AP2006003478A0 - Muscarinic acetylcholine receptor antagonists. - Google Patents
Muscarinic acetylcholine receptor antagonists.Info
- Publication number
- AP2006003478A0 AP2006003478A0 AP2006003478A AP2006003478A AP2006003478A0 AP 2006003478 A0 AP2006003478 A0 AP 2006003478A0 AP 2006003478 A AP2006003478 A AP 2006003478A AP 2006003478 A AP2006003478 A AP 2006003478A AP 2006003478 A0 AP2006003478 A0 AP 2006003478A0
- Authority
- AP
- ARIPO
- Prior art keywords
- receptor antagonists
- acetylcholine receptor
- muscarinic acetylcholine
- muscarinic
- antagonists
- Prior art date
Links
- 229940121683 Acetylcholine receptor antagonist Drugs 0.000 title 1
- 102000014415 Muscarinic acetylcholine receptor Human genes 0.000 title 1
- 108050003473 Muscarinic acetylcholine receptor Proteins 0.000 title 1
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D451/00—Heterocyclic compounds containing 8-azabicyclo [3.2.1] octane, 9-azabicyclo [3.3.1] nonane, or 3-oxa-9-azatricyclo [3.3.1.0<2,4>] nonane ring systems, e.g. tropane or granatane alkaloids, scopolamine; Cyclic acetals thereof
- C07D451/02—Heterocyclic compounds containing 8-azabicyclo [3.2.1] octane, 9-azabicyclo [3.3.1] nonane, or 3-oxa-9-azatricyclo [3.3.1.0<2,4>] nonane ring systems, e.g. tropane or granatane alkaloids, scopolamine; Cyclic acetals thereof containing not further condensed 8-azabicyclo [3.2.1] octane or 3-oxa-9-azatricyclo [3.3.1.0<2,4>] nonane ring systems, e.g. tropane; Cyclic acetals thereof
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
- A61K31/46—8-Azabicyclo [3.2.1] octane; Derivatives thereof, e.g. atropine, cocaine
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P11/00—Drugs for disorders of the respiratory system
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P11/00—Drugs for disorders of the respiratory system
- A61P11/02—Nasal agents, e.g. decongestants
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P11/00—Drugs for disorders of the respiratory system
- A61P11/06—Antiasthmatics
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P11/00—Drugs for disorders of the respiratory system
- A61P11/08—Bronchodilators
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P37/00—Drugs for immunological or allergic disorders
- A61P37/08—Antiallergic agents
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
Landscapes
- Health & Medical Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Animal Behavior & Ethology (AREA)
- Medicinal Chemistry (AREA)
- Pharmacology & Pharmacy (AREA)
- Life Sciences & Earth Sciences (AREA)
- General Health & Medical Sciences (AREA)
- Public Health (AREA)
- Veterinary Medicine (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- General Chemical & Material Sciences (AREA)
- Engineering & Computer Science (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Pulmonology (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Epidemiology (AREA)
- Emergency Medicine (AREA)
- Immunology (AREA)
- Otolaryngology (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
- Nitrogen Condensed Heterocyclic Rings (AREA)
- Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
Applications Claiming Priority (2)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
US48798103P | 2003-07-17 | 2003-07-17 | |
PCT/US2004/022947 WO2005009439A1 (en) | 2003-07-17 | 2004-07-16 | Muscarinic acetylcholine receptor antagonists |
Publications (1)
Publication Number | Publication Date |
---|---|
AP2006003478A0 true AP2006003478A0 (en) | 2006-02-28 |
Family
ID=34102735
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
AP2006003478A AP2006003478A0 (en) | 2003-07-17 | 2004-07-16 | Muscarinic acetylcholine receptor antagonists. |
Country Status (21)
Country | Link |
---|---|
US (1) | US20060178395A1 (es) |
EP (1) | EP1648460A4 (es) |
JP (1) | JP2007523877A (es) |
KR (1) | KR20060063890A (es) |
CN (1) | CN1822838A (es) |
AP (1) | AP2006003478A0 (es) |
AR (1) | AR045913A1 (es) |
AU (1) | AU2004259232A1 (es) |
BR (1) | BRPI0412716A (es) |
CA (1) | CA2532375A1 (es) |
EA (1) | EA200600267A1 (es) |
EC (1) | ECSP056254A (es) |
IL (1) | IL172822A0 (es) |
IS (1) | IS8302A (es) |
MA (1) | MA27900A1 (es) |
MX (1) | MXPA06000662A (es) |
NO (1) | NO20060775L (es) |
PE (1) | PE20050327A1 (es) |
TW (1) | TW200523261A (es) |
UY (1) | UY28417A1 (es) |
WO (1) | WO2005009439A1 (es) |
Families Citing this family (19)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
PE20050250A1 (es) * | 2003-07-17 | 2005-04-08 | Glaxo Group Ltd | Antagonistas de los receptores muscarinicos de la acetilcolina |
PE20050963A1 (es) | 2003-10-14 | 2006-01-11 | Glaxo Group Ltd | Compuestos derivados de 8-azoniabiciclo [3.2.1]octanos como antagonistas de receptores de acetilcolina muscarinicos |
UY28567A1 (es) * | 2003-10-17 | 2005-05-31 | Glaxo Group Ltd | Antagonistas de receptores de acetilcolina muscarinicos |
PE20050489A1 (es) * | 2003-11-04 | 2005-09-02 | Glaxo Group Ltd | Antagonistas de receptores de acetilcolina muscarinicos |
WO2005087236A1 (en) * | 2004-03-11 | 2005-09-22 | Glaxo Group Limited | Novel m3 muscarinic acetylcholine receptor antagonists |
EP1725238A4 (en) * | 2004-03-17 | 2009-04-01 | Glaxo Group Ltd | ACETYLCHOLINE M 3 MUSCARINIC RECEPTOR ANTAGONISTS |
US7384946B2 (en) * | 2004-03-17 | 2008-06-10 | Glaxo Group Limited | M3 muscarinic acetylcholine receptor antagonists |
UY28871A1 (es) | 2004-04-27 | 2005-11-30 | Glaxo Group Ltd | Antagonistas del receptor de acetilcolina muscarinico |
US7598267B2 (en) * | 2004-05-13 | 2009-10-06 | Glaxo Group Limited | Muscarinic acetylcholine receptor antagonists |
EP1957075A4 (en) * | 2004-11-15 | 2009-11-18 | Glaxo Group Ltd | NOVEL ANTAGONISTS OF ACETYLCHOLINE M3 TYPE MUSCARINIC RECEPTORS |
TWI268704B (en) * | 2005-06-28 | 2006-12-11 | Realtek Semiconductor Corp | Apparatus and method for detecting vertical blanking interval |
US20080234315A1 (en) * | 2005-08-02 | 2008-09-25 | Jakob Busch-Petersen | M3 Muscarinic Acetylcholine Receptor Antagonists |
CL2009000250A1 (es) | 2008-02-06 | 2009-09-11 | Glaxo Group Ltd | Compuestos derivados de pirazolo[3,4-b]piridina carboxamida; composicion farmaceutica que los comprende; y su uso en el tratamiento del asma, epoc y rinitis. |
AR070563A1 (es) | 2008-02-06 | 2010-04-21 | Glaxo Group Ltd | Compuesto de un biciclo condensado pirazol-piridin-amina, composicion farmaceutica que lo comprende y su uso para preparar un medicamento util para el tratamiento de enfermedades respiratorias. |
PE20091553A1 (es) | 2008-02-06 | 2009-10-30 | Glaxo Group Ltd | Farmacoforos duales - antagonistas muscarinicos de pde4 |
WO2010094643A1 (en) | 2009-02-17 | 2010-08-26 | Glaxo Group Limited | Quinoline derivatives and their uses for rhinitis and urticaria |
EP2627317A4 (en) * | 2010-10-15 | 2014-08-20 | Glaxo Group Ltd | MEDICINAL FORMULATIONS FROM AGGREGATED NANOPARTICLES AND THEIR PREPARATION AND USE |
RU2666963C2 (ru) | 2012-04-13 | 2018-09-13 | Глаксосмитклайн Интеллекчуал Проперти Дивелопмент Лимитед | Агрегированные частицы |
CA3173172A1 (en) | 2020-03-26 | 2021-09-30 | Christopher D. Kane | Cathepsin inhibitors for preventing or treating viral infections |
Family Cites Families (11)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US2800481A (en) * | 1955-07-01 | 1957-07-23 | Smith Kline French Lab | Tertiary alcohol derivatives of 8-alkylnortropanes and the acid and quaternary ammonium salts thereof |
US2800482A (en) * | 1955-07-01 | 1957-07-23 | Smith Kline French Lab | Olefinic derivatives of 8-alkylnortropanes and the acid and quaternary ammonium salts thereof |
US2800478A (en) * | 1955-07-01 | 1957-07-23 | Smith Kline French Lab | 3-substituted-8-alkylnortropanes and the acid and quaternary ammonium salts thereof |
US6350758B1 (en) * | 1996-12-02 | 2002-02-26 | Georgetown University | Tropane derivatives and method for their synthesis |
US6248752B1 (en) * | 1998-02-27 | 2001-06-19 | Charles Duane Smith | Azabicyclooctane compositions and methods for enhancing chemotherapy |
US6262066B1 (en) * | 1998-07-27 | 2001-07-17 | Schering Corporation | High affinity ligands for nociceptin receptor ORL-1 |
EP1177196B1 (en) * | 1999-05-04 | 2004-03-10 | Neurosearch A/S | Heteroaryl diazabicycloalkanes, their preparation and use |
ES2165768B1 (es) * | 1999-07-14 | 2003-04-01 | Almirall Prodesfarma Sa | Nuevos derivados de quinuclidina y composiciones farmaceuticas que los contienen. |
CA2415468A1 (en) * | 2000-07-11 | 2003-01-10 | Yoshio Ogino | Ester derivatives |
CN1571787A (zh) * | 2001-10-17 | 2005-01-26 | Ucb公司 | 奎宁环衍生物、制备它们的方法和它们作为m2和/或m3毒蕈碱受体抑制剂的用途 |
JP4851937B2 (ja) * | 2003-11-21 | 2012-01-11 | セラヴァンス, インコーポレーテッド | β2アドレナリン作動性受容体作動薬活性およびムスカリン受容体拮抗薬活性を有する化合物 |
-
2004
- 2004-07-15 TW TW093121062A patent/TW200523261A/zh unknown
- 2004-07-15 PE PE2004000673A patent/PE20050327A1/es not_active Application Discontinuation
- 2004-07-15 AR ARP040102498A patent/AR045913A1/es unknown
- 2004-07-15 UY UY28417A patent/UY28417A1/es not_active Application Discontinuation
- 2004-07-16 AU AU2004259232A patent/AU2004259232A1/en not_active Abandoned
- 2004-07-16 WO PCT/US2004/022947 patent/WO2005009439A1/en active Application Filing
- 2004-07-16 BR BRPI0412716-1A patent/BRPI0412716A/pt not_active IP Right Cessation
- 2004-07-16 CN CNA2004800206494A patent/CN1822838A/zh active Pending
- 2004-07-16 CA CA002532375A patent/CA2532375A1/en not_active Abandoned
- 2004-07-16 JP JP2006520377A patent/JP2007523877A/ja not_active Withdrawn
- 2004-07-16 KR KR1020067001000A patent/KR20060063890A/ko not_active Withdrawn
- 2004-07-16 AP AP2006003478A patent/AP2006003478A0/xx unknown
- 2004-07-16 MX MXPA06000662A patent/MXPA06000662A/es unknown
- 2004-07-16 US US10/565,046 patent/US20060178395A1/en not_active Abandoned
- 2004-07-16 EA EA200600267A patent/EA200600267A1/ru unknown
- 2004-07-16 EP EP04778451A patent/EP1648460A4/en not_active Withdrawn
-
2005
- 2005-12-26 IL IL172822A patent/IL172822A0/en unknown
- 2005-12-27 EC EC2005006254A patent/ECSP056254A/es unknown
-
2006
- 2006-01-06 MA MA28704A patent/MA27900A1/fr unknown
- 2006-02-14 IS IS8302A patent/IS8302A/is unknown
- 2006-02-17 NO NO20060775A patent/NO20060775L/no not_active Application Discontinuation
Also Published As
Publication number | Publication date |
---|---|
CN1822838A (zh) | 2006-08-23 |
BRPI0412716A (pt) | 2006-09-26 |
KR20060063890A (ko) | 2006-06-12 |
TW200523261A (en) | 2005-07-16 |
AR045913A1 (es) | 2005-11-16 |
EP1648460A1 (en) | 2006-04-26 |
PE20050327A1 (es) | 2005-06-08 |
EP1648460A4 (en) | 2009-04-01 |
JP2007523877A (ja) | 2007-08-23 |
NO20060775L (no) | 2006-04-11 |
CA2532375A1 (en) | 2005-02-03 |
MA27900A1 (fr) | 2006-05-02 |
AU2004259232A1 (en) | 2005-02-03 |
IL172822A0 (en) | 2006-06-11 |
IS8302A (is) | 2006-02-14 |
ECSP056254A (es) | 2006-04-19 |
US20060178395A1 (en) | 2006-08-10 |
UY28417A1 (es) | 2005-02-28 |
EA200600267A1 (ru) | 2006-06-30 |
WO2005009439A1 (en) | 2005-02-03 |
MXPA06000662A (es) | 2006-03-30 |
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