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AR112265A1 - Antagonista del receptor de angiotensina ii para la prevención o tratamiento de enfermedades sistémicas en gatos - Google Patents

Antagonista del receptor de angiotensina ii para la prevención o tratamiento de enfermedades sistémicas en gatos

Info

Publication number
AR112265A1
AR112265A1 ARP180101883A AR112265A1 AR 112265 A1 AR112265 A1 AR 112265A1 AR P180101883 A ARP180101883 A AR P180101883A AR 112265 A1 AR112265 A1 AR 112265A1
Authority
AR
Argentina
Prior art keywords
treatment
sartan
angiotensin
amount
prophylaxis
Prior art date
Application number
Other languages
English (en)
Inventor
Tanja Margrit Zimmering
Anne Michelle Traas
Markus Stark
Stefan Johannes Lehner
Saskia Kley
Sven Anke
Balazs Albrecht
Original Assignee
Boehringer Ingelheim Vetmedica Gmbh
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Boehringer Ingelheim Vetmedica Gmbh filed Critical Boehringer Ingelheim Vetmedica Gmbh
Publication of AR112265A1 publication Critical patent/AR112265A1/es

Links

Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/41Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
    • A61K31/41641,3-Diazoles
    • A61K31/41781,3-Diazoles not condensed 1,3-diazoles and containing further heterocyclic rings, e.g. pilocarpine, nitrofurantoin
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/41Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
    • A61K31/41641,3-Diazoles
    • A61K31/41841,3-Diazoles condensed with carbocyclic rings, e.g. benzimidazoles
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/0012Galenical forms characterised by the site of application
    • A61K9/0053Mouth and digestive tract, i.e. intraoral and peroral administration
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00Drugs for disorders of the cardiovascular system
    • A61P9/12Antihypertensives
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/08Solutions

Landscapes

  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Epidemiology (AREA)
  • Engineering & Computer Science (AREA)
  • Cardiology (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Organic Chemistry (AREA)
  • Nutrition Science (AREA)
  • Physiology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Wood Science & Technology (AREA)
  • Zoology (AREA)

Abstract

Reivindicación 1: Un antagonista del receptor 1 de angiotensina II (AT-1) (sartan) para usar en un método para la profilaxis o tratamiento de hipertensión en un gato que necesita tal profilaxis o tratamiento, caracterizado porque el método comprende la administración de una cantidad terapéuticamente efectiva del antagonista del receptor 1 de angiotensina II (AT-1) (sartan) al gato, donde la cantidad terapéuticamente efectiva del sartan se administra en una cantidad de dosis diaria que varia durante un periodo de tratamiento, la cantidad de dosis diaria del sartan durante un primer periodo de tiempo durante el periodo de tratamiento es 1,0 a 5,0 mg/kg de peso corporal, y la cantidad de dosis diaria del sartan disminuye durante un segundo periodo de tiempo posterior al primer período de tiempo durante el periodo de tratamiento. Reivindicación 16: Un kit en partes caracterizado porque comprende: un contenedor que contiene una composición farmacéutica en una formulación líquida que comprende un antagonista del receptor de angiotensina II (AT-1) (sartan) y uno o más diluyentes y/o portadores farmacéuticamente aceptables, la cantidad de sartan que está dentro de la formulación líquida en una cantidad que es terapéuticamente efectiva para la profilaxis o el tratamiento de la hipertensión en un gato que necesita de tal tratamiento; y una jeringa que comprende un cilindro y opcionalmente tiene marcas de graduación volumétricas opcionalmente impresas en esta en incrementos de 0,25 ml o menos o en incrementos de 0,10 ml o menos.
ARP180101883 2017-07-07 2018-07-05 Antagonista del receptor de angiotensina ii para la prevención o tratamiento de enfermedades sistémicas en gatos AR112265A1 (es)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US201762529587P 2017-07-07 2017-07-07

Publications (1)

Publication Number Publication Date
AR112265A1 true AR112265A1 (es) 2019-10-09

Family

ID=62904440

Family Applications (1)

Application Number Title Priority Date Filing Date
ARP180101883 AR112265A1 (es) 2017-07-07 2018-07-05 Antagonista del receptor de angiotensina ii para la prevención o tratamiento de enfermedades sistémicas en gatos

Country Status (23)

Country Link
US (2) US10905676B2 (es)
EP (2) EP4299120A3 (es)
JP (2) JP7050893B2 (es)
KR (3) KR20250007040A (es)
CN (1) CN110785168A (es)
AR (1) AR112265A1 (es)
AU (1) AU2018295387B2 (es)
BR (1) BR112020000194A2 (es)
CA (1) CA3067918A1 (es)
DK (1) DK3648761T3 (es)
EA (1) EA202090205A1 (es)
ES (1) ES2979279T3 (es)
FI (1) FI3648761T3 (es)
HR (1) HRP20240703T1 (es)
HU (1) HUE067255T2 (es)
LT (1) LT3648761T (es)
NZ (1) NZ759782A (es)
PL (1) PL3648761T3 (es)
PT (1) PT3648761T (es)
RS (1) RS65570B1 (es)
SI (1) SI3648761T1 (es)
TW (1) TW201919703A (es)
WO (1) WO2019008077A1 (es)

Families Citing this family (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CA3142877A1 (en) 2019-07-09 2021-01-14 Boehringer Ingelheim Vetmedica Gmbh Telmisartan for the treatment of chronic kidney disease in dogs
CA3142876A1 (en) 2019-07-09 2021-01-14 Boehringer Ingelheim Vetmedica Gmbh Telmisartan for the treatment of chronic kidney disease in dogs

Family Cites Families (30)

* Cited by examiner, † Cited by third party
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JPS5671074A (en) 1979-11-12 1981-06-13 Takeda Chem Ind Ltd 1,2-disubstituted-4-halogenoimidazole-5-acetic acid derivative
CA1334092C (en) 1986-07-11 1995-01-24 David John Carini Angiotensin ii receptor blocking imidazoles
US5015651A (en) 1988-01-07 1991-05-14 E. I. Du Pont De Nemours And Company Treatment of hypertension with 1,2,4-angiotensin II antagonists
CA1338238C (en) 1988-01-07 1996-04-09 David John Carini Angiotensin ii receptor blocking imidazoles and combinations thereof with diuretics and nsaids
US4880804A (en) 1988-01-07 1989-11-14 E. I. Du Pont De Nemours And Company Angiotensin II receptor blocking benzimidazoles
IE70593B1 (en) 1989-09-29 1996-12-11 Eisai Co Ltd Biphenylmethane derivative the use of it and pharmacological compositions containing same
PH30484A (en) 1990-02-19 1997-05-28 Ciba Geigy Acy compounds pharmaceutical composition containing said compound and method of use thereof
IE910913A1 (en) 1990-03-20 1991-09-25 Sanofi Sa N-substituted heterocyclic derivates, their preparation¹and pharmaceutical compositions containing them
US5196444A (en) 1990-04-27 1993-03-23 Takeda Chemical Industries, Ltd. 1-(cyclohexyloxycarbonyloxy)ethyl 2-ethoxy-1-[[2'-(1H-tetrazol-5-yl)biphenyl-4-yl]methyl]benzimidazole-7-carboxylate and compositions and methods of pharmaceutical use thereof
IL99246A0 (en) 1990-09-10 1992-07-15 Abbott Lab Angiotensin ii receptor antagonists and pharmaceutical compositions containing them
GB9027210D0 (en) 1990-12-14 1991-02-06 Smithkline Beecham Plc Medicaments
US6028091A (en) 1990-12-14 2000-02-22 Smithkline Beecham Plc Medicament
SI9210098B (sl) 1991-02-06 2000-06-30 Dr. Karl Thomae Benzimidazoli, zdravila, ki te spojine vsebujejo, in postopek za njihovo pripravo
US5196537A (en) 1991-03-21 1993-03-23 G. D. Searle & Co. 5-apylheteroarylalkyl-1,3,5-trisubstituted-1,2,4-triazole compounds for treatment of circulatory disorders
GB9110636D0 (en) 1991-05-16 1991-07-03 Glaxo Group Ltd Chemical compounds
DE69325574T2 (de) 1992-04-13 2000-03-16 Zeneca Ltd. ANGIOTENSIN-II-ANTAGONISTEN GEGEN ERKRANKUNGEN; DIE MIT EINER EINGESCHRäNKTEN; NEURONALEN LEITUNGSGESCHWINDIGKEIT VERBUNDEN SIND, INSBESONDERE DIABETISCHE NEUROPATHIE
EP0754042A4 (en) 1994-03-29 2004-06-23 Merck & Co Inc TREATING ATHEROSCLEROSIS WITH IMIDAZOLES BLOCKING THE ANGIOTENSIN II RECEPTOR
DE19901921C2 (de) 1999-01-19 2001-01-04 Boehringer Ingelheim Pharma Polymorphe von Telmisartan, Verfahren zu deren Herstellung und deren Verwendung zur Herstellung eines Arzneimittels
US6358986B1 (en) 1999-01-19 2002-03-19 Boehringer Ingelheim Pharma Kg Polymorphs of telmisartan
DE10018401A1 (de) 2000-04-13 2001-10-25 Boehringer Ingelheim Pharma Verwendung von Bradycardica bei der Behandlung von mit Hypertrophie einhergehenden Myocarderkrankungen und neue Arzneimittelkombinationen
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DE10153737A1 (de) 2001-10-31 2003-05-28 Boehringer Ingelheim Pharma Kristallines Natriumsalz des Telmisartans, Verfahren zu dessen Herstellung und dessen Verwendung zur Herstellung eines Arzneimittels
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EP1579862A1 (en) 2004-03-25 2005-09-28 Boehringer Ingelheim Vetmedica Gmbh Use of PDE III inhibitors for the reduction of heart size in mammals suffering from heart failure
US20070026026A1 (en) 2005-08-01 2007-02-01 David Delmarre Oral liquid losartan compositions
EP1908469A1 (en) 2006-10-06 2008-04-09 Boehringer Ingelheim Vetmedica Gmbh Angiotensin II receptor antagonist for the treatment of systemic diseases in cats
CA2653011A1 (en) * 2008-12-03 2010-06-03 Apotex Technologies Inc Method and apparatus for packaging and dispensing pharmaceuticals
SG176585A1 (en) * 2009-05-20 2012-01-30 Boehringer Ingelheim Vetmed Pharmaceutical oral telmisartan solution
WO2016200694A1 (en) * 2015-06-10 2016-12-15 Hackensack University Medical Center Use of telmisartan to prevent and treat graft versus host disease and other alloimmune and autoimmune diseases
JP2019526641A (ja) 2016-09-07 2019-09-19 ソニオナ エー/エス テソフェンシン組成物

Also Published As

Publication number Publication date
PL3648761T3 (pl) 2024-07-22
KR20250007040A (ko) 2025-01-13
JP7402907B2 (ja) 2023-12-21
JP2020526516A (ja) 2020-08-31
BR112020000194A2 (pt) 2020-07-07
DK3648761T3 (da) 2024-06-24
EP3648761A1 (en) 2020-05-13
RS65570B1 (sr) 2024-06-28
AU2018295387A1 (en) 2020-01-02
EA202090205A1 (ru) 2020-06-02
HUE067255T2 (hu) 2024-10-28
TW201919703A (zh) 2019-06-01
CN110785168A (zh) 2020-02-11
SI3648761T1 (sl) 2024-07-31
CA3067918A1 (en) 2019-01-10
US20210106564A1 (en) 2021-04-15
ES2979279T3 (es) 2024-09-25
LT3648761T (lt) 2024-06-10
KR20200026975A (ko) 2020-03-11
US20190008831A1 (en) 2019-01-10
PT3648761T (pt) 2024-06-05
EP3648761B1 (en) 2024-03-13
JP7050893B2 (ja) 2022-04-08
US10905676B2 (en) 2021-02-02
AU2018295387B2 (en) 2024-02-15
NZ759782A (en) 2023-06-30
HRP20240703T1 (hr) 2024-08-16
WO2019008077A1 (en) 2019-01-10
EP4299120A2 (en) 2024-01-03
FI3648761T3 (fi) 2024-05-21
KR20230161541A (ko) 2023-11-27
JP2022075670A (ja) 2022-05-18
EP4299120A3 (en) 2024-03-06

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