BR122017023130A8 - Derivado de tetrazoliloxima, métodos de produção de derivados de tetrazoliloxima - Google Patents
Derivado de tetrazoliloxima, métodos de produção de derivados de tetrazoliloximaInfo
- Publication number
- BR122017023130A8 BR122017023130A8 BR122017023130A BR122017023130A BR122017023130A8 BR 122017023130 A8 BR122017023130 A8 BR 122017023130A8 BR 122017023130 A BR122017023130 A BR 122017023130A BR 122017023130 A BR122017023130 A BR 122017023130A BR 122017023130 A8 BR122017023130 A8 BR 122017023130A8
- Authority
- BR
- Brazil
- Prior art keywords
- tetrazolyloxime derivatives
- group
- tetrazolyloxime
- derivatives
- production
- Prior art date
Links
- 238000004519 manufacturing process Methods 0.000 title abstract 2
- 125000005843 halogen group Chemical group 0.000 abstract 2
- 125000004191 (C1-C6) alkoxy group Chemical group 0.000 abstract 1
- JUJWROOIHBZHMG-UHFFFAOYSA-N Pyridine Chemical group C1=CC=NC=C1 JUJWROOIHBZHMG-UHFFFAOYSA-N 0.000 abstract 1
- 125000002777 acetyl group Chemical group [H]C([H])([H])C(*)=O 0.000 abstract 1
- 125000004453 alkoxycarbonyl group Chemical group 0.000 abstract 1
- 150000001875 compounds Chemical class 0.000 abstract 1
- 125000004093 cyano group Chemical group *C#N 0.000 abstract 1
- 230000000855 fungicidal effect Effects 0.000 abstract 1
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
- C07D401/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
- C07D401/12—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings linked by a chain containing hetero atoms as chain links
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D213/00—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members
- C07D213/02—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members
- C07D213/04—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom
- C07D213/60—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D213/72—Nitrogen atoms
- C07D213/75—Amino or imino radicals, acylated by carboxylic or carbonic acids, or by sulfur or nitrogen analogues thereof, e.g. carbamates
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D405/00—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom
- C07D405/02—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings
- C07D405/12—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings linked by a chain containing hetero atoms as chain links
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Plural Heterocyclic Compounds (AREA)
- Pyridine Compounds (AREA)
- Low-Molecular Organic Synthesis Reactions Using Catalysts (AREA)
- Agricultural Chemicals And Associated Chemicals (AREA)
Abstract
A presente invenção refere-se a um composto contendo um anel de piridina que pode ser sintetizado de uma maneira industrialmente vantajosa, e é útil como um intermediário para produzir derivados de tetrazoliloxima que apresentam atividade fungicida (em que R0 representa um grupo C1-6 alcóxi, grupo C1-6 alcóxi-C1-6 alcóxi ou outros, R1 representa um grupo C1-2 alcoxicarbonila, grupo acetila ou outros, Z representa um átomo de halogênio, grupo ciano ou outros, X representa um átomo de halogênio, e n representa um número inteiro de 0 a 3), e métodos de produção industrialmente vantajosos para produzir o derivado de amino-6-halometilpiridina 2-substituída e os derivados de tetrazoliloxima.
Applications Claiming Priority (8)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| JP2010056718 | 2010-03-12 | ||
| JP2010-056718 | 2010-03-12 | ||
| JP2010-115703 | 2010-05-19 | ||
| JP2010115703 | 2010-05-19 | ||
| JP2010-127207 | 2010-06-02 | ||
| JP2010127207 | 2010-06-02 | ||
| BR112012022823-4A BR112012022823B1 (pt) | 2010-03-12 | 2011-03-11 | Composto contendo anel de piridina |
| PCT/JP2011/055809 WO2011111831A1 (ja) | 2010-03-12 | 2011-03-11 | ピリジン環含有化合物、及びハロゲン化ピコリン誘導体及びテトラゾリルオキシム誘導体の製造方法 |
Publications (3)
| Publication Number | Publication Date |
|---|---|
| BR122017023130A2 BR122017023130A2 (pt) | 2016-08-30 |
| BR122017023130A8 true BR122017023130A8 (pt) | 2018-01-02 |
| BR122017023130B1 BR122017023130B1 (pt) | 2018-03-06 |
Family
ID=44563629
Family Applications (4)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| BR122017023128-6A BR122017023128B1 (pt) | 2010-03-12 | 2011-03-11 | Método para produzir derivado de picolina brominada |
| BR112012022823-4A BR112012022823B1 (pt) | 2010-03-12 | 2011-03-11 | Composto contendo anel de piridina |
| BR122017023123-5A BR122017023123B1 (pt) | 2010-03-12 | 2011-03-11 | Método para produzir derivado de picolina halogenada |
| BR122017023130-8A BR122017023130B1 (pt) | 2010-03-12 | 2011-03-11 | Derivado de tetrazoliloxima, métodos de produção de derivados de tetrazoliloxima |
Family Applications Before (3)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| BR122017023128-6A BR122017023128B1 (pt) | 2010-03-12 | 2011-03-11 | Método para produzir derivado de picolina brominada |
| BR112012022823-4A BR112012022823B1 (pt) | 2010-03-12 | 2011-03-11 | Composto contendo anel de piridina |
| BR122017023123-5A BR122017023123B1 (pt) | 2010-03-12 | 2011-03-11 | Método para produzir derivado de picolina halogenada |
Country Status (10)
| Country | Link |
|---|---|
| US (5) | US8841458B2 (pt) |
| EP (4) | EP2719688B1 (pt) |
| JP (5) | JP5627038B2 (pt) |
| KR (1) | KR101409137B1 (pt) |
| CN (5) | CN104130184B (pt) |
| AU (1) | AU2011225122B8 (pt) |
| BR (4) | BR122017023128B1 (pt) |
| IL (3) | IL221847A (pt) |
| RU (1) | RU2512344C1 (pt) |
| WO (1) | WO2011111831A1 (pt) |
Families Citing this family (7)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| RU2581828C2 (ru) | 2012-03-13 | 2016-04-20 | Ниппон Сода Ко., Лтд. | Производное тетразолилгидроксиимина, способ его очистки и способ его получения |
| AU2013291223B2 (en) * | 2012-07-19 | 2015-08-06 | Nippon Soda Co., Ltd. | Water dispersible granule, and method for producing same |
| CA2972161C (en) | 2015-03-10 | 2018-07-24 | Lonza Ltd | Method for preparation of certain 1,5 disubstituted tetrazoles |
| EP3112344A1 (en) | 2015-06-30 | 2017-01-04 | Lonza Ltd | Method for preparation of certain thioacetamides |
| CN110452220B (zh) * | 2018-04-26 | 2020-08-14 | 东莞市东阳光农药研发有限公司 | 肟衍生物及其在农业中的应用 |
| KR102731001B1 (ko) * | 2019-05-13 | 2024-11-19 | 다이킨 고교 가부시키가이샤 | 플루오로락톤 및 그 제조 방법 |
| EP3782985A1 (en) | 2019-08-19 | 2021-02-24 | BASF Agrochemical Products B.V. | Process for manufacturing 5-methoxymethylpyridine-2,3-dicarboxylic acid derivatives |
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| IL96436A0 (en) | 1989-11-28 | 1991-08-16 | Ishihara Sangyo Kaisha | Pyridylcarbamates,their preparation and biocidal compositions containing them |
| GB2279346A (en) * | 1993-07-01 | 1995-01-04 | Glaxo Group Ltd | Benzofuran intermediates |
| DE4322054A1 (de) | 1993-07-02 | 1995-01-12 | Bayer Ag | Verfahren zur Herstellung von Chlormethylpyridinen |
| DE4446338A1 (de) | 1994-12-23 | 1996-06-27 | Bayer Ag | Verfahren zur Herstellung von Chlormethylpyridinen |
| JPH09268178A (ja) | 1996-04-01 | 1997-10-14 | Shiratori Seiyaku Kk | 光学活性な４，５−ジフェニル−２−イミダゾリジノン誘導体 |
| US5872136A (en) * | 1996-04-03 | 1999-02-16 | Merck & Co., Inc. | Arylheteroaryl inhibitors of farnesyl-protein transferase |
| DE19815946A1 (de) | 1998-04-09 | 1999-10-14 | Basf Ag | N-Vinyleinheiten enthaltende polymere Gerbstoffe |
| NZ531160A (en) | 2001-08-20 | 2005-12-23 | Nippon Soda Co | Tetrazoyl oxime derivative as active ingredient in agricultural chemical to control plant disease |
| JP4330313B2 (ja) | 2001-08-20 | 2009-09-16 | 日本曹達株式会社 | テトラゾイルオキシム誘導体及びこれを有効成分とする農薬 |
| AU2003220122A1 (en) * | 2002-03-12 | 2003-09-29 | Wyeth | Preparation of n1-(2'-pyridyl)-1,2-propanediamine sulfamic acid and its use in the synthesis of biologically active piperazines |
| JP2004131392A (ja) | 2002-10-08 | 2004-04-30 | Sumitomo Chem Co Ltd | テトラゾール化合物およびその用途 |
| JP2004131416A (ja) | 2002-10-10 | 2004-04-30 | Sumitomo Chem Co Ltd | テトラゾール化合物およびその植物病害防除用途 |
| TWI346108B (en) * | 2004-08-23 | 2011-08-01 | Bristol Myers Squibb Co | A method for preparing irbesartan and intermediates thereof |
| AR059339A1 (es) | 2006-02-09 | 2008-03-26 | Chugai Pharmaceutical Co Ltd | Derivados de la cumarina para trastornos proliferativos de celulas, composicion farmaceutica y agente terapeutico que los contiene |
| EP2049490A1 (en) | 2006-06-09 | 2009-04-22 | Astra Zeneca AB | N-(benzoyl)-o- [2- (pyridin- 2 -ylamino) ethyl]-l-tyrosine derivatives and related compounds as a5b1 antagonists for the treatment of solid tumors |
| WO2008006875A1 (en) * | 2006-07-13 | 2008-01-17 | Bayer Cropscience Sa | Fungicide hydroximoyl-tetrazole derivatives |
| BRPI0808523A2 (pt) * | 2007-03-01 | 2014-08-19 | Novartis Vaccines & Diagnostic | Inibidores de pim cinase e métodos de seu uso |
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2011
- 2011-03-11 CN CN201410283542.4A patent/CN104130184B/zh active Active
- 2011-03-11 BR BR122017023128-6A patent/BR122017023128B1/pt active IP Right Grant
- 2011-03-11 CN CN201410283563.6A patent/CN104109150B/zh active Active
- 2011-03-11 BR BR112012022823-4A patent/BR112012022823B1/pt active IP Right Grant
- 2011-03-11 RU RU2012138410/04A patent/RU2512344C1/ru active
- 2011-03-11 EP EP14000071.2A patent/EP2719688B1/en active Active
- 2011-03-11 WO PCT/JP2011/055809 patent/WO2011111831A1/ja active Application Filing
- 2011-03-11 KR KR1020127023288A patent/KR101409137B1/ko active Active
- 2011-03-11 BR BR122017023123-5A patent/BR122017023123B1/pt active IP Right Grant
- 2011-03-11 CN CN201180012762.8A patent/CN102791691B/zh active Active
- 2011-03-11 CN CN201410283225.2A patent/CN104072483B/zh active Active
- 2011-03-11 AU AU2011225122A patent/AU2011225122B8/en active Active
- 2011-03-11 CN CN201410283380.4A patent/CN104072408B/zh active Active
- 2011-03-11 EP EP14000069.6A patent/EP2719686B1/en active Active
- 2011-03-11 US US13/583,733 patent/US8841458B2/en active Active
- 2011-03-11 BR BR122017023130-8A patent/BR122017023130B1/pt active IP Right Grant
- 2011-03-11 JP JP2012504543A patent/JP5627038B2/ja active Active
- 2011-03-11 EP EP11753489.1A patent/EP2546236A4/en not_active Withdrawn
- 2011-03-11 EP EP14000070.4A patent/EP2719687B1/en active Active
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2012
- 2012-09-09 IL IL221847A patent/IL221847A/en active IP Right Grant
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2013
- 2013-12-17 IL IL229967A patent/IL229967A/en active IP Right Grant
- 2013-12-17 IL IL229968A patent/IL229968A/en active IP Right Grant
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2014
- 2014-02-05 US US14/173,330 patent/US9012653B2/en active Active
- 2014-02-05 US US14/173,338 patent/US8962848B2/en active Active
- 2014-02-05 US US14/173,323 patent/US9018385B2/en active Active
- 2014-02-05 US US14/173,352 patent/US9000178B2/en active Active
- 2014-02-13 JP JP2014025952A patent/JP5695233B2/ja active Active
- 2014-02-13 JP JP2014025954A patent/JP5793589B2/ja active Active
- 2014-02-13 JP JP2014025955A patent/JP5695234B2/ja active Active
- 2014-02-13 JP JP2014025953A patent/JP5793588B2/ja active Active
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Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| B15K | Others concerning applications: alteration of classification |
Ipc: C07D 401/12 (1974.07), A01P 7/04 (2006.01) |
|
| B09A | Decision: intention to grant [chapter 9.1 patent gazette] | ||
| B16A | Patent or certificate of addition of invention granted [chapter 16.1 patent gazette] |