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Kakigami et al., 1998 - Google Patents

Synthesis and structure-activity relationship of 3-substituted benzamide, benzo [b] furan-7-carboxamide, 2, 3-dihydrobenzo [b] furan-7-carboxamide, and indole-5 …

Kakigami et al., 1998

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Document ID
7429123690838968380
Author
Kakigami T
Usui T
Tsukamoto K
KATAokA T
Publication year
Publication venue
Chemical and pharmaceutical bulletin

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抄録 The title compounds (6-9) were prepared and evaluated for serotonin 5-HT 4 agonistic activity in in vitro tests. Introducing a propyl or allyl group at the 3-position of benzamide caused only a slight enhancement of agonistic activity. Construction of the benzo [b] furan …
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    • C07D209/04—Indoles; Hydrogenated indoles
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    • C07D207/30—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having two double bonds between ring members or between ring members and non-ring members
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