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YU47783B - SUBSTITUTED PYROLES AND PROCEDURE FOR THEIR PRODUCTION - Google Patents

SUBSTITUTED PYROLES AND PROCEDURE FOR THEIR PRODUCTION

Info

Publication number
YU47783B
YU47783B YU126791A YU126791A YU47783B YU 47783 B YU47783 B YU 47783B YU 126791 A YU126791 A YU 126791A YU 126791 A YU126791 A YU 126791A YU 47783 B YU47783 B YU 47783B
Authority
YU
Yugoslavia
Prior art keywords
bond
sum
together form
piq
chn
Prior art date
Application number
YU126791A
Other languages
Serbo-Croatian (sh)
Serbian (sr)
Other versions
YU126791A (en
Inventor
P.D. Davis
C.H. Hill
G. Lawton
Original Assignee
F. Hoffmann-La Roche Ag.
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by F. Hoffmann-La Roche Ag. filed Critical F. Hoffmann-La Roche Ag.
Publication of YU126791A publication Critical patent/YU126791A/en
Publication of YU47783B publication Critical patent/YU47783B/en

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  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)

Abstract

SUPSTITUISANI PIROLI I POSTUPAK ZA NJIHOVU PROIZVODNJU jedinjenja, naznačena time, što imaju opštu formulu gde R1 i R3 zajedno formiraju vezu, a R2 predstavlja vodonik ili R1 i R2 zajedno formiraju vezu, a R3 predstavlja vodonik; R4, R5, R6 i R7 nezavisno jedan od drugog predstavljaju vodonik, halogen, alkil, haloalkil, alkoksi, nitro, amino, alkanoilamino, aroilamino, alkiltio ili alkilsulfonil; R8 predstavlja vodonik, alkil ili aralkil; X predstavlja -N(R9)- ili -CHN(R10, R11)- pri čemu svaki od R9, R10 i R11 predstavljaju vodonik, alkil, aralkil ili alkanoil; m znači 0-2, a n 1-3, uz uslov da suma m i n bude 1-3; p znači 0-4, a q 0-4, uz uslov da suma p i q bude 2-4 kada X predstavlja -N(R9)-, da suma p i q bude 1-5 kada X predstavlja -CHN(R10, R11)-, a R1 i R2 zajedno predstavljaju vezu, da suma p i q bude 0-4 kada X predstavlja-CHN(R10, R11)-, a R1 i R3 zajedno formiraju vezu i da p bude 1-4 kada X predstavlja -N(R9)-, R1 i R3 zajedno čine vezu, a m znači 0, kao i farmaceutski prihvatljive soli kiseli jedinjenja formule I sa bazama i bazna jedinjenja formule I sa kiselinama. Prijava sadrži još 1 nezavisan i 8 zavisnih zahteva.SUBSTITUTED PYROLES AND A PROCEDURE FOR THEIR PRODUCTION OF THE COMPOUNDS EMI7.1 having the general formula wherein R1 and R3 together form a bond and R2 represents hydrogen or R1 and R2 together form a bond and R3 represents hydrogen; R 4, R 5, R 6 and R 7 independently of one another are hydrogen, halogen, alkyl, haloalkyl, alkoxy, nitro, amino, alkanoylamino, aroylamino, alkylthio or alkylsulfonyl; R 8 represents hydrogen, alkyl or aralkyl; X represents -N (R 9) - or -CHN (R 10, R 11) - wherein each of R 9, R 10 and R 11 represents hydrogen, alkyl, aralkyl or alkanoyl; m is 0-2 and n is 1-3, provided that the sum of m and n is 1-3; p means 0-4, aq 0-4, provided that the sum of piq is 2-4 when X represents -N (R9) -, that the sum of piq is 1-5 when X represents -CHN (R10, R11) -, and R1 and R2 together represent a bond, that the sum of piq is 0-4 when X represents -CHN (R10, R11) -, and R1 and R3 together form a bond and p is 1-4 when X represents -N (R9) -. R1 and R3 together form a bond, am means 0, as well as pharmaceutically acceptable salts of the acidic compounds of formula I with bases and the base compounds of formula I with acids. The application contains 1 more independent and 8 dependent requests.

YU126791A 1990-08-07 1991-07-18 SUBSTITUTED PYROLES AND PROCEDURE FOR THEIR PRODUCTION YU47783B (en)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
GB909017269A GB9017269D0 (en) 1990-08-07 1990-08-07 Substituted pyrroles

Publications (2)

Publication Number Publication Date
YU126791A YU126791A (en) 1994-01-20
YU47783B true YU47783B (en) 1996-01-09

Family

ID=10680268

Family Applications (1)

Application Number Title Priority Date Filing Date
YU126791A YU47783B (en) 1990-08-07 1991-07-18 SUBSTITUTED PYROLES AND PROCEDURE FOR THEIR PRODUCTION

Country Status (5)

Country Link
BR (1) BR9103385A (en)
GB (1) GB9017269D0 (en)
MX (1) MX9100530A (en)
YU (1) YU47783B (en)
ZA (1) ZA916041B (en)

Also Published As

Publication number Publication date
MX9100530A (en) 1992-04-01
GB9017269D0 (en) 1990-09-19
BR9103385A (en) 1992-05-12
ZA916041B (en) 1992-04-29
YU126791A (en) 1994-01-20

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