AU2713100A - Protease inhibitors - Google Patents

Protease inhibitors

Info

Publication number: AU2713100A
Authority: AU; Australia
Prior art keywords: protease inhibitors; protease; inhibitors
Prior art date: 1998-12-23
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.): Abandoned

Application number

AU27131/00A

Inventor

Robert Wells Marquis Jr.

Daniel Frank Veber

Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)

SmithKline Beecham Corp

Original Assignee

SmithKline Beecham Corp

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

1998-12-23

Filing date

1999-12-21

Publication date

2000-07-31

1999-12-21 Application filed by SmithKline Beecham Corp filed Critical SmithKline Beecham Corp

2000-07-31 Publication of AU2713100A publication Critical patent/AU2713100A/en

Status Abandoned legal-status Critical Current

Classifications

- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
- C07D401/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
- C07D401/12—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings linked by a chain containing hetero atoms as chain links
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P19/00—Drugs for skeletal disorders
- A61P19/02—Drugs for skeletal disorders for joint disorders, e.g. arthritis, arthrosis
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P19/00—Drugs for skeletal disorders
- A61P19/04—Drugs for skeletal disorders for non-specific disorders of the connective tissue
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P19/00—Drugs for skeletal disorders
- A61P19/08—Drugs for skeletal disorders for bone diseases, e.g. rachitism, Paget's disease
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P19/00—Drugs for skeletal disorders
- A61P19/08—Drugs for skeletal disorders for bone diseases, e.g. rachitism, Paget's disease
- A61P19/10—Drugs for skeletal disorders for bone diseases, e.g. rachitism, Paget's disease for osteoporosis
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P29/00—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D225/00—Heterocyclic compounds containing rings of more than seven members having one nitrogen atom as the only ring hetero atom
- C07D225/02—Heterocyclic compounds containing rings of more than seven members having one nitrogen atom as the only ring hetero atom not condensed with other rings

Landscapes

Health & Medical Sciences (AREA)
Organic Chemistry (AREA)
Chemical & Material Sciences (AREA)
Physical Education & Sports Medicine (AREA)
General Health & Medical Sciences (AREA)
Animal Behavior & Ethology (AREA)
Medicinal Chemistry (AREA)
Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
Chemical Kinetics & Catalysis (AREA)
Pharmacology & Pharmacy (AREA)
Life Sciences & Earth Sciences (AREA)
General Chemical & Material Sciences (AREA)
Engineering & Computer Science (AREA)
Public Health (AREA)
Veterinary Medicine (AREA)
Rheumatology (AREA)
Bioinformatics & Cheminformatics (AREA)
Orthopedic Medicine & Surgery (AREA)
Pain & Pain Management (AREA)
Immunology (AREA)
Biomedical Technology (AREA)
Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Plural Heterocyclic Compounds (AREA)
Other In-Based Heterocyclic Compounds (AREA)
Peptides Or Proteins (AREA)
Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)

AU27131/00A 1998-12-23 1999-12-21 Protease inhibitors Abandoned AU2713100A (en)

Applications Claiming Priority (3)

Application Number	Priority Date	Filing Date	Title
US11414398P	1998-12-23	1998-12-23
US60114143		1998-12-23
PCT/US1999/030602 WO2000039115A1 (en)	1998-12-23	1999-12-21	Protease inhibitors

Publications (1)

Publication Number	Publication Date
AU2713100A true AU2713100A (en)	2000-07-31

Family

ID=22353596

Family Applications (1)

Application Number	Title	Priority Date	Filing Date
AU27131/00A Abandoned AU2713100A (en)	1998-12-23	1999-12-21	Protease inhibitors

Country Status (9)

Country	Link
EP (1)	EP1140897A4 (en)
JP (1)	JP2002533452A (en)
AR (1)	AR021970A1 (en)
AU (1)	AU2713100A (en)
CO (1)	CO5180541A1 (en)
DZ (1)	DZ2976A1 (en)
HK (1)	HK1041690A1 (en)
PE (1)	PE20001355A1 (en)
WO (1)	WO2000039115A1 (en)

Families Citing this family (9)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
US20030144175A1 (en)	1998-12-23	2003-07-31	Smithkline Beecham Corporation	Protease inhibitors
WO2001034599A1 (en)	1999-11-10	2001-05-17	Smithkline Beecham Corporation	Protease inhibitors
AU1474801A (en)	1999-11-10	2001-06-06	Smithkline Beecham Corporation	Protease inhibitors
JP2003513972A (en)	1999-11-10	2003-04-15	スミスクライン・ビーチャム・コーポレイション	Protease inhibitor
MXPA02009305A (en)	2000-03-21	2003-03-12	Smithkline Beecham Corp	Protease inhibitors.
US6982263B2 (en)	2001-06-08	2006-01-03	Boehringer Ingelheim Pharmaceuticals, Inc.	Nitriles useful as reversible inhibitors of cysteine proteases
EP1483241A4 (en)	2002-03-08	2006-12-13	Bristol Myers Squibb Co	Cyclic derivatives as modulators of chemokine receptor activity
JP2008512461A (en) *	2004-09-07	2008-04-24	スミスクライン・ビーチャム・コーポレイション	New compounds
JP5236293B2 (en) *	2005-01-13	2013-07-17	ブリストル−マイヤーズスクイブカンパニー	Substituted biaryl compounds as XIA factor inhibitors

Family Cites Families (2)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
DZ2285A1 (en) *	1996-08-08	2002-12-25	Smithkline Beecham Corp	Cysteine protease inhibitors.
HUP0001285A3 (en) *	1997-05-08	2000-10-30	Smithkline Beecham Corp Philap	Pyrrolidine derivatives as protease inhibitors, process for producing them and pharmaceutical compositions containing them

1999
- 1999-12-16 CO CO99078651A patent/CO5180541A1/en not_active Application Discontinuation
- 1999-12-21 JP JP2000591026A patent/JP2002533452A/en not_active Withdrawn
- 1999-12-21 EP EP99968936A patent/EP1140897A4/en not_active Withdrawn
- 1999-12-21 AU AU27131/00A patent/AU2713100A/en not_active Abandoned
- 1999-12-21 AR ARP990106647A patent/AR021970A1/en unknown
- 1999-12-21 WO PCT/US1999/030602 patent/WO2000039115A1/en not_active Application Discontinuation
- 1999-12-22 DZ DZ990276A patent/DZ2976A1/en active
- 1999-12-23 PE PE1999001311A patent/PE20001355A1/en not_active Application Discontinuation
2002
- 2002-02-19 HK HK02101209.3A patent/HK1041690A1/en unknown

Also Published As

Publication number	Publication date
EP1140897A1 (en)	2001-10-10
DZ2976A1 (en)	2004-03-15
WO2000039115A1 (en)	2000-07-06
CO5180541A1 (en)	2002-07-30
JP2002533452A (en)	2002-10-08
AR021970A1 (en)	2002-09-04
HK1041690A1 (en)	2002-07-19
PE20001355A1 (en)	2001-01-28
EP1140897A4 (en)	2002-04-03

Publication	Publication Date	Title
PL349192A1 (en)	2002-07-01	Protease inhibitors
AU7127298A (en)	1998-11-11	Serine protease inhibitors
PL336625A1 (en)	2000-07-03	Protease inhibitors
PL336589A1 (en)	2000-07-03	Serinic protease inhibitors
AU4723799A (en)	2000-01-10	Protease inhibitors
AU6007200A (en)	2001-02-19	Cysteine protease inhibitors
IL132088A0 (en)	2001-03-19	Protease inhibitors
AU1795697A (en)	1997-09-16	Serine protease inhibitors
AU7139598A (en)	1998-11-24	Protease inhibitors
PL337755A1 (en)	2000-09-11	Protease inhibitors
AU1877597A (en)	1997-09-16	Serine protease inhibitors
IL132629A0 (en)	2001-03-19	Protease inhibitors
AU9059798A (en)	2000-04-10	Urokinase inhibitors
AU4092799A (en)	1999-12-06	Protease inhibitors
AU1393900A (en)	2000-06-05	Morpholino-ethoxybenzofuran protease inhibitors
AU9110298A (en)	1999-12-06	Protease inhibitors
AU2723099A (en)	1999-08-23	Tryptase inhibitors
AU4229599A (en)	1999-12-20	Protease inhibitor peptides
AU1588901A (en)	2001-06-06	Protease inhibitors
AU4564499A (en)	1999-12-30	Protease inhibitors
AU2713100A (en)	2000-07-31	Protease inhibitors
AU9300298A (en)	1999-03-22	Protease inhibitors
AU1474801A (en)	2001-06-06	Protease inhibitors
AU4066900A (en)	2000-10-16	Protease inhibitors
AU1474601A (en)	2001-06-06	Protease inhibitors

Legal Events

Date	Code	Title	Description
2001-09-20	MK6	Application lapsed section 142(2)(f)/reg. 8.3(3) - pct applic. not entering national phase