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AR088808A2 - Derivados de 2h-piridazin-3-ona, composiciones farmaceuticas que los contienen y un proceso para la preparacion de dichos derivados y el uso de dichos derivados para la preparacion de una composicion farmaceutica - Google Patents

Derivados de 2h-piridazin-3-ona, composiciones farmaceuticas que los contienen y un proceso para la preparacion de dichos derivados y el uso de dichos derivados para la preparacion de una composicion farmaceutica

Info

Publication number
AR088808A2
AR088808A2 ARP120104216A ARP120104216A AR088808A2 AR 088808 A2 AR088808 A2 AR 088808A2 AR P120104216 A ARP120104216 A AR P120104216A AR P120104216 A ARP120104216 A AR P120104216A AR 088808 A2 AR088808 A2 AR 088808A2
Authority
AR
Argentina
Prior art keywords
derivatives
preparation
piridazin
ona
contain
Prior art date
Application number
ARP120104216A
Other languages
English (en)
Original Assignee
Egyt Gyogyszervegyeszeti Gyar
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Egyt Gyogyszervegyeszeti Gyar filed Critical Egyt Gyogyszervegyeszeti Gyar
Publication of AR088808A2 publication Critical patent/AR088808A2/es

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D413/00Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms
    • C07D413/14Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing three or more hetero rings
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/18Antipsychotics, i.e. neuroleptics; Drugs for mania or schizophrenia
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/22Anxiolytics
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/24Antidepressants
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00Drugs for disorders of the cardiovascular system
    • A61P9/06Antiarrhythmics

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Neurology (AREA)
  • Biomedical Technology (AREA)
  • Neurosurgery (AREA)
  • Psychiatry (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Cardiology (AREA)
  • Pain & Pain Management (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)

Abstract

Para ser usado en el tratamiento de la esquizofrenia. Reivindicación 1: Un derivado de 2H-piridazin-3-ona de la fórmula (1) caracterizado porque R representa un átomo de hidrógeno o un grupo alquilo C₁₋₄; X e Y representan, independientemente, un átomo de hidrógeno, un átomo de halógeno o un grupo de fórmula (2), donde uno de X e Y representa siempre un grupo de la fórmula (2), y el otro representa un átomo de hidrógeno o un átomo de halógeno, en el que en la fórmula (2) n tiene un valor de 1 ó 2, y sus sales ácidas de adición farmacéuticamente aceptables.
ARP120104216A 2001-07-26 2012-11-08 Derivados de 2h-piridazin-3-ona, composiciones farmaceuticas que los contienen y un proceso para la preparacion de dichos derivados y el uso de dichos derivados para la preparacion de una composicion farmaceutica AR088808A2 (es)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
HU0103063A HU225955B1 (en) 2001-07-26 2001-07-26 Novel 2h-pyridazin-3-one derivatives, process for their preparation, their use and pharmaceutical compositions containing them

Publications (1)

Publication Number Publication Date
AR088808A2 true AR088808A2 (es) 2014-07-10

Family

ID=89979562

Family Applications (2)

Application Number Title Priority Date Filing Date
ARP020102834A AR036248A1 (es) 2001-07-26 2002-07-26 Derivados de 2h-piridazin-3-ona, composiciones farmaceuticas que los contienen y un proceso para la preparacion de dichos derivados y el uso de dichos derivados para la preparacion de una composicion farmaceutica
ARP120104216A AR088808A2 (es) 2001-07-26 2012-11-08 Derivados de 2h-piridazin-3-ona, composiciones farmaceuticas que los contienen y un proceso para la preparacion de dichos derivados y el uso de dichos derivados para la preparacion de una composicion farmaceutica

Family Applications Before (1)

Application Number Title Priority Date Filing Date
ARP020102834A AR036248A1 (es) 2001-07-26 2002-07-26 Derivados de 2h-piridazin-3-ona, composiciones farmaceuticas que los contienen y un proceso para la preparacion de dichos derivados y el uso de dichos derivados para la preparacion de una composicion farmaceutica

Country Status (28)

Country Link
US (1) US7098210B2 (es)
EP (1) EP1417206B1 (es)
JP (1) JP4249012B2 (es)
KR (1) KR100909514B1 (es)
CN (1) CN1247571C (es)
AR (2) AR036248A1 (es)
AT (1) ATE466859T1 (es)
AU (1) AU2002321669B8 (es)
BR (1) BR0211440A (es)
CA (1) CA2453917C (es)
CY (1) CY1110240T1 (es)
CZ (1) CZ2004123A3 (es)
DE (1) DE60236294D1 (es)
DK (1) DK1417206T3 (es)
EA (1) EA006246B1 (es)
ES (1) ES2345541T3 (es)
HK (1) HK1067626A1 (es)
HU (1) HU225955B1 (es)
MA (1) MA27867A1 (es)
MX (1) MXPA04000814A (es)
NO (1) NO326155B1 (es)
NZ (1) NZ531154A (es)
PL (1) PL206824B1 (es)
PT (1) PT1417206E (es)
SI (1) SI1417206T1 (es)
SK (1) SK552004A3 (es)
WO (1) WO2003010166A1 (es)
ZA (1) ZA200400482B (es)

Families Citing this family (28)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
HU227255B1 (en) 2002-04-26 2010-12-28 Egis Gyogyszergyar Nyilvanosan Muekoedoe Reszvenytarsasag Novel piperidine-alkyl-amino-pyridazine derivatives, pharmaceutical compositions containing the same and process for the preparation of the active ingredient
EP1904995A4 (en) 2005-06-08 2011-01-05 Ignis Innovation Inc METHOD AND SYSTEM FOR CONTROLLING A LIGHT EMITTING DEVICE DISPLAY
US9489891B2 (en) 2006-01-09 2016-11-08 Ignis Innovation Inc. Method and system for driving an active matrix display circuit
US9269322B2 (en) 2006-01-09 2016-02-23 Ignis Innovation Inc. Method and system for driving an active matrix display circuit
WO2007079572A1 (en) 2006-01-09 2007-07-19 Ignis Innovation Inc. Method and system for driving an active matrix display circuit
HUP0600555A3 (en) * 2006-07-03 2008-10-28 Egis Gyogyszergyar Nyrt Use of 4-chloro-5-{2-[4-(6-fluoro-1,2-benz[d]izoxazol-3-yl)piperidin-1-yl]ethylamino}2-methyl-3(2h)-piridazinon for the production of pharmaceutical compositions for influencing cognitive functions and causing neuroprotective effect
US8614652B2 (en) 2008-04-18 2013-12-24 Ignis Innovation Inc. System and driving method for light emitting device display
CA2637343A1 (en) 2008-07-29 2010-01-29 Ignis Innovation Inc. Improving the display source driver
US9370075B2 (en) 2008-12-09 2016-06-14 Ignis Innovation Inc. System and method for fast compensation programming of pixels in a display
US8633873B2 (en) 2009-11-12 2014-01-21 Ignis Innovation Inc. Stable fast programming scheme for displays
CA2687631A1 (en) 2009-12-06 2011-06-06 Ignis Innovation Inc Low power driving scheme for display applications
CA2696778A1 (en) 2010-03-17 2011-09-17 Ignis Innovation Inc. Lifetime, uniformity, parameter extraction methods
US9351368B2 (en) 2013-03-08 2016-05-24 Ignis Innovation Inc. Pixel circuits for AMOLED displays
US9886899B2 (en) 2011-05-17 2018-02-06 Ignis Innovation Inc. Pixel Circuits for AMOLED displays
US20140368491A1 (en) 2013-03-08 2014-12-18 Ignis Innovation Inc. Pixel circuits for amoled displays
CN106898307B (zh) 2011-05-28 2021-04-27 伊格尼斯创新公司 在以交错模式实施的显示器上显示图像的方法
US9747834B2 (en) 2012-05-11 2017-08-29 Ignis Innovation Inc. Pixel circuits including feedback capacitors and reset capacitors, and display systems therefore
US9336717B2 (en) 2012-12-11 2016-05-10 Ignis Innovation Inc. Pixel circuits for AMOLED displays
US9786223B2 (en) 2012-12-11 2017-10-10 Ignis Innovation Inc. Pixel circuits for AMOLED displays
WO2014124755A1 (de) 2013-02-18 2014-08-21 Jürgen Von Der Ohe Verfahren und vorrichtung zum kaltstrahlreinigen
US9721505B2 (en) 2013-03-08 2017-08-01 Ignis Innovation Inc. Pixel circuits for AMOLED displays
CA2894717A1 (en) 2015-06-19 2016-12-19 Ignis Innovation Inc. Optoelectronic device characterization in array with shared sense line
CA2873476A1 (en) 2014-12-08 2016-06-08 Ignis Innovation Inc. Smart-pixel display architecture
CA2886862A1 (en) 2015-04-01 2016-10-01 Ignis Innovation Inc. Adjusting display brightness for avoiding overheating and/or accelerated aging
US10373554B2 (en) 2015-07-24 2019-08-06 Ignis Innovation Inc. Pixels and reference circuits and timing techniques
US10657895B2 (en) 2015-07-24 2020-05-19 Ignis Innovation Inc. Pixels and reference circuits and timing techniques
CA2898282A1 (en) 2015-07-24 2017-01-24 Ignis Innovation Inc. Hybrid calibration of current sources for current biased voltage progra mmed (cbvp) displays
CA2908285A1 (en) 2015-10-14 2017-04-14 Ignis Innovation Inc. Driver with multiple color pixel structure

Family Cites Families (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
IE62890B1 (en) * 1988-12-06 1995-03-08 Hafslund Nycomed Pharma New piperazinylalkyl-3(2h)-pyridazinones process for the preparation thereof and the use thereof as agents lowering blood pressure
IL117646A (en) * 1995-04-12 2000-06-01 Ferrer Int 7-¬3-¬4-(6-fluoro-1,2-benzisoxazole-3-YL)piperidin-1-YL¾propoxy¾3-alkyl-chromen-4-ones their preparation their uses and pharmaceutical compositions comprising them

Also Published As

Publication number Publication date
AR036248A1 (es) 2004-08-25
KR100909514B1 (ko) 2009-07-27
CA2453917A1 (en) 2003-02-06
US7098210B2 (en) 2006-08-29
EP1417206A1 (en) 2004-05-12
PL367447A1 (en) 2005-02-21
US20040171619A1 (en) 2004-09-02
DE60236294D1 (de) 2010-06-17
EA006246B1 (ru) 2005-10-27
JP2004538293A (ja) 2004-12-24
ES2345541T3 (es) 2010-09-27
SI1417206T1 (sl) 2010-09-30
NZ531154A (en) 2005-09-30
MA27867A1 (fr) 2006-05-02
HUP0103063A3 (en) 2005-06-28
CZ2004123A3 (cs) 2004-05-12
KR20040030862A (ko) 2004-04-09
AU2002321669B2 (en) 2008-05-15
PL206824B1 (pl) 2010-09-30
NO326155B1 (no) 2008-10-13
HU0103063D0 (en) 2001-10-28
HUP0103063A2 (hu) 2003-02-28
NO20040268L (no) 2004-03-23
AU2002321669B8 (en) 2008-06-05
EA200400223A1 (ru) 2004-12-30
CN1247571C (zh) 2006-03-29
JP4249012B2 (ja) 2009-04-02
PT1417206E (pt) 2010-07-29
CY1110240T1 (el) 2015-01-14
CA2453917C (en) 2009-06-23
CN1545513A (zh) 2004-11-10
ATE466859T1 (de) 2010-05-15
HK1067626A1 (en) 2005-04-15
HU225955B1 (en) 2008-01-28
WO2003010166A1 (en) 2003-02-06
SK552004A3 (en) 2004-08-03
MXPA04000814A (es) 2004-05-21
AU2002321669A2 (en) 2003-02-17
ZA200400482B (en) 2005-05-25
EP1417206B1 (en) 2010-05-05
BR0211440A (pt) 2004-07-20
DK1417206T3 (da) 2010-08-16

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