Agonists induce conformational changes in transmembrane domains III and VI of the beta2 adrenoceptor (Q33887729)

29 July 2017

title

Agonists induce conformational changes in transmembrane domains III and VI of the beta2 adrenoceptor (English)

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29 July 2017

main subject

transmembrane protein

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B K Kobilka

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29 July 2017

U Gether

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29 July 2017

S Lin

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29 July 2017

P Ghanouni

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29 July 2017

J A Ballesteros

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29 July 2017

H Weinstein

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29 July 2017

language of work or name

English

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publication date

1 November 1997

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29 July 2017

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29 July 2017

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29 July 2017

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29 July 2017

page(s)

6737-6747

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Optimization by Simulated Annealing

29 July 2017

cites work

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5 July 2018

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5 July 2018

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5 July 2018

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5 July 2018

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5 July 2018

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5 July 2018

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5 July 2018

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5 July 2018

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5 July 2018

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5 July 2018

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5 July 2018

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Evidence for essential disulfide bonds in beta1-adrenergic receptors of turkey erythrocyte membranes. Inactivation by dithiothreitol

5 July 2018

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Structural features and light-dependent changes in the cytoplasmic interhelical E-F loop region of rhodopsin: a site-directed spin-labeling study

5 July 2018

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29 October 2018

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Mapping of the amino acids in membrane-embedded helices that interact with the retinal chromophore in bovine rhodopsin.

29 October 2018

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Modeling of G-protein coupled receptors with bacteriorhodopsin as a template. A novel approach based on interaction energy differences

29 October 2018

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12 December 2020

The high affinity state of the beta 2-adrenergic receptor requires unique interaction between conserved and non-conserved extracellular loop cysteines

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12 December 2020

Projection structure of rhodopsin

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Fluorescent labeling of purified beta 2 adrenergic receptor. Evidence for ligand-specific conformational changes

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A reciprocal mutation supports helix 2 and helix 7 proximity in the gonadotropin-releasing hormone receptor

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Signal transduction by a 5-HT2 receptor: a mechanistic hypothesis from molecular dynamics simulations of the three-dimensional model of the receptor complexed to ligands

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Requirement of rigid-body motion of transmembrane helices for light activation of rhodopsin

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Differential ergoline and ergopeptine binding to 5-hydroxytryptamine2A receptors: ergolines require an aromatic residue at position 340 for high affinity binding

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Three-dimensional structure for the β2 adrenergic receptor protein based on computer modeling studies

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Modeling of transmembrane seven helix bundles

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Molecular dynamics simulations of m3-muscarinic receptor activation and QSAR analysis

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Identifiers

DOI

10.1093/EMBOJ/16.22.6737

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29 July 2017

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29 July 2017

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