[go: up one dir, main page]

BR112014012942A2 - uso de derivados de aril para controle de ectoparasitas - Google Patents

uso de derivados de aril para controle de ectoparasitas

Info

Publication number
BR112014012942A2
BR112014012942A2 BR112014012942A BR112014012942A BR112014012942A2 BR 112014012942 A2 BR112014012942 A2 BR 112014012942A2 BR 112014012942 A BR112014012942 A BR 112014012942A BR 112014012942 A BR112014012942 A BR 112014012942A BR 112014012942 A2 BR112014012942 A2 BR 112014012942A2
Authority
BR
Brazil
Prior art keywords
animal
aryl derivatives
ectoparasite control
control
medicament
Prior art date
Application number
BR112014012942A
Other languages
English (en)
Inventor
Kablitz Caroline
Desevaux Cyril
Jung Martin
Nanchen Steve
Original Assignee
Novartis Ag
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Novartis Ag filed Critical Novartis Ag
Publication of BR112014012942A2 publication Critical patent/BR112014012942A2/pt

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D413/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms
    • C07D413/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings
    • C07D413/04—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings directly linked by a ring-member-to-ring-member bond
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/41—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
    • A61K31/42—Oxazoles
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/0087—Galenical forms not covered by A61K9/02 - A61K9/7023
    • A61K9/0095—Drinks; Beverages; Syrups; Compositions for reconstitution thereof, e.g. powders or tablets to be dispersed in a glass of water; Veterinary drenches
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/08—Solutions
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P33/00—Antiparasitic agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P33/00—Antiparasitic agents
    • A61P33/14—Ectoparasiticides, e.g. scabicides
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D261/00—Heterocyclic compounds containing 1,2-oxazole or hydrogenated 1,2-oxazole rings
    • C07D261/02—Heterocyclic compounds containing 1,2-oxazole or hydrogenated 1,2-oxazole rings not condensed with other rings
    • C07D261/04—Heterocyclic compounds containing 1,2-oxazole or hydrogenated 1,2-oxazole rings not condensed with other rings having one double bond between ring members or between a ring member and a non-ring member

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Veterinary Medicine (AREA)
  • Animal Behavior & Ethology (AREA)
  • Public Health (AREA)
  • Medicinal Chemistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Epidemiology (AREA)
  • General Chemical & Material Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Tropical Medicine & Parasitology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Medicinal Preparation (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Fodder In General (AREA)

Abstract

resumo uso de derivados de aril para controle de ectoparasitas a presente invenção refere-se ao uso de compostos de fórmula (i), em que as variáveis são como definidas na descrição, na forma livre ou na forma de sal, para a fabricação de um medicamento para controle de ectoparasitas em um animal de sangue quente, em que dito medicamento é administrado oralmente ao animal em uma dose de 0,1 a 100 mg/kg a partir de 30 minutos antes a 3 horas após a alimentação do animal com uma ração animal.
BR112014012942A 2011-11-29 2012-11-23 uso de derivados de aril para controle de ectoparasitas BR112014012942A2 (pt)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
EP11191133 2011-11-29
PCT/EP2012/073475 WO2013079407A1 (en) 2011-11-29 2012-11-23 Aryl derivatives for controlling ectoparasites

Publications (1)

Publication Number Publication Date
BR112014012942A2 true BR112014012942A2 (pt) 2017-06-13

Family

ID=47216325

Family Applications (1)

Application Number Title Priority Date Filing Date
BR112014012942A BR112014012942A2 (pt) 2011-11-29 2012-11-23 uso de derivados de aril para controle de ectoparasitas

Country Status (7)

Country Link
US (1) US20140343085A1 (pt)
EP (1) EP2785341A1 (pt)
JP (1) JP2014533735A (pt)
AU (1) AU2012344083A1 (pt)
BR (1) BR112014012942A2 (pt)
CA (1) CA2856476A1 (pt)
WO (1) WO2013079407A1 (pt)

Families Citing this family (10)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
EP2833867B2 (en) * 2012-04-04 2023-05-10 Intervet International B.V. Solid oral pharmaceutical compositions for isoxazoline compounds
ES2659974T3 (es) * 2013-06-24 2018-03-20 Merial, Inc. Compuestos de isotiazolina sustituidos con tiofeno o furano como pesticidas
ES2817098T3 (es) * 2013-06-24 2021-04-06 Boehringer Ingelheim Animal Health Usa Inc Compuestos de isotiazolinas sustituidas con naftilo
UY37137A (es) 2016-02-24 2017-09-29 Merial Inc Compuestos antiparasitarios de isoxazolina, formulaciones inyectables de acción prolongada que los comprenden, métodos y usos de los mismos
CA3121202A1 (en) 2018-11-30 2020-06-04 Nuvation Bio Inc. Pyrrole and pyrazole compounds and methods of use thereof
CA3164924A1 (en) 2019-12-18 2021-06-24 Elanco Tiergesundheit Ag Isoxazoline derivatives as pesticides
JP2023536070A (ja) 2020-07-24 2023-08-23 エランコ・ユーエス・インコーポレイテッド イソオキサゾリン化合物及びその中間体を作製するための方法
US20240270729A1 (en) 2021-06-16 2024-08-15 Elanco Tiergesundheit Ag (thi)oxazoline pesticides
CA3223820A1 (en) 2021-06-16 2022-12-22 Elanco Tiergesundheit Ag Isoxazoline pesticides
CA3224701A1 (en) 2021-08-11 2023-02-16 Jingdan Hu Process for making diaryl isoxazoline derivative

Family Cites Families (15)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
WO2005085216A1 (ja) * 2004-03-05 2005-09-15 Nissan Chemical Industries, Ltd. イソキサゾリン置換ベンズアミド化合物及び有害生物防除剤
BRPI0617076B1 (pt) 2005-09-02 2021-07-06 Nissan Chemical Corporation Composto benzamida substituída por isoxazolina da fórmula (1) ou sal do mesmo; composto benzamida substituido por 4-hidroxiiminametila da fórmula (2) ou sal do mesmo; pesticida; agente agroquímico; parasiticida interno ou externo para mamíferos ou aves; inseticida ou acaricida
JP2009519937A (ja) 2005-12-14 2009-05-21 イー・アイ・デュポン・ドウ・ヌムール・アンド・カンパニー 無脊椎有害生物防除用イソオキサゾリン
TW200803740A (en) 2005-12-16 2008-01-16 Du Pont 5-aryl isoxazolines for controlling invertebrate pests
TWI412322B (zh) 2005-12-30 2013-10-21 Du Pont 控制無脊椎害蟲之異唑啉
JP4703445B2 (ja) 2006-03-20 2011-06-15 株式会社エヌ・ティ・ティ・ドコモ 上位局及びパケット送信方法
WO2007123855A2 (en) 2006-04-20 2007-11-01 E. I. Du Pont De Nemours And Company Pyrazolines for controlling invertebrate pests
JP2008044880A (ja) 2006-08-15 2008-02-28 Bayer Cropscience Ag 殺虫性イソオキサゾリン類
CA2700598C (en) 2007-08-10 2012-11-20 Nippon Soda Co., Ltd. Nitrogen-containing heterocyclic compound and pest control agent
TWI556741B (zh) * 2007-08-17 2016-11-11 英特威特國際股份有限公司 異唑啉組成物及其作為抗寄生蟲藥上的應用
US8318757B2 (en) 2007-09-10 2012-11-27 Nissan Chemical Industries, Ltd. Substituted isoxazoline compound and pest control agent
WO2009071500A2 (en) 2007-12-03 2009-06-11 Novartis Ag Organic compounds
TWI411395B (zh) 2007-12-24 2013-10-11 Syngenta Participations Ag 殺蟲化合物
JP2009286773A (ja) 2008-03-14 2009-12-10 Bayer Cropscience Ag 殺虫性縮環式アリール類
ES2395704T3 (es) 2008-12-19 2013-02-14 Novartis Ag Derivados de isoxazolina y su uso como pesticida

Also Published As

Publication number Publication date
US20140343085A1 (en) 2014-11-20
AU2012344083A1 (en) 2014-05-29
CA2856476A1 (en) 2013-06-06
EP2785341A1 (en) 2014-10-08
JP2014533735A (ja) 2014-12-15
WO2013079407A1 (en) 2013-06-06

Similar Documents

Publication Publication Date Title
BR112014012942A2 (pt) uso de derivados de aril para controle de ectoparasitas
BR112013000275A2 (pt) derivados de tetraidro-pirido-pirimidina
BR112019008341A2 (pt) processo para a preparação de pirazolo[1,5-a]pirimidinas e sais dos mesmos
BR112014014909A2 (pt) agonistas de tgr5 não sistêmicos
CR20140301A (es) Derivados de betulina
BR112017019286A2 (pt) composto de fórmula (i) ou um sal farmaceuticamente aceitável deste
BR112014003198A2 (pt) compostos para o tratamento e profilaxia de doença por vírus sincicial respiratório
BR112015028452A2 (pt) agonistas do receptor somastatina subtipo 4 (sstr4)
BR112014018879A8 (pt) Composto e composição farmacêutica e combinação compreendendo dito composto
BR112015023412A8 (pt) 3-pirimidin-4-il-oxazolidin-2-onas como inibidores de idh mutante, sua composição farmacêutica e seu uso.
PE20141038A1 (es) Sales de 2,3-dihidroimidazo[1,2-c]quinazolina substituida
UY32096A (es) Derivados de 2-carboxamida - cicloamino - urea especìficos, sus sales farmacèuticamente aceptables, composiciones contenièndolos, pro-farmacos de los mismos, procesos para su produciòn y aplicaciones
BR112015018738A8 (pt) compostos de tetra-hidropirrolotiazina, seus usos, e composição farmacêutica
BR112014007310A2 (pt) 3-pirimidin-4-il-oxazolidin-2-onas como inibidores de idh mutante
BR112014002946A2 (pt) sistema de travamento mecânico para painéis de piso
MD20140103A2 (ro) Inhibitori ai diacilglicerol aciltransferazei 2
BR112012019762A2 (pt) composto, composição, e, método para tratar uma doença.
BR112013011593A2 (pt) cristal de derivado de morfinan 7-carbamoíla-6,7-insaturada e método para produzir o mesmo
WO2009080705A3 (en) Bis-thiazole derivatives, process for their preparation and their use as medicaments
BR112012012903A2 (pt) compostos de espiropiperidina
CR20150663A (es) Derivados de diazacarbazol como ligandos de tau para pet
CO6680645A2 (es) Inhibidores de oxadiazol de la producción de leucotrieno
BR112015019369A2 (pt) derivados de ácido bisfenil butanóico substituídos como inibidores de nep (endopeptidase neutra)
BR112015020823A2 (pt) 1-hidróxi-benzooxaboróis como agentes antiparasíticos
BR112014026266A2 (pt) derivado de quinazolidinadiona

Legal Events

Date Code Title Description
B11A Dismissal acc. art.33 of ipl - examination not requested within 36 months of filing
B11Y Definitive dismissal - extension of time limit for request of examination expired [chapter 11.1.1 patent gazette]
B25B Requested transfer of rights rejected

Owner name: NOVARTIS AG (CH)

B350 Update of information on the portal [chapter 15.35 patent gazette]