AU1576495A - Inhibitors of serine proteases, bearing a chelating group - Google Patents

Inhibitors of serine proteases, bearing a chelating group

Info

Publication number: AU1576495A
Authority: AU; Australia
Prior art keywords: inhibitors; bearing; serine proteases; chelating group; chelating
Prior art date: 1994-01-26
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.): Abandoned

Application number

AU15764/95A

Inventor

Rainer Metternich

Carlo Tapparelli

Anette Wienand

Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)

Sandoz AG

Original Assignee

Sandoz AG

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

1994-01-26

Filing date

1995-01-25

Publication date

1995-08-15

1995-01-25 Application filed by Sandoz AG filed Critical Sandoz AG

1995-08-15 Publication of AU1576495A publication Critical patent/AU1576495A/en

Status Abandoned legal-status Critical Current

Classifications

- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K51/00—Preparations containing radioactive substances for use in therapy or testing in vivo
- A61K51/02—Preparations containing radioactive substances for use in therapy or testing in vivo characterised by the carrier, i.e. characterised by the agent or material covalently linked or complexing the radioactive nucleus
- A61K51/04—Organic compounds
- A61K51/08—Peptides, e.g. proteins, carriers being peptides, polyamino acids, proteins
- A61K51/088—Peptides, e.g. proteins, carriers being peptides, polyamino acids, proteins conjugates with carriers being peptides, polyamino acids or proteins
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07K—PEPTIDES
- C07K5/00—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof
- C07K5/04—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof containing only normal peptide links
- C07K5/06—Dipeptides
- C07K5/06191—Dipeptides containing heteroatoms different from O, S, or N
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07K—PEPTIDES
- C07K5/00—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof
- C07K5/04—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof containing only normal peptide links
- C07K5/08—Tripeptides
- C07K5/0827—Tripeptides containing heteroatoms different from O, S, or N
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K38/00—Medicinal preparations containing peptides

Landscapes

Chemical & Material Sciences (AREA)
Health & Medical Sciences (AREA)
Life Sciences & Earth Sciences (AREA)
Organic Chemistry (AREA)
Proteomics, Peptides & Aminoacids (AREA)
General Health & Medical Sciences (AREA)
Medicinal Chemistry (AREA)
Genetics & Genomics (AREA)
Molecular Biology (AREA)
Biophysics (AREA)
Biochemistry (AREA)
Epidemiology (AREA)
Optics & Photonics (AREA)
Pharmacology & Pharmacy (AREA)
Physics & Mathematics (AREA)
Animal Behavior & Ethology (AREA)
Public Health (AREA)
Veterinary Medicine (AREA)
Peptides Or Proteins (AREA)
Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
Medicines Containing Antibodies Or Antigens For Use As Internal Diagnostic Agents (AREA)
Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)

AU15764/95A 1994-01-26 1995-01-25 Inhibitors of serine proteases, bearing a chelating group Abandoned AU1576495A (en)

Applications Claiming Priority (3)

Application Number	Priority Date	Filing Date	Title
GB9401483		1994-01-26
GB9401483A GB9401483D0 (en)	1994-01-26	1994-01-26	Organic compounds
PCT/EP1995/000269 WO1995020603A1 (en)	1994-01-26	1995-01-25	Inhibitors of serine proteases, bearing a chelating group

Publications (1)

Publication Number	Publication Date
AU1576495A true AU1576495A (en)	1995-08-15

Family

ID=10749357

Family Applications (1)

Application Number	Title	Priority Date	Filing Date
AU15764/95A Abandoned AU1576495A (en)	1994-01-26	1995-01-25	Inhibitors of serine proteases, bearing a chelating group

Country Status (10)

Country	Link
EP (1)	EP0741747A1 (en)
JP (1)	JPH09509653A (en)
AU (1)	AU1576495A (en)
CA (1)	CA2179889A1 (en)
GB (1)	GB9401483D0 (en)
IL (1)	IL112423A0 (en)
PE (1)	PE45295A1 (en)
SG (1)	SG47079A1 (en)
WO (1)	WO1995020603A1 (en)
ZA (1)	ZA95636B (en)

Families Citing this family (9)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
GB9515489D0 (en) *	1995-07-28	1995-09-27	Sandoz Ltd	Organic compounds
DE10046514A1 (en)	2000-09-15	2002-04-25	Diagnostikforschung Inst	Process for imaging and diagnosis of thrombi using magnetic resonance imaging using particulate contrast media
ES2264515T3 (en)	2002-09-09	2007-01-01	Trigen Limited	BORONIC ACID SALTS USED IN PARENTERAL FORMULATIONS FOR THE SELECTIVE INHIBITION OF THE THROMBIN.
US7223745B2 (en)	2003-08-14	2007-05-29	Cephalon, Inc.	Proteasome inhibitors and methods of using the same
US7576206B2 (en)	2003-08-14	2009-08-18	Cephalon, Inc.	Proteasome inhibitors and methods of using the same
US7468383B2 (en)	2005-02-11	2008-12-23	Cephalon, Inc.	Proteasome inhibitors and methods of using the same
JP5783659B2 (en)	2009-12-22	2015-09-24	セファロン、インク．	Proteasome inhibitors and methods for their preparation, purification and use
US10526315B2 (en)	2016-06-21	2020-01-07	Orion Ophthalmology LLC	Carbocyclic prolinamide derivatives
WO2017222915A1 (en)	2016-06-21	2017-12-28	Inception 4, Inc.	Heterocyclic prolinamide derivatives

Family Cites Families (6)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
US4668503A (en) *	1982-07-26	1987-05-26	Trustees Of University Of Massachusetts	Process for labeling amines with 99m Tc
US5187157A (en) *	1987-06-05	1993-02-16	Du Pont Merck Pharmaceutical Company	Peptide boronic acid inhibitors of trypsin-like proteases
EP0403243B1 (en) *	1989-06-16	1995-11-08	Merck Frosst Canada Inc.	Chelate derivatives of atrial natriuretic factor (ANF)
GB9017694D0 (en) *	1990-08-13	1990-09-26	Sandoz Ltd	Improvements in or relating to organic chemistry
US5252721A (en) *	1990-09-28	1993-10-12	Neorx Corporation	S3 N chelating compounds
AU2175492A (en) *	1991-04-22	1992-11-17	Mallinckrodt Medical, Inc.	Method for detecting and localizing tissues having neurokinine 1 receptors

1994
- 1994-01-26 GB GB9401483A patent/GB9401483D0/en active Pending
1995
- 1995-01-24 IL IL11242395A patent/IL112423A0/en unknown
- 1995-01-24 PE PE1995260194A patent/PE45295A1/en not_active Application Discontinuation
- 1995-01-25 AU AU15764/95A patent/AU1576495A/en not_active Abandoned
- 1995-01-25 EP EP95907611A patent/EP0741747A1/en not_active Ceased
- 1995-01-25 SG SG1996005775A patent/SG47079A1/en unknown
- 1995-01-25 WO PCT/EP1995/000269 patent/WO1995020603A1/en not_active Application Discontinuation
- 1995-01-25 CA CA002179889A patent/CA2179889A1/en not_active Abandoned
- 1995-01-25 JP JP7519884A patent/JPH09509653A/en active Pending
- 1995-01-26 ZA ZA95636A patent/ZA95636B/en unknown

Also Published As

Publication number	Publication date
GB9401483D0 (en)	1994-03-23
PE45295A1 (en)	1995-12-29
EP0741747A1 (en)	1996-11-13
SG47079A1 (en)	1998-03-20
CA2179889A1 (en)	1995-08-03
ZA95636B (en)	1996-07-26
IL112423A0 (en)	1995-03-30
JPH09509653A (en)	1997-09-30
WO1995020603A1 (en)	1995-08-03

Publication	Publication Date	Title
AU7127298A (en)	1998-11-11	Serine protease inhibitors
AU5122196A (en)	1996-10-16	Cysteine protease inhibitor
AU8875398A (en)	1999-03-22	1-amino-7-isoquinoline derivatives as serine protease inhibitors
AU4236796A (en)	1996-05-31	Cysteine protease and serine protease inhibitors
ZA9811830B (en)	2000-06-23	Prodrugs of aspartyl protease inhibitors.
AU2012199A (en)	1999-07-19	Prodrugs of aspartyl protease inhibitors
PL326508A1 (en)	1998-09-28	Protease inhibitors
AU3972697A (en)	1998-02-25	Inhibitors of cysteine protease
HUP9901187A3 (en)	1999-11-29	Serine protease inhibitors
IL142398A0 (en)	2002-03-10	Serine protease inhibitor
AU1795697A (en)	1997-09-16	Serine protease inhibitors
AU1877597A (en)	1997-09-16	Serine protease inhibitors
AU4723799A (en)	2000-01-10	Protease inhibitors
AU7139598A (en)	1998-11-24	Protease inhibitors
AU4092799A (en)	1999-12-06	Protease inhibitors
AU1576495A (en)	1995-08-15	Inhibitors of serine proteases, bearing a chelating group
AUPM982594A0 (en)	1995-01-05	HIV protease inhibitors
AU1893795A (en)	1995-09-25	Novel thiol protease inhibitor
AU4480797A (en)	1998-04-02	Protease m, a novel serine protease
AU9110298A (en)	1999-12-06	Protease inhibitors
AU1393900A (en)	2000-06-05	Morpholino-ethoxybenzofuran protease inhibitors
AU4672996A (en)	1996-09-04	Serine protease inhibitors
AU9300298A (en)	1999-03-22	Protease inhibitors
AU2713100A (en)	2000-07-31	Protease inhibitors
AU4564499A (en)	1999-12-30	Protease inhibitors