[go: up one dir, main page]

YU49796A - Optički aktivni derivat fenil pirimidina - Google Patents

Optički aktivni derivat fenil pirimidina

Info

Publication number
YU49796A
YU49796A YU49796A YU49796A YU49796A YU 49796 A YU49796 A YU 49796A YU 49796 A YU49796 A YU 49796A YU 49796 A YU49796 A YU 49796A YU 49796 A YU49796 A YU 49796A
Authority
YU
Yugoslavia
Prior art keywords
active derivative
optical active
phenyl pyrimidine
pyrimidine
phenyl
Prior art date
Application number
YU49796A
Other languages
English (en)
Inventor
Stuart Nobbs Malcolm
Jane Rodgers Sandra
Original Assignee
Glaxo Group Limited
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Glaxo Group Limited filed Critical Glaxo Group Limited
Publication of YU49796A publication Critical patent/YU49796A/sh

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D239/00Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings
    • C07D239/02Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings
    • C07D239/24Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members
    • C07D239/28Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, directly attached to ring carbon atoms
    • C07D239/46Two or more oxygen, sulphur or nitrogen atoms
    • C07D239/48Two nitrogen atoms
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/495Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A61K31/505Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/04Centrally acting analgesics, e.g. opioids

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • General Health & Medical Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • General Chemical & Material Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Neurosurgery (AREA)
  • Neurology (AREA)
  • Biomedical Technology (AREA)
  • Engineering & Computer Science (AREA)
  • Pain & Pain Management (AREA)
  • Epidemiology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)

Abstract

Pronalazak se odnosi na pirimidin formule (I): i njegove aditivne soli kiselina, koji su korisni kao analgetici, kao sredstva protiv grčeva ili za lečenje sindroma nadraženih creva ili manično depresivnih psihoza.
YU49796A 1995-09-05 1996-09-04 Optički aktivni derivat fenil pirimidina YU49796A (sh)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
GBGB9518027.9A GB9518027D0 (en) 1995-09-05 1995-09-05 Pharmacologically active compound

Publications (1)

Publication Number Publication Date
YU49796A true YU49796A (sh) 1999-07-28

Family

ID=10780172

Family Applications (1)

Application Number Title Priority Date Filing Date
YU49796A YU49796A (sh) 1995-09-05 1996-09-04 Optički aktivni derivat fenil pirimidina

Country Status (32)

Country Link
US (1) US6124308A (sh)
EP (1) EP0879230B1 (sh)
JP (1) JPH11512108A (sh)
KR (1) KR19990044397A (sh)
CN (1) CN1200729A (sh)
AP (1) AP640A (sh)
AR (1) AR004192A1 (sh)
AT (1) ATE203523T1 (sh)
AU (1) AU710091B2 (sh)
BG (1) BG65102B1 (sh)
BR (1) BR9610388A (sh)
CA (1) CA2230362A1 (sh)
CO (1) CO4750651A1 (sh)
CZ (1) CZ65598A3 (sh)
DE (1) DE69614150T2 (sh)
EA (1) EA000695B1 (sh)
ES (1) ES2160834T3 (sh)
GB (1) GB9518027D0 (sh)
HR (1) HRP960399A2 (sh)
HU (1) HUP9901260A3 (sh)
ID (1) ID17274A (sh)
IL (1) IL123414A0 (sh)
IS (1) IS4673A (sh)
NO (1) NO980923L (sh)
NZ (1) NZ318390A (sh)
PL (1) PL325329A1 (sh)
SK (1) SK28598A3 (sh)
TR (1) TR199800386T1 (sh)
TW (1) TW367326B (sh)
WO (1) WO1997009317A2 (sh)
YU (1) YU49796A (sh)
ZA (1) ZA967466B (sh)

Families Citing this family (13)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
AR016212A1 (es) * 1998-04-28 2001-06-20 Astra Ab Uso de compuestos farmaceuticos que tienen una actividad antagonista de nmda para preparar un medicamento para el tratamiento del sindrome de intestino irritable (ibs), y composiciones farmaceuticas
EP1085879A2 (en) * 1998-06-08 2001-03-28 Advanced Medicine, Inc. Multibinding agents that modulate the 5-ht transporter
US6420354B1 (en) 1998-06-08 2002-07-16 Advanced Medicine, Inc. Sodium channel drugs and uses
GB9907965D0 (en) * 1999-04-09 1999-06-02 Glaxo Group Ltd Medical use
US6479498B1 (en) 1999-06-04 2002-11-12 Theravance, Inc. Sodium channel drugs and uses
CZ2003445A3 (cs) * 2000-07-21 2004-08-18 Ortho@Mcneilápharmaceuticalźáinc Karbamátové sloučeniny pro prevenci nebo léčbu neuropatické bolesti a bolesti asociované s histaminovou a migrenózní bolestí hlavy
CA2439468A1 (en) * 2001-02-27 2002-09-06 Teva Pharmaceutical Industries Ltd. New crystal forms of lamotrigine and processes for their preparations
JP4625637B2 (ja) 2002-02-22 2011-02-02 シャイア エルエルシー 活性物質送達系及び活性物質を保護し投与する方法
CA2483103A1 (en) * 2002-04-23 2003-11-06 Teva Pharmaceutical Industries Ltd. Pharmaceutical composition containing lamotrigine particles of defined morphology
EP1596844A2 (en) * 2003-01-30 2005-11-23 Dynogen Pharmaceuticals Inc. Use of sodium channel modulators for treating gastrointestinal tract disorders
GB0603087D0 (en) * 2006-02-15 2006-03-29 Glaxo Group Ltd Novel use
JP2010516731A (ja) 2007-01-24 2010-05-20 グラクソ グループ リミテッド 2−メトキシ−5−(5−トリフルオロメチル−テトラゾール−1−イル)−ベンジル]−(2s−フェニル−ピペリジン−3s−イル)−アミンを含む医薬組成物
GB201111712D0 (en) 2011-07-08 2011-08-24 Gosforth Ct Holdings Pty Ltd Pharmaceutical compositions

Family Cites Families (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DK153787C (da) * 1979-06-01 1989-01-16 Wellcome Found Analogifremgangsmaade til fremstilling af substituerede 3,5-diamino-6-phenyl-1,2,4-triaziner og alfa-cyanobenzyliden-aminoguanidinforbindelser til anvendelse som mellemprodukter herved
FI895821A0 (fi) * 1988-12-07 1989-12-05 Wellcome Found Farmaceutiskt aktiva cns foereningar.

Also Published As

Publication number Publication date
TW367326B (en) 1999-08-21
WO1997009317A3 (en) 1997-04-03
AP640A (en) 1998-04-14
MX9801680A (es) 1998-05-31
DE69614150T2 (de) 2001-11-22
BG102342A (en) 1998-09-30
HUP9901260A2 (hu) 1999-09-28
WO1997009317A2 (en) 1997-03-13
AR004192A1 (es) 1998-11-04
ID17274A (id) 1997-12-18
AP9600857A0 (en) 1996-10-31
SK28598A3 (en) 1998-09-09
EP0879230A2 (en) 1998-11-25
GB9518027D0 (en) 1995-11-08
CN1200729A (zh) 1998-12-02
IS4673A (is) 1998-02-23
AU710091B2 (en) 1999-09-16
EP0879230B1 (en) 2001-07-25
NZ318390A (en) 1999-02-25
HUP9901260A3 (en) 2001-04-28
HRP960399A2 (en) 1998-04-30
JPH11512108A (ja) 1999-10-19
AU6986596A (en) 1997-03-27
DE69614150D1 (de) 2001-08-30
CZ65598A3 (cs) 1998-07-15
BR9610388A (pt) 1999-07-06
BG65102B1 (bg) 2007-02-28
ES2160834T3 (es) 2001-11-16
EA199800189A1 (ru) 1998-10-29
CO4750651A1 (es) 1999-03-31
NO980923D0 (no) 1998-03-04
EA000695B1 (ru) 2000-02-28
ZA967466B (en) 1998-04-06
PL325329A1 (en) 1998-07-20
US6124308A (en) 2000-09-26
NO980923L (no) 1998-05-04
TR199800386T1 (xx) 1998-05-21
KR19990044397A (ko) 1999-06-25
IL123414A0 (en) 1998-09-24
ATE203523T1 (de) 2001-08-15
CA2230362A1 (en) 1997-03-13

Similar Documents

Publication Publication Date Title
EA200401157A1 (ru) N-аминоацетилпирролидин-2-карбонитрилы и их применение в качестве ингибиторов ddp-iv
YU49796A (sh) Optički aktivni derivat fenil pirimidina
EA200100412A1 (ru) Замещенные 3-цианохинолины в качестве ингибиторов протеинтирозинкиназ
TR199901905T2 (xx) 2-(P�rin-9-il)-tetrahidrofuran-3,4-diol t�revleri.
ATE284690T1 (de) Antithrombotische diamine
MY138335A (en) Antimicrobial quinolones, their compositions and uses
ATE298750T1 (de) 3-(heteroarylacetamido)-2-oxo-azetidin-1- sulfonsäure derivate als antibakterielle mittel
ATE273690T1 (de) Zusammensetzung zur hautdesinfizierung
EA199901016A1 (ru) 9-оксим-производные эритромицина
BR9713338A (pt) Benzonaftiridinas como terapêuticos brÈnquicos.
ES2193241T3 (es) Nuevas n-2-oxo2.3.4.5-tetrajodrp-1h-1,5-benzodiazepin-3-il)-3-amidas.
SE9901077D0 (sv) Novel use
ATE297903T1 (de) Substituierte phenyluracile
EA200000204A1 (ru) Производные пирролопирролона в качестве ингибиторов эластазы нейтрофилов
PT828721E (pt) 2-amino-benxoxazinonas para o tratamento de infeccoes virais
SE9801494D0 (sv) Novel use
YU60101A (sh) Derivati rezorcinola
YU44301A (sh) 5ht1 antagonisti za antidepresantnu terapiju
EA200100807A1 (ru) Производные алкинилсодержащих гидроксамовых кислот и их применение в качестве ингибиторов tace
DE69819539D1 (de) Antithrombotische mittel
PT98604A (pt) Processo para a preparacao de uma solucao estavel de hipoclorito de sodio
ATE335739T1 (de) Cak inhibitoren und deren verwendungen
ATE416174T1 (de) Substituierte homopiperidylbenzimidazolanaloga als fundusrelaxantien
ES2076838T3 (es) Nuevo derivado de la isoindolinona, su preparacion y las composiciones farmaceuticas que le contienen.
DE69524064D1 (de) Indan-2-mercaptoacetylamid disulfidderivate als enkephalinase inhibitoren