AR018825A1 - Antagonistas del receptor de bradiquinina no peptidica para uso en el tratamiento de trastornos y enfermedades oftalmicas - Google Patents
Antagonistas del receptor de bradiquinina no peptidica para uso en el tratamiento de trastornos y enfermedades oftalmicasInfo
- Publication number
- AR018825A1 AR018825A1 ARP990101487A ARP990101487A AR018825A1 AR 018825 A1 AR018825 A1 AR 018825A1 AR P990101487 A ARP990101487 A AR P990101487A AR P990101487 A ARP990101487 A AR P990101487A AR 018825 A1 AR018825 A1 AR 018825A1
- Authority
- AR
- Argentina
- Prior art keywords
- treatment
- disorders
- bradiquinine
- antigonists
- peptidic
- Prior art date
Links
- 208000037265 diseases, disorders, signs and symptoms Diseases 0.000 title abstract 4
- 201000010099 disease Diseases 0.000 title abstract 2
- 239000000203 mixture Substances 0.000 abstract 4
- 108090000765 processed proteins & peptides Proteins 0.000 abstract 3
- 239000005557 antagonist Substances 0.000 abstract 2
- UYRCOTSOPWOSJK-JXTBTVDRSA-N bradykinin antagonist Chemical compound C1C2=CC=CC=C2CC1[C@@H](NC(=O)C(CO)NC(=O)C(NC(=O)CNC(=O)[C@H]1N(C[C@H](O)C1)C(=O)C1N(CCC1)C(=O)C(CCCNC(N)=N)NC(=O)[C@@H](CCCNC(N)=N)NC(=N)CCCCCCC(=N)N[C@H](CCCNC(N)=N)C(=O)NC(CCCNC(N)=N)C(=O)N1C(CCC1)C(=O)N1[C@@H](C[C@@H](O)C1)C(=O)NCC(=O)NC(C1CC2=CC=CC=C2C1)C(=O)NC(CO)C(=O)N[C@H](C1CC2=CC=CC=C2C1)C(=O)N1C2CCCCC2CC1C(=O)NC(CCCNC(N)=N)C(O)=O)C1CC2=CC=CC=C2C1)C(=O)N1C2CCCCC2CC1C(=O)NC(CCCNC(=N)N)C(O)=O UYRCOTSOPWOSJK-JXTBTVDRSA-N 0.000 abstract 1
- 239000003152 bradykinin antagonist Substances 0.000 abstract 1
- 208000035475 disorder Diseases 0.000 abstract 1
- 239000003814 drug Substances 0.000 abstract 1
- 238000004519 manufacturing process Methods 0.000 abstract 1
Classifications
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
- A61K31/47—Quinolines; Isoquinolines
- A61K31/4709—Non-condensed quinolines and containing further heterocyclic rings
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
- A61K31/44—Non condensed pyridines; Hydrogenated derivatives thereof
- A61K31/4427—Non condensed pyridines; Hydrogenated derivatives thereof containing further heterocyclic ring systems
- A61K31/4439—Non condensed pyridines; Hydrogenated derivatives thereof containing further heterocyclic ring systems containing a five-membered ring with nitrogen as a ring hetero atom, e.g. omeprazole
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/66—Phosphorus compounds
Landscapes
- Health & Medical Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Pharmacology & Pharmacy (AREA)
- Epidemiology (AREA)
- Life Sciences & Earth Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- General Health & Medical Sciences (AREA)
- Public Health (AREA)
- Veterinary Medicine (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
Abstract
Composiciones y uso de una composicion que comprende un antagonista de bradiquina no peptídica para la fabricacion de un medicamento para elojo o para el tratamiento de trastornos o enfermedades oftálmicas, que comprende una composicion que incluye una cantidad terapéuticamente efectivade un antagonista de bradiquinina no peptídica en un vehículo oftálmico farmacéuticamente aceptable. Las composiciones comprenden antagonistas debradiquinina no peptídica.
Applications Claiming Priority (1)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
US8000398P | 1998-04-03 | 1998-04-03 |
Publications (1)
Publication Number | Publication Date |
---|---|
AR018825A1 true AR018825A1 (es) | 2001-12-12 |
Family
ID=22154279
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
ARP990101487A AR018825A1 (es) | 1998-04-03 | 1999-03-31 | Antagonistas del receptor de bradiquinina no peptidica para uso en el tratamiento de trastornos y enfermedades oftalmicas |
Country Status (4)
Country | Link |
---|---|
US (1) | US6531480B1 (es) |
AR (1) | AR018825A1 (es) |
AU (1) | AU2985499A (es) |
WO (1) | WO1999051245A1 (es) |
Families Citing this family (3)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
AU680870B2 (en) | 1993-04-28 | 1997-08-14 | Astellas Pharma Inc. | New heterocyclic compounds |
US20070225225A1 (en) * | 2006-02-28 | 2007-09-27 | Sharif Najam A | Use of natriuretic peptide receptor antagonists to treat ocular, otic and nasal edemetous conditions |
US20080160366A1 (en) * | 2006-12-29 | 2008-07-03 | Allen Glenn M | Porous plate for a fuel cell |
Family Cites Families (3)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
FR2646773B1 (fr) | 1989-05-12 | 1994-05-13 | Chauvin Sa Laboratoire | Composition pharmaceutique a base de paracetamol |
EP0529499A1 (de) * | 1991-08-22 | 1993-03-03 | Hoechst Aktiengesellschaft | Pharmazeutische Zusammensetzungen enthaltend Bradykinin-Antagonisten zur lokalen Anwendung an Nase und Auge |
JPH10316677A (ja) * | 1997-05-19 | 1998-12-02 | Fujisawa Pharmaceut Co Ltd | 結 晶 |
-
1999
- 1999-03-04 US US09/647,640 patent/US6531480B1/en not_active Expired - Fee Related
- 1999-03-04 AU AU29854/99A patent/AU2985499A/en not_active Abandoned
- 1999-03-04 WO PCT/US1999/004866 patent/WO1999051245A1/en active Application Filing
- 1999-03-31 AR ARP990101487A patent/AR018825A1/es unknown
Also Published As
Publication number | Publication date |
---|---|
WO1999051245A1 (en) | 1999-10-14 |
US6531480B1 (en) | 2003-03-11 |
AU2985499A (en) | 1999-10-25 |
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Legal Events
Date | Code | Title | Description |
---|---|---|---|
FB | Suspension of granting procedure |