UY27324A1 - Nuevas sales de napsilato i - Google Patents
Nuevas sales de napsilato iInfo
- Publication number
- UY27324A1 UY27324A1 UY27324A UY27324A UY27324A1 UY 27324 A1 UY27324 A1 UY 27324A1 UY 27324 A UY27324 A UY 27324A UY 27324 A UY27324 A UY 27324A UY 27324 A1 UY27324 A1 UY 27324A1
- Authority
- UY
- Uruguay
- Prior art keywords
- napsilate
- salts
- new
- solvates
- stereoisomers
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C309/00—Sulfonic acids; Halides, esters, or anhydrides thereof
- C07C309/01—Sulfonic acids
- C07C309/28—Sulfonic acids having sulfo groups bound to carbon atoms of six-membered aromatic rings of a carbon skeleton
- C07C309/33—Sulfonic acids having sulfo groups bound to carbon atoms of six-membered aromatic rings of a carbon skeleton of six-membered aromatic rings being part of condensed ring systems
- C07C309/34—Sulfonic acids having sulfo groups bound to carbon atoms of six-membered aromatic rings of a carbon skeleton of six-membered aromatic rings being part of condensed ring systems formed by two rings
- C07C309/35—Naphthalene sulfonic acids
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07F—ACYCLIC, CARBOCYCLIC OR HETEROCYCLIC COMPOUNDS CONTAINING ELEMENTS OTHER THAN CARBON, HYDROGEN, HALOGEN, OXYGEN, NITROGEN, SULFUR, SELENIUM OR TELLURIUM
- C07F9/00—Compounds containing elements of Groups 5 or 15 of the Periodic Table
- C07F9/02—Phosphorus compounds
- C07F9/28—Phosphorus compounds with one or more P—C bonds
- C07F9/48—Phosphonous acids [RP(OH)2] including [RHP(=O)(OH)]; Thiophosphonous acids including [RP(SH)2], [RHP(=S)(SH)]; Derivatives thereof
- C07F9/4808—Phosphonous acids [RP(OH)2] including [RHP(=O)(OH)]; Thiophosphonous acids including [RP(SH)2], [RHP(=S)(SH)]; Derivatives thereof the acid moiety containing a substituent or structure which is considered as characteristic
- C07F9/4816—Acyclic saturated acids or derivatices which can have further substituents on alkyl
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Health & Medical Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
- Biochemistry (AREA)
- General Health & Medical Sciences (AREA)
- Molecular Biology (AREA)
- Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
- Nitrogen Condensed Heterocyclic Rings (AREA)
Abstract
Novedosas sales napsilato de fórmula I, o solvatos de las mismas y estereoisómeros de las mismas, así como también un proceso para la preparación de los mismos, composiciones farmacéuticas que contienen la sal de napsilato terapéuticamente activa y el uso de los mencionados compuestos activos en tratamientos.
Applications Claiming Priority (1)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
SE0102057A SE0102057D0 (sv) | 2001-06-08 | 2001-06-08 | New Salts I |
Publications (1)
Publication Number | Publication Date |
---|---|
UY27324A1 true UY27324A1 (es) | 2003-02-28 |
Family
ID=20284432
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
UY27324A UY27324A1 (es) | 2001-06-08 | 2002-06-07 | Nuevas sales de napsilato i |
Country Status (3)
Country | Link |
---|---|
SE (1) | SE0102057D0 (es) |
UY (1) | UY27324A1 (es) |
WO (1) | WO2002100869A1 (es) |
Families Citing this family (10)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US7494985B2 (en) | 2004-11-03 | 2009-02-24 | Xenoport, Inc. | Acyloxyalkyl carbamate prodrugs, methods of synthesis, and use |
US7566738B2 (en) | 2004-11-03 | 2009-07-28 | Xenoport, Inc. | Acyloxyalkyl carbamate prodrugs of sulfinic acids, methods of synthesis, and use |
WO2006071186A1 (en) * | 2004-12-27 | 2006-07-06 | Astrazeneca Ab | Use of gabab receptor agonists |
US20060160777A1 (en) * | 2004-12-27 | 2006-07-20 | Anders Lehmann | New use of GABAbeta receptor agonists |
US7585996B2 (en) | 2006-09-15 | 2009-09-08 | Xenoport, Inc. | Acyloxyalkyl carbamate prodrugs, methods of synthesis and use |
CN101743011A (zh) * | 2007-07-25 | 2010-06-16 | 阿斯利康(瑞典)有限公司 | (3-氨基-2-氟丙基)次膦酸用于治疗非糜烂性反流病的用途 |
EP2235026A4 (en) * | 2007-12-21 | 2011-08-17 | Astrazeneca Ab | NEW PROCESS FOR THE PREPARATION OF (2R) - (3-AMINO-2-FLUORO-PROPYL) PHOSPHIC ACID FORM A |
PE20091176A1 (es) * | 2007-12-21 | 2009-09-03 | Astrazeneca Ab | Nueva forma cristalina c del acido (2r)-(3-amino-2-fluoropropil)fosfinico |
WO2009082345A1 (en) * | 2007-12-21 | 2009-07-02 | Astrazeneca Ab | Novel crystalline form b of (2r)-(3-amino-2-fluoropropyl)phosphinic acid |
US20120016021A1 (en) | 2010-07-15 | 2012-01-19 | Xenoport, Inc. | Methods of treating fragile x syndrome, down's syndrome, autism and related disorders |
Family Cites Families (1)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
SE9603408D0 (sv) * | 1996-09-18 | 1996-09-18 | Astra Ab | Medical use |
-
2001
- 2001-06-08 SE SE0102057A patent/SE0102057D0/xx unknown
-
2002
- 2002-06-04 WO PCT/SE2002/001083 patent/WO2002100869A1/en not_active Application Discontinuation
- 2002-06-07 UY UY27324A patent/UY27324A1/es unknown
Also Published As
Publication number | Publication date |
---|---|
SE0102057D0 (sv) | 2001-06-08 |
WO2002100869A1 (en) | 2002-12-19 |
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Legal Events
Date | Code | Title | Description |
---|---|---|---|
DESI | Application deemed to be withdrawn |
Effective date: 20111129 |