Opposing orientations of the anti-psychotic drug trifluoperazine selected by alternate conformations of M144 in calmodulin (Q35450179)

25694384

8 August 2017

title

Opposing orientations of the anti-psychotic drug trifluoperazine selected by alternate conformations of M144 in calmodulin (English)

1 reference

8 August 2017

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3 June 2020

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https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:25694384%20AND%20SRC:MED&resulttype=core&format=json

3 June 2020

Michael D Feldkamp

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3 June 2020

Nisha Pandey

series ordinal

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3 June 2020

language of work or name

English

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publication date

25 March 2015

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8 August 2017

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inferred from page(s)

published in

Proteins

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3 June 2020

volume

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issue

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page(s)

989-996

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Fluorinated compounds in medicinal chemistry: recent applications, synthetic advances and matched-pair analyses

3 June 2020

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Ca2+-bound calmodulin forms a compact globular structure on binding four trifluoperazine molecules in solution

12 July 2018

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12 July 2018

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12 July 2018

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12 July 2018

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12 July 2018

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The energetics and dynamics of molecular recognition by calmodulin

12 July 2018

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Drug binding by calmodulin: crystal structure of a calmodulin-trifluoperazine complex

12 July 2018

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12 July 2018

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12 July 2018

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Different developmental functions for calmodulin in dictyostelium: Trifluoperazine and R24571 both inhibit cell and pronuclear fusion but enhance gamete formation*1

12 July 2018

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12 July 2018

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12 July 2018

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12 July 2018

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12 July 2018

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The treatment of schizophrenia with long-acting oral neuroleptics: a six-month double-blind investigation of penfluridol versus trifluoperazine

12 July 2018

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12 July 2018

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Oxidation of Met144 and Met145 in calmodulin blocks calmodulin dependent activation of the plasma membrane Ca-ATPase

26 September 2018

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26 September 2018

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26 September 2018

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Bacterial expression and characterization of proteins derived from the chicken calmodulin cDNA and a calmodulin processed gene

26 September 2018

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Structure of calmodulin refined at 2.2 A resolution

26 September 2018

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Crossref

https://api.crossref.org/works/10.1002%2FPROT.24781

The Trifluoromethyl Group in Medical Chemistry

21 January 2018

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Crossref

https://api.crossref.org/works/10.1002%2FPROT.24781

Quantitative endoproteinase GluC footprinting of cooperative Ca2+ binding to calmodulin: proteolytic susceptibility of E31 and E87 indicates interdomain interactions

21 January 2018

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12 December 2020

Novel interaction of the voltage-dependent sodium channel (VDSC) with calmodulin: does VDSC acquire calmodulin-mediated Ca2+-sensitivity?

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Identifiers

DOI

10.1002/PROT.24781

1 reference

https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:25694384%20AND%20SRC:MED&resulttype=core&format=json

3 June 2020

1 reference

https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:25694384%20AND%20SRC:MED&resulttype=core&format=json

3 June 2020

25694384

1 reference

https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:25694384%20AND%20SRC:MED&resulttype=core&format=json