Welcome to our Ligands and Bioactive Small Molecules section, meticulously crafted for the dynamic realm of scientific services and research and development (R&D) in chemistry and life sciences. Explore our comprehensive collection of high-quality ligands and small molecules meticulously engineered to drive innovation and propel advancements across various industries. From receptor agonists and antagonists to enzyme inhibitors and modulators, our selection serves as the foundation for cutting-edge projects in drug discovery, chemical biology, and molecular pharmacology. Whether you're elucidating biological pathways, screening for potential therapeutics, or probing protein-ligand interactions, our Ligands and Bioactive Small Molecules offer versatility, reliability, and precision for your scientific services and R&D endeavors. Discover the potential of ligands and small molecules in your next breakthrough project. Small molecules, drug targets, and ligands are all key terms in the world of pharmacology and drug discovery.
Bioactive Small Molecules
- Compound Libraries
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- Metabolites
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- PROTACs, molecular glues and other degraders
- Fluorescence Imaging
- Antimalarial ligands
- Approved Ligands
- WHO
- Synthetic organic ligands
- Endogenous peptide in human, mouse or rat
- Other peptides
- Antibodies
- Labelled Ligands
- Ligands of Immunopharmacology
- Antibacterial ligands
- Sertaconazole nitrate, Cytochrome P450 51 inhibitor
Specifications & Purity: ≥98%
CAS No.: 99592-39-9
Starting at $48.90
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- Compound Libraries81item
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- Fluorescence Imaging69item
- Antimalarial ligands175item
- Approved Ligands534item
- WHO295item
- Synthetic organic ligands8526item
- Endogenous peptide in human, mouse or rat869item
- Other peptides1384item
- Antibodies613item
- Labelled Ligands78item
- Ligands of Immunopharmacology1047item
- Antibacterial ligands283item
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Antibody Type
Application
Reactive species
- Baboon1 item
- Canine1 item
- Chicken1 item
- Cotton Rat1 item
- Cow1 item
- Cynomolgus256item
- Cynomolgus monkey2item
- Dog3item
- Human567item
- Mouse164item
- Pig2item
- Rabbit16item
- Rat40item
- Respiratory syncytial virus1 item
- Rhesus Macaque35item
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- Turkey1 item
- Zaire Ebola virus3item
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Host species
Clonality
Conjugation
Tag
- 5-HT Receptor79item
- 5-HT1A receptor Agonist64item
- 5-HT1A receptor Antagonist42item
- 5-HT1B receptor Agonist47item
- 5-HT1B receptor Antagonist24item
- 5-HT1D receptor Agonist47item
- 5-HT1D receptor Antagonist21item
- 5-ht1e receptor Agonist27item
- 5-HT1F receptor Agonist25item
- 5-HT2A receptor Agonist39item
- 5-HT2A receptor Antagonist88item
- 5-HT2B receptor Agonist36item
- 5-HT2B receptor Antagonist52item
- 5-HT2C receptor Agonist33item
- 5-HT2C receptor Antagonist56item
- 5-HT3A Antagonist19item
- 5-HT4 receptor Agonist23item
- 5-HT4 receptor Antagonist18item
- 5-HT6 receptor Agonist25item
- 5-HT6 receptor Antagonist41item
- 5-HT7 receptor Agonist25item
- 5-HT7 receptor Antagonist40item
- A1 receptor Agonist31item
- A1 receptor Antagonist59item
- A2A receptor Agonist31item
- A2A receptor Antagonist60item
- A2B receptor Agonist17item
- A2B receptor Antagonist58item
- A3 receptor Agonist33item
- A3 receptor Antagonist57item
- ABL proto-oncogene 1,non-receptor tyrosine kinase Inhibitor29item
- Accession#:Q1511621item
- Acids53item
- Acyltransferase26item
- ADC Cytotoxin51item
- Adenosine Receptor31item
- Adrenergic Receptor55item
- Akt73item
- AKT serine/threonine kinase 1 Inhibitor14item
- Aldehydes53item
- ALK receptor tyrosine kinase Inhibitor25item
- alkaloid16item
- Alkaloids Other Alkaloids19item
- Ammonium salt20item
- AMPK39item
- AMY1 receptor Agonist15item
- AMY3 receptor Agonist14item
- Amyloid-β58item
- Anaplastic lymphoma kinase (ALK)17item
- Androgen Receptor63item
- Angiotensin Receptor44item
- Angiotensin-converting Enzyme (ACE)29item
- Angiotensin-converting enzyme Inhibitor31item
- Anti-infection665item
- Antibiotic16item
- Antibody-drug Conjugate/ADC Related138item
- apelin receptor Agonist29item
- Apoptosis485item
- Arenavirus16item
- Aryl Hydrocarbon Receptor18item
- AT1 receptor Antagonist33item
- Aurora Kinase18item
- aurora kinase A Inhibitor36item
- aurora kinase B Inhibitor34item
- Autophagy115item
- AXL receptor tyrosine kinase Inhibitor19item
- azole16item
- B-Raf proto-oncogene,serine/threonine kinase Inhibitor19item
- B1 receptor Agonist17item
- B1 receptor Antagonist20item
- B2 receptor Antagonist15item
- Bacterial69item
- BB1 receptor Agonist16item
- BB2 receptor Agonist19item
- BB2 receptor Antagonist23item
- BB3 receptor Agonist19item
- Bcl-2 Family74item
- beta-secretase 1 Inhibitor33item
- beta-secretase 2 Inhibitor15item
- bromodomain containing 2 Inhibitor14item
- bromodomain containing 4 Inhibitor42item
- Bruton tyrosine kinase Inhibitor51item
- Btk51item
- c-Fms28item
- c-Kit21item
- c-Met/HGFR17item
- C3a receptor Agonist14item
- C5a1 receptor Antagonist16item
- Calcium Channel61item
- Cannabinoid Receptor30item
- Carbonyl compound20item
- carboxylic acid32item
- Casein Kinase26item
- Caspase41item
- Cathepsin35item
- CB1 receptor Agonist17item
- CB1 receptor Antagonist17item
- CB2 receptor Agonist20item
- CCK1 receptor Agonist23item
- CCK1 receptor Antagonist21item
- CCK2 receptor Agonist35item
- CCK2 receptor Antagonist30item
- CCR52item
- CCR1 Agonist17item
- CCR2 Agonist17item
- CCR2 Antagonist16item
- CCR3 Agonist20item
- CCR3 Antagonist20item
- CCR5 Agonist26item
- CCR5 Antagonist20item
- CDK124item
- Cell Cycle/DNA Damage1058item
- Cell signal transduction and Neuroscience46item
- checkpoint kinase 1 Inhibitor16item
- Chemical Biology20item
- Cholinesterase (ChE)37item
- colony stimulating factor 1 receptor Inhibitor32item
- Complement System38item
- CoV 3C-like (main) protease Inhibitor67item
- COX54item
- COX-1 Inhibitor15item
- COX-2 Inhibitor26item
- CRF1 receptor Antagonist15item
- CT receptor Agonist15item
- CXCR2 Agonist22item
- CXCR3 Agonist18item
- CXCR3 Antagonist14item
- CXCR4 Agonist14item
- CXCR4 Antagonist16item
- cyclin dependent kinase 1 Inhibitor47item
- cyclin dependent kinase 2 Inhibitor48item
- cyclin dependent kinase 4 Inhibitor39item
- cyclin dependent kinase 5 Inhibitor24item
- cyclin dependent kinase 6 Inhibitor21item
- cyclin dependent kinase 9 Inhibitor30item
- Cytochrome P45082item
- Cytoskeleton228item
- D1 receptor Agonist20item
- D2 receptor Agonist33item
- D2 receptor Antagonist56item
- D3 receptor Agonist24item
- D3 receptor Antagonist36item
- D4 receptor Antagonist36item
- D5 receptor Agonist14item
- Deubiquitinase50item
- Dihydroorotate Dehydrogenase19item
- Dipeptidyl Peptidase19item
- DNA Alkylator/Crosslinker21item
- DNA Stain16item
- DNA/RNA Synthesis119item
- Dopamine Receptor78item
- DP1 receptor Agonist17item
- Drug Metabolite101item
- Drug-Linker Conjugates for ADC79item
- DYRK27item
- E1/E2/E3 Enzyme60item
- E3 Ligase Ligand-Linker Conjugates24item
- EGFR96item
- Element classified compounds36item
- Endogenous Metabolite120item
- Enterovirus20item
- EP1 receptor Agonist15item
- EP2 receptor Agonist24item
- EP3 receptor Agonist29item
- EP4 receptor Agonist27item
- EP4 receptor Antagonist17item
- epidermal growth factor receptor Inhibitor71item
- Epigenetic Reader Domain158item
- Epigenetics679item
- erb-b2 receptor tyrosine kinase 2 Inhibitor27item
- ERK55item
- Estrogen Receptor/ERR73item
- ETA receptor Antagonist21item
- Eukaryotic Initiation Factor (eIF)28item
- FAK18item
- farnesyl diphosphate synthase Inhibitor18item
- Farnesyl Transferase16item
- Fatty acid amide hydrolase Inhibitor21item
- Fatty Acid Synthase (FASN)18item
- Ferroptosis41item
- FGFR45item
- fibroblast growth factor receptor 1 Inhibitor37item
- fibroblast growth factor receptor 2 Inhibitor17item
- fibroblast growth factor receptor 3 Inhibitor20item
- fibroblast growth factor receptor 4 Inhibitor14item
- Five-Membered Heterocyclic Compounds109item
- FKBP21item
- Flavonoids Flavones Phenols Polyphenols18item
- Flavonoids Flavonols Phenols Polyphenols17item
- FLT344item
- Fluorescent Dye68item
- fms related receptor tyrosine kinase 1 Inhibitor30item
- fms related receptor tyrosine kinase 3 Inhibitor57item
- fms related receptor tyrosine kinase 4 Inhibitor30item
- FP receptor Agonist24item
- FPR1 Agonist25item
- FPR2/ALX Agonist44item
- Free Fatty Acid Receptor30item
- Functional group compounds17item
- Fungal55item
- GABA Receptor58item
- GABAA receptor α1 subunit Allosteric modulator15item
- GABAA receptor α2 subunit Allosteric modulator15item
- GABAA receptor α3 subunit Allosteric modulator14item
- GABAA receptor α5 subunit Allosteric modulator19item
- GAL1 receptor Agonist52item
- GAL2 receptor Agonist63item
- GAL3 receptor Agonist28item
- GCGR47item
- Gene ID:513321item
- geranylgeranyl diphosphate synthase Inhibitor17item
- GHRH receptor Antagonist18item
- Glucocorticoid receptor Agonist37item
- Glucosidase28item
- Glycine Receptor (All subtypes) Subunit-specific18item
- glycogen synthase kinase 3 beta Inhibitor42item
- GnRH1 receptor Agonist24item
- GnRH1 receptor Antagonist23item
- GPCR/G Protein1232item
- GPR119 Agonist36item
- GPR55 Agonist25item
- GSK-341item
- H1 receptor Antagonist64item
- H3 receptor Agonist23item
- H3 receptor Antagonist31item
- H4 receptor Agonist21item
- H4 receptor Antagonist15item
- HBV43item
- HCA2 receptor Agonist19item
- HCV86item
- HDAC66item
- HIF/HIF Prolyl-Hydroxylase48item
- Histamine Receptor46item
- Histamine receptor antagonists27item
- Histone Acetyltransferase35item
- histone deacetylase 1 Inhibitor28item
- histone deacetylase 2 Inhibitor21item
- histone deacetylase 3 Inhibitor28item
- histone deacetylase 6 Inhibitor34item
- histone deacetylase 8 Inhibitor21item
- Histone Demethylase57item
- Histone Methyltransferase104item
- HIV72item
- HSP57item
- HSV24item
- hydroxymethylglutaryl-CoA reductase Inhibitor70item
- IAP15item
- iGluR82item
- IKK16item
- Imidazoles20item
- Immunology/Inflammation724item
- Indoleamine 2,3-Dioxygenase (IDO)34item
- Influenza Virus60item
- inhibitor23item
- Integrin47item
- Interferon-α/β receptor Agonist14item
- Interleukin Related52item
- IP receptor Agonist20item
- IRAK27item
- Isotope-Labeled Compounds79item
- JAK73item
- JAK/STAT Signaling230item
- Janus kinase 1 Inhibitor52item
- Janus kinase 2 Inhibitor74item
- Janus kinase 3 Inhibitor54item
- JNK16item
- Keap1-Nrf243item
- Ketones43item
- kinase insert domain receptor Inhibitor83item
- KIT proto-oncogene,receptor tyrosine kinase Inhibitor51item
- lanosterol synthase Inhibitor16item
- LCK proto-oncogene,Src family tyrosine kinase Inhibitor26item
- leucine rich repeat kinase 2 Inhibitor25item
- Leukotriene Receptor19item
- Ligands for Target Protein for PROTAC31item
- Liposome42item
- Lipoxygenase22item
- LPA1 receptor Antagonist18item
- LPL Receptor41item
- M1 receptor Agonist28item
- M1 receptor Allosteric modulator28item
- M1 receptor Antagonist48item
- M2 receptor Agonist16item
- M2 receptor Allosteric modulator17item
- M2 receptor Antagonist51item
- M3 receptor Agonist16item
- M3 receptor Antagonist43item
- M4 receptor Agonist16item
- M4 receptor Allosteric modulator16item
- M4 receptor Antagonist47item
- M5 receptor Antagonist36item
- mAChR69item
- MAPK/ERK Pathway222item
- MCH1 receptor Antagonist23item
- MDM-2/p5350item
- mechanistic target of rapamycin kinase Inhibitor44item
- MEK23item
- Melanocortin Receptor27item
- Membrane Transporter/Ion Channel584item
- MET proto-oncogene,receptor tyrosine kinase Inhibitor39item
- Metabolic Enzyme/Protease1792item
- mGlu1 receptor Allosteric modulator61item
- mGlu2 receptor Allosteric modulator31item
- mGlu4 receptor Allosteric modulator18item
- mGlu5 receptor Allosteric modulator80item
- mGluR66item
- Microtubule/Tubulin94item
- Mitochondrial Metabolism38item
- mitogen-activated protein kinase 14 Inhibitor26item
- MMP49item
- Molecular Glues16item
- Monoamine Oxidase40item
- motilin receptor Agonist24item
- MT1 receptor Agonist29item
- MT2 receptor Agonist33item
- mTOR59item
- nAChR51item
- NAMPT16item
- Natural product15item
- NET Inhibitor29item
- Neuronal Signaling1109item
- Neuropeptide Y Receptor18item
- neurotrophic receptor tyrosine kinase 1 Inhibitor25item
- NF-κB200item
- NK1 receptor Antagonist30item
- NK2 receptor Antagonist14item
- NK3 receptor Antagonist18item
- NMU1 receptor Agonist16item
- NMU2 receptor Agonist16item
- NO Synthase31item
- NOD-like Receptor (NLR)22item
- Non heterocyclic block18item
- NOP receptor Agonist23item
- Notch19item
- NPFF2 receptor Agonist14item
- NTS1 receptor Agonist18item
- Nucleoside Antimetabolite/Analog75item
- Opioid Receptor48item
- Orexin Receptor (OX Receptor)17item
- OT receptor Antagonist34item
- Others65item
- OX1 receptor Antagonist25item
- OX2 receptor Antagonist27item
- P-glycoprotein21item
- P2X Receptor26item
- P2Y1 receptor Antagonist19item
- P2Y12 receptor Antagonist16item
- p38 MAPK56item
- PAC1 receptor Agonist15item
- PAF receptor Antagonist33item
- Parasite85item
- PARP48item
- PD-1/PD-L141item
- PD117item
- PDCD118item
- PDGFR45item
- PEG30item
- PEG derivatives28item
- Peptide Linkers54item
- Peroxisome proliferator-activated receptor-α Agonist31item
- Peroxisome proliferator-activated receptor-γ Agonist47item
- Pharmaceutical ingredients240item
- Phenols Polyphenols38item
- Phenylpropanoids61item
- Phosphatase113item
- phosphatidylinositol-4,5-bisphosphate 3-kinase catalytic subunit alpha Inhibitor76item
- phosphatidylinositol-4,5-bisphosphate 3-kinase catalytic subunit beta Inhibitor60item
- phosphatidylinositol-4,5-bisphosphate 3-kinase catalytic subunit delta Inhibitor71item
- phosphatidylinositol-4,5-bisphosphate 3-kinase catalytic subunit gamma Inhibitor68item
- Phosphodiesterase (PDE)136item
- phosphodiesterase 5A Inhibitor14item
- Phospholipase39item
- PI3K86item
- PI3K/Akt/mTOR298item
- Pim-1 proto-oncogene,serine/threonine kinase Inhibitor17item
- PKC35item
- platelet derived growth factor receptor alpha Inhibitor24item
- platelet derived growth factor receptor beta Inhibitor47item
- Potassium Channel65item
- PPAR59item
- Pregnane X receptor Agonist14item
- Prostaglandin Receptor60item
- PROTAC249item
- PROTAC Linkers35item
- PROTACs132item
- Protease Activated Receptor (PAR)27item
- Proteasome35item
- Protein Tyrosine Kinase/RTK585item
- Proton Pump18item
- PTH1 receptor Agonist33item
- PTH2 receptor Agonist15item
- Pyridines24item
- Pyrimidines34item
- quinolines17item
- Raf29item
- Raf-1 proto-oncogene,serine/threonine kinase Inhibitor20item
- RAR-related orphan receptor-γ Agonist14item
- RAR/RXR27item
- Ras79item
- Reactive Oxygen Species55item
- receptor interacting serine/threonine kinase 1 Inhibitor26item
- ret proto-oncogene Inhibitor26item
- Reverse Transcriptase21item
- Rho associated coiled-coil containing protein kinase 2 Inhibitor18item
- RIP kinase44item
- ROCK32item
- ROR28item
- RSV29item
- RXFP1 Agonist17item
- RXFP2 Agonist14item
- RXFP3 Agonist24item
- RXFP4 Agonist27item
- S1P1 receptor Agonist30item
- S1P4 receptor Agonist17item
- S1P5 receptor Agonist17item
- SARS-CoV97item
- Ser/Thr Protease32item
- Serotonin Transporter20item
- SERT Inhibitor31item
- Seven membered ring compound19item
- SHP216item
- Sigma Receptor32item
- Sirtuin37item
- Six membered carbocyclic compound14item
- Six-Membered Heterocyclic Compounds148item
- Sodium Channel82item
- spleen associated tyrosine kinase Inhibitor18item
- squalene synthase Inhibitor80item
- Src43item
- SRC proto-oncogene,non-receptor tyrosine kinase Inhibitor28item
- SST1 receptor Agonist20item
- SST2 receptor Agonist63item
- SST2 receptor Antagonist16item
- SST3 receptor Agonist44item
- SST4 receptor Agonist25item
- SST5 receptor Agonist36item
- Stable isotope15item
- STAT69item
- Stem Cell/Wnt447item
- Steroids102item
- STING30item
- TAS2R14 Agonist21item
- terpenes78item
- Terpenoids Diterpenoids29item
- Terpenoids Sesquiterpenes22item
- Terpenoids Triterpenes110item
- TGF-beta/Smad116item
- TGF-β Receptor35item
- Thyroid Hormone Receptor18item
- TNF Receptor43item
- Toll-like Receptor (TLR)94item
- Topoisomerase54item
- TP receptor Agonist21item
- TP receptor Antagonist20item
- TRP Channel58item
- TRPA1 Activator34item
- TRPC5 Channel blocker16item
- TRPC6 Channel blocker17item
- TRPM8 Activator15item
- TRPV1 Activator17item
- TRPV1 Channel blocker18item
- Tyrosinase15item
- tyrosine kinase 2 Inhibitor40item
- V1A receptor Agonist20item
- V1A receptor Antagonist40item
- V1B receptor Antagonist18item
- V2 receptor Agonist20item
- V2 receptor Antagonist35item
- VD/VDR21item
- VEGFR61item
- Virus Protease17item
- Vitamin D Related/Nuclear Receptor346item
- VPAC1 receptor Agonist23item
- VPAC2 receptor Agonist22item
- VRAC Channel blocker14item
- Wnt39item
- Y1 receptor Agonist19item
- Y2 receptor Agonist28item
- Y4 receptor Agonist23item
- YAP24item
- α1A-adrenoceptor Antagonist37item
- α1B-adrenoceptor Antagonist31item
- α1D-adrenoceptor Antagonist32item
- α2A-adrenoceptor Antagonist20item
- α2B-adrenoceptor Antagonist21item
- α2C-adrenoceptor Antagonist24item
- β-catenin22item
- β1-adrenoceptor Agonist23item
- β1-adrenoceptor Antagonist29item
- β2-adrenoceptor Agonist28item
- β2-adrenoceptor Antagonist23item
- β3-adrenoceptor Agonist18item
- γ-secretase26item
- δ receptor Agonist38item
- δ receptor Antagonist19item
- κ receptor Agonist48item
- κ receptor Antagonist17item
- μ receptor Agonist42item
- μ receptor Antagonist23item
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Active
Source
Grade
- 1mg/ml in methyl acetate1 item
- ACS2item
- ActiBioPure™1 item
- analytical standard24item
- Animal Free5item
- AR2item
- Azide Free579item
- Bioactive1 item
- BioReagent4item
- BP1 item
- Carrier Free580item
- Contains 10-15% Methanol as stabilizer1 item
- CP1 item
- ExactAb™576item
- for plant cell culture1 item
- granular1 item
- Isomer mixture1 item
- Low Endotoxin566item
- MW 20001 item
- Ph. Eur.1 item
- Ph.Eur1 item
- pharmaceutical grade3item
- pharmacopedia grade1 item
- PharmPure™1 item
- purified grade1 item
- Reagent grade2item
- Recombinant577item
- RValidatedant1 item
- sublimed grade1 item
- Technical Grade1 item
- Ultra pure2item
- UltraBio™2item
- USP1 item
- Validated579item
- viscosity 45-55 cP3item
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Species reactivity(Predicted to work with)
Action Type
- ACTIVATOR322item
- AGONIST3093item
- ALLOSTERIC ANTAGONIST1 item
- ALLOSTERIC MODULATOR467item
- ANTAGONIST2368item
- ANTIBODY25item
- ANTISENSE INHIBITOR1 item
- BINDING AGENT59item
- BLOCKER87item
- CHANNEL BLOCKER340item
- CHELATING AGENT5item
- CROSS-LINKING AGENT16item
- DEGRADER4item
- DISRUPTING AGENT20item
- FUSION PROTEIN1 item
- GATING INHIBITOR75item
- INHIBITOR4171item
- INVERSE AGONIST9item
- MODULATOR69item
- NEGATIVE ALLOSTERIC MODULATOR11item
- NEGATIVE MODULATOR4item
- OPENER7item
- OTHER12item
- PARTIAL AGONIST35item
- POSITIVE ALLOSTERIC MODULATOR30item
- POSITIVE MODULATOR15item
- REDUCING AGENT1 item
- RELEASING AGENT4item
- RNAI INHIBITOR1 item
- SEQUESTERING AGENT3item
- STABILISER16item
- SUBSTRATE6item
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Purity
- ≥75%2item
- ≥80%1 item
- ≥80.0%(GC)1 item
- ≥85%2item
- ≥85%(HPLC)1 item
- ≥88%1 item
- ≥90%6item
- ≥90%(HPLC)1 item
- ≥90%(SDS-PAGE&SEC)30item
- ≥93%1 item
- ≥94%1 item
- ≥95%169item
- ≥95%(HPLC)2item
- ≥95%(mixture of polymers)1 item
- ≥95%(SDS-PAGE&SEC)547item
- ≥95%(SDS-PAGE)2item
- ≥95%,≥95 atom% D1 item
- ≥96%24item
- ≥96%(HPLC)1 item
- ≥97%110item
- ≥97%,≥98atom%D2item
- ≥97.0%1 item
- ≥98 atom% D,≥98%3item
- ≥98%573item
- ≥98% metals basis1 item
- ≥98%(HPLC)14item
- ≥98%(sum of isomers)1 item
- ≥98%,≥98 atom% D2item
- ≥98%,≥98% atom% D1 item
- ≥98%,≥98atom%D7item
- ≥98.0%3item
- ≥99%69item
- ≥99%(CP),≥99 atom % D1 item
- ≥99%(HPLC)1 item
- ≥99%(SDS-PAGE)1 item
- ≥99%,≥98atom%D2item
- ≥99%,≥99 atom % ¹³C1 item
- ≥99.5%2item
- ≥99.5% metals basis1 item
- ≥99.5%(GC)1 item
- ≥99.5%(HPLC)1 item
- ≥99.5%(T)1 item
- ≥99.7%1 item
- ≥99.8%1 item
- ≥99.9% metals basis3item
- ≥99.99%1 item
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Physical form
Price
Species
Carrier free
Animal free
Protein length
Immunogen species
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