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UY30676A1 - Microemulsion aceite/agua de propofol estable y lista para uso - Google Patents

Microemulsion aceite/agua de propofol estable y lista para uso

Info

Publication number
UY30676A1
UY30676A1 UY30676A UY30676A UY30676A1 UY 30676 A1 UY30676 A1 UY 30676A1 UY 30676 A UY30676 A UY 30676A UY 30676 A UY30676 A UY 30676A UY 30676 A1 UY30676 A1 UY 30676A1
Authority
UY
Uruguay
Prior art keywords
ready
propofol
oil
water microemulsion
c17h35coo
Prior art date
Application number
UY30676A
Other languages
English (en)
Inventor
Marisa Dutra Rodriguez
Roberto Debom Moreira
Ogari De Castro Pacheco
Original Assignee
Cristalia Prod Quimicos Farm
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Cristalia Prod Quimicos Farm filed Critical Cristalia Prod Quimicos Farm
Publication of UY30676A1 publication Critical patent/UY30676A1/es

Links

Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/02Halogenated hydrocarbons
    • A61K31/025Halogenated hydrocarbons carbocyclic
    • A61K31/03Halogenated hydrocarbons carbocyclic aromatic
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/045Hydroxy compounds, e.g. alcohols; Salts thereof, e.g. alcoholates
    • A61K31/05Phenols
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/10Dispersions; Emulsions
    • A61K9/107Emulsions ; Emulsion preconcentrates; Micelles
    • A61K9/1075Microemulsions or submicron emulsions; Preconcentrates or solids thereof; Micelles, e.g. made of phospholipids or block copolymers
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P23/00Anaesthetics
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P23/00Anaesthetics
    • A61P23/02Local anaesthetics
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/20Hypnotics; Sedatives

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • General Health & Medical Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Medicinal Chemistry (AREA)
  • Epidemiology (AREA)
  • Anesthesiology (AREA)
  • Organic Chemistry (AREA)
  • General Chemical & Material Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Biophysics (AREA)
  • Dispersion Chemistry (AREA)
  • Molecular Biology (AREA)
  • Neurosurgery (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Biomedical Technology (AREA)
  • Neurology (AREA)
  • Medicinal Preparation (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)

Abstract

La presente invencion describe una nueva composicion farmacéutica anestésica conteniendo propofol para administracion parenteral, estando en la forma de micro emulsion oleo/agua en la cual la fase oleosa es constituida por el propofol bajo la forma de partículas con diámetro comprendido entre 1 y 100 nm utilizando un unico surfactante seleccionado del gripo constituido por estearatos de polietileno glocol poseyendo la formula general C17H35COO. (OCH2CH2) nH o C17H35COO. (OCH2CH2) nÀCOOC17H35À
UY30676A 2006-10-27 2007-10-30 Microemulsion aceite/agua de propofol estable y lista para uso UY30676A1 (es)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
BRPI0604377-1A BRPI0604377A (pt) 2006-10-27 2006-10-27 microemulsão óleo/água de propofol estável e pronta-para-uso

Publications (1)

Publication Number Publication Date
UY30676A1 true UY30676A1 (es) 2008-05-31

Family

ID=39324037

Family Applications (1)

Application Number Title Priority Date Filing Date
UY30676A UY30676A1 (es) 2006-10-27 2007-10-30 Microemulsion aceite/agua de propofol estable y lista para uso

Country Status (9)

Country Link
US (1) US20100041769A1 (es)
EP (1) EP2097073A4 (es)
CN (1) CN101553215B (es)
AR (1) AR063397A1 (es)
BR (1) BRPI0604377A (es)
CL (1) CL2007003075A1 (es)
HK (1) HK1135029A1 (es)
UY (1) UY30676A1 (es)
WO (1) WO2008049178A1 (es)

Families Citing this family (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US8242158B1 (en) 2012-01-04 2012-08-14 Hospira, Inc. Dexmedetomidine premix formulation
WO2014033751A2 (en) * 2012-08-16 2014-03-06 Emcure Pharmaceuticals Limited Pharmaceutical composition of propofol
WO2017002117A1 (en) * 2015-07-01 2017-01-05 Yissum Research Development Company Of The Hebrew University Of Jerusalem Ltd Delivery systems for propofol

Family Cites Families (11)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB8912391D0 (en) * 1989-05-30 1989-07-12 Unilever Plc Shampoo composition
DE4039602A1 (de) * 1990-12-12 1992-06-17 Bauer Kurt Heinz Prof Dr Pharmazeutische formulierungen
US5962536A (en) * 1998-07-31 1999-10-05 Komer; Gene Injectable propofol formulations
CN1149984C (zh) * 1999-06-21 2004-05-19 健一制药株式会社 用于静脉注射的含有普鲁泊福的麻醉组合物
KR20010055736A (ko) * 1999-12-13 2001-07-04 이규현 프로포폴의 마이크로에멀젼 주사제 조성물
IN188917B (es) * 2000-12-07 2002-11-23 Bharat Surums & Vaccines Ltd
US20040220283A1 (en) * 2002-07-29 2004-11-04 Transform Pharmaceuticals, Inc. Aqueous 2,6-diisopropylphenol pharmaceutical compositions
NZ526347A (en) * 2003-04-30 2005-07-29 Parnell Lab Aust Pty Ltd Formulations containing propofol for anaesthetic use
US7326735B2 (en) * 2003-04-30 2008-02-05 Parnell Laboratories (Aust) Pty Limited Formulations for anaesthetic use
WO2005079758A1 (en) * 2004-02-13 2005-09-01 Bioavailability, Inc. A microemulsion preparation of high concentration propofol for anesthetic uses
MX2008001746A (es) * 2005-08-05 2008-04-07 Bharat Serums & Vaccines Ltd Composiciones de emulsion de propofol intravenosas que tienen eficacia de conservacion.

Also Published As

Publication number Publication date
CN101553215A (zh) 2009-10-07
CN101553215B (zh) 2013-04-10
CL2007003075A1 (es) 2008-03-14
WO2008049178A1 (en) 2008-05-02
EP2097073A1 (en) 2009-09-09
US20100041769A1 (en) 2010-02-18
HK1135029A1 (en) 2010-05-28
EP2097073A4 (en) 2013-09-18
WO2008049178A8 (en) 2008-06-12
AR063397A1 (es) 2009-01-28
BRPI0604377A (pt) 2008-06-24

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Legal Events

Date Code Title Description
109 Application deemed to be withdrawn

Effective date: 20170727