BR0110642A - Processo para preparação de sais de sulfonilbenzoilguanidìnio - Google Patents
Processo para preparação de sais de sulfonilbenzoilguanidìnioInfo
- Publication number
- BR0110642A BR0110642A BR0110642-2A BR0110642A BR0110642A BR 0110642 A BR0110642 A BR 0110642A BR 0110642 A BR0110642 A BR 0110642A BR 0110642 A BR0110642 A BR 0110642A
- Authority
- BR
- Brazil
- Prior art keywords
- salts
- preparation
- sulfonylbenzoylguanidium
- sulphonylbenzoilguanidine
- alkyl
- Prior art date
Links
- 150000003839 salts Chemical class 0.000 title abstract 3
- 238000000034 method Methods 0.000 title abstract 2
- 239000002253 acid Substances 0.000 abstract 1
- 125000000217 alkyl group Chemical group 0.000 abstract 1
- 125000004432 carbon atom Chemical group C* 0.000 abstract 1
- 150000001875 compounds Chemical class 0.000 abstract 1
- 238000004519 manufacturing process Methods 0.000 abstract 1
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C315/00—Preparation of sulfones; Preparation of sulfoxides
- C07C315/04—Preparation of sulfones; Preparation of sulfoxides by reactions not involving the formation of sulfone or sulfoxide groups
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C315/00—Preparation of sulfones; Preparation of sulfoxides
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Abstract
Patente de Invenção: "PROCESSO PARA PREPARAçãO DE SAIS DE SULFONILBENZOILGUANIDìNIO". A invenção refere-se a um processo para a preparação de sais de adição ácidos dos compostos de fórmula(I) em que R^ 1^, R^ 2^ e R^ 3^ são alquila tendo de 1 a 12 átomos de carbono.
Applications Claiming Priority (2)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
DE10023405A DE10023405A1 (de) | 2000-05-12 | 2000-05-12 | Verfahren zur Herstellung von Sulfonyl-benzoylguanidinum-Salzen |
PCT/EP2001/004294 WO2001085679A1 (de) | 2000-05-12 | 2001-04-17 | Verfahren zur herstellung von sulfonyl-benzoylguanidinium-salzen |
Publications (1)
Publication Number | Publication Date |
---|---|
BR0110642A true BR0110642A (pt) | 2003-03-18 |
Family
ID=7641866
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
BR0110642-2A BR0110642A (pt) | 2000-05-12 | 2001-04-17 | Processo para preparação de sais de sulfonilbenzoilguanidìnio |
Country Status (24)
Country | Link |
---|---|
US (1) | US6706921B2 (pt) |
EP (1) | EP1282598B1 (pt) |
JP (1) | JP2003532704A (pt) |
KR (1) | KR20030007599A (pt) |
CN (1) | CN1193011C (pt) |
AR (1) | AR028442A1 (pt) |
AT (1) | ATE280151T1 (pt) |
AU (1) | AU783369B2 (pt) |
BR (1) | BR0110642A (pt) |
CA (1) | CA2408640A1 (pt) |
CZ (1) | CZ20023647A3 (pt) |
DE (2) | DE10023405A1 (pt) |
DK (1) | DK1282598T3 (pt) |
ES (1) | ES2228897T3 (pt) |
HU (1) | HUP0301936A2 (pt) |
MX (1) | MXPA02011069A (pt) |
MY (1) | MY133941A (pt) |
NO (1) | NO20025385D0 (pt) |
PL (1) | PL358690A1 (pt) |
PT (1) | PT1282598E (pt) |
RU (1) | RU2258699C2 (pt) |
SK (1) | SK15812002A3 (pt) |
WO (1) | WO2001085679A1 (pt) |
ZA (1) | ZA200210050B (pt) |
Families Citing this family (2)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
WO2004037815A1 (ja) * | 2002-10-28 | 2004-05-06 | Kaneka Corporation | 光学活性n−(2,3−エポキシプロパンー1−イル)フタルイミドの製造法 |
DK2271327T3 (en) | 2008-05-09 | 2015-07-13 | Merck Patent Gmbh | Pharmaceutical composition comprising rhymeporide for the treatment of diseases associated with beta-cell dysfunction |
Family Cites Families (8)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
JPS6248648A (ja) * | 1985-08-28 | 1987-03-03 | Fujisawa Pharmaceut Co Ltd | ジアルコキシ酢酸エステル化合物の製造法 |
DE59305042D1 (de) * | 1992-09-22 | 1997-02-20 | Hoechst Ag | Benzoylguanidine, Verfahren zu ihrer Herstellung, sowie ihre Verwendung als Antiarrhythmika |
DE4437874A1 (de) * | 1994-10-22 | 1996-04-25 | Merck Patent Gmbh | Alkyl-5-methylsulfonyl-benzoylguanidin-Derivate |
DE19502644A1 (de) * | 1995-01-28 | 1996-08-01 | Merck Patent Gmbh | 4-Amino-benzoylguanidin-Derivate |
DE19529612A1 (de) | 1995-08-11 | 1997-02-13 | Merck Patent Gmbh | Sulfonyl- oder Sulfinyl-benzoylguanidin-Derivate |
DE19621482A1 (de) * | 1996-05-29 | 1997-12-04 | Hoechst Ag | Substituierte 1-Naphthoylguanidine, Verfahren zu ihrer Herstellung, ihre Verwendung als Medikament oder Diagnostikum sowie sie enthaltendes Medikament |
DE19951418A1 (de) * | 1999-10-26 | 2001-05-03 | Merck Patent Gmbh | Verfahren zur Herstellung von N-(4,5-Bismethansulfonyl-2-methyl-benzoyl) -guanidin, Hydrochlorid |
JP2001247557A (ja) * | 1999-12-27 | 2001-09-11 | Sagami Chem Res Center | 5−オキシ−7−オキサビシクロ[4.1.0]ヘプト−3−エン−3−カルボン酸エステルの製造方法 |
-
2000
- 2000-05-12 DE DE10023405A patent/DE10023405A1/de active Pending
-
2001
- 2001-04-17 AU AU68969/01A patent/AU783369B2/en not_active Ceased
- 2001-04-17 AT AT01947223T patent/ATE280151T1/de not_active IP Right Cessation
- 2001-04-17 CA CA002408640A patent/CA2408640A1/en not_active Abandoned
- 2001-04-17 SK SK1581-2002A patent/SK15812002A3/sk unknown
- 2001-04-17 DK DK01947223T patent/DK1282598T3/da active
- 2001-04-17 DE DE50104219T patent/DE50104219D1/de not_active Expired - Lifetime
- 2001-04-17 CZ CZ20023647A patent/CZ20023647A3/cs unknown
- 2001-04-17 PT PT01947223T patent/PT1282598E/pt unknown
- 2001-04-17 KR KR1020027015038A patent/KR20030007599A/ko not_active Application Discontinuation
- 2001-04-17 MX MXPA02011069A patent/MXPA02011069A/es active IP Right Grant
- 2001-04-17 ES ES01947223T patent/ES2228897T3/es not_active Expired - Lifetime
- 2001-04-17 PL PL01358690A patent/PL358690A1/xx unknown
- 2001-04-17 BR BR0110642-2A patent/BR0110642A/pt not_active Application Discontinuation
- 2001-04-17 EP EP01947223A patent/EP1282598B1/de not_active Expired - Lifetime
- 2001-04-17 JP JP2001582280A patent/JP2003532704A/ja active Pending
- 2001-04-17 US US10/275,484 patent/US6706921B2/en not_active Expired - Fee Related
- 2001-04-17 CN CNB018094058A patent/CN1193011C/zh not_active Expired - Fee Related
- 2001-04-17 HU HU0301936A patent/HUP0301936A2/hu unknown
- 2001-04-17 RU RU2002133235/04A patent/RU2258699C2/ru not_active IP Right Cessation
- 2001-04-17 WO PCT/EP2001/004294 patent/WO2001085679A1/de active IP Right Grant
- 2001-05-09 MY MYPI20012143 patent/MY133941A/en unknown
- 2001-05-11 AR ARP010102230A patent/AR028442A1/es unknown
-
2002
- 2002-11-11 NO NO20025385A patent/NO20025385D0/no not_active Application Discontinuation
- 2002-12-11 ZA ZA200210050A patent/ZA200210050B/en unknown
Also Published As
Publication number | Publication date |
---|---|
EP1282598A1 (de) | 2003-02-12 |
CA2408640A1 (en) | 2002-11-08 |
AR028442A1 (es) | 2003-05-07 |
DE10023405A1 (de) | 2001-11-15 |
ATE280151T1 (de) | 2004-11-15 |
RU2258699C2 (ru) | 2005-08-20 |
PT1282598E (pt) | 2005-03-31 |
PL358690A1 (en) | 2004-08-09 |
CZ20023647A3 (cs) | 2003-02-12 |
US20030162999A1 (en) | 2003-08-28 |
DE50104219D1 (de) | 2004-11-25 |
SK15812002A3 (sk) | 2003-03-04 |
HUP0301936A2 (hu) | 2003-09-29 |
NO20025385L (no) | 2002-11-11 |
AU783369B2 (en) | 2005-10-20 |
MXPA02011069A (es) | 2003-03-10 |
WO2001085679A1 (de) | 2001-11-15 |
MY133941A (en) | 2007-11-30 |
CN1193011C (zh) | 2005-03-16 |
DK1282598T3 (da) | 2005-02-07 |
EP1282598B1 (de) | 2004-10-20 |
AU6896901A (en) | 2001-11-20 |
US6706921B2 (en) | 2004-03-16 |
KR20030007599A (ko) | 2003-01-23 |
CN1429207A (zh) | 2003-07-09 |
ZA200210050B (en) | 2003-09-10 |
ES2228897T3 (es) | 2005-04-16 |
JP2003532704A (ja) | 2003-11-05 |
NO20025385D0 (no) | 2002-11-11 |
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Legal Events
Date | Code | Title | Description |
---|---|---|---|
B07A | Application suspended after technical examination (opinion) [chapter 7.1 patent gazette] | ||
B09B | Patent application refused [chapter 9.2 patent gazette] | ||
B09B | Patent application refused [chapter 9.2 patent gazette] |
Free format text: MANTIDO O INDEFERIMENTO UMA VEZ QUE NAO FOI APRESENTADO RECURSO DENTRO DO PRAZO LEGAL. |