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ATE191711T1 - Neue selektive inhibitoren viraler oder bakterieller neuraminidasen - Google Patents

Neue selektive inhibitoren viraler oder bakterieller neuraminidasen

Info

Publication number
ATE191711T1
ATE191711T1 AT96912404T AT96912404T ATE191711T1 AT E191711 T1 ATE191711 T1 AT E191711T1 AT 96912404 T AT96912404 T AT 96912404T AT 96912404 T AT96912404 T AT 96912404T AT E191711 T1 ATE191711 T1 AT E191711T1
Authority
AT
Austria
Prior art keywords
viral
selective inhibitors
neuraminidase
compounds
new selective
Prior art date
Application number
AT96912404T
Other languages
English (en)
Inventor
Norbert W Bischofberger
Choung U Kim
Willard Lew
Hongtao Liu
Matthew A Williams
Original Assignee
Gilead Sciences Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=27410155&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=ATE191711(T1) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Priority claimed from US08/476,946 external-priority patent/US5866601A/en
Application filed by Gilead Sciences Inc filed Critical Gilead Sciences Inc
Application granted granted Critical
Publication of ATE191711T1 publication Critical patent/ATE191711T1/de

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D309/00—Heterocyclic compounds containing six-membered rings having one oxygen atom as the only ring hetero atom, not condensed with other rings
    • C07D309/16—Heterocyclic compounds containing six-membered rings having one oxygen atom as the only ring hetero atom, not condensed with other rings having one double bond between ring members or between a ring member and a non-ring member
    • C07D309/28—Heterocyclic compounds containing six-membered rings having one oxygen atom as the only ring hetero atom, not condensed with other rings having one double bond between ring members or between a ring member and a non-ring member with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04—Antibacterial agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/12—Antivirals
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/12—Antivirals
    • A61P31/14—Antivirals for RNA viruses
    • A61P31/16—Antivirals for RNA viruses for influenza or rhinoviruses
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • Y—GENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
    • Y02—TECHNOLOGIES OR APPLICATIONS FOR MITIGATION OR ADAPTATION AGAINST CLIMATE CHANGE
    • Y02P—CLIMATE CHANGE MITIGATION TECHNOLOGIES IN THE PRODUCTION OR PROCESSING OF GOODS
    • Y02P20/00—Technologies relating to chemical industry
    • Y02P20/50—Improvements relating to the production of bulk chemicals
    • Y02P20/55—Design of synthesis routes, e.g. reducing the use of auxiliary or protecting groups

Landscapes

  • Chemical & Material Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • Organic Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Virology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Oncology (AREA)
  • Communicable Diseases (AREA)
  • Engineering & Computer Science (AREA)
  • Pulmonology (AREA)
  • Molecular Biology (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Saccharide Compounds (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Measuring Or Testing Involving Enzymes Or Micro-Organisms (AREA)
  • Epoxy Compounds (AREA)
  • Heterocyclic Compounds That Contain Two Or More Ring Oxygen Atoms (AREA)
  • Pyrane Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Pyrrole Compounds (AREA)
  • Thiazole And Isothizaole Compounds (AREA)
  • Pyridine Compounds (AREA)
  • Polyesters Or Polycarbonates (AREA)
  • Preparation Of Compounds By Using Micro-Organisms (AREA)
AT96912404T 1995-02-27 1996-02-26 Neue selektive inhibitoren viraler oder bakterieller neuraminidasen ATE191711T1 (de)

Applications Claiming Priority (4)

Application Number Priority Date Filing Date Title
US39524595A 1995-02-27 1995-02-27
US08/476,946 US5866601A (en) 1995-02-27 1995-06-06 Carbocyclic compounds
US58056795A 1995-12-29 1995-12-29
PCT/US1996/002882 WO1996026933A1 (en) 1995-02-27 1996-02-26 Novel selective inhibitors of viral or bacterial neuraminidases

Publications (1)

Publication Number Publication Date
ATE191711T1 true ATE191711T1 (de) 2000-04-15

Family

ID=27410155

Family Applications (2)

Application Number Title Priority Date Filing Date
AT99117934T ATE305453T1 (de) 1995-02-27 1996-02-26 Selektive inhibitoren viraler oder bakterieller neuraminidase
AT96912404T ATE191711T1 (de) 1995-02-27 1996-02-26 Neue selektive inhibitoren viraler oder bakterieller neuraminidasen

Family Applications Before (1)

Application Number Title Priority Date Filing Date
AT99117934T ATE305453T1 (de) 1995-02-27 1996-02-26 Selektive inhibitoren viraler oder bakterieller neuraminidase

Country Status (27)

Country Link
US (3) US5952375A (de)
EP (1) EP0759917B1 (de)
JP (3) JP3300365B2 (de)
KR (1) KR100447096B1 (de)
CN (2) CN1185223C (de)
AT (2) ATE305453T1 (de)
AU (1) AU720933B2 (de)
BR (2) BR9607098B8 (de)
CZ (1) CZ297945B6 (de)
DE (4) DE69607704T2 (de)
DK (1) DK0759917T3 (de)
ES (2) ES2249863T3 (de)
GR (1) GR3033914T3 (de)
HK (1) HK1026893A1 (de)
HU (1) HU228450B1 (de)
LU (1) LU90991I2 (de)
MX (1) MX9706496A (de)
NL (1) NL300105I2 (de)
NO (1) NO318455B1 (de)
NZ (1) NZ306625A (de)
PL (1) PL194173B1 (de)
PT (1) PT759917E (de)
RU (1) RU2181357C2 (de)
SG (1) SG45864A1 (de)
SI (1) SI9620042A (de)
UA (1) UA56128C2 (de)
WO (1) WO1996026933A1 (de)

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PT759917E (pt) 2000-10-31
WO1996026933A1 (en) 1996-09-06
AU720933B2 (en) 2000-06-15
EP0759917B1 (de) 2000-04-12
NZ306625A (en) 2001-04-27
CZ297945B6 (cs) 2007-05-02
NL300105I1 (nl) 2003-01-06
DK0759917T3 (da) 2000-07-31
NO973908D0 (no) 1997-08-26
SG45864A1 (en) 1999-04-27
NO318455B1 (no) 2005-03-21
KR100447096B1 (ko) 2005-10-11
UA56128C2 (uk) 2003-05-15
DE10299052I1 (de) 2003-05-22
HUP9800026A2 (hu) 1999-09-28
KR19980703600A (ko) 1998-12-05
GR3033914T3 (en) 2000-11-30
DE69607704T2 (de) 2000-12-28
MX9706496A (es) 1997-11-29
PL322000A1 (en) 1998-01-05
CZ269097A3 (en) 1997-11-12
US5952375A (en) 1999-09-14
US20050176758A1 (en) 2005-08-11
DE69635231T2 (de) 2006-07-13
RU2181357C2 (ru) 2002-04-20
JP4234917B2 (ja) 2009-03-04
HU228450B1 (en) 2013-03-28
SI9620042A (sl) 1998-12-31
NO973908L (no) 1997-10-27
JP2006036770A (ja) 2006-02-09
LU90991I2 (fr) 2003-02-11
HK1026893A1 (en) 2000-12-29
CN1147813A (zh) 1997-04-16
CN1347693A (zh) 2002-05-08
CN100409844C (zh) 2008-08-13
DE69607704D1 (de) 2000-05-18
EP0759917A1 (de) 1997-03-05
JP2002161074A (ja) 2002-06-04
DE759917T1 (de) 1998-10-22
ATE305453T1 (de) 2005-10-15
US6225341B1 (en) 2001-05-01
ES2118674T3 (es) 2000-08-16
BR9607098B8 (pt) 2014-11-18
CN1185223C (zh) 2005-01-19
HUP9800026A3 (en) 2002-04-29
BR9607098A (pt) 1997-11-04
NL300105I2 (nl) 2003-02-03
ES2249863T3 (es) 2006-04-01
JPH11501908A (ja) 1999-02-16
DE69635231D1 (de) 2006-02-09
JP3300365B2 (ja) 2002-07-08
AU5357196A (en) 1996-09-18
PL194173B1 (pl) 2007-05-31
ES2118674T1 (es) 1998-10-01

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