TR200604349A2 - Aripiprazol içeren farmasötik bileşimler - Google Patents
Aripiprazol içeren farmasötik bileşimlerInfo
- Publication number
- TR200604349A2 TR200604349A2 TR2006/04349A TR200604349A TR200604349A2 TR 200604349 A2 TR200604349 A2 TR 200604349A2 TR 2006/04349 A TR2006/04349 A TR 2006/04349A TR 200604349 A TR200604349 A TR 200604349A TR 200604349 A2 TR200604349 A2 TR 200604349A2
- Authority
- TR
- Turkey
- Prior art keywords
- pharmaceutical compositions
- compositions containing
- aripiprazole
- containing aripiprazole
- disintegrant
- Prior art date
Links
- CEUORZQYGODEFX-UHFFFAOYSA-N Aripirazole Chemical compound ClC1=CC=CC(N2CCN(CCCCOC=3C=C4NC(=O)CCC4=CC=3)CC2)=C1Cl CEUORZQYGODEFX-UHFFFAOYSA-N 0.000 title abstract 3
- 229960004372 aripiprazole Drugs 0.000 title abstract 3
- 239000008194 pharmaceutical composition Substances 0.000 title 1
- 239000013543 active substance Substances 0.000 abstract 1
- 239000011230 binding agent Substances 0.000 abstract 1
- 239000007884 disintegrant Substances 0.000 abstract 1
- 238000004090 dissolution Methods 0.000 abstract 1
- 239000000945 filler Substances 0.000 abstract 1
- 239000000314 lubricant Substances 0.000 abstract 1
- 239000000546 pharmaceutical excipient Substances 0.000 abstract 1
- 150000003839 salts Chemical class 0.000 abstract 1
- 239000007916 tablet composition Substances 0.000 abstract 1
Classifications
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
- A61K31/47—Quinolines; Isoquinolines
- A61K31/4704—2-Quinolinones, e.g. carbostyril
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
- A61K31/496—Non-condensed piperazines containing further heterocyclic rings, e.g. rifampin, thiothixene or sparfloxacin
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/20—Pills, tablets, discs, rods
- A61K9/2004—Excipients; Inactive ingredients
- A61K9/2013—Organic compounds, e.g. phospholipids, fats
- A61K9/2018—Sugars, or sugar alcohols, e.g. lactose, mannitol; Derivatives thereof, e.g. polysorbates
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/18—Antipsychotics, i.e. neuroleptics; Drugs for mania or schizophrenia
Landscapes
- Health & Medical Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
- Pharmacology & Pharmacy (AREA)
- Veterinary Medicine (AREA)
- Public Health (AREA)
- Chemical & Material Sciences (AREA)
- General Health & Medical Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- Medicinal Chemistry (AREA)
- Epidemiology (AREA)
- Engineering & Computer Science (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Neurosurgery (AREA)
- Organic Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- General Chemical & Material Sciences (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Neurology (AREA)
- Biomedical Technology (AREA)
- Psychiatry (AREA)
- Biophysics (AREA)
- Molecular Biology (AREA)
- Medicinal Preparation (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Abstract
Buluş konusu uygun dissolüsyon ve stabilite değerlerine sahip aripiprazol tablet formülasyonu, aripiprazol etken maddesini veya farmasötik açıdan uygun bir tuzunu ve yardımcı madde olarak en az bir dolgu maddesini, en az bir dağıtıcıyı, en az bir bağlayıcıyı ve en az bir kaydırıcı içermektedir.
Priority Applications (3)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
TR2006/04349A TR200604349A2 (tr) | 2006-08-15 | 2006-08-15 | Aripiprazol içeren farmasötik bileşimler |
PCT/TR2007/000076 WO2008020820A2 (en) | 2006-08-15 | 2007-08-15 | Pharmaceutical compositions comprising aripiprazole |
EP07835588.0A EP2051694B1 (en) | 2006-08-15 | 2007-08-15 | Pharmaceutical compositions comprising aripiprazole |
Applications Claiming Priority (1)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
TR2006/04349A TR200604349A2 (tr) | 2006-08-15 | 2006-08-15 | Aripiprazol içeren farmasötik bileşimler |
Publications (1)
Publication Number | Publication Date |
---|---|
TR200604349A2 true TR200604349A2 (tr) | 2008-03-21 |
Family
ID=39082470
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
TR2006/04349A TR200604349A2 (tr) | 2006-08-15 | 2006-08-15 | Aripiprazol içeren farmasötik bileşimler |
Country Status (3)
Country | Link |
---|---|
EP (1) | EP2051694B1 (tr) |
TR (1) | TR200604349A2 (tr) |
WO (1) | WO2008020820A2 (tr) |
Families Citing this family (12)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US7799790B2 (en) | 2006-07-20 | 2010-09-21 | Helm Ag | Amorphous aripiprazole and process for the preparation thereof |
EP1880714A1 (en) | 2006-07-20 | 2008-01-23 | Helm AG | Amorphous Aripiprazole and Process for the Preparation thereof |
TR201000948A1 (tr) * | 2010-02-09 | 2011-08-22 | Sanovel İlaç San.Ve Ti̇c.A.Ş. | Aripiprazol formülasyonları. |
WO2013100878A1 (en) * | 2011-12-27 | 2013-07-04 | Mahmut Bilgic | Pharmaceutical formulations comprising aripiprazole |
WO2014104989A1 (en) * | 2011-12-27 | 2014-07-03 | Mahmut Bilgic | Pharmaceutical compositions comprising aripiprazole |
WO2013175508A2 (en) * | 2012-05-24 | 2013-11-28 | Medreich Limited | Stable pharmaceutical composition of aripiprazole |
GR1008186B (el) | 2013-04-22 | 2014-05-08 | "Φαρματεν Α.Β.Ε.Ε.", | Φαρμακευτικο σκευασμα περιεχον ενα ατυπο αντιψυχωσικο παραγοντα και μεθοδος για την παρασκευη αυτου |
US9051268B2 (en) | 2013-04-30 | 2015-06-09 | Otsuka Pharmaceutical Co., Ltd. | Oral solid preparation comprising aripiprazole and method for producing oral solid preparation comprising aripiprazole |
EP2838513B1 (en) * | 2013-04-30 | 2017-04-05 | Otsuka Pharmaceutical Co., Ltd. | Oral solid preparation comprising aripiprazole and method for producing oral solid preparation comprising aripiprazole |
US20150093441A1 (en) * | 2013-09-30 | 2015-04-02 | Otsuka Pharmaceutical Co., Ltd | Oral solid preparation comprising aripiprazole and method for producing oral solid preparation comprising aripiprazole |
GR1008442B (el) | 2014-01-16 | 2015-03-05 | "Φαρματεν Α.Β.Ε.Ε.", | Φαρμακευτικο σκευασμα περιεχον αριπιπραζολη ή αλας αυτης |
WO2016189504A1 (en) * | 2015-05-28 | 2016-12-01 | Leiutis Pharmaceuticals Pvt Ltd | Non-lyophilized compositions of aripiprazole and methods of preparation thereof |
Family Cites Families (9)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US5006528A (en) | 1988-10-31 | 1991-04-09 | Otsuka Pharmaceutical Co., Ltd. | Carbostyril derivatives |
WO2003030868A1 (en) | 2001-10-09 | 2003-04-17 | Bristol-Myers Squibb Company | Flashmelt oral dosage formulation |
AR033485A1 (es) | 2001-09-25 | 2003-12-26 | Otsuka Pharma Co Ltd | Sustancia medicinal de aripiprazol de baja higroscopicidad y proceso para la preparacion de la misma |
TWI324074B (en) * | 2001-10-09 | 2010-05-01 | Bristol Myers Squibb Co | Flashmelt oral dosage formulation |
NZ546063A (en) * | 2003-10-23 | 2009-05-31 | Otsuka Pharma Co Ltd | Controlled release sterile injectable aripiprazole (7-{4-[4-(2,3-dichlorophenyl)-1-piperazinyl]-butoxy]-3,4-dihydro-2(1H)-quinolinone) formulation and method |
CN100336509C (zh) | 2004-06-18 | 2007-09-12 | 成都康弘科技实业(集团)有限公司 | 阿立哌唑的口腔崩解片制剂及其制备方法 |
WO2006097344A1 (en) | 2005-03-17 | 2006-09-21 | Synthon B.V. | Pharmaceutical tablets of crystalline type ii aripiprazole |
EP2036545A1 (en) | 2006-01-05 | 2009-03-18 | Teva Pharmaceutical Industries Ltd. | Aripiprazole tablets |
JP2008531738A (ja) | 2006-01-05 | 2008-08-14 | テバ ファーマシューティカル インダストリーズ リミティド | アリピプラゾールの乾燥製剤 |
-
2006
- 2006-08-15 TR TR2006/04349A patent/TR200604349A2/tr unknown
-
2007
- 2007-08-15 EP EP07835588.0A patent/EP2051694B1/en not_active Revoked
- 2007-08-15 WO PCT/TR2007/000076 patent/WO2008020820A2/en active Application Filing
Also Published As
Publication number | Publication date |
---|---|
WO2008020820A3 (en) | 2008-05-29 |
EP2051694A2 (en) | 2009-04-29 |
WO2008020820A2 (en) | 2008-02-21 |
EP2051694B1 (en) | 2017-10-18 |
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