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UY27324A1 - Nuevas sales de napsilato i - Google Patents

Nuevas sales de napsilato i

Info

Publication number
UY27324A1
UY27324A1 UY27324A UY27324A UY27324A1 UY 27324 A1 UY27324 A1 UY 27324A1 UY 27324 A UY27324 A UY 27324A UY 27324 A UY27324 A UY 27324A UY 27324 A1 UY27324 A1 UY 27324A1
Authority
UY
Uruguay
Prior art keywords
napsilate
salts
new
solvates
stereoisomers
Prior art date
Application number
UY27324A
Other languages
English (en)
Inventor
Taylor Lynne
Original Assignee
Astrazeneca Ab
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Astrazeneca Ab filed Critical Astrazeneca Ab
Publication of UY27324A1 publication Critical patent/UY27324A1/es

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07CACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C309/00Sulfonic acids; Halides, esters, or anhydrides thereof
    • C07C309/01Sulfonic acids
    • C07C309/28Sulfonic acids having sulfo groups bound to carbon atoms of six-membered aromatic rings of a carbon skeleton
    • C07C309/33Sulfonic acids having sulfo groups bound to carbon atoms of six-membered aromatic rings of a carbon skeleton of six-membered aromatic rings being part of condensed ring systems
    • C07C309/34Sulfonic acids having sulfo groups bound to carbon atoms of six-membered aromatic rings of a carbon skeleton of six-membered aromatic rings being part of condensed ring systems formed by two rings
    • C07C309/35Naphthalene sulfonic acids
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07FACYCLIC, CARBOCYCLIC OR HETEROCYCLIC COMPOUNDS CONTAINING ELEMENTS OTHER THAN CARBON, HYDROGEN, HALOGEN, OXYGEN, NITROGEN, SULFUR, SELENIUM OR TELLURIUM
    • C07F9/00Compounds containing elements of Groups 5 or 15 of the Periodic Table
    • C07F9/02Phosphorus compounds
    • C07F9/28Phosphorus compounds with one or more P—C bonds
    • C07F9/48Phosphonous acids [RP(OH)2] including [RHP(=O)(OH)]; Thiophosphonous acids including [RP(SH)2], [RHP(=S)(SH)]; Derivatives thereof
    • C07F9/4808Phosphonous acids [RP(OH)2] including [RHP(=O)(OH)]; Thiophosphonous acids including [RP(SH)2], [RHP(=S)(SH)]; Derivatives thereof the acid moiety containing a substituent or structure which is considered as characteristic
    • C07F9/4816Acyclic saturated acids or derivatices which can have further substituents on alkyl

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Biochemistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Molecular Biology (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)

Abstract

Novedosas sales napsilato de fórmula I, o solvatos de las mismas y estereoisómeros de las mismas, así como también un proceso para la preparación de los mismos, composiciones farmacéuticas que contienen la sal de napsilato terapéuticamente activa y el uso de los mencionados compuestos activos en tratamientos.
UY27324A 2001-06-08 2002-06-07 Nuevas sales de napsilato i UY27324A1 (es)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
SE0102057A SE0102057D0 (sv) 2001-06-08 2001-06-08 New Salts I

Publications (1)

Publication Number Publication Date
UY27324A1 true UY27324A1 (es) 2003-02-28

Family

ID=20284432

Family Applications (1)

Application Number Title Priority Date Filing Date
UY27324A UY27324A1 (es) 2001-06-08 2002-06-07 Nuevas sales de napsilato i

Country Status (3)

Country Link
SE (1) SE0102057D0 (es)
UY (1) UY27324A1 (es)
WO (1) WO2002100869A1 (es)

Families Citing this family (10)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US7494985B2 (en) 2004-11-03 2009-02-24 Xenoport, Inc. Acyloxyalkyl carbamate prodrugs, methods of synthesis, and use
US7566738B2 (en) 2004-11-03 2009-07-28 Xenoport, Inc. Acyloxyalkyl carbamate prodrugs of sulfinic acids, methods of synthesis, and use
WO2006071186A1 (en) * 2004-12-27 2006-07-06 Astrazeneca Ab Use of gabab receptor agonists
US20060160777A1 (en) * 2004-12-27 2006-07-20 Anders Lehmann New use of GABAbeta receptor agonists
US7585996B2 (en) 2006-09-15 2009-09-08 Xenoport, Inc. Acyloxyalkyl carbamate prodrugs, methods of synthesis and use
CN101743011A (zh) * 2007-07-25 2010-06-16 阿斯利康(瑞典)有限公司 (3-氨基-2-氟丙基)次膦酸用于治疗非糜烂性反流病的用途
EP2235026A4 (en) * 2007-12-21 2011-08-17 Astrazeneca Ab NEW PROCESS FOR THE PREPARATION OF (2R) - (3-AMINO-2-FLUORO-PROPYL) PHOSPHIC ACID FORM A
PE20091176A1 (es) * 2007-12-21 2009-09-03 Astrazeneca Ab Nueva forma cristalina c del acido (2r)-(3-amino-2-fluoropropil)fosfinico
WO2009082345A1 (en) * 2007-12-21 2009-07-02 Astrazeneca Ab Novel crystalline form b of (2r)-(3-amino-2-fluoropropyl)phosphinic acid
US20120016021A1 (en) 2010-07-15 2012-01-19 Xenoport, Inc. Methods of treating fragile x syndrome, down's syndrome, autism and related disorders

Family Cites Families (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
SE9603408D0 (sv) * 1996-09-18 1996-09-18 Astra Ab Medical use

Also Published As

Publication number Publication date
SE0102057D0 (sv) 2001-06-08
WO2002100869A1 (en) 2002-12-19

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Legal Events

Date Code Title Description
DESI Application deemed to be withdrawn

Effective date: 20111129