ZA792729B - Novel aminothiazoles - Google Patents

Novel aminothiazoles

Info

Publication number: ZA792729B
Authority: ZA; South Africa
Prior art keywords: aminothiazoles; novel; novel aminothiazoles
Prior art date: 1978-06-02

Application number

ZA792729A

Other languages

English (en)

Inventor

J Lombardino

Original Assignee

Pfizer

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

1978-06-02

Filing date

1979-06-01

Publication date

1981-03-25

1979-06-01 Application filed by Pfizer filed Critical Pfizer

1981-03-25 Publication of ZA792729B publication Critical patent/ZA792729B/xx

Classifications

- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D307/00—Heterocyclic compounds containing five-membered rings having one oxygen atom as the only ring hetero atom
- C07D307/02—Heterocyclic compounds containing five-membered rings having one oxygen atom as the only ring hetero atom not condensed with other rings
- C07D307/34—Heterocyclic compounds containing five-membered rings having one oxygen atom as the only ring hetero atom not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
- C07D307/38—Heterocyclic compounds containing five-membered rings having one oxygen atom as the only ring hetero atom not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with substituted hydrocarbon radicals attached to ring carbon atoms
- C07D307/52—Radicals substituted by nitrogen atoms not forming part of a nitro radical
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P29/00—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P37/00—Drugs for immunological or allergic disorders
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P37/00—Drugs for immunological or allergic disorders
- A61P37/02—Immunomodulators
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D277/00—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings
- C07D277/02—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings
- C07D277/20—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
- C07D277/32—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D277/38—Nitrogen atoms
- C07D277/42—Amino or imino radicals substituted by hydrocarbon or substituted hydrocarbon radicals
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D333/00—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom
- C07D333/02—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom not condensed with other rings
- C07D333/04—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom not condensed with other rings not substituted on the ring sulphur atom
- C07D333/06—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom not condensed with other rings not substituted on the ring sulphur atom with only hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, directly attached to the ring carbon atoms
- C07D333/14—Radicals substituted by singly bound hetero atoms other than halogen
- C07D333/20—Radicals substituted by singly bound hetero atoms other than halogen by nitrogen atoms
- F—MECHANICAL ENGINEERING; LIGHTING; HEATING; WEAPONS; BLASTING
- F16—ENGINEERING ELEMENTS AND UNITS; GENERAL MEASURES FOR PRODUCING AND MAINTAINING EFFECTIVE FUNCTIONING OF MACHINES OR INSTALLATIONS; THERMAL INSULATION IN GENERAL
- F16B—DEVICES FOR FASTENING OR SECURING CONSTRUCTIONAL ELEMENTS OR MACHINE PARTS TOGETHER, e.g. NAILS, BOLTS, CIRCLIPS, CLAMPS, CLIPS OR WEDGES; JOINTS OR JOINTING
- F16B15/00—Nails; Staples
- F16B15/0023—Nail plates
- F16B2015/0076—Nail plates with provisions for additional fastening means, e.g. hooks, holes for separate screws or nails, adhesive

Landscapes

Chemical & Material Sciences (AREA)
Organic Chemistry (AREA)
Health & Medical Sciences (AREA)
Pharmacology & Pharmacy (AREA)
Animal Behavior & Ethology (AREA)
Chemical Kinetics & Catalysis (AREA)
General Chemical & Material Sciences (AREA)
Medicinal Chemistry (AREA)
Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
Veterinary Medicine (AREA)
Immunology (AREA)
Life Sciences & Earth Sciences (AREA)
Public Health (AREA)
General Health & Medical Sciences (AREA)
Bioinformatics & Cheminformatics (AREA)
Engineering & Computer Science (AREA)
Pain & Pain Management (AREA)
Rheumatology (AREA)
Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Thiazole And Isothizaole Compounds (AREA)
Plural Heterocyclic Compounds (AREA)

ZA792729A 1978-06-02 1979-06-01 Novel aminothiazoles ZA792729B (en)

Applications Claiming Priority (1)

Application Number	Priority Date	Filing Date	Title
US91183078A	1978-06-02	1978-06-02

Publications (1)

Publication Number	Publication Date
ZA792729B true ZA792729B (en)	1981-03-25

Family

ID=25430923

Family Applications (1)

Application Number	Title	Priority Date	Filing Date
ZA792729A ZA792729B (en)	1978-06-02	1979-06-01	Novel aminothiazoles

Country Status (36)

Country	Link
JP (1)	JPS5936988B2 (xx)
AR (1)	AR226285A1 (xx)
AT (1)	AT373248B (xx)
AU (1)	AU511242B2 (xx)
BE (1)	BE876732A (xx)
CA (1)	CA1117949A (xx)
CH (1)	CH639653A5 (xx)
CS (1)	CS216927B2 (xx)
DD (1)	DD144055A5 (xx)
DE (1)	DE2922523C2 (xx)
DK (1)	DK150068C (xx)
EG (1)	EG14354A (xx)
ES (1)	ES481220A1 (xx)
FI (1)	FI68820C (xx)
FR (1)	FR2427333A1 (xx)
GB (1)	GB2022085B (xx)
GR (1)	GR73142B (xx)
HK (1)	HK66487A (xx)
HU (1)	HU180045B (xx)
IE (1)	IE48426B1 (xx)
IL (1)	IL57450A (xx)
IT (1)	IT1121238B (xx)
KE (1)	KE3459A (xx)
LU (1)	LU81349A1 (xx)
MY (1)	MY8500318A (xx)
NL (1)	NL178421C (xx)
NO (1)	NO150760C (xx)
NZ (1)	NZ190623A (xx)
PH (1)	PH17020A (xx)
PL (1)	PL117515B1 (xx)
PT (1)	PT69718A (xx)
SE (1)	SE438333B (xx)
SG (1)	SG56184G (xx)
SU (1)	SU843746A3 (xx)
YU (1)	YU40997B (xx)
ZA (1)	ZA792729B (xx)

Families Citing this family (32)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
JPS57501565A (xx) *	1980-10-24	1982-09-02
JPS57136579A (en) *	1981-01-21	1982-08-23	Mitsui Toatsu Chem Inc	Thiazolylurea derivative, its preparation, and pharmaceutical composition containing the same
DE3264595D1 (en) *	1981-01-08	1985-08-14	Mitsui Toatsu Chemicals	N-(4-phenyl-2-thiazolyl)carbamate derivatives, process for their preparation, and medicinal composition containing same
JPS57116067A (en) *	1981-01-12	1982-07-19	Sankyo Kagaku Kk	Novel 8-quinolinesulfonyl derivative, its synthesis and use
WO1982002386A1 (en) *	1981-01-13	1982-07-22	Sakano Isao	Aminothiazole derivatives,process for their preparation,and medicinal composition containing same
DE3273781D1 (en) *	1981-01-13	1986-11-20	Mitsui Toatsu Chemicals	Novel thiazole compounds, process for their preparation, and medicinal composition containing same
JPS57154175A (en) *	1981-03-16	1982-09-22	Mitsui Toatsu Chem Inc	2-thiazoleamine derivative, its preparation, and drug composition comprising it
DE3227329A1 (de) *	1982-07-22	1984-01-26	Basf Ag, 6700 Ludwigshafen	Verfahren zur herstellung von 2-n,n-disubstituierten aminothiazolen
WO1986003203A1 (en) *	1984-11-22	1986-06-05	Yoshitomi Pharmaceutical Industries, Ltd.	Thienylthiazole derivatives
FR2581063B1 (fr) *	1985-04-30	1987-07-17	Chauvin Blache Lab	Amino-2 thiazoles n-substitues, leur procede de preparation et leur application en therapeutique
JPS63152368A (ja) *	1986-06-03	1988-06-24	Sumitomo Pharmaceut Co Ltd	新規なアミノアゾ−ル誘導体およびその酸付加塩
JPH075579B2 (ja) *	1986-09-01	1995-01-25	吉富製薬株式会社	アミノチアゾ−ル化合物
JPH0753666B2 (ja) *	1987-09-14	1995-06-07	久光製薬株式会社	置換ジフェニルチアゾール誘導体からなる抗炎症剤
DK0486543T3 (da) *	1989-08-10	1998-07-20	Commw Scient Ind Res Org	Fremgangsmåde til fremstilling af en elektrosuspension af mikropartikler
WO1992015570A1 (fr) *	1991-03-07	1992-09-17	Hisamitsu Pharmaceutical Co., Inc.	Nouveau derive de diphenylthiazole
FR2692893B1 (fr) *	1992-06-24	1994-09-02	Sanofi Elf	Dérivés alkylamino ramifiés du thiazole, leurs procédés de préparation et les compositions pharmaceutiques qui les contiennent.
JPH10504542A (ja) *	1994-07-27	1998-05-06	ジー．ディー．サールアンドカンパニー	炎症処置用の置換チアゾール化合物
FR2754258B1 (fr)	1996-10-08	1998-12-31	Sanofi Sa	Derives d'aminothiazole, leur procede de preparation et les compositions pharmaceutiques les contenant
AU3740101A (en)	2000-03-01	2001-09-12	Janssen Pharmaceutica Nv	2,4-disubstituted thiazolyl derivatives
WO2003015777A1 (en) *	2001-08-13	2003-02-27	Lion Bioscience Ag	Nr1h4 nuclear receptor binding compounds
WO2003027105A1 (en) *	2001-09-26	2003-04-03	Bayer Pharmaceuticals Corporation	Substituted 3-pyridyl thiophenes as c17,20 lyase inhibitors
MXPA04006709A (es)	2002-01-11	2004-10-04	Sankyo Co	Derivados de aminoalcohol o derivados de acido fosfonico y composiciones farmaceuticas que los contienen.
EP1555264A1 (en) *	2004-01-15	2005-07-20	Sireen AG	Five-membered heterocyclic compounds as inhibitors of SRC family protein kinase.
JP2005272453A (ja)	2004-02-24	2005-10-06	Sankyo Co Ltd	アミノアルコール化合物
AP2358A (en)	2005-05-09	2012-01-30	Achillion Pharmaceuticals Inc	Thiazole compounds and methods of use.
EP1981884B1 (en)	2006-01-18	2012-06-13	Amgen, Inc	Thiazole compounds as protein kinase b (pkb) inhibitors
JP2010533715A (ja)	2007-07-17	2010-10-28	アムジエン・インコーポレーテツド	複素環系ｐｋｂ調節剤
US7919504B2 (en)	2007-07-17	2011-04-05	Amgen Inc.	Thiadiazole modulators of PKB
US20120316182A1 (en)	2011-06-10	2012-12-13	Calcimedica, Inc.	Compounds that modulate intracellular calcium
WO2012170951A2 (en) *	2011-06-10	2012-12-13	Calcimedica, Inc.	Compounds that modulate intracellular calcium
WO2013059677A1 (en)	2011-10-19	2013-04-25	Calcimedica, Inc.	Compounds that modulate intracellular calcium
CN110590785B (zh) *	2019-09-23	2021-02-02	武汉大学	一种氨基噻唑类化合物及其制备方法与抗肠道病毒71型的应用

Family Cites Families (1)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
US3458526A (en) *	1966-09-26	1969-07-29	Upjohn Co	Certain 2-amino-4,5-bis(p-methoxyphenyl)thiazoles

1979
- 1979-04-30 DK DK177679A patent/DK150068C/da not_active IP Right Cessation
- 1979-05-23 GB GB7917872A patent/GB2022085B/en not_active Expired
- 1979-05-29 CH CH501679A patent/CH639653A5/fr not_active IP Right Cessation
- 1979-05-30 EG EG333/79A patent/EG14354A/xx active
- 1979-05-30 CS CS793728A patent/CS216927B2/cs unknown
- 1979-05-31 SE SE7904798A patent/SE438333B/sv not_active IP Right Cessation
- 1979-05-31 HU HU79PI679A patent/HU180045B/hu not_active IP Right Cessation
- 1979-05-31 YU YU1288/79A patent/YU40997B/xx unknown
- 1979-05-31 SU SU792773929A patent/SU843746A3/ru active
- 1979-05-31 PH PH22588A patent/PH17020A/en unknown
- 1979-05-31 LU LU81349A patent/LU81349A1/xx unknown
- 1979-05-31 CA CA000328805A patent/CA1117949A/en not_active Expired
- 1979-05-31 IL IL57450A patent/IL57450A/xx unknown
- 1979-05-31 AU AU47634/79A patent/AU511242B2/en not_active Ceased
- 1979-06-01 AR AR276782A patent/AR226285A1/es active
- 1979-06-01 FI FI791754A patent/FI68820C/fi not_active IP Right Cessation
- 1979-06-01 JP JP54068781A patent/JPS5936988B2/ja not_active Expired
- 1979-06-01 DD DD79213371A patent/DD144055A5/de not_active IP Right Cessation
- 1979-06-01 ZA ZA792729A patent/ZA792729B/xx unknown
- 1979-06-01 BE BE0/195534A patent/BE876732A/xx not_active IP Right Cessation
- 1979-06-01 IT IT23228/79A patent/IT1121238B/it active
- 1979-06-01 PL PL1979216030A patent/PL117515B1/pl unknown
- 1979-06-01 ES ES481220A patent/ES481220A1/es not_active Expired
- 1979-06-01 AT AT0401679A patent/AT373248B/de not_active IP Right Cessation
- 1979-06-01 NO NO791831A patent/NO150760C/no unknown
- 1979-06-01 DE DE2922523A patent/DE2922523C2/de not_active Expired
- 1979-06-01 NL NLAANVRAGE7904337,A patent/NL178421C/xx not_active IP Right Cessation
- 1979-06-01 PT PT69718A patent/PT69718A/pt unknown
- 1979-06-01 NZ NZ190623A patent/NZ190623A/en unknown
- 1979-06-01 FR FR7914164A patent/FR2427333A1/fr active Granted
- 1979-06-01 GR GR59240A patent/GR73142B/el unknown
- 1979-08-08 IE IE1069/79A patent/IE48426B1/en unknown
1984
- 1984-08-13 SG SG561/84A patent/SG56184G/en unknown
- 1984-09-24 KE KE3459A patent/KE3459A/xx unknown
1985
- 1985-12-30 MY MY318/85A patent/MY8500318A/xx unknown
1987
- 1987-09-17 HK HK664/87A patent/HK66487A/xx unknown

Also Published As

Publication number	Publication date
JPS54160369A (en)	1979-12-19
ATA401679A (de)	1983-05-15
NO150760C (no)	1984-12-12
GB2022085B (en)	1983-01-12
CA1117949A (en)	1982-02-09
YU40997B (en)	1986-10-31
IT1121238B (it)	1986-03-26
EG14354A (en)	1984-06-30
SE7904798L (sv)	1979-12-03
IE791069L (en)	1979-12-02
FI791754A (fi)	1979-11-26
FI68820C (fi)	1985-11-11
PL216030A1 (xx)	1980-03-10
MY8500318A (en)	1985-12-31
LU81349A1 (fr)	1979-12-07
BE876732A (fr)	1979-12-03
AU4763479A (en)	1979-12-06
FI68820B (fi)	1985-07-31
GR73142B (xx)	1984-02-09
IE48426B1 (en)	1985-01-23
AU511242B2 (en)	1980-08-07
ES481220A1 (es)	1980-09-01
IL57450A (en)	1982-11-30
NO150760B (no)	1984-09-03
YU128879A (en)	1982-10-31
CS216927B2 (en)	1982-12-31
NO791831L (no)	1979-12-04
AT373248B (de)	1983-12-27
NL178421B (nl)	1985-10-16
JPS5936988B2 (ja)	1984-09-06
NL7904337A (nl)	1979-12-04
DK177679A (da)	1979-12-03
HU180045B (en)	1983-01-28
NZ190623A (en)	1984-07-06
DK150068B (da)	1986-12-01
FR2427333B1 (xx)	1983-05-20
NL178421C (nl)	1986-03-17
GB2022085A (en)	1979-12-12
PL117515B1 (en)	1981-08-31
PT69718A (en)	1979-07-01
SG56184G (en)	1985-03-08
AR226285A1 (es)	1982-06-30
KE3459A (en)	1984-10-12
IL57450A0 (en)	1979-09-30
FR2427333A1 (fr)	1979-12-28
HK66487A (en)	1987-09-25
DE2922523A1 (de)	1979-12-06
DK150068C (da)	1987-06-29
IT7923228A0 (it)	1979-06-01
DD144055A5 (de)	1980-09-24
DE2922523C2 (de)	1982-10-21
SU843746A3 (ru)	1981-06-30
PH17020A (en)	1984-05-11
CH639653A5 (fr)	1983-11-30
SE438333B (sv)	1985-04-15

Publication	Publication Date	Title
GB2022085B (en)	1983-01-12	Aminothiazoles
EG13913A (en)	1982-09-30	Novel n-heterocyclyl-4-piperidinamines
CS520079A2 (en)	1984-02-13	Nosna soustava snimaci hlavice
ZA794379B (en)	1980-08-27	Novel spiro-oxazolidindiones
BG27580A1 (en)	1979-12-12	Two- poled pelvis- thight articulation- set
CS74479A2 (en)	1987-03-12	Omezovac nadmerne proudove vodivosti televizni reprodukcni obrazovky
CS761579A2 (en)	1984-02-13	Elektricky vypinac se samocinnym zhasenim elektrickeho oblouku
CS333379A2 (en)	1988-04-15	Upinaci zarizeni
JPS554499A (en)	1980-01-12	Extension
JPS54154730A (en)	1979-12-06	Novel dialkoxybenzamides
CS353979A2 (en)	1985-05-15	Zpusob extrakce organickych slozek z rostlinnych materialu
CS615079A2 (en)	1985-08-15	Zpusob vyroby inhibitoru enzymu
CS613879A2 (en)	1985-06-13	Zpusob vyroby fenylchinolizidinu
CS846479A2 (en)	1985-08-15	Tkaci stroj
CS290179A2 (en)	1984-01-16	Plynova vybojka
PH17031A (en)	1984-05-17	Novel phenoxyalkyloxazolines
ZA793391B (en)	1980-06-25	Aminothiazole compounds
JPS54110080A (en)	1979-08-29	Insideepainted can
MY8400085A (en)	1984-12-31	Phenoxyalkanamides
CS556679A2 (en)	1985-08-15	Zpusob vyroby derivatu chlorambucilu
CS839779A2 (en)	1985-08-15	Zpusob vyroby benzimidazol-karbamatu
BG31541A1 (en)	1982-02-15	Ornitopter
CA43944S (en)	1978-07-24	Compositiontable
CS702378A2 (en)	1985-06-13	Budova sestavena z nosnych kontejneru
CS576984A2 (en)	1988-07-15	Zpusob vyroby 2-pyridylmethylsulfinylbenzimidazolu