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UY34730A - Formulaciones farmacéuticas que comprenden antagonistas de ccr3 - Google Patents

Formulaciones farmacéuticas que comprenden antagonistas de ccr3

Info

Publication number
UY34730A
UY34730A UY0001034730A UY34730A UY34730A UY 34730 A UY34730 A UY 34730A UY 0001034730 A UY0001034730 A UY 0001034730A UY 34730 A UY34730 A UY 34730A UY 34730 A UY34730 A UY 34730A
Authority
UY
Uruguay
Prior art keywords
pharmaceutical formulations
ccr3 antagonists
include ccr3
antagonists
formulations
Prior art date
Application number
UY0001034730A
Other languages
English (en)
Inventor
Fetscher Alfred
Jochen Matthias Scher
Original Assignee
Boehringer Ingelheim Int
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=49292482&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=UY34730(A) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Boehringer Ingelheim Int filed Critical Boehringer Ingelheim Int
Publication of UY34730A publication Critical patent/UY34730A/es

Links

Classifications

    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
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    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/44—Non condensed pyridines; Hydrogenated derivatives thereof
    • A61K31/445—Non condensed piperidines, e.g. piperocaine
    • A61K31/4523—Non condensed piperidines, e.g. piperocaine containing further heterocyclic ring systems
    • A61K31/4545—Non condensed piperidines, e.g. piperocaine containing further heterocyclic ring systems containing a six-membered ring with nitrogen as a ring hetero atom, e.g. pipamperone, anabasine
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    • A61K9/14—Particulate form, e.g. powders, Processes for size reducing of pure drugs or the resulting products, Pure drug nanoparticles
    • A61K9/16—Agglomerates; Granulates; Microbeadlets ; Microspheres; Pellets; Solid products obtained by spray drying, spray freeze drying, spray congealing,(multiple) emulsion solvent evaporation or extraction
    • A61K9/1605—Excipients; Inactive ingredients
    • A61K9/1617—Organic compounds, e.g. phospholipids, fats
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    • A61K9/2013—Organic compounds, e.g. phospholipids, fats
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    • A61K9/2013—Organic compounds, e.g. phospholipids, fats
    • A61K9/2018—Sugars, or sugar alcohols, e.g. lactose, mannitol; Derivatives thereof, e.g. polysorbates
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Landscapes

  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Epidemiology (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Organic Chemistry (AREA)
  • Immunology (AREA)
  • Molecular Biology (AREA)
  • Biophysics (AREA)
  • Pulmonology (AREA)
  • Inorganic Chemistry (AREA)
  • Rheumatology (AREA)
  • Physical Education & Sports Medicine (AREA)
  • Orthopedic Medicine & Surgery (AREA)
  • Physiology (AREA)
  • Nutrition Science (AREA)
  • Oncology (AREA)
  • Dermatology (AREA)
  • Pain & Pain Management (AREA)
  • Neurology (AREA)
  • Communicable Diseases (AREA)
  • Cardiology (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Transplantation (AREA)
  • Otolaryngology (AREA)
  • Urology & Nephrology (AREA)
  • Ophthalmology & Optometry (AREA)
  • Diabetes (AREA)
  • Hematology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)

Abstract

La presente invención se refiere a composiciones farmacéuticas que contienen compuestos de la fórmula 1 en donde: R1 es H, alquilo C1-6, alquil C0-4- cicloalquilo C3-6, haloalquilo C1-6; R2 es H, alquilo C1-6; X es un anión seleccionado del grupo que consiste en cloruro o ½ dibenzoiltartrato j es 1 ó 2. a procesos para su preparación y a su uso para tratar enfermedades conectadas con el receptor CCR3.
UY0001034730A 2012-04-04 2013-04-04 Formulaciones farmacéuticas que comprenden antagonistas de ccr3 UY34730A (es)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
EP12163078 2012-04-04

Publications (1)

Publication Number Publication Date
UY34730A true UY34730A (es) 2013-10-31

Family

ID=49292482

Family Applications (1)

Application Number Title Priority Date Filing Date
UY0001034730A UY34730A (es) 2012-04-04 2013-04-04 Formulaciones farmacéuticas que comprenden antagonistas de ccr3

Country Status (31)

Country Link
US (3) US10213421B2 (es)
EP (3) EP3970693A1 (es)
JP (4) JP6320990B2 (es)
KR (2) KR102138709B1 (es)
CN (1) CN104203213A (es)
AR (1) AR090596A1 (es)
AU (1) AU2013245028B2 (es)
BR (1) BR112014024479A8 (es)
CA (1) CA2869058C (es)
CL (1) CL2014002524A1 (es)
CY (1) CY1121137T1 (es)
DK (2) DK2833864T3 (es)
EA (1) EA027627B1 (es)
ES (2) ES2898179T3 (es)
HR (1) HRP20190069T1 (es)
HU (2) HUE056943T2 (es)
IL (1) IL234299A (es)
IN (1) IN2014DN07082A (es)
LT (1) LT2833864T (es)
MX (1) MX358307B (es)
NZ (1) NZ628993A (es)
PH (1) PH12014502241A1 (es)
PL (2) PL3524230T3 (es)
PT (2) PT3524230T (es)
RS (1) RS58360B1 (es)
SI (1) SI2833864T1 (es)
SM (1) SMT201900121T1 (es)
TR (1) TR201821285T4 (es)
TW (1) TW201400115A (es)
UY (1) UY34730A (es)
WO (1) WO2013149987A1 (es)

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US8278302B2 (en) 2009-04-08 2012-10-02 Boehringer Ingelheim International Gmbh Substituted piperidines as CCR3 antagonists
UA109290C2 (uk) 2010-10-07 2015-08-10 Спільні кристали і солі інгібіторів ccr3
US8680280B2 (en) 2012-04-02 2014-03-25 Boehringer Ingelheim International Gmbh Process for the manufacturing of CRR inhibitors
US20130261153A1 (en) * 2012-04-03 2013-10-03 Boehringer Ingelheim International Gmbh Use of ccr3-inhibitors
US10213421B2 (en) * 2012-04-04 2019-02-26 Alkahest, Inc. Pharmaceutical formulations comprising CCR3 antagonists
SG11201909207VA (en) * 2017-04-05 2019-11-28 Alkahest Inc Methods and compositions for treating retina-associated disease using ccr3-inhibitors
EP3606525A4 (en) * 2017-04-05 2020-09-09 Alkahest, Inc. METHODS AND COMPOSITIONS FOR TREATING AGING-ASSOCIATED DISORDERS USING CCR3 INHIBITORS
CA3076017A1 (en) * 2017-10-13 2019-04-18 Alkahest, Inc. Methods and compositions for treating pruritus, xerosis, and associated disease using ccr3-inhibitors
CN112469439A (zh) 2018-05-15 2021-03-09 万能溶剂有限公司 用白三烯a4水解酶调节剂治疗衰老相关性疾病
EA202190463A1 (ru) * 2018-09-26 2021-06-29 Алкахест, Инк. Способы и композиции для лечения ассоциированных со старением нарушений с применением ccr3-ингибиторов
KR20230056017A (ko) 2020-08-27 2023-04-26 에이지씨 가부시키가이샤 무알칼리 유리 및 유리판
US11957671B2 (en) 2021-11-01 2024-04-16 Alkahest, Inc. Benzodioxane modulators of leukotriene A4 hydrolase (LTA4H) for prevention and treatment of aging-associated diseases

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