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BE2024C511I2 - - Google Patents

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Publication number
BE2024C511I2
BE2024C511I2 BE2024C511C BE2024C511C BE2024C511I2 BE 2024C511 I2 BE2024C511 I2 BE 2024C511I2 BE 2024C511 C BE2024C511 C BE 2024C511C BE 2024C511 C BE2024C511 C BE 2024C511C BE 2024C511 I2 BE2024C511 I2 BE 2024C511I2
Authority
BE
Belgium
Application number
BE2024C511C
Other languages
Dutch (nl)
Original Assignee
Japan Tobacco Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=35079161&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=BE2024C511(I2) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Japan Tobacco Inc filed Critical Japan Tobacco Inc
Publication of BE2024C511I2 publication Critical patent/BE2024C511I2/nl

Links

Classifications

    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/47—Quinolines; Isoquinolines
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/12—Antivirals
    • A61P31/14—Antivirals for RNA viruses
    • A61P31/18—Antivirals for RNA viruses for HIV
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D215/00—Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems
    • C07D215/02—Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen atoms or carbon atoms directly attached to the ring nitrogen atom
    • C07D215/16—Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen atoms or carbon atoms directly attached to the ring nitrogen atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D215/48—Carbon atoms having three bonds to hetero atoms with at the most one bond to halogen
    • C07D215/54—Carbon atoms having three bonds to hetero atoms with at the most one bond to halogen attached in position 3
    • C07D215/56—Carbon atoms having three bonds to hetero atoms with at the most one bond to halogen attached in position 3 with oxygen atoms in position 4

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • General Health & Medical Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Virology (AREA)
  • General Chemical & Material Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Oncology (AREA)
  • Communicable Diseases (AREA)
  • Molecular Biology (AREA)
  • Tropical Medicine & Parasitology (AREA)
  • AIDS & HIV (AREA)
  • Epidemiology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Quinoline Compounds (AREA)
BE2024C511C 2004-05-20 2024-03-15 BE2024C511I2 (en)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
JP2004150979 2004-05-20

Publications (1)

Publication Number Publication Date
BE2024C511I2 true BE2024C511I2 (en) 2024-10-08

Family

ID=35079161

Family Applications (1)

Application Number Title Priority Date Filing Date
BE2024C511C BE2024C511I2 (en) 2004-05-20 2024-03-15

Country Status (33)

Country Link
US (7) US7635704B2 (en)
EP (4) EP3281939B1 (en)
JP (1) JP3754064B2 (en)
KR (1) KR20080064909A (en)
CN (1) CN1956961B (en)
AR (2) AR049280A1 (en)
AU (1) AU2005245296B2 (en)
BE (1) BE2024C511I2 (en)
BR (1) BRPI0510114B8 (en)
CA (1) CA2566922C (en)
CY (4) CY1113010T1 (en)
DK (2) DK3281939T3 (en)
ES (2) ES2388441T3 (en)
FI (2) FI3281939T3 (en)
FR (1) FR23C1040I1 (en)
HR (2) HRP20231588T3 (en)
HU (2) HUE064615T2 (en)
IL (1) IL179250A0 (en)
LT (1) LT3281939T (en)
LU (1) LUC00334I2 (en)
MX (1) MXPA06013405A (en)
MY (1) MY134672A (en)
NO (7) NO339223B1 (en)
NZ (1) NZ551839A (en)
PE (2) PE20060358A1 (en)
PL (2) PL1636190T3 (en)
PT (2) PT3281939T (en)
RS (2) RS52375B (en)
RU (1) RU2330845C1 (en)
SI (2) SI1636190T1 (en)
TW (1) TWI329015B (en)
WO (1) WO2005113508A1 (en)
ZA (1) ZA200610647B (en)

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US20090233964A1 (en) * 2005-12-30 2009-09-17 Gilead Sciences, Inc. Methods for improving the pharmacokinetics of hiv integrase inhibitors
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EA018544B1 (en) * 2005-12-30 2013-08-30 Джилид Сайэнс, Инк. Method for treating retroviral infection
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WO2007092802A1 (en) * 2006-02-09 2007-08-16 Boehringer Ingelheim International Gmbh Method for treating hiv infection through co-administration of tipranavir and gs 9137
CN101437801B (en) 2006-03-06 2013-02-06 日本烟草产业株式会社 Process for preparing 4-oxoquinoline compounds
JP4669040B2 (en) * 2006-03-06 2011-04-13 日本たばこ産業株式会社 Process for producing 4-oxoquinoline compound
EA020489B1 (en) 2006-07-07 2014-11-28 Джилид Сайэнс, Инк. Modulators of pharmacokinetic properties of therapeutics
HRP20090213B1 (en) 2006-09-12 2016-12-02 Gilead Sciences, Inc. PROCEDURE AND INTERMEDIATES IN PREPARATION OF INTEGRASE INHIBITOR
EA019893B1 (en) * 2007-02-23 2014-07-30 Джилид Сайэнс, Инк. Pharmaceutical composition and method for treating hiv infection
US20090093467A1 (en) * 2007-06-29 2009-04-09 Gilead Sciences, Inc. Therapeutic compositions and methods
SG182228A1 (en) * 2007-06-29 2012-07-30 Gilead Sciences Inc Therapeutic compositions and uses thereof
AR068403A1 (en) * 2007-09-11 2009-11-18 Gilead Sciences Inc PROCESS AND INTERMEDIARIES FOR THE PREPARATION OF INTEGRASA INHIBITORS
BRPI0911871A8 (en) 2008-05-02 2018-03-06 Gilead Sciences Inc use of solid carrier particles to improve processability of a pharmaceutical agent
CA2750521A1 (en) 2009-02-06 2010-08-12 Gilead Sciences, Inc. Tablets for combination therapy
WO2010137032A2 (en) * 2009-05-14 2010-12-02 Matrix Laboratories Ltd. Novel polymorphic forms of elvitegravir and its pharmaceutically acceptable salts
WO2011004389A2 (en) * 2009-06-18 2011-01-13 Matrix Laboratories Ltd An improved process for the preparation of elvitegravir
CN102212032B (en) * 2011-04-20 2013-07-31 复旦大学 5-hyroxyquinolone derivatives, and preparation method and application thereof
CA2878478A1 (en) 2012-07-06 2014-01-09 Genentech, Inc. N-substituted benzamides and methods of use thereof
BR112015002275A2 (en) 2012-08-03 2017-07-04 Gilead Sciences Inc processes and intermediates for the preparation of integrase inhibitors
CN103819402B (en) * 2012-11-17 2016-03-30 上海迪赛诺化学制药有限公司 Dust is for drawing Wei intermediate and its preparation method and application
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MY164352A (en) 2012-12-21 2017-12-15 Gilead Sciences Inc Polycyclic-carbamoylpyridone compounds and their pharmaceutical use
SI3019503T1 (en) 2013-07-12 2017-11-30 Gilead Sciences, Inc. Polycyclic-carbamoylpyridone compounds and their use for the treatment of hiv infections
NO2865735T3 (en) 2013-07-12 2018-07-21
CN105315203A (en) * 2014-06-06 2016-02-10 上海迪赛诺化学制药有限公司 V-type elvitegravir crystal and preparation method thereof
TWI744723B (en) 2014-06-20 2021-11-01 美商基利科學股份有限公司 Synthesis of polycyclic-carbamoylpyridone compounds
NO2717902T3 (en) 2014-06-20 2018-06-23
TW201613936A (en) 2014-06-20 2016-04-16 Gilead Sciences Inc Crystalline forms of(2R,5S,13aR)-8-hydroxy-7,9-dioxo-n-(2,4,6-trifluorobenzyl)-2,3,4,5,7,9,13,13a-octahydro-2,5-methanopyrido[1',2':4,5]pyrazino[2,1-b][1,3]oxazepine-10-carboxamide
TWI695003B (en) 2014-12-23 2020-06-01 美商基利科學股份有限公司 Polycyclic-carbamoylpyridone compounds and their pharmaceutical use
SI3466490T1 (en) 2015-04-02 2020-12-31 Gilead Sciences, Inc. Polycyclic-carbamoylpyridone compounds and their pharmaceutical use
CN106008195B (en) * 2016-05-19 2018-08-03 绍兴文理学院 The preparation method of 2,4- of one kind, bis- fluoro- 5- iodo-benzoic acids
EP3984536B1 (en) * 2020-10-19 2025-06-25 Centre national de la recherche scientifique Inhibition of the hiv-1 replication by compounds directed against a new target of the viral cycle

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Also Published As

Publication number Publication date
CY2015009I1 (en) 2024-09-20
DK1636190T3 (en) 2012-09-24
CY1113010T1 (en) 2016-04-13
CY2024008I2 (en) 2024-09-20
US20190185433A1 (en) 2019-06-20
FIC20240008I1 (en) 2024-03-20
US20250091995A1 (en) 2025-03-20
NO339223B1 (en) 2016-11-21
SI3281939T1 (en) 2024-02-29
NO20220690A1 (en) 2007-02-07
LT3281939T (en) 2023-11-27
EP4299563A3 (en) 2024-02-28
CA2566922A1 (en) 2005-12-01
HK1083341A1 (en) 2006-06-30
HRP20231588T3 (en) 2024-03-15
IL179250A0 (en) 2007-03-08
AU2005245296B2 (en) 2010-08-12
CN1956961B (en) 2010-05-26
HUE064615T2 (en) 2024-04-28
AR096100A2 (en) 2015-12-09
NO20230913A1 (en) 2007-02-07
EP1636190A1 (en) 2006-03-22
EP4299563A2 (en) 2024-01-03
US20100204271A1 (en) 2010-08-12
SI1636190T1 (en) 2012-09-28
EP2514746A1 (en) 2012-10-24
US20150361044A1 (en) 2015-12-17
PE20060358A1 (en) 2006-05-12
PT1636190E (en) 2012-08-20
US7635704B2 (en) 2009-12-22
EP3281939A1 (en) 2018-02-14
US8981103B2 (en) 2015-03-17
DK3281939T3 (en) 2024-01-22
NO20200873A1 (en) 2007-02-07
AR049280A1 (en) 2006-07-12
ES2960824T3 (en) 2024-03-06
RS52375B (en) 2012-12-31
LUC00334I2 (en) 2024-07-01
NO20065790L (en) 2007-02-07
US20180029989A1 (en) 2018-02-01
FI3281939T3 (en) 2023-10-23
RU2330845C1 (en) 2008-08-10
CY2024008I1 (en) 2024-09-20
PL1636190T3 (en) 2012-10-31
WO2005113508A1 (en) 2005-12-01
US20060030710A1 (en) 2006-02-09
CY2015009I2 (en) 2024-09-20
NO20240384A1 (en) 2007-02-07
EP1636190B1 (en) 2012-06-27
NO20190051A1 (en) 2007-02-07
NO347902B1 (en) 2024-05-06
BRPI0510114A (en) 2007-09-25
RS64845B1 (en) 2023-12-29
PL3281939T3 (en) 2024-03-18
US20220235009A1 (en) 2022-07-28
JP3754064B2 (en) 2006-03-08
CY1126560T1 (en) 2024-09-20
MXPA06013405A (en) 2007-03-01
EP3281939B1 (en) 2023-10-18
ES2388441T3 (en) 2012-10-15
FR23C1040I1 (en) 2023-12-29
BRPI0510114B8 (en) 2021-05-25
MY134672A (en) 2007-12-31
NO20161297A1 (en) 2007-02-07
PT3281939T (en) 2023-11-22
TW200600097A (en) 2006-01-01
ZA200610647B (en) 2008-06-25
TWI329015B (en) 2010-08-21
HRP20120681T1 (en) 2012-09-30
KR20080064909A (en) 2008-07-09
NZ551839A (en) 2009-11-27
JP2006001927A (en) 2006-01-05
HUS2400006I1 (en) 2024-04-28
AU2005245296A1 (en) 2005-12-01
CA2566922C (en) 2011-01-11
PE20120361A1 (en) 2012-05-03
BRPI0510114B1 (en) 2020-09-15
CN1956961A (en) 2007-05-02

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