Protean agonism at histamine H3 receptors in vitro and in vivo (Q34228615)

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7 November 2019

title

Protean agonism at histamine H3 receptors in vitro and in vivo (English)

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7 November 2019

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7 November 2019

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7 November 2019

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7 November 2019

Florence Gbahou

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7 November 2019

Agnès Rouleau

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7 November 2019

Régis Parmentier

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7 November 2019

Jian-Sheng Lin

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7 November 2019

Joël Tardivel-Lacombe

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7 November 2019

Holger Stark

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7 November 2019

Walter Schunack

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7 November 2019

C Robin Ganellin

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7 November 2019

Jean-Charles Schwartz

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7 November 2019

Jean-Michel Arrang

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7 November 2019

language of work or name

English

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publication date

5 September 2003

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7 November 2019

number of pages

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Proceedings of the National Academy of Sciences of the United States of America

inferred from page(s)

published in

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7 November 2019

volume

100

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7 November 2019

issue

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7 November 2019

page(s)

11086-11091

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Anatomical, physiological, and pharmacological characteristics of histidine decarboxylase knock-out mice: evidence for the role of brain histamine in behavioral and sleep-wake control

7 November 2019

cites work

1 reference

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Evidence for protean agonism of RX 831003 at alpha 2A-adrenoceptors by co-expression with different G alpha protein subunits

5 July 2018

1 reference

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Histamine H3-receptor-mediated [35S]GTP gamma[S] binding: evidence for constitutive activity of the recombinant and native rat and human H3 receptors.

5 July 2018

1 reference

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Inverse, protean, and ligand-selective agonism: matters of receptor conformation

5 July 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=196931

The rat H3 receptor: gene organization and multiple isoforms.

5 July 2018

1 reference

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High constitutive activity of native H3 receptors regulates histamine neurons in brain.

5 July 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=196931

Distinct pharmacology of rat and human histamine H(3) receptors: role of two amino acids in the third transmembrane domain

5 July 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=196931

Cloning and functional expression of the human histamine H3 receptor

5 July 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=196931

On the mechanism of histaminergic inhibition of glutamate release in the rat dentate gyrus

5 July 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=196931

Neurochemical and behavioral effects of ciproxifan, a potent histamine H3-receptor antagonist

5 July 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=196931

Protean effects of a natural peptide agonist of the G protein-coupled secretin receptor demonstrated by receptor mutagenesis.

5 July 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=196931

The cubic ternary complex receptor-occupancy model. III. resurrecting efficacy

5 July 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=196931

Agonist-induced modulation of inverse agonist efficacy at the beta 2-adrenergic receptor

5 July 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=196931

Constitutive activity of receptors coupled to guanine nucleotide regulatory proteins

5 July 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=196931

A mutation-induced activated state of the beta 2-adrenergic receptor. Extending the ternary complex model

5 July 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=196931

Inverse agonist activity of beta-adrenergic antagonists.

5 July 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=196931

Physiological effects of inverse agonists in transgenic mice with myocardial overexpression of the beta 2-adrenoceptor

5 July 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=196931

The two-state model of receptor activation

5 July 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=196931

Auto-inhibition of brain histamine release mediated by a novel class (H3) of histamine receptor

5 July 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=196931

Autoregulation of histamine release in brain by presynaptic H3-receptors

5 July 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=196931

Highly potent and selective ligands for histamine H3-receptors

5 July 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=196931

Antagonists with negative intrinsic activity at delta opioid receptors coupled to GTP-binding proteins

5 July 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=196931

Involvement of histaminergic neurons in arousal mechanisms demonstrated with H3-receptor ligands in the cat.

5 July 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=196931

S-[2-(4-imidazolyl)ethyl]isothiourea, a highly specific and potent histamine H3 receptor agonist

5 July 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=196931

Expression analysis of the histamine H(3) receptor in developing rat tissues

5 July 2018

1 reference

Crossref

https://api.crossref.org/works/10.1073%2FPNAS.1932276100

Histamine modulates high-voltage-activated calcium channels in neurons dissociated from the rat tuberomammillary nucleus

21 January 2018

1 reference

Crossref

https://api.crossref.org/works/10.1073%2FPNAS.1932276100

Identification of rat H3 receptor isoforms with different brain expression and signaling properties.

21 January 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=196931

Effects of histamine H3-receptor ligands on various biochemical indices of histaminergic neuron activity in rat brain

28 October 2018

1 reference

12 December 2020

[125I]iodoproxyfan, a new antagonist to label and visualize cerebral histamine H3 receptors

1 reference

12 December 2020

Inverse agonism: pharmacological curiosity or potential therapeutic strategy?

1 reference

12 December 2020

Pharmacological proteus?

1 reference

12 December 2020

Protean agonism at alpha2A-adrenoceptors

1 reference

12 December 2020

Anti-inflammatory and antinociceptive properties of BP 2-94, a histamine H(3)-receptor agonist prodrug

1 reference

12 December 2020

Identifiers

DOI

10.1073/PNAS.1932276100

1 reference

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7 November 2019

0 references

1 reference

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7 November 2019

PubMed publication ID

12960366

1 reference

https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:12960366%20AND%20SRC:MED&resulttype=core&format=json