AU8736691A - Cyclopeptides, a method of preparing them, and their use as drugs - Google Patents

Cyclopeptides, a method of preparing them, and their use as drugs

Info

Publication number: AU8736691A
Authority: AU; Australia
Prior art keywords: cyclopeptides; drugs; preparing
Prior art date: 1990-10-11
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.): Abandoned

Application number

AU87366/91A

Inventor

Stefan Heinrichs

Rainer Palluk

Gerd Schnorrenberg

Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)

Boehringer Ingelheim International GmbH

Original Assignee

Boehringer Ingelheim International GmbH

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

1990-10-11

Filing date

1991-10-10

Publication date

1992-05-20

1990-10-11 Priority claimed from DE19904032268 external-priority patent/DE4032268A1/en

1990-10-11 Priority claimed from DE19904032271 external-priority patent/DE4032271A1/en

1990-10-11 Priority claimed from DE19904032269 external-priority patent/DE4032269A1/en

1991-05-30 Priority claimed from DE19914117733 external-priority patent/DE4117733A1/en

1991-10-10 Application filed by Boehringer Ingelheim International GmbH filed Critical Boehringer Ingelheim International GmbH

1992-05-20 Publication of AU8736691A publication Critical patent/AU8736691A/en

Status Abandoned legal-status Critical Current

Classifications

- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07K—PEPTIDES
- C07K7/00—Peptides having 5 to 20 amino acids in a fully defined sequence; Derivatives thereof
- C07K7/50—Cyclic peptides containing at least one abnormal peptide link
- C07K7/54—Cyclic peptides containing at least one abnormal peptide link with at least one abnormal peptide link in the ring
- C07K7/56—Cyclic peptides containing at least one abnormal peptide link with at least one abnormal peptide link in the ring the cyclisation not occurring through 2,4-diamino-butanoic acid
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07K—PEPTIDES
- C07K14/00—Peptides having more than 20 amino acids; Gastrins; Somatostatins; Melanotropins; Derivatives thereof
- C07K14/435—Peptides having more than 20 amino acids; Gastrins; Somatostatins; Melanotropins; Derivatives thereof from animals; from humans
- C07K14/575—Hormones
- C07K14/58—Atrial natriuretic factor complex; Atriopeptin; Atrial natriuretic peptide [ANP]; Cardionatrin; Cardiodilatin
- C07K14/582—Atrial natriuretic factor complex; Atriopeptin; Atrial natriuretic peptide [ANP]; Cardionatrin; Cardiodilatin at least 1 amino acid in D-form
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P7/00—Drugs for disorders of the blood or the extracellular fluid
- A61P7/10—Antioedematous agents; Diuretics
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
- A61P9/08—Vasodilators for multiple indications
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
- A61P9/12—Antihypertensives
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K38/00—Medicinal preparations containing peptides

Landscapes

Health & Medical Sciences (AREA)
Chemical & Material Sciences (AREA)
Organic Chemistry (AREA)
Life Sciences & Earth Sciences (AREA)
General Health & Medical Sciences (AREA)
Medicinal Chemistry (AREA)
General Chemical & Material Sciences (AREA)
Animal Behavior & Ethology (AREA)
Chemical Kinetics & Catalysis (AREA)
Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
Cardiology (AREA)
Pharmacology & Pharmacy (AREA)
Bioinformatics & Cheminformatics (AREA)
Veterinary Medicine (AREA)
Engineering & Computer Science (AREA)
Public Health (AREA)
Biochemistry (AREA)
Heart & Thoracic Surgery (AREA)
Proteomics, Peptides & Aminoacids (AREA)
Molecular Biology (AREA)
Genetics & Genomics (AREA)
Biophysics (AREA)
Diabetes (AREA)
Gastroenterology & Hepatology (AREA)
Zoology (AREA)
Toxicology (AREA)
Endocrinology (AREA)
Hematology (AREA)
Peptides Or Proteins (AREA)
Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)

AU87366/91A 1990-10-11 1991-10-10 Cyclopeptides, a method of preparing them, and their use as drugs Abandoned AU8736691A (en)

Applications Claiming Priority (8)

Application Number	Priority Date	Filing Date	Title
DE19904032268 DE4032268A1 (en)	1990-10-11	1990-10-11	CYCLOPEPTIDES, METHOD FOR THE PRODUCTION THEREOF AND THEIR USE AS MEDICINAL PRODUCTS
DE19904032271 DE4032271A1 (en)	1990-10-11	1990-10-11	New cyclo:peptide(s) are atrial natriuretic factor agonists - useful as hypotensives, vasodilators, spasmolytics and broncholytics, and as ligands in receptor binding assays
DE4032269		1990-10-11
DE4032271		1990-10-11
DE19904032269 DE4032269A1 (en)	1990-10-11	1990-10-11	CYCLOPEPTIDES, METHOD FOR THE PRODUCTION THEREOF AND THEIR USE AS MEDICINAL PRODUCTS
DE4032268		1990-10-11
DE19914117733 DE4117733A1 (en)	1991-05-30	1991-05-30	CYCLOPEPTIDES, METHOD FOR THE PRODUCTION THEREOF AND THEIR USE AS MEDICINAL PRODUCTS
DE4117733		1991-05-30

Publications (1)

Publication Number	Publication Date
AU8736691A true AU8736691A (en)	1992-05-20

Family

ID=27435038

Family Applications (1)

Application Number	Title	Priority Date	Filing Date
AU87366/91A Abandoned AU8736691A (en)	1990-10-11	1991-10-10	Cyclopeptides, a method of preparing them, and their use as drugs

Country Status (12)

Country	Link
EP (1)	EP0552238A1 (en)
JP (1)	JPH06501950A (en)
KR (1)	KR930702395A (en)
AU (1)	AU8736691A (en)
CA (1)	CA2089747A1 (en)
CZ (1)	CZ61893A3 (en)
FI (1)	FI931499A0 (en)
HU (1)	HUT63859A (en)
IE (1)	IE913582A1 (en)
PL (1)	PL168456B1 (en)
SK (1)	SK32693A3 (en)
WO (1)	WO1992006998A1 (en)

Families Citing this family (29)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
US6525022B1 (en)	1993-11-12	2003-02-25	Genentech, Inc.	Receptor specific atrial natriuretic peptides
US5665704A (en) *	1993-11-12	1997-09-09	Genentech, Inc.	Receptor specific atrial natriuretic peptides
US5846932A (en) *	1993-11-12	1998-12-08	Genentech, Inc.	Receptor specific atrial natriuretic peptides
US6337385B1 (en)	1998-06-24	2002-01-08	The Rockefeller University	Staphylococcus peptides for bacterial interference
WO1999067286A2 (en) *	1998-06-24	1999-12-29	The Rockefeller University	Novel staphylococcus peptides for bacterial interference
FR2797689B1 (en) *	1999-08-16	2003-06-27	Pasteur Sanofi Diagnostics	USE OF SYNTHETIC COMPOUNDS FOR IMMUNODAYS
US6455587B1 (en) *	2000-03-15	2002-09-24	Pharmacor Inc.	Amino acid derivatives as HIV aspartyl protease inhibitors
CA2518265A1 (en)	2003-03-17	2004-09-30	Albany Molecular Research, Inc.	Novel cyclosporins
US7388008B2 (en)	2004-08-02	2008-06-17	Ambrilia Biopharma Inc.	Lysine based compounds
JP2008514701A (en)	2004-09-29	2008-05-08	エーエムアールテクノロジーインコーポレイテッド	Cyclosporine alkyne analogs and their pharmaceutical use
US7511013B2 (en)	2004-09-29	2009-03-31	Amr Technology, Inc.	Cyclosporin analogues and their pharmaceutical uses
US7361636B2 (en)	2004-10-06	2008-04-22	Amr Technology, Inc.	Cyclosporin alkynes and their utility as pharmaceutical agents
ES2452718T3 (en)	2005-11-30	2014-04-02	Taimed Biologics, Inc.	Lysine-based prodrugs of aspartyl protease inhibitors and processes for their preparation
US8580746B2 (en)	2006-03-30	2013-11-12	Palatin Technologies, Inc.	Amide linkage cyclic natriuretic peptide constructs
WO2007115182A2 (en)	2006-03-30	2007-10-11	Palatin Technologies, Inc.	Linear natriuretic peptide constructs
BRPI0709427A2 (en)	2006-03-30	2011-07-12	Palatin Technologies Inc	"Cyclic construct, pharmaceutical composition and use of a compound
ES2628730T3 (en)	2006-09-21	2017-08-03	Taimed Biologics, Inc.	Protease inhibitors
CA2939778C (en)	2007-01-31	2019-01-29	Dana-Farber Cancer Institute, Inc.	Stabilized p53 peptides and uses thereof
EP2142562B1 (en)	2007-03-28	2013-07-03	President and Fellows of Harvard College	Stitched polypeptides
CN108570097A (en)	2010-08-13	2018-09-25	爱勒让治疗公司	Peptidomimetic macrocyclic compound
CN108929375A (en)	2011-10-18	2018-12-04	爱勒让治疗公司	Peptidomimetic macrocyclic compound
NZ627528A (en)	2012-02-15	2016-05-27	Aileron Therapeutics Inc	Peptidomimetic macrocycles
EP2819688A4 (en)	2012-02-15	2015-10-28	Aileron Therapeutics Inc	TRIAZOL AND THIOETHER-COUPLED PEPTIDOMIMETIC MACROCYCLES
SG11201503052RA (en)	2012-11-01	2015-05-28	Aileron Therapeutics Inc	Disubstituted amino acids and methods of preparation and use thereof
WO2015179438A1 (en)	2014-05-20	2015-11-26	Ohio State Innovation Foundation	Small molecule rac or rho inhibitors
MX2017003797A (en)	2014-09-24	2017-06-15	Aileron Therapeutics Inc	Peptidomimetic macrocycles and uses thereof.
CA2961029A1 (en)	2014-09-24	2016-03-31	Aileron Therapeutics, Inc.	Peptidomimetic macrocycles and formulations thereof
CA2979847A1 (en)	2015-03-20	2016-09-29	Aileron Therapeutics, Inc.	Peptidomimetic macrocycles and uses thereof
WO2017044633A1 (en)	2015-09-10	2017-03-16	Aileron Therapeutics, Inc.	Peptidomimetic macrocycles as modulators of mcl-1

Family Cites Families (3)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
CA1337891C (en) *	1987-12-16	1996-01-02	John Dimaio	Anf derivatives with novel bridging
US4935492A (en) *	1987-12-24	1990-06-19	California Biotechnology Inc.	Cyclic analogs of atrial natriuretic peptides
DK380288D0 (en) *	1988-07-07	1988-07-07	Novo Industri As	HOW TO UNKNOWN PEPTIDES

1991
- 1991-10-10 EP EP91918322A patent/EP0552238A1/en not_active Withdrawn
- 1991-10-10 SK SK32693A patent/SK32693A3/en unknown
- 1991-10-10 AU AU87366/91A patent/AU8736691A/en not_active Abandoned
- 1991-10-10 WO PCT/EP1991/001934 patent/WO1992006998A1/en not_active Application Discontinuation
- 1991-10-10 CA CA002089747A patent/CA2089747A1/en not_active Abandoned
- 1991-10-10 HU HU931054A patent/HUT63859A/en unknown
- 1991-10-10 CZ CS93618A patent/CZ61893A3/en unknown
- 1991-10-10 JP JP3516845A patent/JPH06501950A/en active Pending
- 1991-10-10 PL PL91299317A patent/PL168456B1/en unknown
- 1991-10-16 IE IE358291A patent/IE913582A1/en not_active Application Discontinuation
1993
- 1993-04-02 FI FI931499A patent/FI931499A0/en not_active Application Discontinuation
- 1993-04-10 KR KR1019930701088A patent/KR930702395A/en not_active Withdrawn

Also Published As

Publication number	Publication date
FI931499L (en)	1993-04-02
PL168456B1 (en)	1996-02-29
HUT63859A (en)	1993-10-28
CZ61893A3 (en)	1994-01-19
KR930702395A (en)	1993-09-09
SK32693A3 (en)	1993-09-09
CA2089747A1 (en)	1992-04-12
WO1992006998A1 (en)	1992-04-30
EP0552238A1 (en)	1993-07-28
JPH06501950A (en)	1994-03-03
FI931499A0 (en)	1993-04-02
HU9301054D0 (en)	1993-07-28
IE913582A1 (en)	1992-04-22

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