ATE185348T1 - Glykosidierungsverfahren - Google Patents

Glykosidierungsverfahren

Info

Publication number: ATE185348T1
Authority: AT; Austria
Prior art keywords: steroidal; activity; pyranoside; glycosylated; steroid
Prior art date: 1991-07-22

Application number

AT92917211T

Other languages

English (en)

Inventor

R Erich Klemke

Masata Koreeda

Original Assignee

Harrier Inc

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

1991-07-22

Filing date

1992-07-21

Publication date

1999-10-15

1992-07-21 Application filed by Harrier Inc filed Critical Harrier Inc

1999-10-15 Application granted granted Critical

1999-10-15 Publication of ATE185348T1 publication Critical patent/ATE185348T1/de

Links

238000000034 method Methods 0.000 title abstract 2
238000005858 glycosidation reaction Methods 0.000 title 1
230000000694 effects Effects 0.000 abstract 4
HVYWMOMLDIMFJA-DPAQBDIFSA-N cholesterol Chemical compound C1C=C2C[C@@H](O)CC[C@]2(C)[C@@H]2[C@@H]1[C@@H]1CC[C@H]([C@H](C)CCCC(C)C)[C@@]1(C)CC2 HVYWMOMLDIMFJA-DPAQBDIFSA-N 0.000 abstract 2
230000000144 pharmacologic effect Effects 0.000 abstract 2
229930002534 steroid glycoside Natural products 0.000 abstract 2
150000008143 steroidal glycosides Chemical class 0.000 abstract 2
230000003637 steroidlike Effects 0.000 abstract 2
150000003431 steroids Chemical class 0.000 abstract 2
DKVBOUDTNWVDEP-NJCHZNEYSA-N teicoplanin aglycone Chemical class N([C@H](C(N[C@@H](C1=CC(O)=CC(O)=C1C=1C(O)=CC=C2C=1)C(O)=O)=O)[C@H](O)C1=CC=C(C(=C1)Cl)OC=1C=C3C=C(C=1O)OC1=CC=C(C=C1Cl)C[C@H](C(=O)N1)NC([C@H](N)C=4C=C(O5)C(O)=CC=4)=O)C(=O)[C@@H]2NC(=O)[C@@H]3NC(=O)[C@@H]1C1=CC5=CC(O)=C1 DKVBOUDTNWVDEP-NJCHZNEYSA-N 0.000 abstract 2
230000003110 anti-inflammatory effect Effects 0.000 abstract 1
125000003178 carboxy group Chemical group [H]OC(*)=O 0.000 abstract 1
239000007809 chemical reaction catalyst Substances 0.000 abstract 1
235000012000 cholesterol Nutrition 0.000 abstract 1
FSMCJUNYLQOAIM-UQBZCTSOSA-N cholesteryl beta-D-glucoside Chemical compound O([C@@H]1CC2=CC[C@H]3[C@@H]4CC[C@@H]([C@]4(CC[C@@H]3[C@@]2(C)CC1)C)[C@H](C)CCCC(C)C)[C@@H]1O[C@H](CO)[C@@H](O)[C@H](O)[C@H]1O FSMCJUNYLQOAIM-UQBZCTSOSA-N 0.000 abstract 1
125000000524 functional group Chemical group 0.000 abstract 1
229930182470 glycoside Natural products 0.000 abstract 1
150000002338 glycosides Chemical class 0.000 abstract 1
230000013595 glycosylation Effects 0.000 abstract 1
238000006206 glycosylation reaction Methods 0.000 abstract 1
229910052736 halogen Inorganic materials 0.000 abstract 1
150000002367 halogens Chemical class 0.000 abstract 1
230000004957 immunoregulator effect Effects 0.000 abstract 1
230000001506 immunosuppresive effect Effects 0.000 abstract 1
238000001727 in vivo Methods 0.000 abstract 1
230000003211 malignant effect Effects 0.000 abstract 1
RYVMUASDIZQXAA-UHFFFAOYSA-N pyranoside Natural products O1C2(OCC(C)C(OC3C(C(O)C(O)C(CO)O3)O)C2)C(C)C(C2(CCC3C4(C)CC5O)C)C1CC2C3CC=C4CC5OC(C(C1O)O)OC(CO)C1OC(C1OC2C(C(OC3C(C(O)C(O)C(CO)O3)O)C(O)C(CO)O2)O)OC(CO)C(O)C1OC1OCC(O)C(O)C1O RYVMUASDIZQXAA-UHFFFAOYSA-N 0.000 abstract 1
230000004936 stimulating effect Effects 0.000 abstract 1

Classifications

- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07H—SUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
- C07H15/00—Compounds containing hydrocarbon or substituted hydrocarbon radicals directly attached to hetero atoms of saccharide radicals
- C07H15/20—Carbocyclic rings
- C07H15/24—Condensed ring systems having three or more rings
- C07H15/256—Polyterpene radicals
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P35/00—Antineoplastic agents
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P35/00—Antineoplastic agents
- A61P35/02—Antineoplastic agents specific for leukemia
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07H—SUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
- C07H17/00—Compounds containing heterocyclic radicals directly attached to hetero atoms of saccharide radicals
- C07H17/04—Heterocyclic radicals containing only oxygen as ring hetero atoms
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07J—STEROIDS
- C07J17/00—Normal steroids containing carbon, hydrogen, halogen or oxygen, having an oxygen-containing hetero ring not condensed with the cyclopenta(a)hydrophenanthrene skeleton
- C07J17/005—Glycosides
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07J—STEROIDS
- C07J9/00—Normal steroids containing carbon, hydrogen, halogen or oxygen substituted in position 17 beta by a chain of more than two carbon atoms, e.g. cholane, cholestane, coprostane
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07J—STEROIDS
- C07J9/00—Normal steroids containing carbon, hydrogen, halogen or oxygen substituted in position 17 beta by a chain of more than two carbon atoms, e.g. cholane, cholestane, coprostane
- C07J9/005—Normal steroids containing carbon, hydrogen, halogen or oxygen substituted in position 17 beta by a chain of more than two carbon atoms, e.g. cholane, cholestane, coprostane containing a carboxylic function directly attached or attached by a chain containing only carbon atoms to the cyclopenta[a]hydrophenanthrene skeleton

Landscapes

Chemical & Material Sciences (AREA)
Organic Chemistry (AREA)
Health & Medical Sciences (AREA)
General Health & Medical Sciences (AREA)
Life Sciences & Earth Sciences (AREA)
Chemical Kinetics & Catalysis (AREA)
Public Health (AREA)
Genetics & Genomics (AREA)
Molecular Biology (AREA)
Biochemistry (AREA)
Veterinary Medicine (AREA)
Biotechnology (AREA)
Engineering & Computer Science (AREA)
General Chemical & Material Sciences (AREA)
Medicinal Chemistry (AREA)
Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
Pharmacology & Pharmacy (AREA)
Animal Behavior & Ethology (AREA)
Oncology (AREA)
Hematology (AREA)
Steroid Compounds (AREA)
Saccharide Compounds (AREA)
Medicines Containing Material From Animals Or Micro-Organisms (AREA)
Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)

AT92917211T 1991-07-22 1992-07-21 Glykosidierungsverfahren ATE185348T1 (de)

Applications Claiming Priority (2)

Application Number	Priority Date	Filing Date	Title
US73391591A	1991-07-22	1991-07-22
US81569192A	1992-01-24	1992-01-24

Publications (1)

Publication Number	Publication Date
ATE185348T1 true ATE185348T1 (de)	1999-10-15

Family

ID=27112641

Family Applications (1)

Application Number	Title	Priority Date	Filing Date
AT92917211T ATE185348T1 (de)	1991-07-22	1992-07-21	Glykosidierungsverfahren

Country Status (10)

Country	Link
EP (1)	EP0597018B1 (de)
JP (1)	JPH06501499A (de)
CN (1)	CN1031643C (de)
AT (1)	ATE185348T1 (de)
AU (1)	AU2401192A (de)
CA (1)	CA2113819C (de)
DE (1)	DE69230104T2 (de)
IL (1)	IL102566A0 (de)
TW (1)	TW202455B (de)
WO (1)	WO1993001821A1 (de)

Families Citing this family (3)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
CN107056878B (zh) *	2017-03-24	2019-07-05	昆明理工大学	一个d-吡喃环孕甾烷糖苷化合物及其应用
KR102124470B1 (ko) *	2019-12-13	2020-06-18	주식회사 큐라클	신규 혈관누출 차단제의 고수율 제조방법
CN116217642A (zh) *	2023-03-09	2023-06-06	西北大学	木樨榄苷类化合物及其在制备抗肿瘤药物中的应用

Family Cites Families (3)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
FI46067C (fi) *	1968-04-06	1972-12-11	Hoechst Ag	Menetelmä digitoksigeniiniglykosidien valmistamiseksi.
US4415731A (en) *	1981-03-30	1983-11-15	Merck & Co., Inc.	Process for the preparation of methyl 2,6-dideoxy-α-D-arabino-hexopyranoside
DE4001895A1 (de) *	1990-01-23	1991-07-25	Harrier Gmbh	Herstellung von insbesondere steroidglykosiden

1992
- 1992-07-20 IL IL102566A patent/IL102566A0/xx unknown
- 1992-07-21 AU AU24011/92A patent/AU2401192A/en not_active Abandoned
- 1992-07-21 CA CA002113819A patent/CA2113819C/en not_active Expired - Fee Related
- 1992-07-21 CN CN92109745A patent/CN1031643C/zh not_active Expired - Fee Related
- 1992-07-21 DE DE69230104T patent/DE69230104T2/de not_active Expired - Fee Related
- 1992-07-21 AT AT92917211T patent/ATE185348T1/de not_active IP Right Cessation
- 1992-07-21 EP EP92917211A patent/EP0597018B1/de not_active Expired - Lifetime
- 1992-07-21 WO PCT/US1992/006063 patent/WO1993001821A1/en active IP Right Grant
- 1992-07-21 JP JP5503027A patent/JPH06501499A/ja active Pending
- 1992-08-14 TW TW081106445A patent/TW202455B/zh active

Also Published As

Publication number	Publication date
DE69230104D1 (de)	1999-11-11
AU2401192A (en)	1993-02-23
CA2113819A1 (en)	1993-02-04
CN1031643C (zh)	1996-04-24
IL102566A0 (en)	1993-01-14
CN1073179A (zh)	1993-06-16
TW202455B (de)	1993-03-21
DE69230104T2 (de)	2000-08-24
WO1993001821A1 (en)	1993-02-04
EP0597018A1 (de)	1994-05-18
EP0597018B1 (de)	1999-10-06
CA2113819C (en)	2009-01-06
EP0597018A4 (de)	1996-02-07
JPH06501499A (ja)	1994-02-17

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Legal Events

Date	Code	Title	Description
2000-04-15	RER	Ceased as to paragraph 5 lit. 3 law introducing patent treaties