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BR0009886A - Método para a fabricação de ácidos 2-(n-fenilamino) benzóicos - Google Patents

Método para a fabricação de ácidos 2-(n-fenilamino) benzóicos

Info

Publication number
BR0009886A
BR0009886A BR0009886-8A BR0009886A BR0009886A BR 0009886 A BR0009886 A BR 0009886A BR 0009886 A BR0009886 A BR 0009886A BR 0009886 A BR0009886 A BR 0009886A
Authority
BR
Brazil
Prior art keywords
manufacture
phenylamino
benzoic acids
benzoic
acids
Prior art date
Application number
BR0009886-8A
Other languages
English (en)
Inventor
Michael Huai Gu Chen
Javier Mangano
Original Assignee
Warner Lambert Co
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Warner Lambert Co filed Critical Warner Lambert Co
Publication of BR0009886A publication Critical patent/BR0009886A/pt

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07CACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C227/00Preparation of compounds containing amino and carboxyl groups bound to the same carbon skeleton
    • C07C227/04Formation of amino groups in compounds containing carboxyl groups
    • C07C227/06Formation of amino groups in compounds containing carboxyl groups by addition or substitution reactions, without increasing the number of carbon atoms in the carbon skeleton of the acid
    • C07C227/08Formation of amino groups in compounds containing carboxyl groups by addition or substitution reactions, without increasing the number of carbon atoms in the carbon skeleton of the acid by reaction of ammonia or amines with acids containing functional groups

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)

Abstract

Patente de Invenção: "MéTODO PARA A FABRICAçãO DE áCIDOS 2-(N-FENILAMINO)BENZóICOS". A presente invenção refere-se a um método para a fabricação de ácidos 2-(N-fenilamino)benzóicos mediante o acoplamento de um ácido benzóico e uma anilina usando uma hexametildissilazida de metal alcalino como uma base.
BR0009886-8A 1999-04-21 2000-02-16 Método para a fabricação de ácidos 2-(n-fenilamino) benzóicos BR0009886A (pt)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US13038499P 1999-04-21 1999-04-21
PCT/US2000/003982 WO2000064856A1 (en) 1999-04-21 2000-02-16 Method for making 2-(n-phenylamino)benzoic acids

Publications (1)

Publication Number Publication Date
BR0009886A true BR0009886A (pt) 2002-01-22

Family

ID=22444462

Family Applications (1)

Application Number Title Priority Date Filing Date
BR0009886-8A BR0009886A (pt) 1999-04-21 2000-02-16 Método para a fabricação de ácidos 2-(n-fenilamino) benzóicos

Country Status (34)

Country Link
EP (1) EP1171418B1 (pt)
JP (1) JP3769192B2 (pt)
KR (1) KR20010108521A (pt)
CN (1) CN1213997C (pt)
AP (1) AP2001002328A0 (pt)
AT (1) ATE286015T1 (pt)
AU (1) AU773096B2 (pt)
BG (1) BG106132A (pt)
BR (1) BR0009886A (pt)
CA (1) CA2368807A1 (pt)
CR (1) CR6486A (pt)
CU (1) CU22996A3 (pt)
DE (1) DE60017109T2 (pt)
DK (1) DK1171418T3 (pt)
EA (1) EA004209B1 (pt)
EE (1) EE200100546A (pt)
ES (1) ES2235843T3 (pt)
GE (1) GEP20033089B (pt)
HK (1) HK1045682B (pt)
HR (1) HRP20010850A2 (pt)
HU (1) HUP0200932A3 (pt)
IL (1) IL146056A0 (pt)
MA (1) MA25412A1 (pt)
NO (1) NO20015095D0 (pt)
NZ (1) NZ515120A (pt)
OA (1) OA11861A (pt)
PL (1) PL351085A1 (pt)
PT (1) PT1171418E (pt)
SK (1) SK14732001A3 (pt)
TR (1) TR200103015T2 (pt)
UA (1) UA70995C2 (pt)
WO (1) WO2000064856A1 (pt)
YU (1) YU73701A (pt)
ZA (1) ZA200107834B (pt)

Families Citing this family (6)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
BR0113520A (pt) * 2000-08-25 2003-06-24 Warner Lambert Co Processo de preparação de ácidos n-aril-antranìlicos e seus derivados
JP5025466B2 (ja) * 2005-04-06 2012-09-12 中外製薬株式会社 2,3,4−トリフルオロ−5−(ヨード又はブロモ)安息香酸の製造方法
JPWO2007021001A1 (ja) * 2005-08-18 2009-02-26 宇部興産株式会社 2,3,4−トリフルオロ−5−置換安息香酸化合物及びその製法
CA2789373A1 (en) * 2010-02-19 2011-08-25 Centre National De La Recherche Scientifique Process for preparing chemical compounds of interest by nucleophilic aromatic substitution of aromatic carboxylic acid derivatives supporting at least one electro-attractive group
EP2536683A1 (fr) * 2010-02-19 2012-12-26 Centre National De La Recherche Scientifique Procédé de préparation de composés chimiques d'intérêt par substitution nucléophile aromatique
JP2016034900A (ja) * 2012-11-26 2016-03-17 中外製薬株式会社 5−置換−2−フェニルアミノ−ベンズアミド類の製造方法

Family Cites Families (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
BR9810366A (pt) * 1997-07-01 2000-08-29 Warner Lambert Co Derivados de ácido 4-bromo ou 4-iodo fenilamino benzidroxîmico e seu uso como inibidores de mek

Also Published As

Publication number Publication date
EE200100546A (et) 2003-02-17
HK1045682B (zh) 2006-04-07
SK14732001A3 (sk) 2002-05-09
DK1171418T3 (da) 2005-05-09
CU22996A3 (es) 2004-10-12
HRP20010850A2 (en) 2002-12-31
ES2235843T3 (es) 2005-07-16
OA11861A (en) 2006-03-02
DE60017109D1 (de) 2005-02-03
NO20015095L (no) 2001-10-19
AU3492800A (en) 2000-11-10
UA70995C2 (uk) 2004-11-15
CN1213997C (zh) 2005-08-10
ATE286015T1 (de) 2005-01-15
HUP0200932A3 (en) 2002-11-28
NZ515120A (en) 2003-08-29
MA25412A1 (fr) 2002-04-01
IL146056A0 (en) 2002-07-25
JP2002543055A (ja) 2002-12-17
YU73701A (sh) 2005-06-10
AU773096B2 (en) 2004-05-13
JP3769192B2 (ja) 2006-04-19
EA200101113A1 (ru) 2002-04-25
NO20015095D0 (no) 2001-10-19
EP1171418A1 (en) 2002-01-16
EP1171418B1 (en) 2004-12-29
EA004209B1 (ru) 2004-02-26
KR20010108521A (ko) 2001-12-07
BG106132A (en) 2002-06-28
HK1045682A1 (en) 2002-12-06
CN1347403A (zh) 2002-05-01
AP2001002328A0 (en) 2001-12-31
WO2000064856A1 (en) 2000-11-02
ZA200107834B (en) 2002-12-23
GEP20033089B (en) 2003-10-27
CA2368807A1 (en) 2000-11-02
DE60017109T2 (de) 2006-01-12
TR200103015T2 (tr) 2002-01-21
PL351085A1 (en) 2003-03-24
CR6486A (es) 2004-03-11
PT1171418E (pt) 2005-02-28
HUP0200932A2 (hu) 2002-07-29

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Legal Events

Date Code Title Description
B08F Application dismissed because of non-payment of annual fees [chapter 8.6 patent gazette]

Free format text: REFERENTE A 8A E 9A ANUIDADES.

B08K Patent lapsed as no evidence of payment of the annual fee has been furnished to inpi [chapter 8.11 patent gazette]

Free format text: REFERENTE AO DESPACHO 8.6 NA RPI2003 DE 26/05/2009.