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AR074982A1 - Metodos para la preparacion de fungicidas - Google Patents

Metodos para la preparacion de fungicidas

Info

Publication number
AR074982A1
AR074982A1 ARP090105106A ARP090105106A AR074982A1 AR 074982 A1 AR074982 A1 AR 074982A1 AR P090105106 A ARP090105106 A AR P090105106A AR P090105106 A ARP090105106 A AR P090105106A AR 074982 A1 AR074982 A1 AR 074982A1
Authority
AR
Argentina
Prior art keywords
independently
formula
alkyl
compound
fungicides
Prior art date
Application number
ARP090105106A
Other languages
English (en)
Original Assignee
Syngenta Ltd
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Syngenta Ltd filed Critical Syngenta Ltd
Publication of AR074982A1 publication Critical patent/AR074982A1/es

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D333/00—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom
    • C07D333/02—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom not condensed with other rings
    • C07D333/04—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom not condensed with other rings not substituted on the ring sulphur atom
    • C07D333/26—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom not condensed with other rings not substituted on the ring sulphur atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D333/28—Halogen atoms
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C25/00—Compounds containing at least one halogen atom bound to a six-membered aromatic ring
    • C07C25/18—Polycyclic aromatic halogenated hydrocarbons
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C251/00—Compounds containing nitrogen atoms doubly-bound to a carbon skeleton
    • C07C251/72—Hydrazones
    • C07C251/82—Hydrazones having doubly-bound carbon atoms of hydrazone groups bound to carbon atoms of rings other than six-membered aromatic rings
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C43/00—Ethers; Compounds having groups, groups or groups
    • C07C43/02—Ethers
    • C07C43/18—Ethers having an ether-oxygen atom bound to a carbon atom of a ring other than a six-membered aromatic ring
    • C07C43/192—Ethers having an ether-oxygen atom bound to a carbon atom of a ring other than a six-membered aromatic ring containing halogen
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C49/00—Ketones; Ketenes; Dimeric ketenes; Ketonic chelates
    • C07C49/587—Unsaturated compounds containing a keto groups being part of a ring
    • C07C49/687—Unsaturated compounds containing a keto groups being part of a ring containing halogen
    • C07C49/693—Unsaturated compounds containing a keto groups being part of a ring containing halogen polycyclic
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D231/00—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings
    • C07D231/02—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings
    • C07D231/10—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
    • C07D231/14—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Low-Molecular Organic Synthesis Reactions Using Catalysts (AREA)
  • Catalysts (AREA)
  • Agricultural Chemicals And Associated Chemicals (AREA)

Abstract

Reivindicacion 1: Un método de preparacion de un compuesto de la formula (1): donde: Y es CHCHR6(R7), C=C(A)Z, CY2(R2)Y3(R3) o C=N-NR4(R5); Y2 e Y3 son, de modo independiente, O, S, N; A y Z son, de modo independiente, alquilo C1-6; R1 es CF3 o CF2H; R2 y R3 son, de modo independiente, alquilo C1-8; donde R2 y R3 se unen opcionalmente para formar un anillo de 5-8 miembros; R4 y R5 son, de modo independiente, alquilo C1-8; B es un enlace simple o un enlace doble; R6 y R7 son, de modo independiente, hidrogeno o alquilo C1-6; que comprende la etapa de hacer reaccionar un compuesto de la formula (2): donde X es F, CI, Br, 1 o un sulfonato; Y y B son como se definen para el compuesto de la formula (1); con un compuesto de la formula (3): donde R1 es como se define para el compuesto de la formula (1); en presencia de un catalizador, catalizador que comprende cobre y un ligando. Reivindicacion 15: Un compuesto de la formula (4), (5), (6), (7), (8), (9) o (10) donde Y2 e Y3 son, de modo independiente, O, S, N; R2 y R3 son, de modo independiente, alquilo C1-8, donde R2 y R3 se unen opcionalmente para formar un anillo de 5-8 miembros; R4 y R5 son, de modo independiente, alquilo C1-8; X es F, CI, Br, I o un sulfonato; excluyendo los siguientes compuestos de la formula (9); i. Y2 es O, Y3 es O, R2 es C3H7-(n), R3 es C3H7-(n); ii. Y2 es O, Y3 es O, R2 es C2H5, R3 es C2H5; iii. Y2 es O, Y3 es O, R2 y R3 son juntos -CH2-CH2-.
ARP090105106A 2008-12-24 2009-12-23 Metodos para la preparacion de fungicidas AR074982A1 (es)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US14065008P 2008-12-24 2008-12-24
EP09163256 2009-06-19

Publications (1)

Publication Number Publication Date
AR074982A1 true AR074982A1 (es) 2011-03-02

Family

ID=42286925

Family Applications (2)

Application Number Title Priority Date Filing Date
ARP090105106A AR074982A1 (es) 2008-12-24 2009-12-23 Metodos para la preparacion de fungicidas
ARP090105105A AR075498A1 (es) 2008-12-24 2009-12-23 Metodos para la preparacion de arilamidas

Family Applications After (1)

Application Number Title Priority Date Filing Date
ARP090105105A AR075498A1 (es) 2008-12-24 2009-12-23 Metodos para la preparacion de arilamidas

Country Status (10)

Country Link
US (3) US8637678B2 (es)
EP (2) EP2370412A1 (es)
JP (2) JP5727381B2 (es)
CN (2) CN102264705A (es)
AR (2) AR074982A1 (es)
BR (2) BRPI0923527A2 (es)
IL (2) IL213344A (es)
MX (2) MX2011006426A (es)
TW (2) TW201026647A (es)
WO (2) WO2010072631A1 (es)

Families Citing this family (14)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
MX2011006426A (es) * 2008-12-24 2011-07-20 Syngenta Ltd Metodos para la preparacion de arilamidas.
MX2012012009A (es) * 2010-04-20 2012-12-17 Syngenta Participations Ag Proceso para preparar amidas de acidos carboxilicos pirazolicos.
EP2560957B1 (en) * 2010-04-20 2014-05-07 Syngenta Participations AG Process for the preparation of pyrazole carboxylic acid amides
MX2012012005A (es) * 2010-04-20 2012-12-17 Syngenta Participations Ag Proceso para preparar amidas de acidos carboxilicos pirazolicos.
WO2011131546A1 (en) * 2010-04-20 2011-10-27 Syngenta Participations Ag Process for the preparation of pyrazole carboxylic acid amides
EP2632901B1 (en) * 2010-10-27 2018-09-12 Solvay Sa Process for the preparation of pyrazole-4-carboxamides
TWI534126B (zh) * 2011-01-25 2016-05-21 先正達合夥公司 用於製備吡唑羧酸醯胺之方法
GB201104203D0 (en) 2011-03-11 2011-04-27 Syngenta Ltd Chemical process
CN105047164B (zh) * 2015-08-27 2017-09-29 深圳市华星光电技术有限公司 一种灰阶调整方法及装置
CN107935930A (zh) * 2017-12-01 2018-04-20 浙江工业大学 一种1‑甲基‑3‑二氟甲基‑1h‑吡唑‑4‑酰胺衍生物及其制备方法与应用
CN111138364A (zh) * 2018-11-01 2020-05-12 东莞市东阳光菌阳氢专利农药有限公司 一种氟苯醚酰胺的制备方法
CN110922285B (zh) * 2019-12-06 2022-08-23 上海合全药业股份有限公司 一种金属催化一锅法制备芳基伯酰胺的方法
WO2023044364A1 (en) 2021-09-15 2023-03-23 Enko Chem, Inc. Protoporphyrinogen oxidase inhibitors
WO2024077487A1 (en) * 2022-10-11 2024-04-18 Syngenta Crop Protection Ag Process for the preparation of pyrazole carboxylic acid amides

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DE69618370T2 (de) 1995-04-11 2002-09-26 Mitsui Chemicals, Inc. Substituierte Thiophenderivate und diese als aktiver Bestandteil enthaltenden Fungizide für Land- und Gartenbauwirtschaft
US20020173475A1 (en) 2001-04-16 2002-11-21 Asim Dasgupta Methods to inhibit viral replication
US6759554B2 (en) 2001-04-24 2004-07-06 Massachusetts Institute Of Technology Copper-catalyzed formation of carbon-heteroatom and carbon-carbon bonds
DE10215292A1 (de) 2002-02-19 2003-08-28 Bayer Cropscience Ag Disubstitutierte Pyrazolylcarbocanilide
JP4511191B2 (ja) 2002-03-05 2010-07-28 シンジェンタ パーティシペーションズ アクチェンゲゼルシャフト Ｏ−シクロプロピル−カルボキサニリド及びそれらの殺真菌剤としての使用
AU2003255620A1 (en) * 2002-05-31 2003-12-19 Rhodia Chimie Method of forming a carbon-carbon or carbon-heteroatom linkage
US7202367B2 (en) 2002-05-31 2007-04-10 Rhodia Chimie Process for arylating or vinylating or alkynating a nucleophilic compound
GB0224316D0 (en) 2002-10-18 2002-11-27 Syngenta Participations Ag Chemical compounds
GB0319949D0 (en) * 2003-08-26 2003-09-24 Univ Strathclyde Nucleic acid sequence identification
TW200526626A (en) * 2003-09-13 2005-08-16 Astrazeneca Ab Chemical compounds
CA2562578C (en) * 2004-04-12 2013-04-02 Eisai R&D Management Co., Ltd. Process for production of pyrazole-fused ring derivatives
CA2608540A1 (en) * 2005-05-18 2006-11-23 Wyeth 3-cyanoquinoline inhibitors of tpl2 kinase and methods of making and using the same
KR101416521B1 (ko) 2005-09-02 2014-07-16 닛산 가가쿠 고교 가부시키 가이샤 이속사졸린치환 벤즈아미드 화합물 및 유해 생물 방제제
EP2253622A1 (en) * 2005-09-16 2010-11-24 Syngenta Participations AG. Process for the production of amides
EA014297B1 (ru) * 2005-10-25 2010-10-29 Зингента Партисипейшнс Аг Гетероциклические амиды, применимые в качестве микробиоцидов
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EA013108B1 (ru) * 2006-04-19 2010-02-26 Бёрингер Ингельхайм Интернациональ Гмбх Дигидротиенопиримидины для лечения воспалительных заболеваний
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DE102006033090A1 (de) * 2006-07-14 2008-01-24 Bayer Cropscience Ag Verfahren zum Herstellen von Alkylaniliden aus Halogenbenzolderivaten
CA2659971A1 (en) 2006-08-04 2008-02-07 Takeda Pharmaceutical Company Limited Fused heterocyclic derivative and use thereof
DK2848610T3 (da) 2006-11-15 2017-11-06 Ym Biosciences Australia Pty Hæmmere af kinaseaktivitet
MX2011006426A (es) * 2008-12-24 2011-07-20 Syngenta Ltd Metodos para la preparacion de arilamidas.

Also Published As

Publication number Publication date
JP2012513962A (ja) 2012-06-21
IL213351A0 (en) 2011-07-31
BRPI0923527A2 (pt) 2016-08-09
US20110263869A1 (en) 2011-10-27
EP2370412A1 (en) 2011-10-05
BRPI0923401A2 (pt) 2015-07-28
JP5727381B2 (ja) 2015-06-03
MX2011006426A (es) 2011-07-20
JP2012513961A (ja) 2012-06-21
EP2373625A1 (en) 2011-10-12
WO2010072632A1 (en) 2010-07-01
IL213344A (en) 2016-07-31
CN102300850A (zh) 2011-12-28
EP2373625B1 (en) 2014-10-08
CN102264705A (zh) 2011-11-30
US9169233B2 (en) 2015-10-27
MX2011006425A (es) 2011-07-20
US8637678B2 (en) 2014-01-28
AR075498A1 (es) 2011-04-06
US20110257410A1 (en) 2011-10-20
TW201023742A (en) 2010-07-01
WO2010072631A1 (en) 2010-07-01
BRPI0923401B1 (pt) 2021-11-23
TW201026647A (en) 2010-07-16
IL213344A0 (en) 2011-07-31
US20140107348A1 (en) 2014-04-17

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