atoms as the only ring hetero atoms
    • A01N43/58—1,2-Diazines; Hydrogenated 1,2-diazines
    • A—HUMAN NECESSITIES
    • A01—AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
    • A01N—PRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
    • A01N43/00—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds
    • A01N43/64—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with three nitrogen atoms as the only ring hetero atoms
    • A01N43/647—Triazoles; Hydrogenated triazoles
    • A01N43/653—1,2,4-Triazoles; Hydrogenated 1,2,4-triazoles
    • A—HUMAN NECESSITIES
    • A01—AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
    • A01N—PRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
    • A01N43/00—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds
    • A01N43/90—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having two or more relevant hetero rings, condensed among themselves or with a common carbocyclic ring system
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
    • C07D401/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
    • C07D401/04—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings directly linked by a ring-member-to-ring-member bond

Landscapes

  • Life Sciences & Earth Sciences (AREA)
  • Agronomy & Crop Science (AREA)
  • Pest Control & Pesticides (AREA)
  • Plant Pathology (AREA)
  • Health & Medical Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Dentistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Wood Science & Technology (AREA)
  • Zoology (AREA)
  • Environmental Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Agricultural Chemicals And Associated Chemicals (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)

Abstract

Patente de Invenção: <B>"HERBICIDAS DE N-PIRIDONILA"<D>. Os compostos de fórmula I na qual R~ 1~ é hidrogênio, flúor, cloro, bromo ou metila; R~ 2~ é C~ 1~-C~ 4~alquila, C~ 1~-C~ 4~haloalquila, halogênio, nitro, amino, ciano ou R~ 43~O-; R~ 43~ é hidrogênio, C~ 1~-C~ 8~alquila, C~ 3~-C~ 8~alquenila, C~ 3~-C~ 8~alquinila, C~ 3~-C~ 6~cicloalquila, C~ 1~-C~ 8~haloalquila, ciano-C~ 1~-C~ 8~alquila, C~ 3~-C~ 8~haloalquenila, hidróxi-C~ 1~-C~ 4~alquila, C~ 1~-C~ 4~alcóxi-C~ 1~-C~ 4~alquila, C~ 3~-C~ 6~alquenilóxi-C~ 1~-C~ 4~-alquila, C~ 3~-C~ 6~alquinilóxi-C~ 1~-C~ 4~alquila, C~ 1~-C~ 4~alcóxi-C~ 1~-C~ 4~alcóxi-C~ 1~-C~ 4~alquila, C~ 1~-C~ 4~-alquiltio-C~ 1~-C~ 4~alquila, C~ 1~-C~ 8~alquilcarbonila, C~ 1~-C~ 8~alcoxicarbonila, C~ 3~-C~ 8~alqueniloxicarbonila, benzilóxi-C~ 1~- ou -C~ 2~-alquila, benzilcarbonila, benziloxicarbonila, fenila, fenil-C~ 2~-C~ 8~alquila, benzila, piridila, pirimidinila, pirazinila ou piridazinila, aqueles anéis aromáticos e heteroaromáticos sendo insubstituídos ou mono- a tri-substituídos por halogênio, C~ 1~-C~ 4~alquila ou por C~ 1~-C~ 4~haloalquila; ou R~ 43~ é R~ 44~X~ 16~C(O)-C~ 1~-C~ 8~alquil- ou X~ 16~ é oxigênio, enxofre ou R~ 44~ é hidrogênio, C~ 1~-C~ 8~alquila, C~ 3~-C~ 8~alquenila, C~ 3~-C~ 8~alquinila, C~ 3~-C~ 6~cicloalquila, C~ 1~-C~ 8~haloalquila, C~ 3~-C~ 8~haloalquenila, C~ 1~-C~ 4~alcoxi-C~ 1~-C~ 4~alquila, C~ 3~-C~ 6~alqueniloxi-C~ 1~-C~ 4~alquila, C~ 1~-C~ 4~alquiltio-C~ 1~-C~ 4~alquila, fenila, fenila mono- a tri-substituída por halogênio, C~ 1~-C~ 4~alquila ou por C~ 1~-C~ 4~haloalquila, benzila ou benzila mono- a tri-substituída no anel de fenila por halogênio, C~ 1~-C~ 4~alquila ou por C~ 1~-C~ 4~haloalquila; R~ 45~ é hidrogênio, C~ 1~-C~ 8~alquila, C~ 3~-C~ 8~alquenila, C~ 3~-C~ 8~alquinila, C~ 3~-C~ 6~cicloalquila, C~ 1~-C~ 8~haloalquila ou benzila; R~ 3~ é hidróxi, C~ 1~-C~ 6~alcóxi, C~ 3~-C~ 6~alquenilóxi, C~ 3~-C~ 6~alquinilóxi, C~ 1~-C~ 6~haloalcóxi, C~ 3~-C~ 6~haloalquenilóxi, C~ 1~-C~ 6~alcóxi-C~ 1~-C~ 6~alquila, C~ 3~-C~ 6~alquenilóxi-C~ 1~-C~ 6~alquila, C~ 3~-C~ 6~alquiniloxi-C~ 1~-C~ 6~alquila, C~ 1~-C~ 6~alcoxi-C~ 1~-C~ 6~alcoxi-C~ 1~-C~ 6~alquila, B~ 1~-C~ 1~-C~ 6~alcóxi, R~ 4~(R~ 5~)N-, C~ 1~-C~ 6~alquila, C~ 3~-C~ 6~alquenila, C~ 3~-C~ 6~alquinila, C~ 2~-C~ 6~haloalquila, C~ 3~-C~ 6~háloalquenila, C~ 3~-C~ 6~cicloalquila, C~ 3~-C~ 6~halocicloalquila, B~ 1~-C~ 1~-C~ 6~alquila, OHC-, C~ 1~-C~ 6~alquilcarbonila, C~ 1~-C~ 6~alquilcarbonilóxi, C~ 1~-C~ 6~haloalquilcarbonila, C~ 2~-C~ 6~alquenilcarbonila, C~ 1~-C~ 6~alcoxicarbonila, C~ 1~-C~ 6~alquil-S(O)~ 2~-, C~ 1~-C~ 6~haloalquil-S(O)~ 2~-, C~ 3~-C~ 8~trialquilsililóxi, (C~ 1~-C~ 6~alquil)~ 2~N-N=CH-, B~ 1~CH=N-, (CH~ 3~)~ 2~N-CH=N-, (C~ 1~-C~ 5~hidroxialquil)-CH~ 2~-, (B~ 1~-C~ 1~-C~ 5~hidroxialquil)-CH~ 2~-, (B-C~ 1~-C~ 5~haloalquil)-CH~ 2~-, (Hidróxi-C~ 1~-C~ 5~alquil)-O- ou (B~ 1~-C~ 1~-C~ 5~hidroxialquil)-O-; B~ 1~ é ciano, OHC-, HOC(O)-, C~ 1~-C~ 6~alquilcarbonila, C~ 1~-C~ 6~haloalquilcarbonila, C~ 1~-C~ 6~alcoxicarbonila, C~ 3~-C~ 6~alqueniloxicarbonila, C~ 3~-C~ 6~alquiniloxicarbonila, benzilóxi, benziloxicarbonila, benziloxicarbonila mono- a tri-substituída no anel de fenila por halogênio, C~ 1~-C~ 4~alquila ou por C~ 1~-C~ 4~haloalquila, benziltio, benziltiocarbonila, benziltiocarbonila mono- a tri-substituída no anel de fenila por halogênio, C~ 1~-C~ 4~alquila ou por C~ 1~-C~ 4~haloalquila, C~ 1~-C~ 6~haloalcoxicarbonila, C~ 1~-C~ 6~alquiltio-C(O)-, R~ 6~(R~ 7~)NC(O)-, fenila, fenila mono- a tri-substituída por halogênio, C~ 1~-C~ 4~alquila ou por C~ 1~-C~ 4~haloalquila, C~ 1~-C~ 6~alquil-S(O)~ 2~-, C~ 1~-C~ 6~alquil-S(O)-, C~ 1~-C~ 6~alquiltio-, C~ 3~-C~ 6~cicloalquila, C~ 1~-C~ 6~alcóxi, C~ 3~-C~ 6~alqueniltio ou C~ 3~C~ 6~alquiniltio; R~ 4~ e R~ 5~ são, cada um independentemente do outro, hidrogênio, C~ 1~-C~ 6~alquila, C~ 3~-C~ 6~alquenila, C~ 3~-C~ 6~alquinila, C~ 1~-C~ 6~haloalquila, C~ 3~-C~ 6~haloalquenila, C~ 3~-C~ 6~-cicloalquila, C~ 1~-C~ 6~alcóxi-C~ 1~-C~ 6~alquila, OHC-, C~ 1~-C~ 6~alquilcarbonila, C~ 1~-C~ 6~haloalquilcarbonila, C~ 1~-C~ 6~alquil-S(O)~ 2~- ou C~ 1~-C~ 6~haloalquil-S(O)~ 2~-; R~ 6~ e R~ 7~ são, cada um independentemente do outro, hidrogênio, C~ 1~-C~ 6~alquila, C~ 3~-C~ 6~alquenila, C~ 3~-C~ 6~alquinila, C~ 1~-C~ 6~haloalquila, C~ 3~-C~ 6~haloalquenila, fenila, fenila mono- a tri-substituída por halogênio, C~ 1~-C~ 4~-alquila ou por C~ 1~-C~ 4~haloalquila, benzila ou benzila mono- a tri-substituída no anel de fenila por halogênio, C~ 1~-C~ 4~alquila ou por C~ 1~-C~ 4~haloalquila; X~ 1~ é oxigênio ou enxofre; W é um grupo e R~ 8~ a R~ 32~ e X~ 2~ a X~ 15~ são como definidos na reivindicação 1, e os sais e os estereoisómeros agroquimicamente aceitáveis de tais compostos de fórmula I, são adequados para uso como herbicidas.Invention Patent: <B> "N-PYRIDONILLA HERBICIDES" <D>. The compounds of formula I in which R ~ 1 ~ is hydrogen, fluorine, chlorine, bromine or methyl; R ~ 2 ~ is C ~ 1 ~ -C ~ 4 ~ alkyl, C ~ 1 ~ -C ~ 4 ~ haloalkyl, halogen, nitro, amino, cyano or R ~ 43 ~ O-; R ~ 43 ~ is hydrogen, C ~ 1 ~ -C ~ 8 ~ alkyl, C ~ 3 ~ -C ~ 8 ~ alkenyl, C ~ 3 ~ -C ~ 8 ~ alkynyl, C ~ 3 ~ -C ~ 6 ~ cycloalkyl , C ~ 1 ~ -C ~ 8 ~ haloalkyl, cyano-C ~ 1 ~ -C ~ 8 ~ alkyl, C ~ 3 ~ -C ~ 8 ~ haloalkenyl, hydroxy-C ~ 1 ~ -C ~ 4 ~ alkyl, C ~ 1 ~ -C ~ 4 ~ C-alkoxy ~ 1 ~ -C ~ 4 ~ alkyl, C ~ 3 ~ -C ~ 6 ~ C-alkenyloxy ~ 1 ~ -C ~ 4 ~ -alkyl, C ~ 3 ~ -C ~ 6 ~ C-alkynyloxy ~ 1 ~ -C ~ 4 ~ alkyl, C ~ 1 ~ -C ~ 4 ~ C-alkoxy ~ 1 ~ -C ~ 4 ~ C ~ 1 ~ -C ~ 4 ~ alkoxy, C ~ 1 ~ -C ~ 4 ~ -Alkylthio-C ~ 1 ~ -C ~ 4 ~ alkyl, C ~ 1 ~ -C ~ 8 ~ alkylcarbonyl, C ~ 1 ~ -C ~ 8 ~ alkoxycarbonyl, C ~ 3 ~ -C ~ 8 ~ alkenyloxycarbonyl, benzyloxy-C ~ 1 ~ - or -C ~ 2 ~ -alkyl, benzylcarbonyl, benzyloxycarbonyl, phenyl, phenyl-C ~ 2 ~ -C ~ 8 ~ alkyl, benzyl, pyridyl, pyrimidinyl, pyrazinyl or pyridazinyl, those aromatic and heteroaromatic rings being unsubstituted or mono- to tri-substituted by halogen, C ~ 1 ~ -C ~ 4 ~ alkyl or by C ~ 1 ~ -C ~ 4 ~ haloalkyl; or R ~ 43 ~ is R ~ 44 ~ X ~ 16 ~ C (O) -C ~ 1 ~ -C ~ 8 ~ alkyl- or X ~ 16 ~ is oxygen, sulfur or R ~ 44 ~ is hydrogen, C ~ 1 ~ -C ~ 8 ~ alkyl, C ~ 3 ~ -C ~ 8 ~ alkenyl, C ~ 3 ~ -C ~ 8 ~ alkynyl, C ~ 3 ~ -C ~ 6 ~ cycloalkyl, C ~ 1 ~ -C ~ 8 ~ haloalkyl, C ~ 3 ~ -C ~ 8 ~ haloalkenyl, C ~ 1 ~ -C ~ 4 ~ alkoxy-C ~ 1 ~ -C ~ 4 ~ alkyl, C ~ 3 ~ -C ~ 6 ~ alkenyloxy-C ~ 1 ~ -C ~ 4 ~ alkyl, C ~ 1 ~ -C ~ 4 ~ alkylthio-C ~ 1 ~ -C ~ 4 ~ alkyl, phenyl, phenyl mono- to tri-substituted by halogen, C ~ 1 ~ -C ~ 4 ~ alkyl or by C ~ 1 ~ -C ~ 4 ~ haloalkyl, benzyl or benzyl mono- to tri-substituted on the phenyl ring by halogen, C ~ 1 ~ -C ~ 4 ~ alkyl or by C ~ 1 ~ -C ~ 4 haloalkyl; R ~ 45 ~ is hydrogen, C ~ 1 ~ -C ~ 8 ~ alkyl, C ~ 3 ~ -C ~ 8 ~ alkenyl, C ~ 3 ~ -C ~ 8 ~ alkynyl, C ~ 3 ~ -C ~ 6 ~ cycloalkyl , C ~ 1 ~ -C ~ 8 ~ haloalkyl or benzyl; R ~ 3 ~ is hydroxy, C ~ 1 ~ -C ~ 6 ~ alkoxy, C ~ 3 ~ -C ~ 6 ~ alkenyloxy, C ~ 3 ~ -C ~ 6 ~ alkynyloxy, C ~ 1 ~ -C ~ 6 ~ haloalkoxy , C ~ 3 ~ -C ~ 6 ~ haloalkenyloxy, C ~ 1 ~ -C ~ 6 ~ alkoxy-C ~ 1 ~ -C ~ 6 ~ alkyl, C ~ 3 ~ -C ~ 6 ~ alkenyloxy-C ~ 1 ~ - C ~ 6 ~ alkyl, C ~ 3 ~ -C ~ 6 ~ alkynyloxy-C ~ 1 ~ -C ~ 6 ~ alkyl, C ~ 1 ~ -C ~ 6 ~ alkoxy-C ~ 1 ~ -C ~ 6 ~ alkoxy- C ~ 1 ~ -C ~ 6 ~ alkyl, B ~ 1 ~ -C ~ 1 ~ -C ~ 6 ~ alkoxy, R ~ 4 ~ (R ~ 5 ~) N-, C ~ 1 ~ -C ~ 6 ~ alkyl , C ~ 3 ~ -C ~ 6 ~ alkenyl, C ~ 3 ~ -C ~ 6 ~ alkynyl, C ~ 2 ~ -C ~ 6 ~ haloalkyl, C ~ 3 ~ -C ~ 6 ~ haloalkenyl, C ~ 3 ~ - C ~ 6 ~ cycloalkyl, C ~ 3 ~ -C ~ 6 ~ halocycloalkyl, B ~ 1 ~ -C ~ 1 ~ -C ~ 6 ~ alkyl, OHC-, C ~ 1 ~ -C ~ 6 ~ alkylcarbonyl, C ~ 1 ~ -C ~ 6 ~ alkylcarbonyloxy, C ~ 1 ~ -C ~ 6 ~ haloalkylcarbonyl, C ~ 2 ~ -C ~ 6 ~ alkenylcarbonyl, C ~ 1 ~ -C ~ 6 ~ alkoxycarbonyl, C ~ 1 ~ -C ~ 6 ~ alkyl-S (O) ~ 2 ~ -, C ~ 1 ~ -C ~ 6 ~ haloalkyl-S (O) ~ 2 ~ -, C ~ 3 ~ -C ~ 8 ~ trialkylsilyloxy, (C ~ 1 ~ -C ~ 6 ~ alkyl) ~ 2 ~ NN = CH-, B ~ 1 ~ CH = N-, (CH ~ 3 ~) ~ 2 ~ N-CH = N-, (C ~ 1 ~ -C ~ 5 ~ hydroxyalkyl) - CH ~ 2 ~ -, (B ~ 1 ~ -C ~ 1 ~ -C ~ 5 ~ hydroxyalkyl) -CH ~ 2 ~ -, (BC ~ 1 ~ -C ~ 5 ~ haloalkyl) -CH ~ 2 ~ -, ( C-hydroxy ~ 1 ~ -C ~ 5 ~ alkyl) -O- or (B ~ 1 ~ -C ~ 1 ~ -C ~ 5 ~ hydroxyalkyl) -O-; B ~ 1 ~ is cyano, OHC-, HOC (O) -, C ~ 1 ~ -C ~ 6 ~ alkylcarbonyl, C ~ 1 ~ -C ~ 6 ~ haloalkylcarbonyl, C ~ 1 ~ -C ~ 6 ~ alkoxycarbonyl, C ~ 3 ~ -C ~ 6 ~ alkenyloxycarbonyl, C ~ 3 ~ -C ~ 6 ~ alkynyloxycarbonyl, benzyloxy, benzyloxycarbonyl, benzyloxycarbonyl mono- to tri-substituted on the phenyl ring by halogen, C ~ 1 ~ -C ~ 4 ~ alkyl or with C ~ 1 ~ -C ~ 4 ~ haloalkyl, benzylthio, benzylthiocarbonyl, mono- to tri-substituted benzylthiocarbonyl on the phenyl ring with halogen, C ~ 1 ~ -C ~ 4 ~ alkyl or with C ~ 1 ~ -C ~ 4 ~ haloalkyl, C ~ 1 ~ -C ~ 6 ~ haloalkoxycarbonyl, C ~ 1 ~ -C ~ 6 ~ alkylthio-C (O) -, R ~ 6 ~ (R ~ 7 ~) NC (O) -, phenyl, phenyl mono- to tri-substituted by halogen, C ~ 1 ~ -C ~ 4 ~ alkyl or by C ~ 1 ~ -C ~ 4 ~ haloalkyl, C ~ 1 ~ -C ~ 6 ~ alkyl-S (O) ~ 2 ~ -, C ~ 1 ~ -C ~ 6 ~ alkyl-S (O) -, C ~ 1 ~ -C ~ 6 ~ alkylthio-, C ~ 3 ~ -C ~ 6 ~ cycloalkyl, C ~ 1 ~ -C ~ 6 ~ alkoxy, C ~ 3 ~ -C ~ 6 ~ alkenylthio or C ~ 3 ~ C ~ 6 ~ alkynylthio; R ~ 4 ~ and R ~ 5 ~ are each independently hydrogen, C ~ 1 ~ -C ~ 6 ~ alkyl, C ~ 3 ~ -C ~ 6 ~ alkenyl, C ~ 3 ~ -C ~ 6 ~ alkynyl, C ~ 1 ~ -C ~ 6 ~ haloalkyl, C ~ 3 ~ -C ~ 6 ~ haloalkenyl, C ~ 3 ~ -C ~ 6 ~ -cycloalkyl, C ~ 1 ~ -C ~ 6 ~ alkoxy-C ~ 1 ~ -C ~ 6 ~ alkyl, OHC-, C ~ 1 ~ -C ~ 6 ~ alkylcarbonyl, C ~ 1 ~ -C ~ 6 ~ haloalkylcarbonyl, C ~ 1 ~ -C ~ 6 ~ alkyl-S (O) ~ 2 ~ - or C ~ 1 ~ -C ~ 6 ~ haloalkyl-S (O) ~ 2 ~ -; R ~ 6 ~ and R ~ 7 ~ are each independently hydrogen, C ~ 1 ~ -C ~ 6 ~ alkyl, C ~ 3 ~ -C ~ 6 ~ alkenyl, C ~ 3 ~ -C ~ 6 ~ alkynyl, C ~ 1 ~ -C ~ 6 ~ haloalkyl, C ~ 3 ~ -C ~ 6 ~ haloalkenyl, phenyl, phenyl mono- to tri-substituted by halogen, C ~ 1 ~ -C ~ 4 ~ -alkyl or by C ~ 1 ~ -C ~ 4 ~ haloalkyl, benzyl or benzyl mono- to tri-substituted on the phenyl ring by halogen, C ~ 1 ~ -C ~ 4 ~ alkyl or by C ~ 1 ~ -C ~ 4 ~ haloalkyl; X ~ 1 ~ is oxygen or sulfur; W is a group and R ~ 8 ~ to R ~ 32 ~ and X ~ 2 ~ to X ~ 15 ~ are as defined in claim 1, and the agrochemically acceptable salts and stereoisomers of such compounds of formula I, are suitable for use as herbicides.

BR9909487-8A 1998-04-08 1999-04-06 N-pyridonyl herbicides BR9909487A (en)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
CH84098 1998-04-08
PCT/EP1999/002313 WO1999052893A1 (en) 1998-04-08 1999-04-06 N-pyridonyl herbicides

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BR9909487A true BR9909487A (en) 2000-12-12

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JP (1) JP2002511461A (en)
KR (1) KR20010042521A (en)
CN (1) CN1295570A (en)
AU (1) AU738222B2 (en)
BR (1) BR9909487A (en)
ID (1) ID27165A (en)
WO (1) WO1999052893A1 (en)

Families Citing this family (22)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CA2469435A1 (en) 2001-12-21 2003-07-24 X-Ceptor Therapeutics, Inc. Modulators of lxr
US7482366B2 (en) 2001-12-21 2009-01-27 X-Ceptor Therapeutics, Inc. Modulators of LXR
NZ534395A (en) 2002-02-14 2006-10-27 Pharmacia Corp Substituted pyridinones as modulators of p38 MAP kinase
KR100574350B1 (en) * 2004-08-31 2006-04-27 한국화학연구원 Method for preparing 2-aminopyridine derivative
PE20070522A1 (en) 2005-09-14 2007-07-11 Takeda Pharmaceutical 2- [6- (3-AMINO-PIPERIDIN-1-IL) -3-METHYL-2,4-DIOXO-3,4-DIHYDRO-2H-PYRIMIDIN-1-ILMETHYL] -4-FLUORO-BENZONITRILE AS INHIBITOR OF DIPEPTIDIL PEPTIDASE AND PHARMACEUTICAL COMPOSITIONS CONTAINING IT
TWI417095B (en) 2006-03-15 2013-12-01 Janssen Pharmaceuticals Inc 1,4-disubstituted 3-cyano-pyridone derivatives and their use as positive allosteric modulators of mglur2-receptors
TW200845978A (en) 2007-03-07 2008-12-01 Janssen Pharmaceutica Nv 3-cyano-4-(4-tetrahydropyran-phenyl)-pyridin-2-one derivatives
TW200900065A (en) 2007-03-07 2009-01-01 Janssen Pharmaceutica Nv 3-cyano-4-(4-pyridinyloxy-phenyl)-pyridin-2-one derivatives
CN103342695B (en) 2007-09-14 2015-04-22 杨森制药有限公司 1',3'-disubstituted-4-pheny-3,4,5,6-tetrahydro-2H,1'H-[1,4']bipyridinyl-2'-ones
WO2010025890A1 (en) 2008-09-02 2010-03-11 Ortho-Mcneil-Janssen Pharmaceuticals, Inc 3-azabicyclo[3.1.0]hexyl derivatives as modulators of metabotropic glutamate receptors
EP2373649B1 (en) 2008-11-28 2013-01-23 Janssen Pharmaceuticals, Inc. Indole and benzoxazine derivatives as modulators of metabotropic glutamate receptors
AU2010246609B2 (en) 2009-05-12 2013-09-05 Addex Pharma S.A. 1,2,4-triazolo [4,3-a] pyridine derivatives and their use for the treatment or prevention of neurological and psychiatric disorders
MX2011011962A (en) 2009-05-12 2012-02-28 Janssen Pharmaceuticals Inc 1,2,4-triazolo[4,3-a]pyridine derivatives and their use as positive allosteric modulators of mglur2 receptors.
MY153913A (en) 2009-05-12 2015-04-15 Janssen Pharmaceuticals Inc 7-aryl-1,2,4-triazolo[4,3-a]pyridine derivatives and their use as positive allosteric modulators of mglur2 receptors
CA2814998C (en) 2010-11-08 2019-10-29 Janssen Pharmaceuticals, Inc. 1,2,4-triazolo[4,3-a]pyridine derivatives and their use as positive allosteric modulators of mglur2 receptors
WO2012062750A1 (en) 2010-11-08 2012-05-18 Janssen Pharmaceuticals, Inc. 1,2,4-TRIAZOLO[4,3-a]PYRIDINE DERIVATIVES AND THEIR USE AS POSITIVE ALLOSTERIC MODULATORS OF MGLUR2 RECEPTORS
US8993591B2 (en) 2010-11-08 2015-03-31 Janssen Pharmaceuticals, Inc. 1,2,4-triazolo[4,3-a] pyridine derivatives and their use as positive allosteric modulators of MGLUR2 receptors
WO2014004094A1 (en) * 2012-06-30 2014-01-03 Dow Agrosciences Llc Production of n-substituted sulfoximine pyridine n-oxides
JO3368B1 (en) 2013-06-04 2019-03-13 Janssen Pharmaceutica Nv 6, 7- dihydropyrazolu [5,1-a] pyrazine-4 (5 hands) -on compounds and their use as negative excretory regulators of Miglore 2 receptors.
JO3367B1 (en) 2013-09-06 2019-03-13 Janssen Pharmaceutica Nv 1,2,4-TRIAZOLO[4,3-a]PYRIDINE COMPOUNDS AND THEIR USE AS POSITIVE ALLOSTERIC MODULATORS OF MGLUR2 RECEPTORS
SMT202100103T1 (en) 2014-01-21 2021-03-15 Janssen Pharmaceutica Nv COMBINATION COMPRISING POSITIVE ALLOSTERIC MODULATORS OF THE METABOTROPIC GLUTAMATE RECEPTOR SUBTYPE 2 AND THEIR USE
HUE045610T2 (en) 2014-01-21 2020-01-28 Janssen Pharmaceutica Nv Combinations comprising positive allosteric modulators or orthosteric agonists of metabotropic glutamatergic receptor subtype 2 and their use

Family Cites Families (9)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JPS58213776A (en) * 1982-06-07 1983-12-12 Ishihara Sangyo Kaisha Ltd Pyridazinone compound and fungicide containing the same
JPS62258731A (en) * 1986-05-06 1987-11-11 Kao Corp Oil-in-water-type emulsified composition
DE3917469A1 (en) * 1989-05-30 1990-12-06 Bayer Ag Heterocyclyl-substd. pyridine derivs. - useful as herbicides, e.g. defoliants, desiccants and esp. weed-killers
NO179282C (en) * 1991-01-18 1996-09-11 Rhone Poulenc Agrochimie New 1- (2-pyridyl) pyrazole compounds for control of insect pests
US5726124A (en) * 1992-07-17 1998-03-10 Rohm And Haas Company 2-arylpyrimidines and herbicidal use thereof
JPH06172306A (en) * 1992-10-05 1994-06-21 Nissan Chem Ind Ltd Cyclic amide compound and herbicide
DE19518054A1 (en) * 1995-03-08 1996-09-12 Hoechst Schering Agrevo Gmbh New 1-(phenyl or pyridyl)-pyrazole derivs.
DE19530606A1 (en) * 1995-08-21 1997-02-27 Basf Ag 1- (pyridyl) pyrazole
GB9711753D0 (en) * 1997-06-06 1997-08-06 Merck Sharp & Dohme Therapeutic agents

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