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ATE422198T1 - Arylsulfonylnaphthalinderivate als 5ht2a- antagonisten - Google Patents

Arylsulfonylnaphthalinderivate als 5ht2a- antagonisten

Info

Publication number
ATE422198T1
ATE422198T1 AT05813608T AT05813608T ATE422198T1 AT E422198 T1 ATE422198 T1 AT E422198T1 AT 05813608 T AT05813608 T AT 05813608T AT 05813608 T AT05813608 T AT 05813608T AT E422198 T1 ATE422198 T1 AT E422198T1
Authority
AT
Austria
Prior art keywords
arylsulfonylnaphthaline
derivatives
5ht2a antagonists
antagonists
5ht2a
Prior art date
Application number
AT05813608T
Other languages
English (en)
Inventor
Mark Chambers
Neil CURTIS
Emanuela Gancia
Myra Gilligan
Alexander Humphries
Tamara Ladduwahetty
Robert Maxey
Kevin Merchant
Original Assignee
Merck Sharp & Dohme
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Merck Sharp & Dohme filed Critical Merck Sharp & Dohme
Application granted granted Critical
Publication of ATE422198T1 publication Critical patent/ATE422198T1/de

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    • C07D401/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
    • C07D401/12—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings linked by a chain containing hetero atoms as chain links
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    • C07D213/04—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom
    • C07D213/60—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
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  • Steroid Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Quinoline Compounds (AREA)
  • Thiazole And Isothizaole Compounds (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Pyrrole Compounds (AREA)
  • Heat Sensitive Colour Forming Recording (AREA)
  • Transition And Organic Metals Composition Catalysts For Addition Polymerization (AREA)
AT05813608T 2004-12-01 2005-11-28 Arylsulfonylnaphthalinderivate als 5ht2a- antagonisten ATE422198T1 (de)

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WO2006059149A8 (en) 2006-11-02
EP1824817B1 (de) 2009-02-04
CA2588864A1 (en) 2006-06-08
US7592456B2 (en) 2009-09-22
AU2005311041A1 (en) 2006-06-08
EP1824817A1 (de) 2007-08-29
GB0426313D0 (en) 2005-01-05
JP2008521872A (ja) 2008-06-26
US20070281952A1 (en) 2007-12-06
WO2006059149A1 (en) 2006-06-08
DE602005012634D1 (en) 2009-03-19
CN101068776A (zh) 2007-11-07

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