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YU171682A - Process for obtaining pyridazine derivatives - Google Patents

Process for obtaining pyridazine derivatives

Info

Publication number
YU171682A
YU171682A YU01716/82A YU171682A YU171682A YU 171682 A YU171682 A YU 171682A YU 01716/82 A YU01716/82 A YU 01716/82A YU 171682 A YU171682 A YU 171682A YU 171682 A YU171682 A YU 171682A
Authority
YU
Yugoslavia
Prior art keywords
obtaining
pyridazine derivatives
pyridazine
derivatives
obtaining pyridazine
Prior art date
Application number
YU01716/82A
Other languages
English (en)
Inventor
C Wermuth
J P Chambon
Original Assignee
Societe Anonyme Dite
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Societe Anonyme Dite filed Critical Societe Anonyme Dite
Publication of YU171682A publication Critical patent/YU171682A/xx

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D237/00Heterocyclic compounds containing 1,2-diazine or hydrogenated 1,2-diazine rings
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D237/00Heterocyclic compounds containing 1,2-diazine or hydrogenated 1,2-diazine rings
    • C07D237/26Heterocyclic compounds containing 1,2-diazine or hydrogenated 1,2-diazine rings condensed with carbocyclic rings or ring systems
    • C07D237/30Phthalazines
    • C07D237/34Phthalazines with nitrogen atoms directly attached to carbon atoms of the nitrogen-containing ring, e.g. hydrazine radicals
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/08Antiepileptics; Anticonvulsants
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/18Antipsychotics, i.e. neuroleptics; Drugs for mania or schizophrenia
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D237/00Heterocyclic compounds containing 1,2-diazine or hydrogenated 1,2-diazine rings
    • C07D237/02Heterocyclic compounds containing 1,2-diazine or hydrogenated 1,2-diazine rings not condensed with other rings
    • C07D237/06Heterocyclic compounds containing 1,2-diazine or hydrogenated 1,2-diazine rings not condensed with other rings having three double bonds between ring members or between ring members and non-ring members
    • C07D237/10Heterocyclic compounds containing 1,2-diazine or hydrogenated 1,2-diazine rings not condensed with other rings having three double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D237/20Nitrogen atoms

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Animal Behavior & Ethology (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Neurology (AREA)
  • Neurosurgery (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Biomedical Technology (AREA)
  • Veterinary Medicine (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Psychiatry (AREA)
  • Pain & Pain Management (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Low-Molecular Organic Synthesis Reactions Using Catalysts (AREA)
  • Plural Heterocyclic Compounds (AREA)
YU01716/82A 1981-08-11 1982-08-06 Process for obtaining pyridazine derivatives YU171682A (en)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
FR8115546A FR2511366A1 (fr) 1981-08-11 1981-08-11 Nouveaux derives de la pyridazine, leur procede de preparation et les medicaments, actifs sur le systeme nerveux central, qui en contiennent

Publications (1)

Publication Number Publication Date
YU171682A true YU171682A (en) 1985-03-20

Family

ID=9261385

Family Applications (1)

Application Number Title Priority Date Filing Date
YU01716/82A YU171682A (en) 1981-08-11 1982-08-06 Process for obtaining pyridazine derivatives

Country Status (30)

Country Link
US (1) US4710499A (xx)
EP (1) EP0073161B1 (xx)
JP (1) JPS5838263A (xx)
KR (1) KR880002711B1 (xx)
AR (1) AR231537A1 (xx)
AT (1) ATE23042T1 (xx)
AU (1) AU579570B2 (xx)
CA (1) CA1179347A (xx)
CS (1) CS239929B2 (xx)
DD (1) DD202550A5 (xx)
DE (1) DE3273893D1 (xx)
DK (1) DK148596C (xx)
EG (1) EG15749A (xx)
ES (1) ES514887A0 (xx)
FI (1) FI72970C (xx)
FR (1) FR2511366A1 (xx)
GR (1) GR76236B (xx)
HU (1) HU189608B (xx)
IE (1) IE53493B1 (xx)
IL (1) IL66424A (xx)
MA (1) MA19559A1 (xx)
NO (1) NO158871C (xx)
NZ (1) NZ201553A (xx)
OA (1) OA07179A (xx)
PH (1) PH18921A (xx)
PL (1) PL137200B1 (xx)
PT (1) PT75372B (xx)
SU (1) SU1356960A3 (xx)
YU (1) YU171682A (xx)
ZA (1) ZA825515B (xx)

Families Citing this family (16)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
FR2539741A1 (fr) * 1983-01-21 1984-07-27 Sanofi Sa Composes a noyau heterocyclique diazote, leur procede de preparation et les medicaments, actifs sur le systeme nerveux central, qui en contiennent
US5001125A (en) * 1984-03-26 1991-03-19 Janssen Pharmaceutica N.V. Anti-virally active pyridazinamines
JPS60218377A (ja) * 1984-04-16 1985-11-01 Mitsubishi Yuka Yakuhin Kk 4−フエニルフタラジン誘導体及びそれを有効成分とする循環改善剤
DE3664772D1 (en) * 1985-01-14 1989-09-07 Boehringer Ingelheim Kg 12-amino pyridazinoû4',5':3,4¨pyrroloû2,1-a¨isoquinolines, process for their preparation and use
US5106973A (en) * 1987-11-23 1992-04-21 Janssen Pharmaceutica N.V. Pyridzainamine derivatives
ATE163412T1 (de) * 1993-06-08 1998-03-15 Sanofi Sa Pyridazine als interleukin-1-beta verwandlungsenzym inhibitoren
US20100210590A1 (en) * 1995-09-27 2010-08-19 Northwestern University Compositions and treatments for seizure-related disorders
GB9707693D0 (en) * 1997-04-16 1997-06-04 Smithkline Beecham Plc Novel method of treatment
EP2264014A1 (en) * 2001-08-31 2010-12-22 Université Louis Pasteur Substituted pyridazines as anti-inflammatory agents and protein kinase inhibitors
CA2589102C (en) * 2004-11-02 2013-08-13 Northwestern University Pyridazine compounds and methods for using the compounds to treat inflammatory diseases
JP5337375B2 (ja) 2004-11-02 2013-11-06 ノースウェスタン ユニバーシティ ピリダジン化合物、組成物および方法
EP2015751A2 (en) * 2006-04-28 2009-01-21 Northwestern University Salts of pyridazine compounds
EP2015750A2 (en) * 2006-04-28 2009-01-21 Northwestern University Compositions and treatments using pyridazine compounds and cholinesterase inhibitors
CN101754762A (zh) 2006-04-28 2010-06-23 西北大学 用于治疗神经炎症性疾病的包含哒嗪化合物的制剂
EP2131839A2 (en) * 2007-03-02 2009-12-16 Northwestern University Compositions comprising derivatives of 3-phenylpyridazine for treating seizure-related disorders
WO2024148148A1 (en) * 2023-01-04 2024-07-11 The Trustees Of Columbia University In The City Of New York Pyridazine based small molecule inhibitor of cognitive impairment

Family Cites Families (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB1345880A (en) * 1971-06-18 1974-02-06 Cepbepe Pyridazine derivatives
FR2473522A1 (fr) * 1980-01-16 1981-07-17 Synthelabo Nouveaux derives substitues de dihydro-2,3 imidazo(1,2-b)pyridazines et les medicaments, utiles notamment comme antidepresseurs, qui en contiennent

Also Published As

Publication number Publication date
DE3273893D1 (en) 1986-11-27
HU189608B (en) 1986-07-28
NO158871C (no) 1988-11-09
US4710499A (en) 1987-12-01
IE53493B1 (en) 1988-11-23
IL66424A0 (en) 1982-11-30
ZA825515B (en) 1983-06-29
JPS5838263A (ja) 1983-03-05
PL137200B1 (en) 1986-05-31
FR2511366A1 (fr) 1983-02-18
FR2511366B1 (xx) 1984-12-14
FI72970C (fi) 1987-08-10
OA07179A (fr) 1984-04-30
AU579570B2 (en) 1988-12-01
FI822768L (fi) 1983-02-11
EP0073161B1 (fr) 1986-10-22
AR231537A1 (es) 1984-12-28
DK148596C (da) 1986-01-13
EP0073161A1 (fr) 1983-03-02
DK358782A (da) 1983-02-12
PT75372A (en) 1982-09-01
ES8305736A1 (es) 1983-04-16
JPH0456032B2 (xx) 1992-09-07
PL237836A1 (en) 1983-02-28
DK148596B (da) 1985-08-12
GR76236B (xx) 1984-08-04
ES514887A0 (es) 1983-04-16
CS239929B2 (en) 1986-01-16
KR880002711B1 (ko) 1988-12-26
AU8702982A (en) 1983-05-12
CA1179347A (en) 1984-12-11
ATE23042T1 (de) 1986-11-15
EG15749A (en) 1986-09-30
FI72970B (fi) 1987-04-30
NO822717L (no) 1983-02-14
NO158871B (no) 1988-08-01
NZ201553A (en) 1985-08-16
MA19559A1 (fr) 1983-04-01
SU1356960A3 (ru) 1987-11-30
KR840001147A (ko) 1984-03-28
FI822768A0 (fi) 1982-08-09
IE821822L (en) 1983-02-11
IL66424A (en) 1985-10-31
PH18921A (en) 1985-11-11
PT75372B (en) 1984-12-10
DD202550A5 (de) 1983-09-21

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