ATE263163T1 - Krytallinischer fungizider polymorph - Google Patents

Krytallinischer fungizider polymorph

Info

Publication number: ATE263163T1
Authority: AT; Austria
Prior art keywords: polymorphous; fungicidal; crystalline; fungicidal polymorphous; crystalline fungicidal
Prior art date: 1997-10-07

Application number

AT98951994T

Other languages

English (en)

Inventor

David R Andrews

William Leong

Anantha R Sudhakar

Original Assignee

Schering Corp

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

1997-10-07

Filing date

1998-10-05

Publication date

2004-04-15

1998-10-05 Application filed by Schering Corp filed Critical Schering Corp

2004-04-15 Application granted granted Critical

2004-04-15 Publication of ATE263163T1 publication Critical patent/ATE263163T1/de

Classifications

- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D405/00—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom
- C07D405/14—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing three or more hetero rings
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
- A61P31/10—Antimycotics

Landscapes

Chemical & Material Sciences (AREA)
Organic Chemistry (AREA)
Health & Medical Sciences (AREA)
Chemical Kinetics & Catalysis (AREA)
Life Sciences & Earth Sciences (AREA)
General Chemical & Material Sciences (AREA)
Medicinal Chemistry (AREA)
Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
Communicable Diseases (AREA)
Pharmacology & Pharmacy (AREA)
Oncology (AREA)
Animal Behavior & Ethology (AREA)
General Health & Medical Sciences (AREA)
Public Health (AREA)
Veterinary Medicine (AREA)
Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Plural Heterocyclic Compounds (AREA)
Agricultural Chemicals And Associated Chemicals (AREA)
Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)

AT98951994T 1997-10-07 1998-10-05 Krytallinischer fungizider polymorph ATE263163T1 (de)

Applications Claiming Priority (2)

Application Number	Priority Date	Filing Date	Title
US94618397A	1997-10-07	1997-10-07
PCT/US1998/020476 WO1999018097A1 (en)	1997-10-07	1998-10-05	Crystalline antifungal polymorph

Publications (1)

Publication Number	Publication Date
ATE263163T1 true ATE263163T1 (de)	2004-04-15

Family

ID=25484068

Family Applications (1)

Application Number	Title	Priority Date	Filing Date
AT98951994T ATE263163T1 (de)	1997-10-07	1998-10-05	Krytallinischer fungizider polymorph

Country Status (31)

Country	Link
EP (1)	EP1021439B1 (de)
JP (4)	JP2001519346A (de)
KR (1)	KR100626109B1 (de)
CN (1)	CN1125067C (de)
AR (1)	AR015947A1 (de)
AT (1)	ATE263163T1 (de)
AU (1)	AU759982B2 (de)
BR (1)	BR9812866A (de)
CA (1)	CA2305803C (de)
CO (1)	CO4970829A1 (de)
CZ (1)	CZ299835B6 (de)
DE (1)	DE69822859T2 (de)
DK (1)	DK1021439T3 (de)
ES (1)	ES2217594T3 (de)
HK (1)	HK1029588A1 (de)
HU (1)	HU225233B1 (de)
ID (1)	ID29290A (de)
IL (1)	IL135331A (de)
IN (1)	IN1998CH02232A (de)
MX (1)	MX225999B (de)
MY (1)	MY130126A (de)
NO (1)	NO318827B1 (de)
NZ (1)	NZ503662A (de)
PE (1)	PE120499A1 (de)
PH (1)	PH11998002606B1 (de)
PL (1)	PL189317B1 (de)
PT (1)	PT1021439E (de)
SK (1)	SK285190B6 (de)
TW (1)	TW589310B (de)
WO (1)	WO1999018097A1 (de)
ZA (1)	ZA989063B (de)

Families Citing this family (27)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
EP2130540A1 (de)	2008-06-02	2009-12-09	Sandoz AG	Pharmazeutische Zusammensetzungen mit einer kristallinen Form von Posaconazol
EP2141159A1 (de)	2008-07-03	2010-01-06	Sandoz AG	Kristalline Form von Posaconazol
EP2451805A1 (de)	2009-07-09	2012-05-16	Sandoz AG	Kristalline form von posaconazol
RU2588570C2 (ru)	2010-05-19	2016-07-10	Сандоз Аг	Способ получения хиральных гидразидов
CA2798002C (en) *	2010-05-19	2019-12-03	Sandoz Ag	Process for the preparation of chiral triazolones
CN102892762B (zh)	2010-05-19	2016-04-20	桑多斯股份公司	制备泊沙康唑中间体
MX2012013331A (es)	2010-05-19	2013-02-01	Sandoz Ag	Purificacion de posaconazol y de intermediarios de posaconazol.
US9493428B2 (en)	2011-06-16	2016-11-15	Sandoz Ag	Process for the preparation of a chiral compound
EP2758385B1 (de) *	2011-09-19	2018-03-28	MSN Laboratories Limited	Verfahren zur herstellung von antimykotischen triazolverbindungen , zwischenprodukten davon und polymorphen davon
WO2015011224A1 (en) *	2013-07-25	2015-01-29	Sandoz Ag	Improved process for the preparation of crystalline form iv of posaconazole
ITMI20132114A1 (it)	2013-12-18	2015-06-19	Djada Pharmaceutical Sa	Una forma cristallina di posaconazolo
ITMI20132118A1 (it) *	2013-12-18	2015-06-19	Djada Pharmaceutical Sa	Una forma cristallina di posaconazolo
ITMI20132115A1 (it) *	2013-12-18	2015-06-19	Djada Pharmaceutical Sa	Una forma cristallina di posaconazolo
ITMI20132117A1 (it) *	2013-12-18	2015-06-19	Djada Pharmaceutical Sa	Una forma cristallina di posaconazolo
MX2017005120A (es)	2014-10-21	2018-02-12	Ariad Pharma Inc	Formas cristalinas de 5-cloro-n4-[-2-(dimetilfosforil) fenil]-n2-{2-metoxi-4-[4-(4-metilpiperazin-1-il)piperidin-1-il] pirimidin-2,4-diamina.
CN104387374A (zh) *	2014-10-21	2015-03-04	江苏恒盛药业有限公司	泊沙康唑晶型i的制备工艺
CN104370894A (zh) *	2014-10-21	2015-02-25	江苏恒盛药业有限公司	无定型泊沙康唑的制备工艺
WO2017025292A1 (en)	2015-08-08	2017-02-16	Alfred E. Tiefenbacher (Gmbh & Co. Kg)	Gastro-resistant formulation containing posaconazole
US10836745B2 (en)	2015-12-24	2020-11-17	Takeda Pharmaceutical Company Limited	Cocrystal, production method thereof, and medicament containing cocrystal
EP4424308A3 (de)	2016-02-26	2024-12-04	Alfred E. Tiefenbacher (GmbH & Co. KG)	Magenresistente formulierung mit posaconazol und einem polymeren fällungshemmer
CN105949278B (zh) *	2016-03-30	2019-12-06	南京曼杰生物科技有限公司	一种取代的四氢呋喃水溶性衍生物及其应用
WO2017032908A1 (en)	2016-07-08	2017-03-02	Synthon B.V.	Pharmaceutical composition comprising amorphous posaconazole
TR201620462A2 (tr)	2016-12-31	2018-07-23	Abdi Ibrahim Ilac Sanayi Ve Ticaret Anonim Sirketi	POSAKONAZOL İÇEREN FARMASÖTİK BİLEŞİMLER ve ÜRETİM YÖNTEMİ
TR201722493A2 (tr)	2017-12-28	2019-07-22	Sanovel Ilac Sanayi Ve Ticaret Anonim Sirketi	Posakonazol i̇çeren kati farmasöti̇k kompozi̇syon
WO2022034232A1 (en)	2020-08-13	2022-02-17	Alfred E. Tiefenbacher (Gmbh & Co. Kg)	Gastro-resistant high-strength formulation containing posaconazole
WO2023012378A1 (en)	2021-11-25	2023-02-09	Alfred E. Tiefenbacher (Gmbh Und Co. Kg)	Granules containing posaconazole
EP4091604B1 (de)	2021-11-25	2024-04-03	Alfred E. Tiefenbacher (GmbH & Co. KG)	Posaconazol-haltige granulate

Family Cites Families (5)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
IL103558A0 (en) *	1991-10-30	1993-03-15	Schering Corp	Tri-substituted tetrahydrofuran antifungals
ATE204875T1 (de) *	1993-12-21	2001-09-15	Schering Corp	Fungizide tetrahydrofurane
ATE186540T1 (de) *	1994-01-24	1999-11-15	Janssen Pharmaceutica Nv	Wasserlösliche azol-antifungus
US5625064A (en) *	1995-04-19	1997-04-29	Schering Corporation	Process for the preparation of triazolones
WO1996038443A1 (en) *	1995-06-02	1996-12-05	Schering Corporation	Tetrahydrofuran antifungals

1998
- 1998-10-05 DE DE69822859T patent/DE69822859T2/de not_active Expired - Lifetime
- 1998-10-05 CZ CZ20001264A patent/CZ299835B6/cs not_active IP Right Cessation
- 1998-10-05 PT PT98951994T patent/PT1021439E/pt unknown
- 1998-10-05 AU AU97803/98A patent/AU759982B2/en not_active Expired
- 1998-10-05 ZA ZA989063A patent/ZA989063B/xx unknown
- 1998-10-05 AR ARP980104957A patent/AR015947A1/es not_active Application Discontinuation
- 1998-10-05 IL IL13533198A patent/IL135331A/xx not_active IP Right Cessation
- 1998-10-05 HU HU0004899A patent/HU225233B1/hu unknown
- 1998-10-05 PL PL98339659A patent/PL189317B1/pl unknown
- 1998-10-05 CN CN98811886A patent/CN1125067C/zh not_active Expired - Lifetime
- 1998-10-05 CA CA002305803A patent/CA2305803C/en not_active Expired - Lifetime
- 1998-10-05 WO PCT/US1998/020476 patent/WO1999018097A1/en active IP Right Grant
- 1998-10-05 PE PE1998000942A patent/PE120499A1/es not_active IP Right Cessation
- 1998-10-05 NZ NZ503662A patent/NZ503662A/xx not_active IP Right Cessation
- 1998-10-05 BR BR9812866-3A patent/BR9812866A/pt not_active Application Discontinuation
- 1998-10-05 EP EP98951994A patent/EP1021439B1/de not_active Expired - Lifetime
- 1998-10-05 ID IDW20000632A patent/ID29290A/id unknown
- 1998-10-05 DK DK98951994T patent/DK1021439T3/da active
- 1998-10-05 SK SK512-2000A patent/SK285190B6/sk not_active IP Right Cessation
- 1998-10-05 JP JP2000514908A patent/JP2001519346A/ja not_active Withdrawn
- 1998-10-05 AT AT98951994T patent/ATE263163T1/de active
- 1998-10-05 KR KR20007003709A patent/KR100626109B1/ko not_active Expired - Lifetime
- 1998-10-05 ES ES98951994T patent/ES2217594T3/es not_active Expired - Lifetime
- 1998-10-05 CO CO98057733A patent/CO4970829A1/es unknown
- 1998-10-06 PH PH11998002606A patent/PH11998002606B1/en unknown
- 1998-10-06 TW TW087116562A patent/TW589310B/zh not_active IP Right Cessation
- 1998-10-06 MY MYPI98004576A patent/MY130126A/en unknown
- 1998-10-06 IN IN2232CH1998 patent/IN1998CH02232A/en unknown
2000
- 2000-04-06 NO NO20001779A patent/NO318827B1/no not_active IP Right Cessation
- 2000-04-06 MX MXPA00003404 patent/MX225999B/es active IP Right Grant
2001
- 2001-01-13 HK HK01100382A patent/HK1029588A1/xx not_active IP Right Cessation
2008
- 2008-01-04 JP JP2008000110A patent/JP2008106075A/ja not_active Withdrawn
2012
- 2012-05-18 JP JP2012114725A patent/JP2012153730A/ja active Pending
- 2012-05-18 JP JP2012114724A patent/JP2012153729A/ja active Pending

Also Published As

Publication number	Publication date
ID29290A (id)	2001-08-16
ZA989063B (en)	1999-04-06
PT1021439E (pt)	2004-07-30
SK285190B6 (sk)	2006-08-03
CZ299835B6 (cs)	2008-12-10
CN1281449A (zh)	2001-01-24
MY130126A (en)	2007-06-29
EP1021439A1 (de)	2000-07-26
SK5122000A3 (en)	2000-09-12
IL135331A (en)	2005-08-31
PL339659A1 (en)	2001-01-02
CA2305803A1 (en)	1999-04-15
CO4970829A1 (es)	2000-11-07
IL135331A0 (en)	2001-05-20
DE69822859T2 (de)	2005-01-27
MXPA00003404A (es)	2000-11-01
AU9780398A (en)	1999-04-27
JP2012153729A (ja)	2012-08-16
CZ20001264A3 (cs)	2000-08-16
HU225233B1 (en)	2006-08-28
NO20001779L (no)	2000-06-06
BR9812866A (pt)	2000-08-08
CN1125067C (zh)	2003-10-22
ES2217594T3 (es)	2004-11-01
TW589310B (en)	2004-06-01
PE120499A1 (es)	1999-12-04
HK1029588A1 (en)	2001-04-06
DK1021439T3 (da)	2004-05-10
JP2008106075A (ja)	2008-05-08
WO1999018097A1 (en)	1999-04-15
AU759982B2 (en)	2003-05-01
MX225999B (es)	2005-02-02
EP1021439B1 (de)	2004-03-31
HUP0004899A2 (hu)	2002-02-28
HUP0004899A3 (en)	2002-03-28
JP2012153730A (ja)	2012-08-16
DE69822859D1 (de)	2004-05-06
PH11998002606B1 (en)	2006-08-10
AR015947A1 (es)	2001-05-30
CA2305803C (en)	2009-12-22
JP2001519346A (ja)	2001-10-23
NO20001779D0 (no)	2000-04-06
KR20010030959A (ko)	2001-04-16
NO318827B1 (no)	2005-05-09
NZ503662A (en)	2002-10-25
PL189317B1 (pl)	2005-07-29
KR100626109B1 (ko)	2006-09-20
IN1998CH02232A (de)	2005-03-04

Publication	Publication Date	Title
ATE263163T1 (de)	2004-04-15	Krytallinischer fungizider polymorph
EE200000437A (et)	2001-06-15	Tselekoksiibiühendid
ID20744A (id)	1999-02-25	Senyawa 2-metoksibenzopenona untuk fungisida
LTC1124961I2 (lt)	2022-03-25	Trombopoetino junginiai
ATE229954T1 (de)	2003-01-15	Betacarbolinverbindungen
ID28266A (id)	2001-05-10	Senyawa-senyawa amidin
PT926158E (pt)	2003-11-28	Hormona paratiroide cristalina
IS5807A (is)	2001-01-12	Þíóbensimídasólafleiður
DE69934788D1 (de)	2007-02-22	Biozide benzylbiphenylderivative
NO20011745L (no)	2001-06-06	Forbindelser
EE200100135A (et)	2002-06-17	EtO2C-CH2-(R)Cgl-Aze-Pab-OH kristalsed vormid
NO20020030L (no)	2002-03-05	Krystallinske 1-metylkarbapenemforbindelser
NO20005006L (no)	2000-10-04	Kalsilytiske forbindelser
NO20006255L (no)	2001-02-12	Krystallinsk efavirenz
NO20006662D0 (no)	2000-12-27	Fluorfenylresin-forbindelser
DE69824331D1 (de)	2004-07-15	Fungizide Zusammensetzung
DK0967869T3 (da)	2003-07-14	Fungicidblandinger
DE59906388D1 (de)	2003-08-28	Fungizide Mischungen
ATE250341T1 (de)	2003-10-15	Fungizide mischungen
DK1224179T3 (da)	2004-10-25	Natrium-hydrogen-udbytter type 1-inhibitorkrystaller
IDP000021790A (id)	1999-07-29	Senyawa-senyawa pirolum tersubstitusi
IDP000021799A (id)	1999-07-29	Senyawa-senyawa pirolum tersubstitusi
SE9800626D0 (sv)	1998-02-27	Compounds
SE9804494D0 (sv)	1998-12-22	Novel compounds
SE9804493D0 (sv)	1998-12-22	Novel compounds

Legal Events

Date	Code	Title	Description
2004-12-15	UEP	Publication of translation of european patent specification	Ref document number: 1021439 Country of ref document: EP

Date

Code

Title

Description

2004-12-15

UEP

Publication of translation of european patent specification

Ref document number: 1021439

Country of ref document: EP