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ATE501125T1 - Verfahren zur herstellung des calciumsalzes von rosuvastatin - Google Patents

Verfahren zur herstellung des calciumsalzes von rosuvastatin

Info

Publication number
ATE501125T1
ATE501125T1 AT03784274T AT03784274T ATE501125T1 AT E501125 T1 ATE501125 T1 AT E501125T1 AT 03784274 T AT03784274 T AT 03784274T AT 03784274 T AT03784274 T AT 03784274T AT E501125 T1 ATE501125 T1 AT E501125T1
Authority
AT
Austria
Prior art keywords
rosuvastatin
producing
calcium salt
calcium
salt
Prior art date
Application number
AT03784274T
Other languages
English (en)
Inventor
John Horbury
Nigel Taylor
Original Assignee
Astrazeneca Uk Ltd
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=9942204&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=ATE501125(T1) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Astrazeneca Uk Ltd filed Critical Astrazeneca Uk Ltd
Application granted granted Critical
Publication of ATE501125T1 publication Critical patent/ATE501125T1/de

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D239/00—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings
    • C07D239/02—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings
    • C07D239/24—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members
    • C07D239/28—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, directly attached to ring carbon atoms
    • C07D239/32—One oxygen, sulfur or nitrogen atom
    • C07D239/42—One nitrogen atom
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00—Drugs for disorders of the metabolism
    • A61P3/06—Antihyperlipidemics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00—Drugs for disorders of the cardiovascular system
    • A61P9/10—Drugs for disorders of the cardiovascular system for treating ischaemic or atherosclerotic diseases, e.g. antianginal drugs, coronary vasodilators, drugs for myocardial infarction, retinopathy, cerebrovascula insufficiency, renal arteriosclerosis

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Animal Behavior & Ethology (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Pharmacology & Pharmacy (AREA)
  • General Health & Medical Sciences (AREA)
  • Urology & Nephrology (AREA)
  • Vascular Medicine (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Cardiology (AREA)
  • Diabetes (AREA)
  • Hematology (AREA)
  • Obesity (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
AT03784274T 2002-08-13 2003-08-07 Verfahren zur herstellung des calciumsalzes von rosuvastatin ATE501125T1 (de)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
GBGB0218781.3A GB0218781D0 (en) 2002-08-13 2002-08-13 Chemical process
PCT/GB2003/003463 WO2004014872A1 (en) 2002-08-13 2003-08-07 Process for preparing the calcium salt of rosuvastatin

Publications (1)

Publication Number Publication Date
ATE501125T1 true ATE501125T1 (de) 2011-03-15

Family

ID=9942204

Family Applications (1)

Application Number Title Priority Date Filing Date
AT03784274T ATE501125T1 (de) 2002-08-13 2003-08-07 Verfahren zur herstellung des calciumsalzes von rosuvastatin

Country Status (30)

Country Link
US (2) US7511140B2 (de)
EP (1) EP1539711B1 (de)
JP (1) JP4588446B2 (de)
KR (1) KR101325827B1 (de)
CN (1) CN100361979C (de)
AR (1) AR040868A1 (de)
AT (1) ATE501125T1 (de)
AU (1) AU2003251369B2 (de)
BR (1) BR0313394A (de)
CA (1) CA2495296C (de)
CY (1) CY1112412T1 (de)
DE (1) DE60336326D1 (de)
DK (1) DK1539711T3 (de)
ES (1) ES2361009T3 (de)
GB (1) GB0218781D0 (de)
HK (1) HK1082735A1 (de)
IL (1) IL166626A (de)
IS (1) IS7728A (de)
MX (1) MXPA05001582A (de)
MY (1) MY135301A (de)
NO (1) NO329439B1 (de)
NZ (1) NZ538070A (de)
PL (1) PL375296A1 (de)
PT (1) PT1539711E (de)
RU (1) RU2326871C2 (de)
SI (1) SI1539711T1 (de)
TW (1) TWI316058B (de)
UA (1) UA83805C2 (de)
WO (1) WO2004014872A1 (de)
ZA (1) ZA200500745B (de)

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TW200831469A (en) * 2006-12-01 2008-08-01 Astrazeneca Uk Ltd Chemical process

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IL166626A0 (en) 2006-01-15
SI1539711T1 (sl) 2011-06-30
MY135301A (en) 2008-03-31
CN100361979C (zh) 2008-01-16
KR101325827B1 (ko) 2013-11-05
US20060116391A1 (en) 2006-06-01
US7842807B2 (en) 2010-11-30
UA83805C2 (uk) 2008-08-26
HK1082735A1 (en) 2006-06-16
DE60336326D1 (de) 2011-04-21
NO20050542L (no) 2005-02-28
TWI316058B (en) 2009-10-21
WO2004014872A1 (en) 2004-02-19
US20090286819A1 (en) 2009-11-19
NO329439B1 (no) 2010-10-18
IL166626A (en) 2011-09-27
KR20050036968A (ko) 2005-04-20
PL375296A1 (en) 2005-11-28
ZA200500745B (en) 2006-03-29
AU2003251369B2 (en) 2007-02-01
EP1539711A1 (de) 2005-06-15
AU2003251369A1 (en) 2004-02-25
MXPA05001582A (es) 2005-04-25
PT1539711E (pt) 2011-05-03
RU2326871C2 (ru) 2008-06-20
NZ538070A (en) 2006-08-31
CA2495296A1 (en) 2004-02-19
IS7728A (is) 2005-03-08
CY1112412T1 (el) 2015-12-09
AR040868A1 (es) 2005-04-20
EP1539711B1 (de) 2011-03-09
BR0313394A (pt) 2005-06-21
DK1539711T3 (da) 2011-05-30
JP4588446B2 (ja) 2010-12-01
GB0218781D0 (en) 2002-09-18
JP2006500347A (ja) 2006-01-05
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US7511140B2 (en) 2009-03-31
CN1688551A (zh) 2005-10-26
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ES2361009T3 (es) 2011-06-13
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