UY30676A1 - Microemulsion aceite/agua de propofol estable y lista para uso - Google Patents
Microemulsion aceite/agua de propofol estable y lista para usoInfo
- Publication number
- UY30676A1 UY30676A1 UY30676A UY30676A UY30676A1 UY 30676 A1 UY30676 A1 UY 30676A1 UY 30676 A UY30676 A UY 30676A UY 30676 A UY30676 A UY 30676A UY 30676 A1 UY30676 A1 UY 30676A1
- Authority
- UY
- Uruguay
- Prior art keywords
- ready
- propofol
- oil
- water microemulsion
- c17h35coo
- Prior art date
Links
Classifications
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/02—Halogenated hydrocarbons
- A61K31/025—Halogenated hydrocarbons carbocyclic
- A61K31/03—Halogenated hydrocarbons carbocyclic aromatic
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/045—Hydroxy compounds, e.g. alcohols; Salts thereof, e.g. alcoholates
- A61K31/05—Phenols
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/10—Dispersions; Emulsions
- A61K9/107—Emulsions ; Emulsion preconcentrates; Micelles
- A61K9/1075—Microemulsions or submicron emulsions; Preconcentrates or solids thereof; Micelles, e.g. made of phospholipids or block copolymers
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P23/00—Anaesthetics
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P23/00—Anaesthetics
- A61P23/02—Local anaesthetics
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/20—Hypnotics; Sedatives
Landscapes
- Health & Medical Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
- Veterinary Medicine (AREA)
- Public Health (AREA)
- General Health & Medical Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- Pharmacology & Pharmacy (AREA)
- Medicinal Chemistry (AREA)
- Epidemiology (AREA)
- Anesthesiology (AREA)
- Organic Chemistry (AREA)
- General Chemical & Material Sciences (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Biophysics (AREA)
- Dispersion Chemistry (AREA)
- Molecular Biology (AREA)
- Neurosurgery (AREA)
- Engineering & Computer Science (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Biomedical Technology (AREA)
- Neurology (AREA)
- Medicinal Preparation (AREA)
- Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
Abstract
La presente invencion describe una nueva composicion farmacéutica anestésica conteniendo propofol para administracion parenteral, estando en la forma de micro emulsion oleo/agua en la cual la fase oleosa es constituida por el propofol bajo la forma de partículas con diámetro comprendido entre 1 y 100 nm utilizando un unico surfactante seleccionado del gripo constituido por estearatos de polietileno glocol poseyendo la formula general C17H35COO. (OCH2CH2) nH o C17H35COO. (OCH2CH2) nÀCOOC17H35À
Applications Claiming Priority (1)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
BRPI0604377-1A BRPI0604377A (pt) | 2006-10-27 | 2006-10-27 | microemulsão óleo/água de propofol estável e pronta-para-uso |
Publications (1)
Publication Number | Publication Date |
---|---|
UY30676A1 true UY30676A1 (es) | 2008-05-31 |
Family
ID=39324037
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
UY30676A UY30676A1 (es) | 2006-10-27 | 2007-10-30 | Microemulsion aceite/agua de propofol estable y lista para uso |
Country Status (9)
Country | Link |
---|---|
US (1) | US20100041769A1 (es) |
EP (1) | EP2097073A4 (es) |
CN (1) | CN101553215B (es) |
AR (1) | AR063397A1 (es) |
BR (1) | BRPI0604377A (es) |
CL (1) | CL2007003075A1 (es) |
HK (1) | HK1135029A1 (es) |
UY (1) | UY30676A1 (es) |
WO (1) | WO2008049178A1 (es) |
Families Citing this family (3)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US8242158B1 (en) | 2012-01-04 | 2012-08-14 | Hospira, Inc. | Dexmedetomidine premix formulation |
WO2014033751A2 (en) * | 2012-08-16 | 2014-03-06 | Emcure Pharmaceuticals Limited | Pharmaceutical composition of propofol |
WO2017002117A1 (en) * | 2015-07-01 | 2017-01-05 | Yissum Research Development Company Of The Hebrew University Of Jerusalem Ltd | Delivery systems for propofol |
Family Cites Families (11)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
GB8912391D0 (en) * | 1989-05-30 | 1989-07-12 | Unilever Plc | Shampoo composition |
DE4039602A1 (de) * | 1990-12-12 | 1992-06-17 | Bauer Kurt Heinz Prof Dr | Pharmazeutische formulierungen |
US5962536A (en) * | 1998-07-31 | 1999-10-05 | Komer; Gene | Injectable propofol formulations |
CN1149984C (zh) * | 1999-06-21 | 2004-05-19 | 健一制药株式会社 | 用于静脉注射的含有普鲁泊福的麻醉组合物 |
KR20010055736A (ko) * | 1999-12-13 | 2001-07-04 | 이규현 | 프로포폴의 마이크로에멀젼 주사제 조성물 |
IN188917B (es) * | 2000-12-07 | 2002-11-23 | Bharat Surums & Vaccines Ltd | |
US20040220283A1 (en) * | 2002-07-29 | 2004-11-04 | Transform Pharmaceuticals, Inc. | Aqueous 2,6-diisopropylphenol pharmaceutical compositions |
NZ526347A (en) * | 2003-04-30 | 2005-07-29 | Parnell Lab Aust Pty Ltd | Formulations containing propofol for anaesthetic use |
US7326735B2 (en) * | 2003-04-30 | 2008-02-05 | Parnell Laboratories (Aust) Pty Limited | Formulations for anaesthetic use |
WO2005079758A1 (en) * | 2004-02-13 | 2005-09-01 | Bioavailability, Inc. | A microemulsion preparation of high concentration propofol for anesthetic uses |
MX2008001746A (es) * | 2005-08-05 | 2008-04-07 | Bharat Serums & Vaccines Ltd | Composiciones de emulsion de propofol intravenosas que tienen eficacia de conservacion. |
-
2006
- 2006-10-27 BR BRPI0604377-1A patent/BRPI0604377A/pt not_active Application Discontinuation
-
2007
- 2007-10-23 CN CN2007800427185A patent/CN101553215B/zh not_active Expired - Fee Related
- 2007-10-23 US US12/447,247 patent/US20100041769A1/en not_active Abandoned
- 2007-10-23 EP EP07815724.5A patent/EP2097073A4/en not_active Withdrawn
- 2007-10-23 WO PCT/BR2007/000283 patent/WO2008049178A1/en active Application Filing
- 2007-10-25 AR ARP070104732A patent/AR063397A1/es not_active Application Discontinuation
- 2007-10-25 CL CL200703075A patent/CL2007003075A1/es unknown
- 2007-10-30 UY UY30676A patent/UY30676A1/es not_active Application Discontinuation
-
2010
- 2010-02-18 HK HK10101737.4A patent/HK1135029A1/xx not_active IP Right Cessation
Also Published As
Publication number | Publication date |
---|---|
CN101553215A (zh) | 2009-10-07 |
CN101553215B (zh) | 2013-04-10 |
CL2007003075A1 (es) | 2008-03-14 |
WO2008049178A1 (en) | 2008-05-02 |
EP2097073A1 (en) | 2009-09-09 |
US20100041769A1 (en) | 2010-02-18 |
HK1135029A1 (en) | 2010-05-28 |
EP2097073A4 (en) | 2013-09-18 |
WO2008049178A8 (en) | 2008-06-12 |
AR063397A1 (es) | 2009-01-28 |
BRPI0604377A (pt) | 2008-06-24 |
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Legal Events
Date | Code | Title | Description |
---|---|---|---|
109 | Application deemed to be withdrawn |
Effective date: 20170727 |