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ATE312116T1 - Verfahren zur herstellung von nukleosid-derivaten - Google Patents

Verfahren zur herstellung von nukleosid-derivaten

Info

Publication number
ATE312116T1
ATE312116T1 AT99900359T AT99900359T ATE312116T1 AT E312116 T1 ATE312116 T1 AT E312116T1 AT 99900359 T AT99900359 T AT 99900359T AT 99900359 T AT99900359 T AT 99900359T AT E312116 T1 ATE312116 T1 AT E312116T1
Authority
AT
Austria
Prior art keywords
hydroxyl group
nucleoside derivatives
sugar moiety
fluorine atom
purine riboside
Prior art date
Application number
AT99900359T
Other languages
English (en)
Inventor
Satoshi Takamatsu
Satoshi Katayama
Naoko Hirose
Kunisuke Izawa
Tokumi Maruyama
Original Assignee
Ajinomoto Kk
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Ajinomoto Kk filed Critical Ajinomoto Kk
Application granted granted Critical
Publication of ATE312116T1 publication Critical patent/ATE312116T1/de

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07H—SUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
    • C07H19/00—Compounds containing a hetero ring sharing one ring hetero atom with a saccharide radical; Nucleosides; Mononucleotides; Anhydro-derivatives thereof
    • C07H19/02—Compounds containing a hetero ring sharing one ring hetero atom with a saccharide radical; Nucleosides; Mononucleotides; Anhydro-derivatives thereof sharing nitrogen
    • C07H19/04—Heterocyclic radicals containing only nitrogen atoms as ring hetero atom
    • C07H19/16—Purine radicals
    • Y—GENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
    • Y02—TECHNOLOGIES OR APPLICATIONS FOR MITIGATION OR ADAPTATION AGAINST CLIMATE CHANGE
    • Y02P—CLIMATE CHANGE MITIGATION TECHNOLOGIES IN THE PRODUCTION OR PROCESSING OF GOODS
    • Y02P20/00—Technologies relating to chemical industry
    • Y02P20/50—Improvements relating to the production of bulk chemicals
    • Y02P20/55—Design of synthesis routes, e.g. reducing the use of auxiliary or protecting groups

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Biochemistry (AREA)
  • Biotechnology (AREA)
  • General Health & Medical Sciences (AREA)
  • Genetics & Genomics (AREA)
  • Molecular Biology (AREA)
  • Saccharide Compounds (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
AT99900359T 1998-01-30 1999-01-19 Verfahren zur herstellung von nukleosid-derivaten ATE312116T1 (de)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
JP10019138A JPH11217396A (ja) 1998-01-30 1998-01-30 ヌクレオシド誘導体の製造方法
PCT/JP1999/000169 WO1999038879A1 (fr) 1998-01-30 1999-01-19 Procede servant a preparer des derives de nucleosides

Publications (1)

Publication Number Publication Date
ATE312116T1 true ATE312116T1 (de) 2005-12-15

Family

ID=11991103

Family Applications (1)

Application Number Title Priority Date Filing Date
AT99900359T ATE312116T1 (de) 1998-01-30 1999-01-19 Verfahren zur herstellung von nukleosid-derivaten

Country Status (6)

Country Link
EP (1) EP1052265B1 (de)
JP (1) JPH11217396A (de)
AT (1) ATE312116T1 (de)
CA (1) CA2318277A1 (de)
DE (1) DE69928772D1 (de)
WO (1) WO1999038879A1 (de)

Families Citing this family (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JP2002293792A (ja) * 1998-12-25 2002-10-09 Ajinomoto Co Inc ヌクレオシド又は糖のフッ素化誘導体の製造方法
SE0402461D0 (sv) * 2004-10-08 2004-10-08 Astrazeneca Ab New process

Family Cites Families (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4751221A (en) * 1985-10-18 1988-06-14 Sloan-Kettering Institute For Cancer Research 2-fluoro-arabinofuranosyl purine nucleosides
HU906976D0 (en) * 1989-11-13 1991-05-28 Bristol Myers Squibb Co Process for producing 2', 3'-didesoxy-2'-fluoarabinonucleoside analogues
AU7558491A (en) * 1990-04-04 1991-10-30 Nycomed Imaging As Nucleoside derivatives
WO1992011276A1 (en) * 1990-12-18 1992-07-09 Sloan-Kettering Institute For Cancer Research Novel synthesis of 2'-'up' fluorinated 2''-deoxy-arabinofuranosylpurines

Also Published As

Publication number Publication date
CA2318277A1 (en) 1999-08-05
EP1052265A4 (de) 2002-10-16
WO1999038879A1 (fr) 1999-08-05
DE69928772D1 (de) 2006-01-12
EP1052265B1 (de) 2005-12-07
JPH11217396A (ja) 1999-08-10
EP1052265A1 (de) 2000-11-15

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Legal Events

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