BR9207024A - Processo e utilizações para 4,5-DI-hidrogeldanamicina e sua hidroquinona - Google Patents
Processo e utilizações para 4,5-DI-hidrogeldanamicina e sua hidroquinonaInfo
- Publication number
- BR9207024A BR9207024A BR9207024A BR9207024A BR9207024A BR 9207024 A BR9207024 A BR 9207024A BR 9207024 A BR9207024 A BR 9207024A BR 9207024 A BR9207024 A BR 9207024A BR 9207024 A BR9207024 A BR 9207024A
- Authority
- BR
- Brazil
- Prior art keywords
- hydrogeldanamycin
- hydroquinone
- Prior art date
Links
- QIGBRXMKCJKVMJ-UHFFFAOYSA-N Hydroquinone Chemical compound OC1=CC=C(O)C=C1 QIGBRXMKCJKVMJ-UHFFFAOYSA-N 0.000 title 2
Classifications
-
- C—CHEMISTRY; METALLURGY
- C12—BIOCHEMISTRY; BEER; SPIRITS; WINE; VINEGAR; MICROBIOLOGY; ENZYMOLOGY; MUTATION OR GENETIC ENGINEERING
- C12P—FERMENTATION OR ENZYME-USING PROCESSES TO SYNTHESISE A DESIRED CHEMICAL COMPOUND OR COMPOSITION OR TO SEPARATE OPTICAL ISOMERS FROM A RACEMIC MIXTURE
- C12P17/00—Preparation of heterocyclic carbon compounds with only O, N, S, Se or Te as ring hetero atoms
- C12P17/10—Nitrogen as only ring hetero atom
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
- A61P31/04—Antibacterial agents
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
- A61P31/12—Antivirals
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P37/00—Drugs for immunological or allergic disorders
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D225/00—Heterocyclic compounds containing rings of more than seven members having one nitrogen atom as the only ring hetero atom
- C07D225/04—Heterocyclic compounds containing rings of more than seven members having one nitrogen atom as the only ring hetero atom condensed with carbocyclic rings or ring systems
- C07D225/06—Heterocyclic compounds containing rings of more than seven members having one nitrogen atom as the only ring hetero atom condensed with carbocyclic rings or ring systems condensed with one six-membered ring
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Health & Medical Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
- Chemical Kinetics & Catalysis (AREA)
- General Chemical & Material Sciences (AREA)
- Engineering & Computer Science (AREA)
- General Health & Medical Sciences (AREA)
- Zoology (AREA)
- Wood Science & Technology (AREA)
- Veterinary Medicine (AREA)
- Animal Behavior & Ethology (AREA)
- Pharmacology & Pharmacy (AREA)
- Public Health (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Medicinal Chemistry (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Communicable Diseases (AREA)
- Oncology (AREA)
- Microbiology (AREA)
- Biochemistry (AREA)
- Biotechnology (AREA)
- General Engineering & Computer Science (AREA)
- Genetics & Genomics (AREA)
- Immunology (AREA)
- Virology (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Preparation Of Compounds By Using Micro-Organisms (AREA)
- Saccharide Compounds (AREA)
- Heterocyclic Carbon Compounds Containing A Hetero Ring Having Oxygen Or Sulfur (AREA)
Applications Claiming Priority (2)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
US81723592A | 1992-01-06 | 1992-01-06 | |
PCT/US1992/010189 WO1993014215A1 (en) | 1992-01-06 | 1992-12-03 | Process and uses for 4,5-dihydrogeldanamycin and its hydroquinone |
Publications (1)
Publication Number | Publication Date |
---|---|
BR9207024A true BR9207024A (pt) | 1995-12-05 |
Family
ID=25222638
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
BR9207024A BR9207024A (pt) | 1992-01-06 | 1992-12-03 | Processo e utilizações para 4,5-DI-hidrogeldanamicina e sua hidroquinona |
Country Status (15)
Country | Link |
---|---|
JP (1) | JPH06510913A (sv) |
KR (1) | KR940703923A (sv) |
CN (1) | CN1074937A (sv) |
AU (1) | AU3225693A (sv) |
BR (1) | BR9207024A (sv) |
CA (1) | CA2127457A1 (sv) |
CZ (1) | CZ390592A3 (sv) |
FI (1) | FI943207A0 (sv) |
HU (1) | HU9401936D0 (sv) |
IL (1) | IL104289A0 (sv) |
MX (1) | MX9300011A (sv) |
NO (1) | NO942532D0 (sv) |
PT (1) | PT101169A (sv) |
WO (1) | WO1993014215A1 (sv) |
ZA (1) | ZA9333B (sv) |
Families Citing this family (26)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
CA2166320A1 (en) * | 1993-06-29 | 1995-01-12 | Randall James Gallaschun | Ansamycin derivatives as antioncogene and anticancer agents |
US5932566A (en) * | 1994-06-16 | 1999-08-03 | Pfizer Inc. | Ansamycin derivatives as antioncogene and anticancer agents |
US6852496B1 (en) | 1997-08-12 | 2005-02-08 | Oregon Health And Science University | Methods of screening for agents that promote nerve cell growth |
US6872715B2 (en) | 2001-08-06 | 2005-03-29 | Kosan Biosciences, Inc. | Benzoquinone ansamycins |
CA2460498A1 (en) | 2001-09-24 | 2003-04-03 | Conforma Therapeutics Corporation | Process for preparing 17-allyl amino geldanamycin (17-aag) and other ansamycins |
EP1923061A1 (en) | 2001-09-24 | 2008-05-21 | Conforma Therapeutic Corporation | Process for preparing 17-Allyl amino geldanamycin (17-AAG) and other ansamycins |
DE60327994D1 (de) | 2002-02-08 | 2009-07-30 | Conforma Therapeutics Corp | Ansamycine mit verbesserten pharmakologischen und biologischen eigenschaften |
TW200303363A (en) * | 2002-02-25 | 2003-09-01 | Upjohn Co | Process to prepare and isolate geldanamycin |
WO2005009345A2 (en) | 2003-06-13 | 2005-02-03 | Kosan Biosciences, Inc. | 2-desmethyl ansamycin compounds |
US6870049B1 (en) | 2003-11-12 | 2005-03-22 | Kosan Biosciences, Inc. | 11-O-methylgeldanamycin compounds |
US6855705B1 (en) | 2003-11-12 | 2005-02-15 | Kosan Biosciences, Inc. | 11-O-methylgeldanamycin compounds |
US6887993B1 (en) | 2003-11-12 | 2005-05-03 | Kosan Biosciences, Inc. | 11-O-methylgeldanamycin compounds |
US6875863B1 (en) | 2003-11-12 | 2005-04-05 | Kosan Biosciences, Inc. | 11-O-methylgeldanamycin compounds |
JP2007512369A (ja) * | 2003-11-26 | 2007-05-17 | エンテロス・インコーポレーテッド | 低酸素誘導因子1αアンタゴニストを用いる慢性関節リウマチの処置 |
CN1898212B (zh) * | 2003-12-23 | 2012-06-13 | 无限发现公司 | 用于治疗癌症的包含苯醌的安沙霉素类似物 |
US20060019941A1 (en) * | 2003-12-23 | 2006-01-26 | Infinity Pharmaceuticals, Inc. | Analogs of benzoquinone-containing ansamycins and methods of use thereof |
BRPI0418147A (pt) | 2003-12-23 | 2007-04-17 | Infinity Pharmaceuticals Inc | análogos de ansamicinas contendo benzoquinona e seus métodos de uso |
KR20080004550A (ko) | 2005-03-30 | 2008-01-09 | 콘포마 세러퓨틱스 코포레이션 | Hsp90-억제제로서 알키닐 피롤로피리미딘 및 관련유사체 |
AU2007319014B2 (en) * | 2006-11-09 | 2013-03-28 | Bristol-Myers Squibb Company | Novel compounds and methods for their production |
PE20081506A1 (es) | 2006-12-12 | 2008-12-09 | Infinity Discovery Inc | Formulaciones de ansamicina |
CN100500668C (zh) * | 2006-12-19 | 2009-06-17 | 中国人民解放军军事医学科学院毒物药物研究所 | 格尔德霉素衍生物及其制备方法和制备药物的用途 |
EP2121957A4 (en) | 2007-01-26 | 2010-11-10 | Kosan Biosciences Inc | MACROLACTAMES OBTAINED BY MODIFIED BIOSYNTHESIS |
EP2297109A4 (en) * | 2008-04-21 | 2011-06-22 | Biocon Ltd | METHOD FOR ISOLATING AND PURIFYING GELDANAMYCIN |
WO2010045442A1 (en) | 2008-10-15 | 2010-04-22 | Infinity Discovery, Inc. | Ansamycin hydroquinone compositions |
CN102030764B (zh) * | 2010-11-12 | 2012-07-04 | 中国医学科学院医药生物技术研究所 | 4,5双氢噻嗪酮格尔德霉素及其制备方法 |
CN103305563B (zh) * | 2013-06-14 | 2014-12-03 | 湖南农业大学 | 一种以链霉菌提制阿里沙霉素的方法 |
Family Cites Families (1)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US3595955A (en) * | 1969-03-26 | 1971-07-27 | Upjohn Co | Geldanamycin and process for producing same |
-
1992
- 1992-12-03 AU AU32256/93A patent/AU3225693A/en not_active Abandoned
- 1992-12-03 HU HU9401936A patent/HU9401936D0/hu unknown
- 1992-12-03 BR BR9207024A patent/BR9207024A/pt not_active Application Discontinuation
- 1992-12-03 KR KR1019940702334A patent/KR940703923A/ko not_active Application Discontinuation
- 1992-12-03 WO PCT/US1992/010189 patent/WO1993014215A1/en active Application Filing
- 1992-12-03 JP JP5512423A patent/JPH06510913A/ja active Pending
- 1992-12-03 CA CA002127457A patent/CA2127457A1/en not_active Abandoned
- 1992-12-15 CN CN92113885A patent/CN1074937A/zh active Pending
- 1992-12-28 CZ CS923905A patent/CZ390592A3/cs unknown
- 1992-12-31 IL IL104289A patent/IL104289A0/xx unknown
-
1993
- 1993-01-04 PT PT101169A patent/PT101169A/pt not_active Application Discontinuation
- 1993-01-05 MX MX9300011A patent/MX9300011A/es unknown
- 1993-01-05 ZA ZA9333A patent/ZA9333B/xx unknown
-
1994
- 1994-07-05 FI FI943207A patent/FI943207A0/sv unknown
- 1994-07-05 NO NO942532A patent/NO942532D0/no unknown
Also Published As
Publication number | Publication date |
---|---|
ZA9333B (en) | 1994-07-05 |
CA2127457A1 (en) | 1993-07-22 |
JPH06510913A (ja) | 1994-12-08 |
NO942532L (no) | 1994-07-05 |
FI943207L (sv) | 1994-07-05 |
MX9300011A (es) | 1993-12-01 |
IL104289A0 (en) | 1993-05-13 |
CN1074937A (zh) | 1993-08-04 |
FI943207A0 (sv) | 1994-07-05 |
NO942532D0 (no) | 1994-07-05 |
PT101169A (pt) | 1994-03-31 |
KR940703923A (ko) | 1994-12-12 |
AU3225693A (en) | 1993-08-03 |
WO1993014215A1 (en) | 1993-07-22 |
CZ390592A3 (en) | 1993-08-11 |
HU9401936D0 (en) | 1994-09-28 |
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Legal Events
Date | Code | Title | Description |
---|---|---|---|
FA1 | Application withdrawn (art. 18(2)) |